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Found 2726 with Last Name = 'luo' and Initial = 'j'
TargetSomatostatin receptor type 2(RAT)
University Of Cambridge

Curated by PDSP Ki Database
LigandPNGBDBM81767(15-28-Somatostatin-28 | CAS_38916-34-6 | CB6417646...)
Affinity DataKi:  0.0410nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 2(Homo sapiens (Human))
University Of Cambridge

Curated by PDSP Ki Database
LigandPNGBDBM81767(15-28-Somatostatin-28 | CAS_38916-34-6 | CB6417646...)
Affinity DataKi:  0.0680nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 2(RAT)
University Of Cambridge

Curated by PDSP Ki Database
LigandPNGBDBM81767(15-28-Somatostatin-28 | CAS_38916-34-6 | CB6417646...)
Affinity DataKi:  0.0680nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 5(Homo sapiens (Human))
University Of Cambridge

Curated by PDSP Ki Database
LigandPNGBDBM81767(15-28-Somatostatin-28 | CAS_38916-34-6 | CB6417646...)
Affinity DataKi:  0.320nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Homo sapiens (Human))
University Of Helsinki

Curated by ChEMBL
LigandPNGBDBM50258529(CHEMBL449158 | bryostatin 1)
Affinity DataKi:  0.440nMAssay Description:Displacement of [3H]PDBu from human recombinant PKCdelta expressed in Sf9 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 1(Homo sapiens (Human))
University Of Cambridge

Curated by PDSP Ki Database
LigandPNGBDBM81767(15-28-Somatostatin-28 | CAS_38916-34-6 | CB6417646...)
Affinity DataKi:  0.560nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 3(Homo sapiens (Human))
University Of Cambridge

Curated by PDSP Ki Database
LigandPNGBDBM81767(15-28-Somatostatin-28 | CAS_38916-34-6 | CB6417646...)
Affinity DataKi:  0.620nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
National University Of Singapore

Curated by ChEMBL
LigandPNGBDBM50252860((S)-N-((S)-1,6-diamino-1-oxohexan-2-yl)-1-((S)-5-g...)
Affinity DataKi:  0.823nMAssay Description:Displacement of [3H]U69593 from kappa opioid receptor in guinea pig brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
National University Of Singapore

Curated by ChEMBL
LigandPNGBDBM50252855((4S,7S,13S)-13-[(S)-3-(4-Carbamoyl-2,6-dimethyl-ph...)
Affinity DataKi:  1.02nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 4(Homo sapiens (Human))
University Of Cambridge

Curated by PDSP Ki Database
LigandPNGBDBM81767(15-28-Somatostatin-28 | CAS_38916-34-6 | CB6417646...)
Affinity DataKi:  1.20nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein ENL(Homo sapiens)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50459745(CHEMBL4210431)
Affinity DataKi:  1.40nMAssay Description:Binding affinity to MBP-tagged human recombinant ENL (489 to 559 residues) incubated for 40 mins by measuring fluorescence polarization by microplate...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetMu-type opioid receptor(GUINEA PIG)
National University Of Singapore

Curated by ChEMBL
LigandPNGBDBM50252864(CHEMBL454035 | antanal 2)
Affinity DataKi:  1.52nMAssay Description:Antagonist activity against mu opioid receptor in guinea pig ileum assessed as effect on TAPP-induced responseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
National University Of Singapore

Curated by ChEMBL
LigandPNGBDBM50252856((4S,7S,13S)-13-[(S)-3-(4-Hydroxy-2,6-dimethyl-phen...)
Affinity DataKi:  2.23nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
National University Of Singapore

Curated by ChEMBL
LigandPNGBDBM50252858((S)-2-({(4R,7S,13S)-7-(4-Fluoro-benzyl)-13-[(S)-3-...)
Affinity DataKi:  2.32nMAssay Description:Displacement of [3H]DSLET from delta opioid receptor in rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
National University Of Singapore

Curated by ChEMBL
LigandPNGBDBM50252863(CHEMBL507442 | antanal 1)
Affinity DataKi:  2.38nMAssay Description:Antagonist activity against mu opioid receptor in guinea pig ileum assessed as effect on TAPP-induced responseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 2(Homo sapiens (Human))
University Of Cambridge

Curated by PDSP Ki Database
LigandPNGBDBM85671(CAS_183658-72-2 | CYN 154806 | CYN-154806)
Affinity DataKi:  2.63nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
National University Of Singapore

Curated by ChEMBL
LigandPNGBDBM50252857((S)-2-{[(4R,7S,13S)-13-[(S)-3-(4-Carbamoyl-2,6-dim...)
Affinity DataKi:  2.92nMAssay Description:Displacement of [3H]DSLET from delta opioid receptor in rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein ENL(Homo sapiens)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50606137(CHEMBL5187921)
Affinity DataKi:  3.40nMAssay Description:Binding affinity to MBP-tagged human recombinant ENL (489 to 559 residues) incubated for 40 mins by measuring fluorescence polarization by microplate...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
National University Of Singapore

