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Found 74 with Last Name = 'mertes' and Initial = 'mp'
TargetThymidylate synthase(Lactobacillus casei)
TBA

Curated by ChEMBL
LigandPNGBDBM50022238((R)-5-Fluoro-1-((4S,5R)-4-hydroxy-5-methylphosphat...)
Affinity DataKi:  14nMAssay Description:Competitive inhibition of thymidylate synthase purified from methotrexate-resistant Lactobacillus casei using 2'-deoxy[5-3H]uridine 5'-phosphate by r...More data for this Ligand-Target Pair
TargetThymidylate synthase(Lactobacillus casei)
TBA

Curated by ChEMBL
LigandPNGBDBM50010241(CHEMBL1234672)
Affinity DataKi:  29nMAssay Description:Competitive inhibition of thymidylate synthase purified from methotrexate-resistant Lactobacillus casei using 2'-deoxy[5-3H]uridine 5'-phosphate by r...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidylate synthase(Lactobacillus casei)
TBA

Curated by ChEMBL
LigandPNGBDBM50010236(CHEMBL3144200)
Affinity DataKi:  39nMAssay Description:Competitive inhibition of thymidylate synthase purified from methotrexate-resistant Lactobacillus casei using 2'-deoxy[5-3H]uridine 5'-phosphate by r...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidylate synthase(Lactobacillus casei)
TBA

Curated by ChEMBL
LigandPNGBDBM50000038(CHEMBL3228321)
Affinity DataKi:  40nMAssay Description:Competitive inhibition of thymidylate synthase purified from methotrexate-resistant Lactobacillus casei using 2'-deoxy[5-3H]uridine 5'-phosphate by r...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidylate synthase(Lactobacillus casei)
TBA

Curated by ChEMBL
LigandPNGBDBM50010239(CHEMBL1236538)
Affinity DataKi:  190nMAssay Description:Competitive inhibition of thymidylate synthase purified from methotrexate-resistant Lactobacillus casei using 2'-deoxy[5-3H]uridine 5'-phosphate by r...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidylate synthase(Lactobacillus casei)
TBA

Curated by ChEMBL
LigandPNGBDBM50023636(CHEMBL3144190 | Phosphoric acid mono-{5-[5-(4-benz...)
Affinity DataKi:  310nMAssay Description:Inhibitory effect on Lactobacillus casei thymidylate synthaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidylate synthase(Lactobacillus casei)
TBA

Curated by ChEMBL
LigandPNGBDBM50027919(5-fluoro-deoxyuridinemonophosphate | CHEMBL416879)
Affinity DataKi:  500nMAssay Description:Inactivation of thymidylate synthetase measured asKi at 6.8 pH 30 degrees centigrade tempMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidylate synthase(Lactobacillus casei)
TBA

Curated by ChEMBL
LigandPNGBDBM50404974(5-NITRO-DUMP | CHEMBL2051758)
Affinity DataKi:  500nMAssay Description:Inactivation of thymidylate synthetase measured asKi at 6.8 pH 30 degrees centigrade tempMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidylate synthase(Lactobacillus casei)
TBA

Curated by ChEMBL
LigandPNGBDBM50010240(CHEMBL3246102)
Affinity DataKi:  550nMAssay Description:Competitive inhibition of thymidylate synthase purified from methotrexate-resistant Lactobacillus casei using 2'-deoxy[5-3H]uridine 5'-phosphate by r...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidylate synthase(Lactobacillus casei)
TBA

Curated by ChEMBL
LigandPNGBDBM50226709(CHEMBL3143111)
Affinity DataKi:  590nMAssay Description:Ability to inhibit the thymidylate synthase from L. casei was determined and expressed as inhibition constant(Ki)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidylate synthase(Lactobacillus casei)
TBA

Curated by ChEMBL
LigandPNGBDBM50021750(CHEMBL3143104 | Phosphoric acid mono-{3-hydroxy-5-...)
Affinity DataKi:  610nMAssay Description:Ability to inhibit the thymidylate synthase from L. casei was determined and expressed as inhibition constant(Ki)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidylate synthase(Lactobacillus casei)
TBA

