Affinity DataKi: 0.530nMAssay Description:Compound was evaluated for the binding affinity of Opioid receptor mu 1 by displacing the radioligand [3H]DAMGO from rat brain membraneMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Institute Of Bioorganic Chemistry Ras
Curated by ChEMBL
Institute Of Bioorganic Chemistry Ras
Curated by ChEMBL
Affinity DataKi: 380nMAssay Description:Concentration required to displace 0.4 nM [3H]-SR-141,716A from CB1 receptor in rat brain preparations in the presence of 0.1 mM phenylmethyl sulphon...More data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Institute Of Bioorganic Chemistry Ras
Curated by ChEMBL
Institute Of Bioorganic Chemistry Ras
Curated by ChEMBL
Affinity DataKi: 620nMAssay Description:Concentration required to displace 0.4 nM [3H]-SR-141,716A from CB1 receptor in rat brain preparations in the presence of 0.1 mM phenylmethyl sulphon...More data for this Ligand-Target Pair
Affinity DataKi: 720nMAssay Description:Compound was evaluated for the binding affinity of Opioid receptor mu 1 by displacing the radioligand [3H]DAMGO from rat brain membraneMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Institute Of Bioorganic Chemistry Ras
Curated by ChEMBL
Institute Of Bioorganic Chemistry Ras
Curated by ChEMBL
Affinity DataKi: 800nMAssay Description:Concentration required to displace 0.4 nM [3H]-SR-141,716A from CB1 receptor in rat brain preparations in the presence of 0.1 mM phenylmethyl sulphon...More data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Institute Of Bioorganic Chemistry Ras
Curated by ChEMBL
Institute Of Bioorganic Chemistry Ras
Curated by ChEMBL
Affinity DataKi: 1.37E+3nMAssay Description:Concentration required to displace 0.4 nM [3H]-SR-141,716A from CB1 receptor in rat brain preparations in the presence of 0.1 mM phenylmethyl sulphon...More data for this Ligand-Target Pair
Affinity DataKi: 1.44E+3nMAssay Description:Compound was evaluated for the binding affinity of Opioid receptor mu 1 by displacing the radioligand [3H]DAMGO from rat brain membraneMore data for this Ligand-Target Pair
Affinity DataKi: 1.62E+3nMAssay Description:Compound was evaluated for the binding affinity of Opioid receptor mu 1 by displacing the radioligand [3H]DAMGO from rat brain membraneMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Institute Of Bioorganic Chemistry Ras
Curated by ChEMBL
Institute Of Bioorganic Chemistry Ras
Curated by ChEMBL
Affinity DataKi: 1.72E+3nMAssay Description:Concentration required to displace 0.4 nM [3H]-SR-141,716A from CB1 receptor in rat brain preparations in the presence of 0.1 mM phenylmethyl sulphon...More data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Institute Of Bioorganic Chemistry Ras
Curated by ChEMBL
Institute Of Bioorganic Chemistry Ras
Curated by ChEMBL
Affinity DataKi: 2.43E+3nMAssay Description:Concentration required to displace 0.4 nM [3H]-SR-141,716A from CB1 receptor in rat brain preparations in the presence of 0.1 mM phenylmethyl sulphon...More data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Institute Of Bioorganic Chemistry Ras
Curated by ChEMBL
Institute Of Bioorganic Chemistry Ras
Curated by ChEMBL
Affinity DataKi: 3.13E+3nMAssay Description:Concentration required to displace 0.4 nM [3H]-SR-141,716A from CB1 receptor in rat brain preparations in the presence of 0.1 mM phenylmethyl sulphon...More data for this Ligand-Target Pair
Affinity DataKi: 7.54E+3nMAssay Description:Compound was evaluated for the binding affinity of Opioid receptor mu 1 by displacing the radioligand [3H]DAMGO from rat brain membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibitory concentration against [3H]DAMGO binding to Opioid receptor mu 1 in rat brain membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 4.00E+3nMAssay Description:Inhibitory concentration against [3H]DAMGO binding to Opioid receptor mu 1 in rat brain membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 4.50E+3nMAssay Description:Inhibitory concentration against [3H]DAMGO binding to Opioid receptor mu 1 in rat brain membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibitory concentration against [3H]DAMGO binding to Opioid receptor mu 1 in rat brain membraneMore data for this Ligand-Target Pair