Curated by ChEMBL
LigandPNGBDBM50252856((4S,7S,13S)-13-[(S)-3-(4-Hydroxy-2,6-dimethyl-phen...)
Affinity DataKi:  3.61nMAssay Description:Displacement of [3H]DSLET from delta opioid receptor in rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
University Of Helsinki

Curated by ChEMBL
LigandPNGBDBM50000092((-)-(etorphine) | (-)-morphine | (1S,5R,13R,14S)-1...)
Affinity DataKi:  4nMAssay Description:Displacement of [3H]diprenorphine from human MOR expressed in African green monkey COS1 cell membranes incubated for 1 hr by scintillation counting m...More data for this Ligand-Target Pair
TargetSomatostatin receptor type 2(RAT)
University Of Cambridge

Curated by PDSP Ki Database
LigandPNGBDBM85671(CAS_183658-72-2 | CYN 154806 | CYN-154806)
Affinity DataKi:  4.47nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
National University Of Singapore

Curated by ChEMBL
LigandPNGBDBM50252864(CHEMBL454035 | antanal 2)
Affinity DataKi:  7.74nMAssay Description:Antagonist activity against delta opioid receptor in mouse vas deference assessed as effect on DPDPE-induced responseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 2(RAT)
University Of Cambridge

Curated by PDSP Ki Database
LigandPNGBDBM85671(CAS_183658-72-2 | CYN 154806 | CYN-154806)
Affinity DataKi:  7.94nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein AF-9(Homo sapiens)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50606139(CHEMBL5198951)
Affinity DataKi:  9nMAssay Description:Binding affinity to MBP-tagged human recombinant AF9 (487 to 568 residues) incubated for 40 mins by measuring fluorescence polarization by microplate...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetProtein AF-9(Homo sapiens)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50606141(CHEMBL5187149)
Affinity DataKi:  9nMAssay Description:Binding affinity to MBP-tagged human recombinant AF9 (487 to 568 residues) incubated for 40 mins by measuring fluorescence polarization by microplate...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetProtein AF-9(Homo sapiens)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50606142(CHEMBL5197715)
Affinity DataKi:  13nMAssay Description:Binding affinity to MBP-tagged human recombinant AF9 (487 to 568 residues) incubated for 40 mins by measuring fluorescence polarization by microplate...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetProtein AF-9(Homo sapiens)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50606140(CHEMBL5184570)
Affinity DataKi:  15nMAssay Description:Binding affinity to MBP-tagged human recombinant AF9 (487 to 568 residues) incubated for 40 mins by measuring fluorescence polarization by microplate...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetMu-type opioid receptor(GUINEA PIG)
National University Of Singapore

Curated by ChEMBL
LigandPNGBDBM50252862((5S,8S,14R)-8-Benzyl-14-[(S)-2-[3-(4-hydroxy-2,6-d...)
Affinity DataKi:  15.5nMAssay Description:Antagonist activity against mu opioid receptor in guinea pig ileum assessed as effect on TAPP-induced responseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein AF-9(Homo sapiens)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50606146(CHEMBL5206253)
Affinity DataKi:  17nMAssay Description:Binding affinity to MBP-tagged human recombinant AF9 (487 to 568 residues) incubated for 40 mins by measuring fluorescence polarization by microplate...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetDelta-type opioid receptor(MOUSE)
National University Of Singapore

Curated by ChEMBL
LigandPNGBDBM50252863(CHEMBL507442 | antanal 1)
Affinity DataKi:  17.4nMAssay Description:Antagonist activity against delta opioid receptor in mouse vas deference assessed as effect on DPDPE-induced responseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUDP-glucuronosyltransferase 2B7(Homo sapiens (Human))
University Of Helsinki

Curated by ChEMBL
LigandPNGBDBM50211740((1R)-phenyl-[(1R,2S,7S,8S,9S)-3,3,7-trimethyltricy...)
Affinity DataKi:  18.4nMAssay Description:Inhibition of human UGT2B7 assessed as reduction of estriol glucuronidationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
National University Of Singapore