Curated by ChEMBL
LigandPNGBDBM50023645(CHEMBL3144187 | Phosphoric acid mono-[5-(2,4-dioxo...)
Affinity DataKi:  610nMAssay Description:Inhibitory effect on Lactobacillus casei thymidylate synthaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidylate synthase(Lactobacillus casei)
TBA

Curated by ChEMBL
LigandPNGBDBM50023647(CHEMBL3144186 | Phosphoric acid mono-[5-(2,4-dioxo...)
Affinity DataKi:  960nMAssay Description:Inhibitory effect on Lactobacillus casei thymidylate synthaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidylate synthase(Lactobacillus casei)
TBA

Curated by ChEMBL
LigandPNGBDBM50023637(CHEMBL3144189 | Phosphoric acid mono-{5-[5-(4-amin...)
Affinity DataKi:  1.13E+3nMAssay Description:Inhibitory effect on Lactobacillus casei thymidylate synthaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidylate synthase(Lactobacillus casei)
TBA

Curated by ChEMBL
LigandPNGBDBM50023640(CHEMBL3144188 | Phosphoric acid mono-{3-hydroxy-5-...)
Affinity DataKi:  1.21E+3nMAssay Description:Inhibitory effect on Lactobacillus casei thymidylate synthaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidylate synthase(Lactobacillus casei)
TBA

Curated by ChEMBL
LigandPNGBDBM50021748(CHEMBL3143138 | Phosphoric acid mono-{5-[5-(4,5-di...)
Affinity DataKi:  1.30E+3nMAssay Description:Ability to inhibit the thymidylate synthase from L. casei was determined and expressed as inhibition constant(Ki)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidylate synthase(Lactobacillus casei)
TBA

Curated by ChEMBL
LigandPNGBDBM50021746(CHEMBL3143107 | Phosphoric acid mono-{5-[5-(2,5-di...)
Affinity DataKi:  1.40E+3nMAssay Description:Ability to inhibit the thymidylate synthase from L. casei was determined and expressed as inhibition constant(Ki)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidylate synthase(Lactobacillus casei)
TBA

Curated by ChEMBL
LigandPNGBDBM50010238(CHEMBL1160593)
Affinity DataKi:  1.40E+3nMAssay Description:Competitive inhibition of thymidylate synthase purified from methotrexate-resistant Lactobacillus casei using 2'-deoxy[5-3H]uridine 5'-phosphate by r...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidylate synthase(Lactobacillus casei)
TBA

Curated by ChEMBL
LigandPNGBDBM50023639(CHEMBL3144192 | Phosphoric acid mono-{5-[5-(4-dime...)
Affinity DataKi:  1.41E+3nMAssay Description:Inhibitory effect on Lactobacillus casei thymidylate synthaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidylate synthase(Lactobacillus casei)
TBA

Curated by ChEMBL
LigandPNGBDBM50010242(CHEMBL1160594)
Affinity DataKi:  1.60E+3nMAssay Description:Competitive inhibition of thymidylate synthase purified from methotrexate-resistant Lactobacillus casei using 2'-deoxy[5-3H]uridine 5'-phosphate by r...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidylate synthase(Lactobacillus casei)
TBA

Curated by ChEMBL
LigandPNGBDBM50023641(CHEMBL3144196 | Phosphoric acid mono-{5-[5-(4-brom...)
Affinity DataKi:  1.81E+3nMAssay Description:Inhibitory effect on Lactobacillus casei thymidylate synthaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidylate synthase(Mus musculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50021750(CHEMBL3143104 | Phosphoric acid mono-{3-hydroxy-5-...)
Affinity DataKi:  1.90E+3nMAssay Description:Ability to inhibit the thymidylate synthase from murine leukemia L1210 cells was determined and expressed as inhibition constant(Ki)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidylate synthase(Lactobacillus casei)
TBA

Curated by ChEMBL
LigandPNGBDBM50027920(5-quinonyl-deoxyuridinemonophosphate | CHEMBL8016)
Affinity DataKi:  2.00E+3nMAssay Description:Inactivation of thymidylate synthetase measured asKi at 6.8 pH 30 degrees centigrade tempMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidylate synthase(Lactobacillus casei)
TBA

