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Found 95 with Last Name = 'morley' and Initial = 'rm'
TargetGlutamate receptor ionotropic, NMDA 1/2A(Rattus norvegicus (Rat))
University Walk

Curated by ChEMBL
LigandPNGBDBM50111396(CHEMBL273636 | [[(S)-1-(4-Bromo-phenyl)-ethylamino...)
Affinity DataKi:  5.40nMAssay Description:Inhibitory constant against (S)-glutamate and glycine evoked currents mediated by N-methyl-D-aspartate glutamate receptor NR1a/NR2A expressed in Xeno...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1/2C(RAT)
University Walk

Curated by ChEMBL
LigandPNGBDBM50111396(CHEMBL273636 | [[(S)-1-(4-Bromo-phenyl)-ethylamino...)
Affinity DataKi:  11.6nMAssay Description:Inhibitory constant against (S)-glutamate and glycine evoked currents mediated by N-methyl-D-aspartate glutamate receptor NR1a/NR2C expressed in Xeno...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1/2A(Rattus norvegicus (Rat))
University Walk

Curated by ChEMBL
LigandPNGBDBM50050704((R)-4-(3-Phosphono-propyl)-piperazine-2-carboxylic...)
Affinity DataKi:  41nMAssay Description:Inhibitory constant against (S)-glutamate and glycine evoked currents mediated by N-methyl-D-aspartate glutamate receptor NR1a/NR2A expressed in Xeno...More data for this Ligand-Target Pair
TargetGlutamate receptor ionotropic, NMDA 1/2B(Rattus norvegicus (Rat))
University Walk

Curated by ChEMBL
LigandPNGBDBM50111396(CHEMBL273636 | [[(S)-1-(4-Bromo-phenyl)-ethylamino...)
Affinity DataKi:  67nMAssay Description:Inhibitory constant against (S)-glutamate and glycine evoked currents mediated by N-methyl-D-aspartate glutamate receptor NR1a/NR2B expressed in Xeno...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1/2C(RAT)
University Walk

Curated by ChEMBL
LigandPNGBDBM50164540((2R,3S)-1-(Phenanthrene-2-carbonyl)-piperazine-2,3...)
Affinity DataKi:  96nMAssay Description:Inhibitory constant against (S)-glutamate and glycine evoked currents mediated by N-methyl-D-aspartate glutamate receptor NR1a/NR2C expressed in Xeno...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1/2C(RAT)
University Walk

Curated by ChEMBL
LigandPNGBDBM50164549((2R,3S)-1-(7-Bromo-phenanthrene-2-carbonyl)-pipera...)
Affinity DataKi:  99.4nMAssay Description:Inhibitory constant against (S)-glutamate and glycine evoked currents mediated by N-methyl-D-aspartate glutamate receptor NR1a/NR2C expressed in Xeno...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1/2B(Rattus norvegicus (Rat))
University Walk

Curated by ChEMBL
LigandPNGBDBM50164549((2R,3S)-1-(7-Bromo-phenanthrene-2-carbonyl)-pipera...)
Affinity DataKi:  250nMAssay Description:Inhibitory constant against (S)-glutamate and glycine evoked currents mediated by N-methyl-D-aspartate glutamate receptor NR1a/NR2B expressed in Xeno...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1/2B(Rattus norvegicus (Rat))
University Walk

Curated by ChEMBL
LigandPNGBDBM50050704((R)-4-(3-Phosphono-propyl)-piperazine-2-carboxylic...)
Affinity DataKi:  270nMAssay Description:Inhibitory constant against (S)-glutamate and glycine evoked currents mediated by N-methyl-D-aspartate glutamate receptor NR1a/NR2B expressed in Xeno...More data for this Ligand-Target Pair
TargetGlutamate receptor ionotropic, NMDA 1/2A(Rattus norvegicus (Rat))
University Walk

Curated by ChEMBL
LigandPNGBDBM50004897((APV)2-Amino-5-phosphono-pentanoic acid | (R)-2-Am...)
Affinity DataKi:  280nMAssay Description:Inhibitory constant against (S)-glutamate and glycine evoked currents mediated by N-methyl-D-aspartate glutamate receptor NR1a/NR2A expressed in Xeno...More data for this Ligand-Target Pair
TargetGlutamate receptor ionotropic, NMDA 1/2C(RAT)
University Walk

