Affinity DataKi: 0.710nMAssay Description:Displacement of [3H]-NPA from rat brain Dopamine receptor D2More data for this Ligand-Target Pair
Affinity DataKi: 2.10nMAssay Description:Displacement of [3H]-NPA from rat brain Dopamine receptor D2More data for this Ligand-Target Pair
Affinity DataKi: 3nMAssay Description:Displacement of [3H]-NPA from rat brain Dopamine receptor D2More data for this Ligand-Target Pair
Affinity DataKi: 3.10nMAssay Description:Displacement of [3H]-NPA from rat brain Dopamine receptor D2More data for this Ligand-Target Pair
Affinity DataKi: 3.70nMAssay Description:Displacement of [3H]-NPA from rat brain Dopamine receptor D2More data for this Ligand-Target Pair
Affinity DataKi: 3.80nMAssay Description:Displacement of [3H]-NPA from rat brain Dopamine receptor D2More data for this Ligand-Target Pair
Affinity DataKi: 4.20nMAssay Description:Displacement of [3H]-NPA from rat brain Dopamine receptor D2More data for this Ligand-Target Pair
Affinity DataKi: 4.20nMAssay Description:Displacement of [3H]-NPA from rat brain Dopamine receptor D2More data for this Ligand-Target Pair
Affinity DataKi: 4.80nMAssay Description:Displacement of [3H]-NPA from rat brain Dopamine receptor D2More data for this Ligand-Target Pair
Affinity DataKi: 5.10nMAssay Description:Displacement of [3H]-NPA from rat brain Dopamine receptor D2More data for this Ligand-Target Pair
Affinity DataKi: 6.30nMAssay Description:Displacement of [3H]-NPA from rat brain Dopamine receptor D2More data for this Ligand-Target Pair
Affinity DataKi: 32nMAssay Description:Inhibition of thrombin (unknown origin) by chromogenic substrate assayMore data for this Ligand-Target Pair
Affinity DataKi: 35nMAssay Description:Inhibition of thrombin (unknown origin) by chromogenic substrate assayMore data for this Ligand-Target Pair
Affinity DataKi: 36nMAssay Description:Inhibition of thrombin (unknown origin) by chromogenic substrate assayMore data for this Ligand-Target Pair
Affinity DataKi: 45nMAssay Description:In vitro ability of the compound to displace [3H]-ketanserin from 5-hydroxytryptamine 2A receptor in rat brain.More data for this Ligand-Target Pair
Affinity DataKi: 78nMAssay Description:Inhibition of thrombin (unknown origin) by chromogenic substrate assayMore data for this Ligand-Target Pair
Affinity DataKi: 83nMAssay Description:Displacement of [3H]-NPA from rat brain Dopamine receptor D2More data for this Ligand-Target Pair
Affinity DataKi: 110nMAssay Description:Inhibition of thrombin (unknown origin) by chromogenic substrate assayMore data for this Ligand-Target Pair
Affinity DataKi: 130nMAssay Description:Inhibition of thrombin (unknown origin) by chromogenic substrate assayMore data for this Ligand-Target Pair
Affinity DataKi: 150nMAssay Description:Inhibition of thrombin (unknown origin) by chromogenic substrate assayMore data for this Ligand-Target Pair
Affinity DataKi: 160nMAssay Description:Inhibition of thrombin (unknown origin) by chromogenic substrate assayMore data for this Ligand-Target Pair
Affinity DataKi: 170nMAssay Description:Inhibition of thrombin (unknown origin) by chromogenic substrate assayMore data for this Ligand-Target Pair
Affinity DataKi: 200nMAssay Description:Inhibition of thrombin (unknown origin) by chromogenic substrate assayMore data for this Ligand-Target Pair
Affinity DataKi: 210nMAssay Description:Inhibition of thrombin (unknown origin) by chromogenic substrate assayMore data for this Ligand-Target Pair
Affinity DataKi: 220nMAssay Description:Inhibition of thrombin (unknown origin) by chromogenic substrate assayMore data for this Ligand-Target Pair
Affinity DataKi: 220nMAssay Description:Inhibition of thrombin (unknown origin) by chromogenic substrate assayMore data for this Ligand-Target Pair
Affinity DataKi: 220nMAssay Description:Inhibition of thrombin (unknown origin) by chromogenic substrate assayMore data for this Ligand-Target Pair
Affinity DataKi: 220nMAssay Description:Inhibition of thrombin (unknown origin) by chromogenic substrate assayMore data for this Ligand-Target Pair
Affinity DataKi: 230nMAssay Description:Inhibition of thrombin (unknown origin) by chromogenic substrate assayMore data for this Ligand-Target Pair