Curated by ChEMBL
LigandPNGBDBM50021749(CHEMBL3144392 | Phosphoric acid mono-{5-[5-(3,6-di...)
Affinity DataKi:  2.00E+3nMAssay Description:Ability to inhibit the thymidylate synthase from L. casei was determined and expressed as inhibition constant(Ki)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidylate synthase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50021749(CHEMBL3144392 | Phosphoric acid mono-{5-[5-(3,6-di...)
Affinity DataKi:  2.00E+3nMAssay Description:Binding affinity of the compound against thymidylateSynthaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidylate synthase(Lactobacillus casei)
TBA

Curated by ChEMBL
LigandPNGBDBM50024666((1,4-Dimethoxy-3-methyl-naphthalen-2-yl)-phosphoni...)
Affinity DataKi:  2.40E+3nMAssay Description:Binding affinity towards L. casei thymidylate synthase was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidylate synthase(Lactobacillus casei)
TBA

Curated by ChEMBL
LigandPNGBDBM50021751(CHEMBL3143106 | Phosphoric acid mono-{5-[5-(1,4-di...)
Affinity DataKi:  2.40E+3nMAssay Description:Ability to inhibit the thymidylate synthase from L. casei was determined and expressed as inhibition constant(Ki)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidylate synthase(Lactobacillus casei)
TBA

Curated by ChEMBL
LigandPNGBDBM50000019(CHEMBL3144338)
Affinity DataKi:  2.80E+3nMAssay Description:Competitive inhibition of Lactobacillus casei thymidylate synthetase using dTMP as substrate assessed as release of water after 15 mins by double rec...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidylate synthase(Bos taurus)
TBA

Curated by ChEMBL
LigandPNGBDBM50010328(CHEMBL3248468)
Affinity DataKi:  3.10E+3nMAssay Description:Competitive inhibition of purified calf thymus thymidylate synthetase using 5-[3H]-2'-deoxyuridine 5'-phosphate as substrate after 7 mins by double r...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidylate synthase(Lactobacillus casei)
TBA

Curated by ChEMBL
LigandPNGBDBM50021752(CHEMBL3143105 | Phosphoric acid mono-{5-[5-(2,5-di...)
Affinity DataKi:  3.60E+3nMAssay Description:Ability to inhibit the thymidylate synthase from L. casei was determined and expressed as inhibition constant (Ki)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidylate synthase(Lactobacillus casei)
TBA

Curated by ChEMBL
LigandPNGBDBM50023635(4-[1-(4-Hydroxy-5-phosphonooxymethyl-tetrahydro-fu...)
Affinity DataKi:  3.99E+3nMAssay Description:Inhibitory effect on Lactobacillus casei thymidylate synthaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidylate synthase(Lactobacillus casei)
TBA

Curated by ChEMBL
LigandPNGBDBM50404975(CHEMBL2051976)
Affinity DataKi:  4.00E+3nMAssay Description:Inactivation of thymidylate synthetase measured as Ki at 6.8 pH 30 degrees centigrade tempMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidylate synthase(Lactobacillus casei)
TBA

Curated by ChEMBL
LigandPNGBDBM50023638(CHEMBL3144194 | Phosphoric acid mono-{5-[2,4-dioxo...)
Affinity DataKi:  4.93E+3nMAssay Description:Inhibitory effect on Lactobacillus casei thymidylate synthaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidylate synthase(Mus musculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50021748(CHEMBL3143138 | Phosphoric acid mono-{5-[5-(4,5-di...)
Affinity DataKi:  5.10E+3nMAssay Description:Ability to inhibit the thymidylate synthase from murine leukemia L1210 cells was determined and expressed as inhibition constant(Ki)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidylate synthase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50023645(CHEMBL3144187 | Phosphoric acid mono-[5-(2,4-dioxo...)
Affinity DataKi:  5.60E+3nMAssay Description:Inhibitory effect on human lymphoblast (Molt/4F) thymidylate synthaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidylate synthase(Lactobacillus casei)
TBA