Curated by ChEMBL
LigandPNGBDBM50164555((2R,3S)-1-(9,10-Dihydro-phenanthrene-2-carbonyl)-p...)
Affinity DataKi:  290nMAssay Description:Inhibitory constant against (S)-glutamate and glycine evoked currents mediated by N-methyl-D-aspartate glutamate receptor NR1a/NR2C expressed in Xeno...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1/2B(Rattus norvegicus (Rat))
University Walk

Curated by ChEMBL
LigandPNGBDBM50164556((2R,3S)-1-((E)-3-Naphthalen-2-yl-acryloyl)-piperaz...)
Affinity DataKi:  300nMAssay Description:Inhibitory constant against (S)-glutamate and glycine evoked currents mediated by N-methyl-D-aspartate glutamate receptor NR1a/NR2B expressed in Xeno...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1/2B(Rattus norvegicus (Rat))
University Walk

Curated by ChEMBL
LigandPNGBDBM50164540((2R,3S)-1-(Phenanthrene-2-carbonyl)-piperazine-2,3...)
Affinity DataKi:  310nMAssay Description:Inhibitory constant against (S)-glutamate and glycine evoked currents mediated by N-methyl-D-aspartate glutamate receptor NR1a/NR2B expressed in Xeno...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1/2A(Rattus norvegicus (Rat))
University Walk

Curated by ChEMBL
LigandPNGBDBM50164549((2R,3S)-1-(7-Bromo-phenanthrene-2-carbonyl)-pipera...)
Affinity DataKi:  320nMAssay Description:Inhibitory constant against (S)-glutamate and glycine evoked currents mediated by N-methyl-D-aspartate glutamate receptor NR1a/NR2A expressed in Xeno...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1/2B(Rattus norvegicus (Rat))
University Walk

Curated by ChEMBL
LigandPNGBDBM50004897((APV)2-Amino-5-phosphono-pentanoic acid | (R)-2-Am...)
Affinity DataKi:  460nMAssay Description:Inhibitory constant against (S)-glutamate and glycine evoked currents mediated by N-methyl-D-aspartate glutamate receptor NR1a/NR2B expressed in Xeno...More data for this Ligand-Target Pair
TargetGlutamate receptor ionotropic, NMDA 1/2A(Rattus norvegicus (Rat))
University Walk

Curated by ChEMBL
LigandPNGBDBM50017226((R)-2-Amino-7-phosphono-heptanoic acid | 2-Amino-7...)
Affinity DataKi:  490nMAssay Description:Inhibitory constant against (S)-glutamate and glycine evoked currents mediated by N-methyl-D-aspartate glutamate receptor NR1a/NR2A expressed in Xeno...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1/2A(Rattus norvegicus (Rat))
University Walk

Curated by ChEMBL
LigandPNGBDBM50164540((2R,3S)-1-(Phenanthrene-2-carbonyl)-piperazine-2,3...)
Affinity DataKi:  550nMAssay Description:Inhibitory constant against (S)-glutamate and glycine evoked currents mediated by N-methyl-D-aspartate glutamate receptor NR1a/NR2A expressed in Xeno...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1/2C(RAT)
University Walk

Curated by ChEMBL
LigandPNGBDBM50050704((R)-4-(3-Phosphono-propyl)-piperazine-2-carboxylic...)
Affinity DataKi:  630nMAssay Description:Inhibitory constant against (S)-glutamate and glycine evoked currents mediated by N-methyl-D-aspartate glutamate receptor NR1a/NR2C expressed in Xeno...More data for this Ligand-Target Pair
TargetGlutamate receptor ionotropic, NMDA 1/2C(RAT)
University Walk

Curated by ChEMBL
LigandPNGBDBM50164548((2R,3S)-1-(7-Bromo-9,10-dihydro-phenanthrene-2-car...)
Affinity DataKi:  660nMAssay Description:Inhibitory constant against (S)-glutamate and glycine evoked currents mediated by N-methyl-D-aspartate glutamate receptor NR1a/NR2C expressed in Xeno...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1/2B(Rattus norvegicus (Rat))
University Walk

Curated by ChEMBL
LigandPNGBDBM50164555((2R,3S)-1-(9,10-Dihydro-phenanthrene-2-carbonyl)-p...)
Affinity DataKi:  760nMAssay Description:Inhibitory constant against (S)-glutamate and glycine evoked currents mediated by N-methyl-D-aspartate glutamate receptor NR1a/NR2B expressed in Xeno...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1/2A(Rattus norvegicus (Rat))
University Walk

