BindingDB PrimarySearch_ki

Found 818 with Last Name = 'mao' and Initial = 'q'

Xanthine dehydrogenase/oxidase(Homo sapiens (Human))
Shenyang Pharmaceutical University

Curated by ChEMBL

PNG

BDBM50320491(2-(3-CYANO-4-ISOBUTOXY-PHENYL)-4-METHYL-5-THIAZOLE...)

Ki: 0.100nMAssay Description:Mixed-type inhibition of xanthine oxidase (unknown origin) assessed as inhibitory constant of enzyme-substrate complex using xanthine as substrate at...More data for this Ligand-Target Pair

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3D Structure (crystal)

Coagulation factor XI(Homo sapiens (Human))
Shenyang Pharmaceutical University

Curated by ChEMBL

PNG

BDBM50063581(CHEMBL3398612)

Ki: 1.5nMAssay Description:Binding affinity to coagulation factor 11a (unknown origin) assessed as inhibition constant using (p-Glu-Pro-Arg-pNa,HCl) as substrate preincubated f...More data for this Ligand-Target Pair

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Xanthine dehydrogenase/oxidase(Homo sapiens (Human))
Shenyang Pharmaceutical University

Curated by ChEMBL

PNG

BDBM50603070(CHEMBL5197177)

Ki: 3.70nMAssay Description:Mixed-type inhibition of xanthine oxidase (unknown origin) assessed as inhibitory constant of enzyme-substrate complex using xanthine as substrate at...More data for this Ligand-Target Pair

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Xanthine dehydrogenase/oxidase(Homo sapiens (Human))
Shenyang Pharmaceutical University

Curated by ChEMBL

PNG

BDBM50517021(CHEMBL4445985)

Ki: 4.20nMAssay Description:Mixed-type inhibition of xanthine oxidase (unknown origin) assessed as inhibitory constant of enzyme-substrate complex using xanthine as substrate at...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
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Xanthine dehydrogenase/oxidase(Bos taurus (Bovine))
Shenyang Pharmaceutical University

Curated by ChEMBL

PNG

BDBM50517021(CHEMBL4445985)

Ki: 4.20nMAssay Description:Mixed type inhibition of bovine xanthine oxidase using xanthine as substrate preincubated with enzyme for 15 mins followed by substrate addition and ...More data for this Ligand-Target Pair

PDB MMDB KEGG
UniProtKB/SwissProt
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Coagulation factor XI(Homo sapiens (Human))
Shenyang Pharmaceutical University

Curated by ChEMBL

PNG

BDBM50572517(CHEMBL4865339)

Ki: 9nMAssay Description:Binding affinity to coagulation factor 11a (unknown origin) assessed as inhibition constant using (p-Glu-Pro-Arg-pNa,HCl) as substrate preincubated f...More data for this Ligand-Target Pair

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Xanthine dehydrogenase/oxidase(Bos taurus (Bovine))
Shenyang Pharmaceutical University

Curated by ChEMBL

PNG

BDBM50570624(CHEMBL4869246)

Ki: 18nMAssay Description:Mixed type inhibition of bovine milk xanthine oxidase assessed as inhibitory constant using xanthine as substrate preincubated for 15 mins followed b...More data for this Ligand-Target Pair

PDB MMDB KEGG
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Coagulation factor XI(Homo sapiens (Human))
Shenyang Pharmaceutical University

Curated by ChEMBL

PNG

BDBM50572518(CHEMBL4849470)

Ki: 23nMAssay Description:Binding affinity to coagulation factor 11a (unknown origin) assessed as inhibition constant using (p-Glu-Pro-Arg-pNa,HCl) as substrate preincubated f...More data for this Ligand-Target Pair

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Xanthine dehydrogenase/oxidase(Homo sapiens (Human))
Shenyang Pharmaceutical University

Curated by ChEMBL

PNG

BDBM50603060(CHEMBL5186383)

Ki: 24nMAssay Description:Mixed-type inhibition of xanthine oxidase (unknown origin) assessed as inhibitory constant of enzyme-substrate complex using xanthine as substrate at...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
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Coagulation factor XI(Homo sapiens (Human))
Shenyang Pharmaceutical University

Curated by ChEMBL

PNG

BDBM50572513(CHEMBL4862896)

