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Found 131 with Last Name = 'mook-jung' and Initial = 'i'
TargetProtein kinase C alpha type(Homo sapiens (Human))
Research Institute Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50184391((R,Z)-2-(2-(hydroxymethyl)-4-(3-isobutyl-5-methylh...)
Affinity DataKi:  1.5nMAssay Description:Displacement of [20-3H]PDBu from recombinant PKC alpha in presence of phosphatidylserineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Homo sapiens (Human))
Korea Institute Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50159089(CHEMBL180523 | N,N-Dibutyl-2-[6,8-dichloro-2-(4-ch...)
Affinity DataKi:  2.70nMAssay Description:Inhibition of TSPO (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
Research Institute Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50107112((Z) 2,2-Dimethyl-propionic acid 2-hydroxymethyl-4-...)
Affinity DataKi:  2.90nMAssay Description:Displacement of [20-3H]PDBu from recombinant PKC alpha in presence of phosphatidylserineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Homo sapiens (Human))
Korea Institute Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50045877(2-(2-(4-fluorophenyl)-1H-indol-3-yl)-N,N-dihexylac...)
Affinity DataKi:  3.30nMAssay Description:Inhibition of TSPO (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
Research Institute Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50184395(5-hexanoyloxymethyl-5-hydroxymethyl-3-[(Z)-3-isobu...)
Affinity DataKi:  3.80nMAssay Description:Displacement of [20-3H]PDBu from recombinant PKC alpha in presence of phosphatidylserineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
Research Institute Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50107120((E) 2,2-Dimethyl-propionic acid 2-hydroxymethyl-4-...)
Affinity DataKi:  4.5nMAssay Description:Displacement of [20-3H]PDBu from recombinant PKC alpha in presence of phosphatidylserineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
Research Institute Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50107118(3-Isopropyl-4-methyl-pentanoic acid 2-hydroxymethy...)
Affinity DataKi:  4.5nMAssay Description:Displacement of [20-3H]PDBu from recombinant PKC alpha in presence of phosphatidylserineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
Research Institute Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50184385(5-hydroxymethyl-3-[(Z)-3-isobutyl-5-methylhexylide...)
Affinity DataKi:  5nMAssay Description:Displacement of [20-3H]PDBu from recombinant PKC alpha in presence of phosphatidylserineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
Research Institute Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50184380(5-hydroxymethyl-3-[(E)-3-isobutyl-5-methylhexylide...)
Affinity DataKi:  6nMAssay Description:Displacement of [20-3H]PDBu from recombinant PKC alpha in presence of phosphatidylserineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
Research Institute Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50184382(5-hexanoyloxymethyl-5-hydroxymethyl-3-[(E)-3-isobu...)
Affinity DataKi:  6.20nMAssay Description:Displacement of [20-3H]PDBu from recombinant PKC alpha in presence of phosphatidylserineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
Research Institute Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50184390(5-benzoyloxymethyl-5-hydroxymethyl-3-[(Z)-3-isobut...)
Affinity DataKi:  6.70nMAssay Description:Displacement of [20-3H]PDBu from recombinant PKC alpha in presence of phosphatidylserineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
Research Institute Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50107116(3-Isopropyl-4-methyl-pentanoic acid 2-hydroxymethy...)
Affinity DataKi:  6.90nMAssay Description:Displacement of [20-3H]PDBu from recombinant PKC alpha in presence of phosphatidylserineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
Research Institute Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50184388(5-hydroxymethyl-3-[(Z)-3-isobutyl-5-methylhexylide...)
Affinity DataKi:  6.90nMAssay Description:Displacement of [20-3H]PDBu from recombinant PKC alpha in presence of phosphatidylserineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
Korea Institute Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM22032(1-(2-chlorophenyl)-N-methyl-N-(1-methylpropyl)isoq...)
Affinity DataKi:  8.90nMAssay Description:Displacement of [3H]PK11195 from TSPO in Sprague-Dawley rat cerebral cortex membranes after 60 mins by microbeta liquid scintillation counting methodMore data for this Ligand-Target Pair
TargetProtein kinase C alpha type(Homo sapiens (Human))
Research Institute Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50184383(5-benzoyloxymethyl-5-hydroxymethyl-3-[(E)-3-isobut...)
Affinity DataKi:  16nMAssay Description:Displacement of [20-3H]PDBu from recombinant PKC alpha in presence of phosphatidylserineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
Research Institute Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50184392(5-[(E)-3-(tert-butoxy)-3-oxo-1-propenyl]-5-hydroxy...)