Curated by ChEMBL
LigandPNGBDBM50164556((2R,3S)-1-((E)-3-Naphthalen-2-yl-acryloyl)-piperaz...)
Affinity DataKi:  840nMAssay Description:Inhibitory constant against (S)-glutamate and glycine evoked currents mediated by N-methyl-D-aspartate glutamate receptor NR1a/NR2A expressed in Xeno...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1/2C(RAT)
University Walk

Curated by ChEMBL
LigandPNGBDBM50164556((2R,3S)-1-((E)-3-Naphthalen-2-yl-acryloyl)-piperaz...)
Affinity DataKi:  850nMAssay Description:Inhibitory constant against (S)-glutamate and glycine evoked currents mediated by N-methyl-D-aspartate glutamate receptor NR1a/NR2C expressed in Xeno...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 2(Rattus norvegicus)
University Walk

Curated by ChEMBL
LigandPNGBDBM50185321(6-cyano-7-nitroquinoxaline-2,3-dione | 7-nitro-2,3...)
Affinity DataKi:  1.05E+3nMAssay Description:Displacement of [3H]kainate from rat GLUK6 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1/2C(RAT)
University Walk

Curated by ChEMBL
LigandPNGBDBM50164546((2R,3S)-1-(9H-Fluorene-2-carbonyl)-piperazine-2,3-...)
Affinity DataKi:  1.17E+3nMAssay Description:Inhibitory constant against (S)-glutamate and glycine evoked currents mediated by N-methyl-D-aspartate glutamate receptor NR1a/NR2C expressed in Xeno...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1/2A(Rattus norvegicus (Rat))
University Walk

Curated by ChEMBL
LigandPNGBDBM50164555((2R,3S)-1-(9,10-Dihydro-phenanthrene-2-carbonyl)-p...)
Affinity DataKi:  1.54E+3nMAssay Description:Inhibitory constant against (S)-glutamate and glycine evoked currents mediated by N-methyl-D-aspartate glutamate receptor NR1a/NR2A expressed in Xeno...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1/2C(RAT)
University Walk

Curated by ChEMBL
LigandPNGBDBM50004897((APV)2-Amino-5-phosphono-pentanoic acid | (R)-2-Am...)
Affinity DataKi:  1.64E+3nMAssay Description:Inhibitory constant against (S)-glutamate and glycine evoked currents mediated by N-methyl-D-aspartate glutamate receptor NR1a/NR2C expressed in Xeno...More data for this Ligand-Target Pair
TargetGlutamate receptor ionotropic, NMDA 1/2B(Rattus norvegicus (Rat))
University Walk

Curated by ChEMBL
LigandPNGBDBM50164548((2R,3S)-1-(7-Bromo-9,10-dihydro-phenanthrene-2-car...)
Affinity DataKi:  2.15E+3nMAssay Description:Inhibitory constant against (S)-glutamate and glycine evoked currents mediated by N-methyl-D-aspartate glutamate receptor NR1a/NR2B expressed in Xeno...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1/2C(RAT)
University Walk

Curated by ChEMBL
LigandPNGBDBM50164541((2R,3S)-1-Phenanthren-2-ylmethyl-piperazine-2,3-di...)
Affinity DataKi:  2.67E+3nMAssay Description:Inhibitory constant against (S)-glutamate and glycine evoked currents mediated by N-methyl-D-aspartate glutamate receptor NR1a/NR2C expressed in Xeno...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1/2B(Rattus norvegicus (Rat))
University Walk

Curated by ChEMBL
LigandPNGBDBM50164546((2R,3S)-1-(9H-Fluorene-2-carbonyl)-piperazine-2,3-...)
Affinity DataKi:  3.25E+3nMAssay Description:Inhibitory constant against (S)-glutamate and glycine evoked currents mediated by N-methyl-D-aspartate glutamate receptor NR1a/NR2B expressed in Xeno...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, kainate 2(Rattus norvegicus)
University Walk

Curated by ChEMBL
LigandPNGBDBM26431((2R)-2-aminopentanedioic acid | CHEMBL76232 | D-Gl...)
Affinity DataKi:  3.28E+3nMAssay Description:Displacement of [3H]kainate from rat GLUK6 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1/2A(Rattus norvegicus (Rat))
University Walk

Curated by ChEMBL
LigandPNGBDBM50164548((2R,3S)-1-(7-Bromo-9,10-dihydro-phenanthrene-2-car...)
Affinity DataKi:  3.88E+3nMAssay Description:Inhibitory constant against (S)-glutamate and glycine evoked currents mediated by N-methyl-D-aspartate glutamate receptor NR1a/NR2A expressed in Xeno...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1/2C(RAT)
University Walk