Ki: 26nMAssay Description:Binding affinity to coagulation factor 11a (unknown origin) assessed as inhibition constant using (p-Glu-Pro-Arg-pNa,HCl) as substrate preincubated f...More data for this Ligand-Target Pair

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Coagulation factor XI(Homo sapiens (Human))
Shenyang Pharmaceutical University

Curated by ChEMBL

PNG

BDBM50572515(CHEMBL4863349)

Ki: 31nMAssay Description:Binding affinity to coagulation factor 11a (unknown origin) assessed as inhibition constant using (p-Glu-Pro-Arg-pNa,HCl) as substrate preincubated f...More data for this Ligand-Target Pair

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Xanthine dehydrogenase/oxidase(Homo sapiens (Human))
Shenyang Pharmaceutical University

Curated by ChEMBL

PNG

BDBM50603046(CHEMBL5189353)

Ki: 33nMAssay Description:Mixed-type inhibition of xanthine oxidase (unknown origin) assessed as inhibitory constant of enzyme-substrate complex using xanthine as substrate at...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
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Coagulation factor XI(Homo sapiens (Human))
Shenyang Pharmaceutical University

Curated by ChEMBL

PNG

BDBM50572519(CHEMBL4849888)

Ki: 34nMAssay Description:Binding affinity to coagulation factor 11a (unknown origin) assessed as inhibition constant using (p-Glu-Pro-Arg-pNa,HCl) as substrate preincubated f...More data for this Ligand-Target Pair

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Coagulation factor XI(Homo sapiens (Human))
Shenyang Pharmaceutical University

Curated by ChEMBL

PNG

BDBM50572514(CHEMBL4854946)

Ki: 53nMAssay Description:Binding affinity to coagulation factor 11a (unknown origin) assessed as inhibition constant using (p-Glu-Pro-Arg-pNa,HCl) as substrate preincubated f...More data for this Ligand-Target Pair

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Coagulation factor XI(Homo sapiens (Human))
Shenyang Pharmaceutical University

Curated by ChEMBL

PNG

BDBM50572520(CHEMBL4875072)

Ki: 56nMAssay Description:Binding affinity to coagulation factor 11a (unknown origin) assessed as inhibition constant using (p-Glu-Pro-Arg-pNa,HCl) as substrate preincubated f...More data for this Ligand-Target Pair

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Coagulation factor XI(Homo sapiens (Human))
Shenyang Pharmaceutical University

Curated by ChEMBL

PNG

BDBM50572523(CHEMBL4872704)

Ki: 81nMAssay Description:Binding affinity to coagulation factor 11a (unknown origin) assessed as inhibition constant using (p-Glu-Pro-Arg-pNa,HCl) as substrate preincubated f...More data for this Ligand-Target Pair

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Xanthine dehydrogenase/oxidase(Bos taurus (Bovine))
Shenyang Pharmaceutical University

Curated by ChEMBL

PNG

BDBM50517021(CHEMBL4445985)

Ki: 127nMAssay Description:Mixed type inhibition of bovine xanthine oxidase using xanthine as substrate preincubated with enzyme for 15 mins followed by substrate addition and ...More data for this Ligand-Target Pair

PDB MMDB KEGG
UniProtKB/SwissProt
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Xanthine dehydrogenase/oxidase(Bos taurus (Bovine))
Shenyang Pharmaceutical University

Curated by ChEMBL

PNG

BDBM50564058(CHEMBL4792232)

Ki: 138nMAssay Description:Mixed type inhibition of bovine xanthine oxidase assessed as inhibitory constant using xanthine as substrate preincubated for 25 mins followed by sub...More data for this Ligand-Target Pair

PDB MMDB KEGG
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Coagulation factor XI(Homo sapiens (Human))
Shenyang Pharmaceutical University

Curated by ChEMBL

PNG

BDBM50572522(CHEMBL4864164)

Ki: 155nMAssay Description:Binding affinity to coagulation factor 11a (unknown origin) assessed as inhibition constant using (p-Glu-Pro-Arg-pNa,HCl) as substrate preincubated f...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
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Coagulation factor XI(Homo sapiens (Human))
Shenyang Pharmaceutical University

Curated by ChEMBL

PNG

BDBM50572512(CHEMBL4872406)

