TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Hoffmann-La Roche
Curated by ChEMBL
Hoffmann-La Roche
Curated by ChEMBL
Affinity DataKi: 0.5nMAssay Description:Binding affinity to MCHR1More data for this Ligand-Target Pair
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Hoffmann-La Roche
Curated by ChEMBL
Hoffmann-La Roche
Curated by ChEMBL
Affinity DataKi: 3nMAssay Description:Binding affinity to MCHR1More data for this Ligand-Target Pair
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Hoffmann-La Roche
Curated by ChEMBL
Hoffmann-La Roche
Curated by ChEMBL
Affinity DataKi: 5nMAssay Description:Binding affinity to MCHR1More data for this Ligand-Target Pair
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Hoffmann-La Roche
Curated by ChEMBL
Hoffmann-La Roche
Curated by ChEMBL
Affinity DataKi: 5.20nMAssay Description:Binding affinity to MCHR1More data for this Ligand-Target Pair
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Hoffmann-La Roche
Curated by ChEMBL
Hoffmann-La Roche
Curated by ChEMBL
Affinity DataKi: 10nMAssay Description:Binding affinity to MCHR1More data for this Ligand-Target Pair
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Hoffmann-La Roche
Curated by ChEMBL
Hoffmann-La Roche
Curated by ChEMBL
Affinity DataKi: 20nMAssay Description:Binding affinity to MCHR1More data for this Ligand-Target Pair
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Hoffmann-La Roche
Curated by ChEMBL
Hoffmann-La Roche
Curated by ChEMBL
Affinity DataKi: 25nMAssay Description:Binding affinity to MCHR1More data for this Ligand-Target Pair
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Hoffmann-La Roche
Curated by ChEMBL
Hoffmann-La Roche
Curated by ChEMBL
Affinity DataKi: 31nMAssay Description:Binding affinity to MCHR1More data for this Ligand-Target Pair
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Hoffmann-La Roche
Curated by ChEMBL
Hoffmann-La Roche
Curated by ChEMBL
Affinity DataKi: 47nMAssay Description:Binding affinity to MCHR1More data for this Ligand-Target Pair
TargetGlutamine--fructose-6-phosphate aminotransferase [isomerizing] 1(Homo sapiens (Human))
Hoffmann-La Roche
Curated by ChEMBL
Hoffmann-La Roche
Curated by ChEMBL
Affinity DataKi: 300nMAssay Description:Competitive inhibition of GFAT in presence of glutamineMore data for this Ligand-Target Pair
TargetGlutamine--fructose-6-phosphate aminotransferase [isomerizing] 1(Homo sapiens (Human))
Hoffmann-La Roche
Curated by ChEMBL
Hoffmann-La Roche
Curated by ChEMBL
Affinity DataKi: 300nMAssay Description:Noncompetitive inhibition of GFAT in presence of fructose-6-phosphateMore data for this Ligand-Target Pair
Affinity DataIC50: 0.200nMAssay Description:Inhibitory binding concentration against VCAM/VLA-4 in ELISA.More data for this Ligand-Target Pair
Affinity DataIC50: 0.25nMAssay Description:Inhibitory binding concentration against VCAM/VLA-4 in ELISA.More data for this Ligand-Target Pair
Affinity DataIC50: 0.25nMAssay Description:Inhibitory binding concentration against VCAM/VLA-4 in ELISA.More data for this Ligand-Target Pair
Affinity DataIC50: 0.300nMAssay Description:Inhibitory binding concentration against VCAM/VLA-4 in ELISA.More data for this Ligand-Target Pair
Affinity DataIC50: 0.300nMAssay Description:Inhibitory binding concentration against VCAM/VLA-4 in ELISA.More data for this Ligand-Target Pair
Affinity DataIC50: 0.370nMAssay Description:Antagonistic activity against VLA-4 (derived from ramos cells) binding to recombinant human VCAM by ELISA assayMore data for this Ligand-Target Pair
Affinity DataIC50: 0.400nMAssay Description:Inhibitory binding concentration against VCAM/VLA-4 in Ramos.More data for this Ligand-Target Pair
Affinity DataIC50: 0.400nMAssay Description:Inhibitory binding concentration against VCAM/VLA-4 in Ramos.More data for this Ligand-Target Pair
Affinity DataIC50: 0.420nMAssay Description:Inhibitory binding concentration against VCAM/VLA-4 in Ramos.More data for this Ligand-Target Pair
Affinity DataIC50: 0.440nMAssay Description:Inhibitory binding concentration against VCAM/VLA-4 in ELISA.More data for this Ligand-Target Pair
Affinity DataIC50: 0.460nMAssay Description:Inhibitory binding concentration against VCAM/VLA-4 in ELISA.More data for this Ligand-Target Pair
Affinity DataIC50: 0.490nMAssay Description:Inhibitory binding concentration against VCAM/VLA-4 in Ramos.More data for this Ligand-Target Pair