Affinity DataKi:  18nMAssay Description:Displacement of [20-3H]PDBu from recombinant PKC alpha in presence of phosphatidylserineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
Korea Institute Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50210940(CHEMBL3948914)
Affinity DataKi:  23nMAssay Description:Displacement of [3H]PK11195 from TSPO in Sprague-Dawley rat cerebral cortex membranes after 60 mins by microbeta liquid scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
Research Institute Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50184384(6-hydroxymethyl-3-[(Z)-3-isobutyl-5-methylhexylide...)
Affinity DataKi:  28nMAssay Description:Displacement of [20-3H]PDBu from recombinant PKC alpha in presence of phosphatidylserineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
Research Institute Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50184394(6-hydroxymethyl-3-[(E)-3-isobutyl-5-methylhexylide...)
Affinity DataKi:  48nMAssay Description:Displacement of [20-3H]PDBu from recombinant PKC alpha in presence of phosphatidylserineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
Research Institute Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50184386(6-hydroxymethyl-3-[(E)-3-isobutyl-5-methylhexylide...)
Affinity DataKi:  129nMAssay Description:Displacement of [20-3H]PDBu from recombinant PKC alpha in presence of phosphatidylserineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
Research Institute Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50184381(6-hydroxymethyl-3-[(E)-3-isobutyl-5-methylhexylide...)
Affinity DataKi:  147nMAssay Description:Displacement of [20-3H]PDBu from recombinant PKC alpha in presence of phosphatidylserineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
Research Institute Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50184389(5-[(E)-3-(tert-butoxy)-3-oxo-1-propenyl]-5-hydroxy...)
Affinity DataKi:  173nMAssay Description:Displacement of [20-3H]PDBu from recombinant PKC alpha in presence of phosphatidylserineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
Research Institute Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50184387(5-(hydroxymethyl)-5-(pivaloyloxymethyl)-3,3-bis(3-...)
Affinity DataKi:  2.10E+3nMAssay Description:Displacement of [20-3H]PDBu from recombinant PKC alpha in presence of phosphatidylserineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
Research Institute Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50184379(5-(hydroxymethyl)-5-(pivaloyloxymethyl)-3,3-bis(3-...)
Affinity DataKi:  1.83E+4nMAssay Description:Displacement of [20-3H]PDBu from recombinant PKC alpha in presence of phosphatidylserineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
Research Institute Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50184393(5-[(Z)-3-(tert-butoxy)-3-oxo-1-propenyl]-5-hydroxy...)
Affinity DataKi:  2.17E+4nMAssay Description:Displacement of [20-3H]PDBu from recombinant PKC alpha in presence of phosphatidylserineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Homo sapiens (Human))
Korea Institute Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50185957(CHEMBL205767 | N-(2-isopropoxybenzyl)-N-(4-chloro-...)
Affinity DataIC50:  0.920nMAssay Description:Inhibition of TSPO (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Homo sapiens (Human))
Korea Institute Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM22032(1-(2-chlorophenyl)-N-methyl-N-(1-methylpropyl)isoq...)
Affinity DataIC50:  1.10nMAssay Description:Inhibition of TSPO (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
Korea Institute Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM22032(1-(2-chlorophenyl)-N-methyl-N-(1-methylpropyl)isoq...)
Affinity DataIC50:  1.30nMAssay Description:Displacement of [3H]PK11195 from TSPO in Sprague-Dawley rat cerebral cortex membranes after 60 mins by microbeta liquid scintillation counting methodMore data for this Ligand-Target Pair
TargetTranslocator protein(Homo sapiens (Human))
Korea Institute Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50210943(CHEMBL3970955)
Affinity DataIC50:  1.60nMAssay Description:Inhibition of TSPO (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Korea Institute Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50210941(CHEMBL3899686)
Affinity DataIC50:  20nMAssay Description:Inhibition of human ERG expressed in CHOK1 cells by automated patch clamp methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutaminyl-peptide cyclotransferase(Homo sapiens (Human))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50435554(CHEMBL2392817)
Affinity DataIC50:  58nMAssay Description:Inhibition of human glutaminyl cyclase expressed in HEK293 cells using L-glutaminyl-beta-naphthylamine as substrate after 1 hr by fluorometric analys...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
Institute Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50263930(4-(2-(6-methoxybenzofuran-2-yl)vinyl)-N,N-dimethyl...)
Affinity DataIC50:  70nMAssay Description:Inhibition of amyloid beta42 fibril formation by thioflavin T formationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
Korea Institute Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50210940(CHEMBL3948914)
Affinity DataIC50:  74nMAssay Description:Displacement of [3H]PK11195 from TSPO in Sprague-Dawley rat cerebral cortex membranes after 60 mins by microbeta liquid scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
Institute Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50263997(4-(2-(5-methoxybenzofuran-2-yl)vinyl)-N-methylbenz...)