Ki: 156nMAssay Description:Binding affinity to coagulation factor 11a (unknown origin) assessed as inhibition constant using (p-Glu-Pro-Arg-pNa,HCl) as substrate preincubated f...More data for this Ligand-Target Pair

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Plasma kallikrein(Homo sapiens (Human))
Shenyang Pharmaceutical University

Curated by ChEMBL

PNG

BDBM50572517(CHEMBL4865339)

Ki: 192nMAssay Description:Binding affinity to plasma kallikrein (unknown origin) assessed as inhibition constant using D-Pro-Phe,Arg,pNa,2HCl as substrate preincubated for 10 ...More data for this Ligand-Target Pair

PDB Reactome pathway
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E3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
Chengdu University Of Traditional Chinese Medicine

Curated by ChEMBL

PNG

BDBM50569138(CHEMBL4871070)

Ki: 240nMAssay Description:Inhibition of MDM2 (unknown origin) using peptide as substrate incubated for 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair

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Coagulation factor XI(Homo sapiens (Human))
Shenyang Pharmaceutical University

Curated by ChEMBL

PNG

BDBM50572516(CHEMBL4856139)

Ki: 259nMAssay Description:Binding affinity to coagulation factor 11a (unknown origin) assessed as inhibition constant using (p-Glu-Pro-Arg-pNa,HCl) as substrate preincubated f...More data for this Ligand-Target Pair

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E3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
Chengdu University Of Traditional Chinese Medicine

Curated by ChEMBL

PNG

BDBM50569140(CHEMBL4863792)

Ki: 260nMAssay Description:Inhibition of MDM2 (unknown origin) using peptide as substrate incubated for 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
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E3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
Chengdu University Of Traditional Chinese Medicine

Curated by ChEMBL

PNG

BDBM31197(CHEMBL211045 | Nutlin-3 | med.21724, Compound 186)

Ki: 280nMAssay Description:Inhibition of MDM2 (unknown origin) using peptide as substrate incubated for 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair

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3D Structure (crystal)

Coagulation factor XI(Homo sapiens (Human))
Shenyang Pharmaceutical University

Curated by ChEMBL

PNG

BDBM50572507(CHEMBL4854369)

Ki: 356nMAssay Description:Binding affinity to coagulation factor 11a (unknown origin) assessed as inhibition constant using (p-Glu-Pro-Arg-pNa,HCl) as substrate preincubated f...More data for this Ligand-Target Pair

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Coagulation factor XI(Homo sapiens (Human))
Shenyang Pharmaceutical University

Curated by ChEMBL

PNG

BDBM50572521(CHEMBL4868504)

Ki: 366nMAssay Description:Binding affinity to coagulation factor 11a (unknown origin) assessed as inhibition constant using (p-Glu-Pro-Arg-pNa,HCl) as substrate preincubated f...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
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Coagulation factor XI(Homo sapiens (Human))
Shenyang Pharmaceutical University

Curated by ChEMBL

PNG

BDBM50572511(CHEMBL4846470)

Ki: 392nMAssay Description:Binding affinity to coagulation factor 11a (unknown origin) assessed as inhibition constant using (p-Glu-Pro-Arg-pNa,HCl) as substrate preincubated f...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
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Coagulation factor XI(Homo sapiens (Human))
Shenyang Pharmaceutical University

Curated by ChEMBL

PNG

BDBM50572506(CHEMBL4879256)

Ki: 486nMAssay Description:Binding affinity to coagulation factor 11a (unknown origin) assessed as inhibition constant using (p-Glu-Pro-Arg-pNa,HCl) as substrate preincubated f...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
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E3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
Chengdu University Of Traditional Chinese Medicine

Curated by ChEMBL

PNG

BDBM50569136(CHEMBL4874111)

Ki: 490nMAssay Description:Inhibition of MDM2 (unknown origin) using peptide as substrate incubated for 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair

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E3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
Chengdu University Of Traditional Chinese Medicine

Curated by ChEMBL

PNG

BDBM50569137(CHEMBL4860936)

Ki: 680nMAssay Description:Inhibition of MDM2 (unknown origin) using peptide as substrate incubated for 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
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Xanthine dehydrogenase/oxidase(Homo sapiens (Human))
Shenyang Pharmaceutical University

Curated by ChEMBL

PNG

BDBM50140241(Allopurinol | Aloral | Aluline 100 | Aluline 300 |...)