Affinity DataIC50: 0.560nMAssay Description:Inhibitory binding concentration against VCAM/VLA-4 in Ramos.More data for this Ligand-Target Pair
Affinity DataIC50: 0.740nMAssay Description:Antagonistic activity against VLA-4 (derived from ramos cells) binding to recombinant human VCAM by ELISA assayMore data for this Ligand-Target Pair
Affinity DataIC50: 0.75nMAssay Description:Antagonistic activity against VLA-4 (derived from ramos cells) binding to recombinant human VCAM by ELISA assayMore data for this Ligand-Target Pair
Affinity DataIC50: 0.820nMAssay Description:Inhibition of human VCAM and Ramos cell VLA-4 interactionMore data for this Ligand-Target Pair
Affinity DataIC50: 0.870nMAssay Description:Antagonistic activity against VLA-4 (derived from ramos cells) binding to recombinant human VCAM by ELISA assayMore data for this Ligand-Target Pair
Affinity DataIC50: 0.880nMAssay Description:Antagonistic activity against VLA-4 (derived from ramos cells) binding to recombinant human VCAM by ELISA assayMore data for this Ligand-Target Pair
Affinity DataIC50: 0.890nMAssay Description:Inhibitory binding concentration against VCAM/VLA-4 in ELISA.More data for this Ligand-Target Pair
Affinity DataIC50: 1nMAssay Description:Inhibition of [3H]-PAF binding to platelet activating factor receptor citrate-treated dog bloodMore data for this Ligand-Target Pair
Affinity DataIC50: 1.20nMAssay Description:Inhibitory binding concentration against VCAM/VLA-4 in Ramos.More data for this Ligand-Target Pair
Affinity DataIC50: 1.20nMAssay Description:Inhibitory binding concentration against VCAM/VLA-4 in ELISA.More data for this Ligand-Target Pair
Affinity DataIC50: 1.30nMAssay Description:Inhibitory binding concentration against VCAM/VLA-4 in ELISA.More data for this Ligand-Target Pair
Affinity DataIC50: 1.40nMAssay Description:Inhibitory binding concentration against VCAM/VLA-4 in ELISA.More data for this Ligand-Target Pair
Affinity DataIC50: 1.40nMAssay Description:Antagonistic activity against VLA-4 (derived from ramos cells) binding to recombinant human VCAM by ELISA assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.5nMAssay Description:Inhibitory binding concentration against VCAM/VLA-4 in ELISA.More data for this Ligand-Target Pair
Affinity DataIC50: 1.60nMAssay Description:Antagonistic activity against VLA-4 (derived from ramos cells) binding to recombinant human VCAM by ELISA assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.60nMAssay Description:Inhibitory binding concentration against VCAM/VLA-4 in ELISA.More data for this Ligand-Target Pair
Affinity DataIC50: 1.60nMAssay Description:Inhibitory binding concentration against VCAM/VLA-4 in Ramos.More data for this Ligand-Target Pair
Affinity DataIC50: 1.90nMAssay Description:Inhibitory binding concentration against VCAM/VLA-4 in ELISA.More data for this Ligand-Target Pair
Affinity DataIC50: 1.90nMAssay Description:Inhibitory binding concentration against VCAM/VLA-4 in Ramos.More data for this Ligand-Target Pair
Affinity DataIC50: 1.90nMAssay Description:Inhibitory binding concentration against VCAM/VLA-4 in ELISA.More data for this Ligand-Target Pair
Affinity DataIC50: 2nMAssay Description:Inhibitory binding concentration against VCAM/VLA-4 in Ramos.More data for this Ligand-Target Pair
Affinity DataIC50: 2nMAssay Description:Inhibitory binding concentration against VCAM/VLA-4 in ELISA.More data for this Ligand-Target Pair
Affinity DataIC50: 2nMAssay Description:Inhibition of platelet activating factor receptor binding activity in dog platelets using [3H]-PAF as radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 2nMAssay Description:Inhibition of platelet activating factor receptor binding activity in dog platelets using [3H]-PAF as radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 2.20nMAssay Description:Inhibitory binding concentration against VCAM/VLA-4 in Ramos.More data for this Ligand-Target Pair
Affinity DataIC50: 2.20nMAssay Description:Antagonistic activity against VLA-4 binding to recombinant human VCAM by ramos cell assayMore data for this Ligand-Target Pair
Affinity DataIC50: 2.40nMAssay Description:Antagonistic activity against VLA-4 binding to recombinant human VCAM by ramos cell assayMore data for this Ligand-Target Pair