Affinity DataKi: 4nMAssay Description:Affinity for Dopamine receptor D2 using [3H]YM-09151-2 was carried out on bovine retinal membrane preparations (high-affinity)More data for this Ligand-Target Pair
Affinity DataKi: 4nMAssay Description:Affinity for Dopamine receptor D2 using [3H]YM-09151-2 was carried out on bovine retinal membrane preparations (high-affinity)More data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor [16-465]/Alpha-2B adrenergic receptor/Alpha-2C adrenergic receptor(RAT)
Universit£
Curated by ChEMBL
Universit£
Curated by ChEMBL
Affinity DataKi: 4.80nMAssay Description:Compound was evaluated for alpha adrenergic binding affinity towards Alpha-2 adrenergic receptor of rat brainMore data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor [16-465]/Alpha-2B adrenergic receptor/Alpha-2C adrenergic receptor(RAT)
Universit£
Curated by ChEMBL
Universit£
Curated by ChEMBL
Affinity DataKi: 4.80nMAssay Description:Tested for binding affinity against alpha-2 adrenergic receptor in rat brain using [3H]- rauwolscine as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 5nMAssay Description:Affinity for Dopamine receptor D2 using [3H]YM-09151-2 was carried out on bovine retinal membrane preparations (high-affinity)More data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor [16-465]/Alpha-2B adrenergic receptor/Alpha-2C adrenergic receptor(RAT)
Universit£
Curated by ChEMBL
Universit£
Curated by ChEMBL
Affinity DataKi: 7.40nMAssay Description:Tested for binding affinity against alpha-2 adrenergic receptor in rat brain using [3H]- rauwolscine as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 9nMAssay Description:Binding affinity towards cloned human Dopamine receptor D4More data for this Ligand-Target Pair
Affinity DataKi: 15nMAssay Description:Inhibition of [3H]YM-09151-2 binding to bovine retina membrane Dopamine receptor D2, high affinity siteMore data for this Ligand-Target Pair
Affinity DataKi: 19nMAssay Description:Inhibition of [3H]YM-09151-2 binding to bovine retina membrane Dopamine receptor D2, high affinity siteMore data for this Ligand-Target Pair
Affinity DataKi: 25nMAssay Description:Affinity for Dopamine receptor D2 using [3H]YM-09151-2 was carried out on bovine retinal membrane preparations (high-affinity)More data for this Ligand-Target Pair
Affinity DataKi: 26nMAssay Description:Affinity for Dopamine receptor D2 using [3H]YM-09151-2 was carried out on bovine retinal membrane preparations (high-affinity)More data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor [16-465]/Alpha-2B adrenergic receptor/Alpha-2C adrenergic receptor(RAT)
Universit£
Curated by ChEMBL
Universit£
Curated by ChEMBL
Affinity DataKi: 26nMAssay Description:Compound was evaluated for alpha adrenergic binding affinity towards Alpha-2 adrenergic receptor of rat brainMore data for this Ligand-Target Pair
Affinity DataKi: 27nMAssay Description:Affinity for Dopamine receptor D2 using [3H]YM-09151-2 was carried out on bovine retinal membrane preparations (high-affinity)More data for this Ligand-Target Pair
Affinity DataKi: 39nMAssay Description:Affinity for Dopamine receptor D2 using [3H]YM-09151-2 was carried out on bovine retinal membrane preparations (high-affinity)More data for this Ligand-Target Pair
Affinity DataKi: 42nMAssay Description:Affinity for Dopamine receptor D2 using [3H]YM-09151-2 was carried out on bovine retinal membrane preparations (high-affinity)More data for this Ligand-Target Pair
Affinity DataKi: 43nMAssay Description:Inhibition of [3H]YM-09151-2 binding to bovine retina membrane Dopamine receptor D2, high affinity siteMore data for this Ligand-Target Pair
Affinity DataKi: 44nMAssay Description:Affinity for Dopamine receptor D2 using [3H]YM-09151-2 was carried out on bovine retinal membrane preparations (high-affinity)More data for this Ligand-Target Pair
Affinity DataKi: 51nMAssay Description:Binding affinity against beta1-adrenergic receptor in rat brainMore data for this Ligand-Target Pair
Affinity DataKi: 52nMAssay Description:Inhibition of [3H]YM-09151-2 binding to bovine retina membrane Dopamine receptor D2, high affinity siteMore data for this Ligand-Target Pair
Affinity DataKi: 59nMAssay Description:Inhibition of [3H]YM-09151-2 binding to bovine retina membrane Dopamine receptor D2, high affinity siteMore data for this Ligand-Target Pair
Affinity DataKi: 62nMAssay Description:Compound was evaluated for beta adrenergic binding affinity towards Beta-2 adrenergic receptor of bovine lungMore data for this Ligand-Target Pair
Affinity DataKi: 75nMAssay Description:Inhibition of [3H]YM-09151-2 binding to bovine retina membrane Dopamine receptor D2, high affinity siteMore data for this Ligand-Target Pair
Affinity DataKi: 80nMAssay Description:Compound was evaluated for beta adrenergic binding affinity towards Beta-1 adrenergic receptor of rat brainMore data for this Ligand-Target Pair
Affinity DataKi: 80nMAssay Description:Tested for binding affinity against beta-1 adrenergic receptor in rat brain using [3H]-CGP- 26505 as radioligandMore data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor [16-465]/Alpha-2B adrenergic receptor/Alpha-2C adrenergic receptor(RAT)