Ki: 700nMAssay Description:Competitive inhibition of xanthine oxidase (unknown origin) assessed as inhibitory constant of enzyme-substrate complex using xanthine as substrate a...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
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Coagulation factor XI(Homo sapiens (Human))
Shenyang Pharmaceutical University

Curated by ChEMBL

PNG

BDBM50572508(CHEMBL4865716)

Ki: 962nMAssay Description:Binding affinity to coagulation factor 11a (unknown origin) assessed as inhibition constant using (p-Glu-Pro-Arg-pNa,HCl) as substrate preincubated f...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
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E3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
Chengdu University Of Traditional Chinese Medicine

Curated by ChEMBL

PNG

BDBM50569139(CHEMBL4863780)

Ki: 1.02E+3nMAssay Description:Inhibition of MDM2 (unknown origin) using peptide as substrate incubated for 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
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E3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
Chengdu University Of Traditional Chinese Medicine

Curated by ChEMBL

PNG

BDBM50569144(CHEMBL4861981)

Ki: 1.03E+3nMAssay Description:Inhibition of MDM2 (unknown origin) using peptide as substrate incubated for 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
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E3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
Chengdu University Of Traditional Chinese Medicine

Curated by ChEMBL

PNG

BDBM50569143(CHEMBL4876458)

Ki: 1.14E+3nMAssay Description:Inhibition of MDM2 (unknown origin) using peptide as substrate incubated for 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
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E3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
Chengdu University Of Traditional Chinese Medicine

Curated by ChEMBL

PNG

BDBM50569158(CHEMBL4856044)

Ki: 1.19E+3nMAssay Description:Inhibition of MDM2 (unknown origin) using peptide as substrate incubated for 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
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E3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
Chengdu University Of Traditional Chinese Medicine

Curated by ChEMBL

PNG

BDBM50569135(CHEMBL4874952)

Ki: 1.28E+3nMAssay Description:Inhibition of MDM2 (unknown origin) using peptide as substrate incubated for 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
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E3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
Chengdu University Of Traditional Chinese Medicine

Curated by ChEMBL

PNG

BDBM50569159(CHEMBL4870214)

Ki: 1.36E+3nMAssay Description:Inhibition of MDM2 (unknown origin) using peptide as substrate incubated for 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
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E3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
Chengdu University Of Traditional Chinese Medicine

Curated by ChEMBL

PNG

BDBM50569142(CHEMBL4877534)

Ki: 1.42E+3nMAssay Description:Inhibition of MDM2 (unknown origin) using peptide as substrate incubated for 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
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E3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
Chengdu University Of Traditional Chinese Medicine

Curated by ChEMBL

PNG

BDBM50569152(CHEMBL4859985)

Ki: 1.49E+3nMAssay Description:Inhibition of MDM2 (unknown origin) using peptide as substrate incubated for 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
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E3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
Chengdu University Of Traditional Chinese Medicine

Curated by ChEMBL

PNG

BDBM50569149(CHEMBL4877092)

Ki: 1.87E+3nMAssay Description:Inhibition of MDM2 (unknown origin) using peptide as substrate incubated for 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
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E3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
Chengdu University Of Traditional Chinese Medicine

Curated by ChEMBL

PNG

BDBM50569154(CHEMBL4860559)

Ki: 2.26E+3nMAssay Description:Inhibition of MDM2 (unknown origin) using peptide as substrate incubated for 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
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E3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
Chengdu University Of Traditional Chinese Medicine

Curated by ChEMBL

PNG

BDBM50569156(CHEMBL4878727)

Ki: 2.36E+3nMAssay Description:Inhibition of MDM2 (unknown origin) using peptide as substrate incubated for 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
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Multidrug resistance-associated protein 1(Homo sapiens (Human))
Queen'S University

Curated by ChEMBL

PNG

BDBM7462(3,5,7-trihydroxy-2-(4-hydroxyphenyl)-4H-chromen-4-...)