Curated by ChEMBL
LigandPNGBDBM50164551((2R,3S)-1-(Naphthalene-2-carbonyl)-piperazine-2,3-...)
Affinity DataKi:  3.89E+3nMAssay Description:Inhibitory constant against (S)-glutamate and glycine evoked currents mediated by N-methyl-D-aspartate glutamate receptor NR1a/NR2C expressed in Xeno...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1/2B(Rattus norvegicus (Rat))
University Walk

Curated by ChEMBL
LigandPNGBDBM50017226((R)-2-Amino-7-phosphono-heptanoic acid | 2-Amino-7...)
Affinity DataKi:  4.14E+3nMAssay Description:Inhibitory constant against (S)-glutamate and glycine evoked currents mediated by N-methyl-D-aspartate glutamate receptor NR1a/NR2B expressed in Xeno...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1/2C(RAT)
University Walk

Curated by ChEMBL
LigandPNGBDBM50164553((2R,3S)-1-(Phenanthrene-3-carbonyl)-piperazine-2,3...)
Affinity DataKi:  4.22E+3nMAssay Description:Inhibitory constant against (S)-glutamate and glycine evoked currents mediated by N-methyl-D-aspartate glutamate receptor NR1a/NR2C expressed in Xeno...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1/2C(RAT)
University Walk

Curated by ChEMBL
LigandPNGBDBM50164545((2R,3S)-1-(9-Oxo-9H-fluorene-2-carbonyl)-piperazin...)
Affinity DataKi:  4.42E+3nMAssay Description:Inhibitory constant against (S)-glutamate and glycine evoked currents mediated by N-methyl-D-aspartate glutamate receptor NR1a/NR2C expressed in Xeno...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1/2C(RAT)
University Walk

Curated by ChEMBL
LigandPNGBDBM50164543((2R,3R)-1-(Phenanthrene-2-carbonyl)-piperazine-2,3...)
Affinity DataKi:  4.88E+3nMAssay Description:Inhibitory constant against (S)-glutamate and glycine evoked currents mediated by N-methyl-D-aspartate glutamate receptor NR1a/NR2C expressed in Xeno...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1/2B(Rattus norvegicus (Rat))
University Walk

Curated by ChEMBL
LigandPNGBDBM50164552((2R,3S)-1-(Biphenyl-4-carbonyl)-piperazine-2,3-dic...)
Affinity DataKi:  5.01E+3nMAssay Description:Inhibitory constant against (S)-glutamate and glycine evoked currents mediated by N-methyl-D-aspartate glutamate receptor NR1a/NR2B expressed in Xeno...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1/2C(RAT)
University Walk

Curated by ChEMBL
LigandPNGBDBM50017226((R)-2-Amino-7-phosphono-heptanoic acid | 2-Amino-7...)
Affinity DataKi:  6.42E+3nMAssay Description:Inhibitory constant against (S)-glutamate and glycine evoked currents mediated by N-methyl-D-aspartate glutamate receptor NR1a/NR2C expressed in Xeno...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1/2C(RAT)
University Walk

Curated by ChEMBL
LigandPNGBDBM50164550((2R,3S)-1-(4'-Fluoro-biphenyl-4-carbonyl)-piperazi...)
Affinity DataKi:  7.38E+3nMAssay Description:Inhibitory constant against (S)-glutamate and glycine evoked currents mediated by N-methyl-D-aspartate glutamate receptor NR1a/NR2C expressed in Xeno...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1/2A(Rattus norvegicus (Rat))
University Walk

Curated by ChEMBL
LigandPNGBDBM50164545((2R,3S)-1-(9-Oxo-9H-fluorene-2-carbonyl)-piperazin...)
Affinity DataKi:  7.97E+3nMAssay Description:Inhibitory constant against (S)-glutamate and glycine evoked currents mediated by N-methyl-D-aspartate glutamate receptor NR1a/NR2A expressed in Xeno...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1/2C(RAT)
University Walk

Curated by ChEMBL
LigandPNGBDBM50164542((2R,3S)-1-(2'-Bromo-biphenyl-4-carbonyl)-piperazin...)
Affinity DataKi:  8.49E+3nMAssay Description:Inhibitory constant against (S)-glutamate and glycine evoked currents mediated by N-methyl-D-aspartate glutamate receptor NR1a/NR2C expressed in Xeno...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1/2C(RAT)
University Walk

