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Found 124 with Last Name = 'narlawar' and Initial = 'r'
TargetTranslocator protein(Homo sapiens (Human))
University Of New South Wales

Curated by ChEMBL
LigandPNGBDBM50327238(2-[2-(4'-Methoxyphenyl)-5,7-dimethylpyrazolo[1,5-a...)
Affinity DataKi:  6.70nMAssay Description:Displacement of [3H]PK11195 from TSPO in human T98G cell membranes incubated for 90 mins by competition radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Homo sapiens (Human))
University Of New South Wales

Curated by ChEMBL
LigandPNGBDBM50327238(2-[2-(4'-Methoxyphenyl)-5,7-dimethylpyrazolo[1,5-a...)
Affinity DataKi:  8.20nMAssay Description:Inhibition constant against Adenosine A2a receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Homo sapiens (Human))
University Of New South Wales

Curated by ChEMBL
LigandPNGBDBM50131400(CHEMBL3634876)
Affinity DataKi:  28nMAssay Description:Inhibition constant against Adenosine A2a receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Homo sapiens (Human))
University Of New South Wales

Curated by ChEMBL
LigandPNGBDBM50131380(CHEMBL3634878)
Affinity DataKi:  29nMAssay Description:Displacement of [3H]PK11195 from TSPO in human T98G cell membranes incubated for 90 mins by competition radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50315857((2R,3S,4R,5R)-2-(hydroxymethyl)-5-(6-(4-methoxyphe...)
Affinity DataKi:  43nMAssay Description:Displacement of [3H]DPCX from human adenosine A1 receptor expressed in CHO cells at high affinity site by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50315861(CHEMBL1090683 | N6-[2-Amino-3-(3,4-dichlorobenzoyl...)
Affinity DataKi:  114nMAssay Description:Displacement of [3H]DPCX from human adenosine A1 receptor expressed in CHO cells by scintillation counting in presence of 10 uM allosteric modulator ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Homo sapiens (Human))
University Of New South Wales

Curated by ChEMBL
LigandPNGBDBM50131380(CHEMBL3634878)
Affinity DataKi:  144nMAssay Description:Inhibition constant against Adenosine A2a receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50315857((2R,3S,4R,5R)-2-(hydroxymethyl)-5-(6-(4-methoxyphe...)
Affinity DataKi:  195nMAssay Description:Displacement of [3H]DPCX from human adenosine A1 receptor expressed in CHO cells by scintillation counting in presence of 10 uM allosteric modulator ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50315861(CHEMBL1090683 | N6-[2-Amino-3-(3,4-dichlorobenzoyl...)
Affinity DataKi:  214nMAssay Description:Displacement of [3H]DPCX from human adenosine A1 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Homo sapiens (Human))
University Of New South Wales

Curated by ChEMBL
LigandPNGBDBM50131399(CHEMBL3634877)
Affinity DataKi:  224nMAssay Description:Displacement of [3H]PK11195 from TSPO in human T98G cell membranes incubated for 90 mins by competition radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50315859(CHEMBL1090681 | N6-[2-Amino-3-(3,4-dichlorobenzoyl...)
Affinity DataKi:  268nMAssay Description:Displacement of [3H]DPCX from human adenosine A1 receptor expressed in CHO cells by scintillation counting in presence of 10 uM allosteric modulator ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50315862(CHEMBL1090684 | N6-[2-Amino-3-(3,4-dichlorobenzoyl...)
Affinity DataKi:  288nMAssay Description:Displacement of [3H]DPCX from human adenosine A1 receptor expressed in CHO cells by scintillation counting in presence of 10 uM allosteric modulator ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50315860(CHEMBL1090682 | N6-[2-Amino-3-(3,4-dichlorobenzoyl...)
Affinity DataKi:  313nMAssay Description:Displacement of [3H]DPCX from human adenosine A1 receptor expressed in CHO cells by scintillation counting in presence of 10 uM allosteric modulator ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50315853(6-[2-Amino-3-(3,4-dichlorobenzoyl)-4,5,6,7-tetrahy...)
Affinity DataKi:  347nMAssay Description:Displacement of [3H]DPCX from human adenosine A1 receptor expressed in CHO cells by scintillation counting in presence of 10 uM allosteric modulator ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Homo sapiens (Human))
University Of New South Wales