Universit£
Curated by ChEMBL
Universit£
Curated by ChEMBL
Affinity DataKi: 90nMAssay Description:Binding affinity towards Alpha-2 adrenergic receptor of rat brainMore data for this Ligand-Target Pair
Affinity DataKi: 110nMAssay Description:Compound was evaluated for beta adrenergic binding affinity towards beta-2 receptor of bovine lungMore data for this Ligand-Target Pair
Affinity DataKi: 110nMAssay Description:Tested for binding affinity against beta-2 adrenergic receptor in bovine lung using [3H]DHA as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 120nMAssay Description:Compound was evaluated for beta adrenergic binding affinity towards beta-2 receptor of bovine lungMore data for this Ligand-Target Pair
Affinity DataKi: 126nMAssay Description:Compound was evaluated for beta adrenergic binding affinity towards Beta-1 adrenergic receptor of rat brainMore data for this Ligand-Target Pair
Affinity DataKi: 126nMAssay Description:Tested for binding affinity against beta-1 adrenergic receptor in rat brain using [3H]-CGP- 26505 as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 140nMAssay Description:Binding afinity against beta2-adrenergic receptor in bovine lungMore data for this Ligand-Target Pair
Affinity DataKi: 140nMAssay Description:Inhibition of [3H]YM-09151-2 binding to bovine retina membrane Dopamine receptor D2, high affinity siteMore data for this Ligand-Target Pair
Affinity DataKi: 156nMAssay Description:Inhibition of [3H]YM-09151-2 binding to bovine retina membrane Dopamine receptor D2, high affinity siteMore data for this Ligand-Target Pair
Affinity DataKi: 240nMAssay Description:Inhibition of [3H]YM-09151-2 binding to bovine retina membrane Dopamine receptor D2, high affinity siteMore data for this Ligand-Target Pair
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Universit£
Curated by ChEMBL
Universit£
Curated by ChEMBL
Affinity DataKi: 300nMAssay Description:Binding affinity towards Alpha-1 adrenergic receptor of rat brainMore data for this Ligand-Target Pair
Affinity DataKi: 420nMAssay Description:Affinity for Dopamine receptor D2 using [3H]-YM-09151-2 was carried out on bovine striatal membrane preparationsMore data for this Ligand-Target Pair
Affinity DataKi: 449nMAssay Description:Affinity for Dopamine receptor D2 using [3H]YM-09151-2 was carried out on bovine retinal membrane preparations (high-affinity)More data for this Ligand-Target Pair
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Universit£
Curated by ChEMBL
Universit£
Curated by ChEMBL
Affinity DataKi: 450nMAssay Description:Binding affinity towards Alpha-1 adrenergic receptor of rat brainMore data for this Ligand-Target Pair
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Universit£
Curated by ChEMBL
Universit£
Curated by ChEMBL
Affinity DataKi: 450nMAssay Description:Tested for binding affinity against alpha-1 adrenergic receptor in rat brain using [3H]-Prazosin as radioligandMore data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor [16-465]/Alpha-2B adrenergic receptor/Alpha-2C adrenergic receptor(RAT)
Universit£
Curated by ChEMBL
Universit£
Curated by ChEMBL
Affinity DataKi: 500nMAssay Description:Compound was evaluated for alpha adrenergic binding affinity towards Alpha-2 adrenergic receptor of rat brainMore data for this Ligand-Target Pair
Affinity DataKi: 500nMAssay Description:Binding affinity against beta1-adrenergic receptor in rat brainMore data for this Ligand-Target Pair
Affinity DataKi: 530nMAssay Description:Inhibition of [3H]YM-09151-2 binding to bovine retina membrane Dopamine receptor D2, high affinity siteMore data for this Ligand-Target Pair
Affinity DataKi: 540nMAssay Description:Inhibition of [3H]YM-09151-2 binding to bovine retina membrane Dopamine receptor D2, high affinity siteMore data for this Ligand-Target Pair
Affinity DataKi: 617nMAssay Description:Tested for binding affinity against Dopamine receptor D2 like from bovine striatum membranes by using [3H]YM-09151-2 radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 720nMAssay Description:Inhibition of [3H]YM-09151-2 binding to bovine retina membrane Dopamine receptor D2, high affinity siteMore data for this Ligand-Target Pair
Affinity DataKi: 760nMAssay Description:Binding affinity against beta1-adrenergic receptor in rat brainMore data for this Ligand-Target Pair
Affinity DataKi: 760nMAssay Description:Compound was evaluated for beta adrenergic binding affinity towards Beta-1 adrenergic receptor of rat brainMore data for this Ligand-Target Pair
Affinity DataKi: 850nMAssay Description:Binding afinity against beta2-adrenergic receptor in bovine lungMore data for this Ligand-Target Pair
Affinity DataKi: 850nMAssay Description:Binding affinity against beta1-adrenergic receptor in rat brainMore data for this Ligand-Target Pair
Affinity DataKi: 1.04E+3nMAssay Description:Binding affinity against beta1-adrenergic receptor in rat brainMore data for this Ligand-Target Pair