Curated by ChEMBL
LigandPNGBDBM50023643(CHEMBL3144195 | Phosphoric acid mono-{5-[5-(4-carb...)
Affinity DataKi:  5.67E+3nMAssay Description:Inhibitory effect on Lactobacillus casei thymidylate synthaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidylate synthase(Mus musculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50226709(CHEMBL3143111)
Affinity DataKi:  6.10E+3nMAssay Description:Ability to inhibit the thymidylate synthase from murine leukemia L1210 cells was determined and expressed as inhibition constant(Ki)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidylate synthase(Lactobacillus casei)
TBA

Curated by ChEMBL
LigandPNGBDBM50227388(CHEMBL3144092)
Affinity DataKi:  6.42E+3nMAssay Description:Inhibitory effect on Lactobacillus casei thymidylate synthaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidylate synthase(Mus musculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50186267(2'-deoxy-5'-uridylic acid | CHEMBL211312 | dUMP)
Affinity DataKi:  6.50E+3nMAssay Description:Competitive inhibition of purified mouse Ehrlich ascites tumor cell thymidylate synthetase using 5-[3H]-2'-deoxyuridine 5'-phosphate as substrate aft...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidylate synthase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50023647(CHEMBL3144186 | Phosphoric acid mono-[5-(2,4-dioxo...)
Affinity DataKi:  6.80E+3nMAssay Description:Inhibitory effect on human lymphoblast (Molt/4F) thymidylate synthaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidylate synthase(Lactobacillus casei)
TBA

Curated by ChEMBL
LigandPNGBDBM50023644(CHEMBL3144191 | Phosphoric acid mono-{3-hydroxy-5-...)
Affinity DataKi:  7.62E+3nMAssay Description:Inhibitory effect on Lactobacillus casei thymidylate synthaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidylate synthase(Bos taurus)
TBA

Curated by ChEMBL
LigandPNGBDBM50186267(2'-deoxy-5'-uridylic acid | CHEMBL211312 | dUMP)
Affinity DataKi:  8.00E+3nMAssay Description:Competitive inhibition of purified calf thymus thymidylate synthetase using 5-[3H]-2'-deoxyuridine 5'-phosphate as substrate after 7 mins by double r...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidylate synthase(Mus musculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50023645(CHEMBL3144187 | Phosphoric acid mono-[5-(2,4-dioxo...)
Affinity DataKi:  8.30E+3nMAssay Description:Inhibitory effect on murine leukemia (L1210) thymidylate synthaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidylate synthase(Lactobacillus casei)
TBA

Curated by ChEMBL
LigandPNGBDBM50023642(CHEMBL3144193 | Phosphoric acid mono-{5-[5-(4-cyan...)
Affinity DataKi:  8.75E+3nMAssay Description:Inhibitory effect on Lactobacillus casei thymidylate synthaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidylate synthase(Mus musculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50023636(CHEMBL3144190 | Phosphoric acid mono-{5-[5-(4-benz...)
Affinity DataKi:  1.12E+4nMAssay Description:Inhibitory effect on murine leukemia (L1210) thymidylate synthaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidylate synthase(Mus musculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50023637(CHEMBL3144189 | Phosphoric acid mono-{5-[5-(4-amin...)
Affinity DataKi:  1.13E+4nMAssay Description:Inhibitory effect on murine leukemia (L1210) thymidylate synthaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidylate synthase(Mus musculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50023647(CHEMBL3144186 | Phosphoric acid mono-[5-(2,4-dioxo...)
Affinity DataKi:  1.22E+4nMAssay Description:Inhibitory effect on murine leukemia (L1210) thymidylate synthaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidylate synthase(Mus musculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50010328(CHEMBL3248468)
Affinity DataKi:  1.40E+4nMAssay Description:Competitive inhibition of purified mouse Ehrlich ascites tumor cell thymidylate synthetase using 5-[3H]-2'-deoxyuridine 5'-phosphate as substrate aft...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidylate synthase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50023637(CHEMBL3144189 | Phosphoric acid mono-{5-[5-(4-amin...)
Affinity DataKi:  1.54E+4nMAssay Description:Inhibitory effect on human lymphoblast (Molt/4F) thymidylate synthaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidylate synthase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50023641(CHEMBL3144196 | Phosphoric acid mono-{5-[5-(4-brom...)
Affinity DataKi:  2.17E+4nMAssay Description:Inhibitory effect on human lymphoblast (Molt/4F) thymidylate synthaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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