Affinity DataKi: 6.70nMAssay Description:Displacement of [3H]PK11195 from TSPO in human T98G cell membranes incubated for 90 mins by competition radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 8.20nMAssay Description:Inhibition constant against Adenosine A2a receptorMore data for this Ligand-Target Pair
Affinity DataKi: 28nMAssay Description:Inhibition constant against Adenosine A2a receptorMore data for this Ligand-Target Pair
Affinity DataKi: 29nMAssay Description:Displacement of [3H]PK11195 from TSPO in human T98G cell membranes incubated for 90 mins by competition radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 43nMAssay Description:Displacement of [3H]DPCX from human adenosine A1 receptor expressed in CHO cells at high affinity site by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 114nMAssay Description:Displacement of [3H]DPCX from human adenosine A1 receptor expressed in CHO cells by scintillation counting in presence of 10 uM allosteric modulator ...More data for this Ligand-Target Pair
Affinity DataKi: 144nMAssay Description:Inhibition constant against Adenosine A2a receptorMore data for this Ligand-Target Pair
Affinity DataKi: 195nMAssay Description:Displacement of [3H]DPCX from human adenosine A1 receptor expressed in CHO cells by scintillation counting in presence of 10 uM allosteric modulator ...More data for this Ligand-Target Pair
Affinity DataKi: 214nMAssay Description:Displacement of [3H]DPCX from human adenosine A1 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 224nMAssay Description:Displacement of [3H]PK11195 from TSPO in human T98G cell membranes incubated for 90 mins by competition radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 268nMAssay Description:Displacement of [3H]DPCX from human adenosine A1 receptor expressed in CHO cells by scintillation counting in presence of 10 uM allosteric modulator ...More data for this Ligand-Target Pair
Affinity DataKi: 288nMAssay Description:Displacement of [3H]DPCX from human adenosine A1 receptor expressed in CHO cells by scintillation counting in presence of 10 uM allosteric modulator ...More data for this Ligand-Target Pair
Affinity DataKi: 313nMAssay Description:Displacement of [3H]DPCX from human adenosine A1 receptor expressed in CHO cells by scintillation counting in presence of 10 uM allosteric modulator ...More data for this Ligand-Target Pair
Affinity DataKi: 347nMAssay Description:Displacement of [3H]DPCX from human adenosine A1 receptor expressed in CHO cells by scintillation counting in presence of 10 uM allosteric modulator ...More data for this Ligand-Target Pair
Affinity DataKi: 398nMAssay Description:Inhibition constant against Adenosine A2a receptorMore data for this Ligand-Target Pair
Affinity DataKi: 417nMAssay Description:Displacement of [3H]DPCX from human adenosine A1 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 419nMAssay Description:Displacement of [3H]DPCX from human adenosine A1 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 450nMAssay Description:Displacement of [3H]DPCX from human adenosine A1 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 457nMAssay Description:Displacement of [3H]DPCX from human adenosine A1 receptor expressed in CHO cells by scintillation counting in presence of 10 uM allosteric modulator ...More data for this Ligand-Target Pair
Affinity DataKi: 469nMAssay Description:Displacement of [3H]DPCX from human adenosine A1 receptor expressed in CHO cells by scintillation counting in presence of 10 uM allosteric modulator ...More data for this Ligand-Target Pair
Affinity DataKi: 618nMAssay Description:Displacement of [3H]DPCX from human adenosine A1 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 651nMAssay Description:Displacement of [3H]DPCX from human adenosine A1 receptor expressed in CHO cells by scintillation counting in presence of 10 uM allosteric modulator ...More data for this Ligand-Target Pair
Affinity DataKi: 661nMAssay Description:Displacement of [3H]DPCX from human adenosine A1 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 741nMAssay Description:Displacement of [3H]DPCX from human adenosine A1 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 776nMAssay Description:Displacement of [3H]DPCX from human adenosine A1 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 806nMAssay Description:Displacement of [3H]PK11195 from TSPO in human T98G cell membranes incubated for 90 mins by competition radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 832nMAssay Description:Displacement of [3H]DPCX from human adenosine A1 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 1.26E+3nMAssay Description:Displacement of [3H]DPCX from human adenosine A1 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 1.36E+3nMAssay Description:Displacement of [3H]DPCX from human adenosine A1 receptor expressed in CHO cells by scintillation counting in presence of 10 uM allosteric modulator ...More data for this Ligand-Target Pair