Curated by ChEMBL
LigandPNGBDBM50252855((4S,7S,13S)-13-[(S)-3-(4-Carbamoyl-2,6-dimethyl-ph...)
Affinity DataKi:  19nMAssay Description:Displacement of [3H]DSLET from delta opioid receptor in rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein AF-9(Homo sapiens)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50606144(CHEMBL5199592)
Affinity DataKi:  19nMAssay Description:Binding affinity to MBP-tagged human recombinant AF9 (487 to 568 residues) incubated for 40 mins by measuring fluorescence polarization by microplate...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetProtein AF-9(Homo sapiens)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50606147(CHEMBL5203898)
Affinity DataKi:  22nMAssay Description:Binding affinity to MBP-tagged human recombinant AF9 (487 to 568 residues) incubated for 40 mins by measuring fluorescence polarization by microplate...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetProtein AF-9(Homo sapiens)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50459730(CHEMBL4211714)
Affinity DataKi:  23nMAssay Description:Binding affinity to MBP-tagged human recombinant AF9 (487 to 568 residues) incubated for 40 mins by measuring fluorescence polarization by microplate...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetProtein AF-9(Homo sapiens)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50606143(CHEMBL5208460)
Affinity DataKi:  23nMAssay Description:Binding affinity to MBP-tagged human recombinant AF9 (487 to 568 residues) incubated for 40 mins by measuring fluorescence polarization by microplate...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
National University Of Singapore

Curated by ChEMBL
LigandPNGBDBM50252859((S)-1-((S)-2-((2S,3S)-2-((S)-2-((S)-2-((S)-2-((S)-...)
Affinity DataKi:  26nMAssay Description:Displacement of [3H]U69593 from kappa opioid receptor in guinea pig brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
National University Of Singapore

Curated by ChEMBL
LigandPNGBDBM50252859((S)-1-((S)-2-((2S,3S)-2-((S)-2-((S)-2-((S)-2-((S)-...)
Affinity DataKi:  27.2nMAssay Description:Displacement of [3H]DSLET from delta opioid receptor in rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein AF-9(Homo sapiens)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50606145(CHEMBL5190103)
Affinity DataKi:  29nMAssay Description:Binding affinity to MBP-tagged human recombinant AF9 (487 to 568 residues) incubated for 40 mins by measuring fluorescence polarization by microplate...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
National University Of Singapore

Curated by ChEMBL
LigandPNGBDBM50252859((S)-1-((S)-2-((2S,3S)-2-((S)-2-((S)-2-((S)-2-((S)-...)
Affinity DataKi:  29.6nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein AF-9(Homo sapiens)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50606138(CHEMBL5207031)
Affinity DataKi:  32nMAssay Description:Binding affinity to MBP-tagged human recombinant AF9 (487 to 568 residues) incubated for 40 mins by measuring fluorescence polarization by microplate...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
University Of Helsinki

Curated by ChEMBL
LigandPNGBDBM50015677((S)-1-hydroxymethyl-2-octanoyloxy-ethyl ester | 1,...)
Affinity DataKi:  40nMAssay Description:Displacement of [3H]PDBu from human recombinant PKCalpha expressed in Sf9 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit alpha(Homo sapiens (Human))
University Of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50257823(CHEMBL4089551)
Affinity DataKi:  80nMAssay Description:Inhibition of recombinant human N-terminal GST-tagged IKKalpha (1 to 745 residues) expressed in baculovirus expression system using biotinylated IkBa...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
National University Of Singapore

Curated by ChEMBL
LigandPNGBDBM50252856((4S,7S,13S)-13-[(S)-3-(4-Hydroxy-2,6-dimethyl-phen...)
Affinity DataKi:  92.8nMAssay Description:Displacement of [3H]U69593 from kappa opioid receptor in guinea pig brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
University Of Strathclyde

Curated by ChEMBL
LigandPNGBDBM50257884(CHEMBL4065551)
Affinity DataKi:  100nMAssay Description:Inhibition of recombinant full length human IKKbeta expressed in baculovirus infected sf9 insect cells using biotinylated IkBalpha as substrate after...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein ENL(Homo sapiens)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50606139(CHEMBL5198951)
Affinity DataKi:  109nMAssay Description:Binding affinity to MBP-tagged human recombinant ENL (489 to 559 residues) incubated for 40 mins by measuring fluorescence polarization by microplate...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetProtein ENL(Homo sapiens)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50606141(CHEMBL5187149)
Affinity DataKi:  112nMAssay Description:Binding affinity to MBP-tagged human recombinant ENL (489 to 559 residues) incubated for 40 mins by measuring fluorescence polarization by microplate...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetProtein ENL(Homo sapiens)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50606142(CHEMBL5197715)
Affinity DataKi:  157nMAssay Description:Binding affinity to MBP-tagged human recombinant ENL (489 to 559 residues) incubated for 40 mins by measuring fluorescence polarization by microplate...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetProtein AF-9(Homo sapiens)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50459745(CHEMBL4210431)
Affinity DataKi:  160nMAssay Description:Binding affinity to MBP-tagged human recombinant AF9 (487 to 568 residues) incubated for 40 mins by measuring fluorescence polarization by microplate...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetProtein AF-9(Homo sapiens)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50606137(CHEMBL5187921)
Affinity DataKi:  160nMAssay Description:Binding affinity to MBP-tagged human recombinant AF9 (487 to 568 residues) incubated for 40 mins by measuring fluorescence polarization by microplate...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
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