Ki: 2.40E+3nMAssay Description:TP_TRANSPORTER: inhibition of LTC4 uptake in membrane vesicle from MRP1-expressing HeLa cellsMore data for this Ligand-Target Pair

PDB Reactome pathway
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GoogleScholar

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E3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
Chengdu University Of Traditional Chinese Medicine

Curated by ChEMBL

PNG

BDBM50569146(CHEMBL4870252)

Ki: 2.77E+3nMAssay Description:Inhibition of MDM2 (unknown origin) using peptide as substrate incubated for 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
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E3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
Chengdu University Of Traditional Chinese Medicine

Curated by ChEMBL

PNG

BDBM50569148(CHEMBL4848056)

Ki: 2.78E+3nMAssay Description:Inhibition of MDM2 (unknown origin) using peptide as substrate incubated for 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
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Coagulation factor XI(Homo sapiens (Human))
Shenyang Pharmaceutical University

Curated by ChEMBL

PNG

BDBM50572505(CHEMBL4865036)

Ki: 2.82E+3nMAssay Description:Binding affinity to coagulation factor 11a (unknown origin) assessed as inhibition constant using (p-Glu-Pro-Arg-pNa,HCl) as substrate preincubated f...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
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Details Article PubMed

Coagulation factor XI(Homo sapiens (Human))
Shenyang Pharmaceutical University

Curated by ChEMBL

PNG

BDBM50572510(CHEMBL4853234)

Ki: 3.08E+3nMAssay Description:Binding affinity to coagulation factor 11a (unknown origin) assessed as inhibition constant using (p-Glu-Pro-Arg-pNa,HCl) as substrate preincubated f...More data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

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E3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
Chengdu University Of Traditional Chinese Medicine

Curated by ChEMBL

PNG

BDBM50569157(CHEMBL4855468)

Ki: 3.68E+3nMAssay Description:Inhibition of MDM2 (unknown origin) using peptide as substrate incubated for 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
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Details Article PubMed

Displayed 1 to 50 (of 818 total ) | Next | Last >>

Filter my 818 hits

Targets 19▿
- High affinity nerve growth factor receptor 491
- Xanthine dehydrogenase/oxidase 189
- Reverse transcriptase 48
- Coagulation factor XI 36
- E3 ubiquitin-protein ligase Mdm2 31
- Multidrug resistance-associated protein 1 5
- Broad substrate specificity ATP-binding cassette transporter ABCG2 3
- P2Y purinoceptor 12 3
- Integrase 2
- Coagulation factor X 1
- Cytochrome P450 1A2 1
- Cytochrome P450 2E1 1
- Plasma kallikrein 1
- Cytochrome P450 2C9 1
- Cytochrome P450 2C19 1
- Cytochrome P450 2D6 1
- Coagulation factor VII 1
- Cytochrome P450 2A6 1
- Cytochrome P450 3A4 1
- ...
Publications 19▿
- US Patent US9815846 (2017) 228
- US Patent US9914736 (2018) 114
- US Patent US9862707 (2018) 103
- US Patent US9896447 (2018) 46
- Eur J Med Chem 229: (2022) 43
- Eur J Med Chem 220: (2021) 39
- Eur J Med Chem 227: (2022) 38
- Eur J Med Chem 217: (2021) 31
- Bioorg Med Chem 38: (2021) 28
- Eur J Med Chem 181: (2019) 28
- Eur J Med Chem 190: (2020) 27
- Eur J Med Chem 181: (2019) 24
- Eur J Med Chem 102: 215-22 (2015) 21
- Eur J Med Chem 97: 1-9 (2015) 13
- J Med Chem 63: 15752-15772 (2020) 11
- Bioorg Med Chem 23: 3860-8 (2015) 11
- Bioorg Med Chem 23: 4248-4255 (2015) 5
- Mol Pharmacol 59: 1171-80 (2001) 5
- J Pharmacol Exp Ther 310: 334-41 (2004) 3
Institutions 6▿
- Merck Sharp & Dohme 491
- Shenyang Pharmaceutical University 238
- Fudan University 50
- Chengdu University Of Traditional Chinese Medicine 31
- Queen'S University 5
- University Of Washington 3
Affinity: 0.069 to 5.0E+5 nM▿
- Ki 85
- IC50 733
- Affinity ≤ nM
Xtal structures: 7
Docked structures: 0
Catalog Cmpds: 18