Affinity DataKi: 1.86E+3nMAssay Description:Displacement of [3H]DPCX from human adenosine A1 receptor expressed in CHO cells at low affinity site by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition constant against Adenosine A2a receptorMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]PK11195 from TSPO in human T98G cell membranes incubated for 90 mins by competition radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataIC50: 7.10nMAssay Description:Effect on gamma-secretase activity in human H4 cells expressing APP695 assessed as reduction of Amyloid beta42 formation LPECL assayMore data for this Ligand-Target Pair
TargetLutropin-choriogonadotropic hormone receptor(Homo sapiens (Human))
Leiden University
Curated by ChEMBL
Leiden University
Curated by ChEMBL
Affinity DataIC50: 2.30E+3nMAssay Description:Displacement of [3H]Org43553 from human luteinizing hormone receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 2.90E+3nMAssay Description:Effect on gamma-secretase activity in human H4 cells expressing APP695 assessed as reduction of Amyloid beta42 formation LPECL assayMore data for this Ligand-Target Pair
Affinity DataIC50: 2.90E+3nMAssay Description:Effect on gamma-secretase activity in human H4 cells expressing APP695 assessed as reduction of Amyloid beta-42 formation LPECL assayMore data for this Ligand-Target Pair
Affinity DataIC50: 4.50E+3nMAssay Description:Effect on gamma-secretase activity in human H4 cells expressing APP695 assessed as reduction of Amyloid beta-38 formation by LPECL assayMore data for this Ligand-Target Pair
Affinity DataIC50: 5.80E+3nMAssay Description:Effect on gamma-secretase activity in human H4 cells expressing APP695 assessed as increase in Amyloid beta-38 formation by LPECL assayMore data for this Ligand-Target Pair
Affinity DataIC50: 7.50E+3nMAssay Description:Effect on gamma-secretase activity in human H4 cells expressing APP695 assessed as reduction of Amyloid beta-42 formation LPECL assayMore data for this Ligand-Target Pair
Affinity DataIC50: 7.50E+3nMAssay Description:Effect on gamma-secretase activity in human H4 cells expressing APP695 assessed as reduction of Amyloid beta42 formation LPECL assayMore data for this Ligand-Target Pair
Affinity DataIC50: 7.80E+3nMAssay Description:Effect on gamma-secretase activity in human H4 cells expressing APP695 assessed as increase in Amyloid beta-38 formation by LPECL assayMore data for this Ligand-Target Pair
Affinity DataIC50: 8.50E+3nMAssay Description:Effect on gamma-secretase activity in human H4 cells expressing APP695 assessed as reduction of Amyloid beta42 formation LPECL assayMore data for this Ligand-Target Pair
Affinity DataIC50: 8.50E+3nMAssay Description:Effect on gamma-secretase activity in human H4 cells expressing APP695 assessed as reduction of Amyloid beta-42 formation LPECL assayMore data for this Ligand-Target Pair
Affinity DataIC50: 9.30E+3nMAssay Description:Effect on gamma-secretase activity in human H4 cells expressing APP695 assessed as increase in Amyloid beta-38 formation by LPECL assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.10E+4nMAssay Description:Effect on gamma-secretase activity in human H4 cells expressing APP695 assessed as reduction of Amyloid beta-42 formation LPECL assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.10E+4nMAssay Description:Effect on gamma-secretase activity in human H4 cells expressing APP695 assessed as reduction of Amyloid beta42 formation LPECL assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.30E+4nMAssay Description:Effect on gamma-secretase activity in human H4 cells expressing APP695 assessed as increase in Amyloid beta-38 formation by LPECL assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.30E+4nMAssay Description:Effect on gamma-secretase activity in human H4 cells expressing APP695 assessed as increase in Amyloid beta-38 formation by LPECL assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.30E+4nMAssay Description:Effect on gamma-secretase activity in human H4 cells expressing APP695 assessed as increase in Amyloid beta-38 formation by LPECL assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.33E+4nMAssay Description:Effect on gamma-secretase activity in human H4 cells expressing APP695 assessed as reduction of Amyloid beta-38 formation by LPECL assayMore data for this Ligand-Target Pair