Curated by ChEMBL
LigandPNGBDBM50131399(CHEMBL3634877)
Affinity DataKi:  398nMAssay Description:Inhibition constant against Adenosine A2a receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50315859(CHEMBL1090681 | N6-[2-Amino-3-(3,4-dichlorobenzoyl...)
Affinity DataKi:  417nMAssay Description:Displacement of [3H]DPCX from human adenosine A1 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50315862(CHEMBL1090684 | N6-[2-Amino-3-(3,4-dichlorobenzoyl...)
Affinity DataKi:  419nMAssay Description:Displacement of [3H]DPCX from human adenosine A1 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50315853(6-[2-Amino-3-(3,4-dichlorobenzoyl)-4,5,6,7-tetrahy...)
Affinity DataKi:  450nMAssay Description:Displacement of [3H]DPCX from human adenosine A1 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50315854(CHEMBL1090686 | N6-[2-Amino-3-(3,4-dichlorobenzoyl...)
Affinity DataKi:  457nMAssay Description:Displacement of [3H]DPCX from human adenosine A1 receptor expressed in CHO cells by scintillation counting in presence of 10 uM allosteric modulator ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50315858(CHEMBL1090680 | N6-[2-Amino-3-(3,4-dichlorobenzoyl...)
Affinity DataKi:  469nMAssay Description:Displacement of [3H]DPCX from human adenosine A1 receptor expressed in CHO cells by scintillation counting in presence of 10 uM allosteric modulator ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50315860(CHEMBL1090682 | N6-[2-Amino-3-(3,4-dichlorobenzoyl...)
Affinity DataKi:  618nMAssay Description:Displacement of [3H]DPCX from human adenosine A1 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50315855(CHEMBL1090687 | LUF-6258 | N6-[2-Amino-3-(3,4-dich...)
Affinity DataKi:  651nMAssay Description:Displacement of [3H]DPCX from human adenosine A1 receptor expressed in CHO cells by scintillation counting in presence of 10 uM allosteric modulator ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50315855(CHEMBL1090687 | LUF-6258 | N6-[2-Amino-3-(3,4-dich...)
Affinity DataKi:  661nMAssay Description:Displacement of [3H]DPCX from human adenosine A1 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50315858(CHEMBL1090680 | N6-[2-Amino-3-(3,4-dichlorobenzoyl...)
Affinity DataKi:  741nMAssay Description:Displacement of [3H]DPCX from human adenosine A1 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50315854(CHEMBL1090686 | N6-[2-Amino-3-(3,4-dichlorobenzoyl...)
Affinity DataKi:  776nMAssay Description:Displacement of [3H]DPCX from human adenosine A1 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Homo sapiens (Human))
University Of New South Wales

Curated by ChEMBL
LigandPNGBDBM50131400(CHEMBL3634876)
Affinity DataKi:  806nMAssay Description:Displacement of [3H]PK11195 from TSPO in human T98G cell membranes incubated for 90 mins by competition radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50315857((2R,3S,4R,5R)-2-(hydroxymethyl)-5-(6-(4-methoxyphe...)
Affinity DataKi:  832nMAssay Description:Displacement of [3H]DPCX from human adenosine A1 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50315856(CHEMBL1090688 | N6-[2-Amino-3-(3,4-dichlorobenzoyl...)
Affinity DataKi:  1.26E+3nMAssay Description:Displacement of [3H]DPCX from human adenosine A1 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50315856(CHEMBL1090688 | N6-[2-Amino-3-(3,4-dichlorobenzoyl...)
Affinity DataKi:  1.36E+3nMAssay Description:Displacement of [3H]DPCX from human adenosine A1 receptor expressed in CHO cells by scintillation counting in presence of 10 uM allosteric modulator ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50315857((2R,3S,4R,5R)-2-(hydroxymethyl)-5-(6-(4-methoxyphe...)
Affinity DataKi:  1.86E+3nMAssay Description:Displacement of [3H]DPCX from human adenosine A1 receptor expressed in CHO cells at low affinity site by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Homo sapiens (Human))
University Of New South Wales

Curated by ChEMBL
LigandPNGBDBM50131379(CHEMBL3634879)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition constant against Adenosine A2a receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Homo sapiens (Human))
University Of New South Wales

Curated by ChEMBL
LigandPNGBDBM50131379(CHEMBL3634879)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]PK11195 from TSPO in human T98G cell membranes incubated for 90 mins by competition radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPresenilin-1(Homo sapiens (Human))
Darmstadt University Of Technology

Curated by ChEMBL
LigandPNGBDBM50477339(BMS-299897 | CHEMBL247471)
Affinity DataIC50:  7.10nMAssay Description:Effect on gamma-secretase activity in human H4 cells expressing APP695 assessed as reduction of Amyloid beta42 formation LPECL assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLutropin-choriogonadotropic hormone receptor(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50256858(CHEMBL474041 | Cyclopentyl-carbamic acid [1,1',3',...)
Affinity DataIC50:  2.30E+3nMAssay Description:Displacement of [3H]Org43553 from human luteinizing hormone receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPresenilin-1(Homo sapiens (Human))
Darmstadt University Of Technology

Curated by ChEMBL
LigandPNGBDBM50477330(CHEMBL218756)
Affinity DataIC50:  2.90E+3nMAssay Description:Effect on gamma-secretase activity in human H4 cells expressing APP695 assessed as reduction of Amyloid beta42 formation LPECL assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPresenilin-1(Homo sapiens (Human))
Darmstadt University Of Technology

Curated by ChEMBL
LigandPNGBDBM50477330(CHEMBL218756)
Affinity DataIC50:  2.90E+3nMAssay Description:Effect on gamma-secretase activity in human H4 cells expressing APP695 assessed as reduction of Amyloid beta-42 formation LPECL assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPresenilin-1(Homo sapiens (Human))
Darmstadt University Of Technology