Curated by ChEMBL
LigandPNGBDBM50164544((2R,3S)-1-(Biphenyl-4-sulfonyl)-piperazine-2,3-dic...)
Affinity DataKi:  8.67E+3nMAssay Description:Inhibitory constant against (S)-glutamate and glycine evoked currents mediated by N-methyl-D-aspartate glutamate receptor NR1a/NR2C expressed in Xeno...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1/2A(Rattus norvegicus (Rat))
University Walk

Curated by ChEMBL
LigandPNGBDBM50164550((2R,3S)-1-(4'-Fluoro-biphenyl-4-carbonyl)-piperazi...)
Affinity DataKi:  8.78E+3nMAssay Description:Inhibitory constant against (S)-glutamate and glycine evoked currents mediated by N-methyl-D-aspartate glutamate receptor NR1a/NR2A expressed in Xeno...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1/2C(RAT)
University Walk

Curated by ChEMBL
LigandPNGBDBM50164552((2R,3S)-1-(Biphenyl-4-carbonyl)-piperazine-2,3-dic...)
Affinity DataKi:  8.98E+3nMAssay Description:Inhibitory constant against (S)-glutamate and glycine evoked currents mediated by N-methyl-D-aspartate glutamate receptor NR1a/NR2C expressed in Xeno...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1/2B(Rattus norvegicus (Rat))
University Walk

Curated by ChEMBL
LigandPNGBDBM50164543((2R,3R)-1-(Phenanthrene-2-carbonyl)-piperazine-2,3...)
Affinity DataKi:  9.08E+3nMAssay Description:Inhibitory constant against (S)-glutamate and glycine evoked currents mediated by N-methyl-D-aspartate glutamate receptor NR1a/NR2B expressed in Xeno...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1/2B(Rattus norvegicus (Rat))
University Walk

Curated by ChEMBL
LigandPNGBDBM50164545((2R,3S)-1-(9-Oxo-9H-fluorene-2-carbonyl)-piperazin...)
Affinity DataKi:  9.36E+3nMAssay Description:Inhibitory constant against (S)-glutamate and glycine evoked currents mediated by N-methyl-D-aspartate glutamate receptor NR1a/NR2B expressed in Xeno...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1/2A(Rattus norvegicus (Rat))
University Walk

Curated by ChEMBL
LigandPNGBDBM50164551((2R,3S)-1-(Naphthalene-2-carbonyl)-piperazine-2,3-...)
Affinity DataKi:  9.60E+3nMAssay Description:Inhibitory constant against (S)-glutamate and glycine evoked currents mediated by N-methyl-D-aspartate glutamate receptor NR1a/NR2A expressed in Xeno...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1/2B(Rattus norvegicus (Rat))
University Walk

Curated by ChEMBL
LigandPNGBDBM50164541((2R,3S)-1-Phenanthren-2-ylmethyl-piperazine-2,3-di...)
Affinity DataKi:  1.03E+4nMAssay Description:Inhibitory constant against (S)-glutamate and glycine evoked currents mediated by N-methyl-D-aspartate glutamate receptor NR1a/NR2B expressed in Xeno...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1/2A(Rattus norvegicus (Rat))
University Walk

Curated by ChEMBL
LigandPNGBDBM50164543((2R,3R)-1-(Phenanthrene-2-carbonyl)-piperazine-2,3...)
Affinity DataKi:  1.05E+4nMAssay Description:Inhibitory constant against (S)-glutamate and glycine evoked currents mediated by N-methyl-D-aspartate glutamate receptor NR1a/NR2A expressed in Xeno...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1/2A(Rattus norvegicus (Rat))
University Walk

Curated by ChEMBL
LigandPNGBDBM50164541((2R,3S)-1-Phenanthren-2-ylmethyl-piperazine-2,3-di...)
Affinity DataKi:  1.12E+4nMAssay Description:Inhibitory constant against (S)-glutamate and glycine evoked currents mediated by N-methyl-D-aspartate glutamate receptor NR1a/NR2A expressed in Xeno...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1/2A(Rattus norvegicus (Rat))
University Walk

Curated by ChEMBL
LigandPNGBDBM50164554((2R,3S)-1-[(E)-(3-Phenyl-acryloyl)]-piperazine-2,3...)
Affinity DataKi:  1.32E+4nMAssay Description:Inhibitory constant against (S)-glutamate and glycine evoked currents mediated by N-methyl-D-aspartate glutamate receptor NR1a/NR2A expressed in Xeno...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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