Affinity DataIC50:  80nMAssay Description:Inhibition of amyloid beta42 fibril formation by thioflavin T formationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
Institute Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50477454(CHEMBL245688)
Affinity DataIC50:  100nMAssay Description:Inhibition of amyloid beta 42 fibril formation by thioflavin T assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGlutaminyl-peptide cyclotransferase(Homo sapiens (Human))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50299853(1-(3,4-Dimethoxyphenyl)-3-(3-(5-methyl-1H-imidazol...)
Affinity DataIC50:  119nMAssay Description:Inhibition of human glutaminyl cyclase expressed in HEK293 cells using L-glutaminyl-beta-naphthylamine as substrate after 1 hr by fluorometric analys...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutaminyl-peptide cyclotransferase(Homo sapiens (Human))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50435549(CHEMBL2392800)
Affinity DataIC50:  123nMAssay Description:Inhibition of human glutaminyl cyclase expressed in HEK293 cells using L-glutaminyl-beta-naphthylamine as substrate after 1 hr by fluorometric analys...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
Institute Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50263881(CHEMBL509088 | N,N-dimethyl-4-(2-(5-methylbenzofur...)
Affinity DataIC50:  130nMAssay Description:Inhibition of amyloid beta42 fibril formation by thioflavin T formationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutaminyl-peptide cyclotransferase(Homo sapiens (Human))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50435533(CHEMBL2392794)
Affinity DataIC50:  158nMAssay Description:Inhibition of human glutaminyl cyclase expressed in HEK293 cells using L-glutaminyl-beta-naphthylamine as substrate after 1 hr by fluorometric analys...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
Institute Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50263880(2-(4-(dimethylamino)styryl)benzofuran-5-ol | CHEMB...)
Affinity DataIC50:  160nMAssay Description:Inhibition of amyloid beta42 fibril formation by thioflavin T formationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
Institute Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50264047(2-methoxy-4-(2-(5-methoxybenzofuran-2-yl)vinyl)-N,...)
Affinity DataIC50:  160nMAssay Description:Inhibition of amyloid beta42 fibril formation by thioflavin T formationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
Institute Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50263885(4-(2-(5-iodobenzofuran-2-yl)vinyl)-N,N-dimethylben...)
Affinity DataIC50:  170nMAssay Description:Inhibition of amyloid beta42 fibril formation by thioflavin T formationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutaminyl-peptide cyclotransferase(Homo sapiens (Human))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50435561(CHEMBL2392810)
Affinity DataIC50:  185nMAssay Description:Inhibition of human glutaminyl cyclase expressed in HEK293 cells using L-glutaminyl-beta-naphthylamine as substrate after 1 hr by fluorometric analys...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
Institute Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50263883(4-(2-(5-chlorobenzofuran-2-yl)vinyl)-N,N-dimethylb...)
Affinity DataIC50:  200nMAssay Description:Inhibition of amyloid beta42 fibril formation by thioflavin T formationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutaminyl-peptide cyclotransferase(Homo sapiens (Human))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50435558(CHEMBL2392814)
Affinity DataIC50:  208nMAssay Description:Inhibition of human glutaminyl cyclase expressed in HEK293 cells using L-glutaminyl-beta-naphthylamine as substrate after 1 hr by fluorometric analys...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutaminyl-peptide cyclotransferase(Homo sapiens (Human))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50435547(CHEMBL2392803)
Affinity DataIC50:  239nMAssay Description:Inhibition of human glutaminyl cyclase expressed in HEK293 cells using L-glutaminyl-beta-naphthylamine as substrate after 1 hr by fluorometric analys...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutaminyl-peptide cyclotransferase(Homo sapiens (Human))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50435532(CHEMBL2392778)
Affinity DataIC50:  293nMAssay Description:Inhibition of human glutaminyl cyclase expressed in HEK293 cells using L-glutaminyl-beta-naphthylamine as substrate after 1 hr by fluorometric analys...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
Institute Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50477429(CHEMBL248132)
Affinity DataIC50:  300nMAssay Description:Inhibition of amyloid beta 42 fibril formation by thioflavin T assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGlutaminyl-peptide cyclotransferase(Homo sapiens (Human))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50435539(CHEMBL2392786)
Affinity DataIC50:  329nMAssay Description:Inhibition of human glutaminyl cyclase expressed in HEK293 cells using L-glutaminyl-beta-naphthylamine as substrate after 1 hr by fluorometric analys...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutaminyl-peptide cyclotransferase(Homo sapiens (Human))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50435534(CHEMBL2392793)
Affinity DataIC50:  337nMAssay Description:Inhibition of human glutaminyl cyclase expressed in HEK293 cells using L-glutaminyl-beta-naphthylamine as substrate after 1 hr by fluorometric analys...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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