Curated by ChEMBL
LigandPNGBDBM19993(CHEMBL62136 | N-[4-(1,1,1,3,3,3-hexafluoro-2-hydro...)
Affinity DataIC50:  4.50E+3nMAssay Description:Effect on gamma-secretase activity in human H4 cells expressing APP695 assessed as reduction of Amyloid beta-38 formation by LPECL assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPresenilin-1(Homo sapiens (Human))
Darmstadt University Of Technology

Curated by ChEMBL
LigandPNGBDBM50477330(CHEMBL218756)
Affinity DataIC50:  5.80E+3nMAssay Description:Effect on gamma-secretase activity in human H4 cells expressing APP695 assessed as increase in Amyloid beta-38 formation by LPECL assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPresenilin-1(Homo sapiens (Human))
Darmstadt University Of Technology

Curated by ChEMBL
LigandPNGBDBM50477329(CHEMBL392028)
Affinity DataIC50:  7.50E+3nMAssay Description:Effect on gamma-secretase activity in human H4 cells expressing APP695 assessed as reduction of Amyloid beta-42 formation LPECL assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPresenilin-1(Homo sapiens (Human))
Darmstadt University Of Technology

Curated by ChEMBL
LigandPNGBDBM50477329(CHEMBL392028)
Affinity DataIC50:  7.50E+3nMAssay Description:Effect on gamma-secretase activity in human H4 cells expressing APP695 assessed as reduction of Amyloid beta42 formation LPECL assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPresenilin-1(Homo sapiens (Human))
Darmstadt University Of Technology

Curated by ChEMBL
LigandPNGBDBM50477329(CHEMBL392028)
Affinity DataIC50:  7.80E+3nMAssay Description:Effect on gamma-secretase activity in human H4 cells expressing APP695 assessed as increase in Amyloid beta-38 formation by LPECL assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPresenilin-1(Homo sapiens (Human))
Darmstadt University Of Technology

Curated by ChEMBL
LigandPNGBDBM50477327(CHEMBL385554)
Affinity DataIC50:  8.50E+3nMAssay Description:Effect on gamma-secretase activity in human H4 cells expressing APP695 assessed as reduction of Amyloid beta42 formation LPECL assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPresenilin-1(Homo sapiens (Human))
Darmstadt University Of Technology

Curated by ChEMBL
LigandPNGBDBM50477327(CHEMBL385554)
Affinity DataIC50:  8.50E+3nMAssay Description:Effect on gamma-secretase activity in human H4 cells expressing APP695 assessed as reduction of Amyloid beta-42 formation LPECL assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPresenilin-1(Homo sapiens (Human))
Darmstadt University Of Technology

Curated by ChEMBL
LigandPNGBDBM50477327(CHEMBL385554)
Affinity DataIC50:  9.30E+3nMAssay Description:Effect on gamma-secretase activity in human H4 cells expressing APP695 assessed as increase in Amyloid beta-38 formation by LPECL assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPresenilin-1(Homo sapiens (Human))
Darmstadt University Of Technology

Curated by ChEMBL
LigandPNGBDBM50477335(CHEMBL247693)
Affinity DataIC50:  1.10E+4nMAssay Description:Effect on gamma-secretase activity in human H4 cells expressing APP695 assessed as reduction of Amyloid beta-42 formation LPECL assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPresenilin-1(Homo sapiens (Human))
Darmstadt University Of Technology

Curated by ChEMBL
LigandPNGBDBM50477335(CHEMBL247693)
Affinity DataIC50:  1.10E+4nMAssay Description:Effect on gamma-secretase activity in human H4 cells expressing APP695 assessed as reduction of Amyloid beta42 formation LPECL assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPresenilin-1(Homo sapiens (Human))
Darmstadt University Of Technology

Curated by ChEMBL
LigandPNGBDBM50477338(CHEMBL248090)
Affinity DataIC50:  1.30E+4nMAssay Description:Effect on gamma-secretase activity in human H4 cells expressing APP695 assessed as increase in Amyloid beta-38 formation by LPECL assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPresenilin-1(Homo sapiens (Human))
Darmstadt University Of Technology

Curated by ChEMBL
LigandPNGBDBM50477331(CHEMBL396693)
Affinity DataIC50:  1.30E+4nMAssay Description:Effect on gamma-secretase activity in human H4 cells expressing APP695 assessed as increase in Amyloid beta-38 formation by LPECL assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPresenilin-1(Homo sapiens (Human))
Darmstadt University Of Technology

Curated by ChEMBL
LigandPNGBDBM50477325(CHEMBL248089)
Affinity DataIC50:  1.30E+4nMAssay Description:Effect on gamma-secretase activity in human H4 cells expressing APP695 assessed as increase in Amyloid beta-38 formation by LPECL assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPresenilin-1(Homo sapiens (Human))
Darmstadt University Of Technology

Curated by ChEMBL
LigandPNGBDBM50477641(CHEMBL249201)
Affinity DataIC50:  1.33E+4nMAssay Description:Effect on gamma-secretase activity in human H4 cells expressing APP695 assessed as reduction of Amyloid beta-38 formation by LPECL assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
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