Affinity DataKi: 260nMAssay Description:Inhibition of thrombin (unknown origin) by chromogenic substrate assayMore data for this Ligand-Target Pair
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Novo Nordisk
Curated by ChEMBL
Novo Nordisk
Curated by ChEMBL
Affinity DataKi: 270nMpH: 5.5Assay Description:Inhibitory effect against recombinant human protein-tyrosine phosphatase 1B (PTP1B), using p-nitrophenyl phosphate substrate at pH 5.5.More data for this Ligand-Target Pair
Affinity DataKi: 290nMAssay Description:Inhibition of factor-10a (unknown origin) by chromogenic substrate assayMore data for this Ligand-Target Pair
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Novo Nordisk
Curated by ChEMBL
Novo Nordisk
Curated by ChEMBL
Affinity DataKi: 290nMpH: 5.5Assay Description:Inhibitory effect against recombinant human protein-tyrosine phosphatase 1B (PTP1B), using p-nitrophenyl phosphate substrate at pH 5.5.More data for this Ligand-Target Pair
Affinity DataKi: 360nMAssay Description:Inhibition of thrombin (unknown origin) by chromogenic substrate assayMore data for this Ligand-Target Pair
Affinity DataKi: 380nMAssay Description:Inhibition of thrombin (unknown origin) by chromogenic substrate assayMore data for this Ligand-Target Pair
Affinity DataKi: 550nMAssay Description:Inhibition of factor-10a (unknown origin) by chromogenic substrate assayMore data for this Ligand-Target Pair
Affinity DataKi: 650nMAssay Description:Inhibition of factor-10a (unknown origin) by chromogenic substrate assayMore data for this Ligand-Target Pair
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Novo Nordisk
Curated by ChEMBL
Novo Nordisk
Curated by ChEMBL
Affinity DataKi: 700nMpH: 5.5Assay Description:Inhibitory effect against recombinant human protein-tyrosine phosphatase 1B (PTP1B), using p-nitrophenyl phosphate substrate at pH 5.5.More data for this Ligand-Target Pair
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Novo Nordisk
Curated by ChEMBL
Novo Nordisk
Curated by ChEMBL
Affinity DataKi: 900nMpH: 5.5Assay Description:Inhibitory effect against recombinant human protein-tyrosine phosphatase 1B (PTP1B), using p-nitrophenyl phosphate substrate at pH 5.5.More data for this Ligand-Target Pair
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Novo Nordisk
Curated by ChEMBL
Novo Nordisk
Curated by ChEMBL
Affinity DataKi: 1.00E+3nMpH: 5.5Assay Description:Inhibitory effect against recombinant human protein-tyrosine phosphatase 1B (PTP1B), using p-nitrophenyl phosphate substrate at pH 5.5.More data for this Ligand-Target Pair
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Novo Nordisk
Curated by ChEMBL
Novo Nordisk
Curated by ChEMBL
Affinity DataKi: 1.00E+3nMpH: 5.5Assay Description:Inhibitory effect against recombinant human protein-tyrosine phosphatase 1B (PTP1B), using p-nitrophenyl phosphate substrate at pH 5.5.More data for this Ligand-Target Pair
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Novo Nordisk
Curated by ChEMBL
Novo Nordisk
Curated by ChEMBL
Affinity DataKi: 1.00E+3nMpH: 5.5Assay Description:Inhibitory effect against recombinant human protein-tyrosine phosphatase 1B (PTP1B), using p-nitrophenyl phosphate substrate at pH 5.5.More data for this Ligand-Target Pair
Affinity DataKi: 1.00E+3nMAssay Description:Inhibition of factor-10a (unknown origin) by chromogenic substrate assayMore data for this Ligand-Target Pair
Affinity DataKi: 1.10E+3nMAssay Description:Inhibition of factor-10a (unknown origin) by chromogenic substrate assayMore data for this Ligand-Target Pair
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Novo Nordisk
Curated by ChEMBL
Novo Nordisk
Curated by ChEMBL
Affinity DataKi: 1.10E+3nMpH: 5.5Assay Description:Inhibitory effect against recombinant human protein-tyrosine phosphatase 1B (PTP1B), using p-nitrophenyl phosphate substrate at pH 5.5.More data for this Ligand-Target Pair
Affinity DataKi: 1.20E+3nMAssay Description:Inhibition of thrombin (unknown origin) by chromogenic substrate assayMore data for this Ligand-Target Pair
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Novo Nordisk
Curated by ChEMBL
Novo Nordisk
Curated by ChEMBL
Affinity DataKi: 1.30E+3nMpH: 5.5Assay Description:Inhibitory effect against recombinant human protein-tyrosine phosphatase 1B (PTP1B), using p-nitrophenyl phosphate substrate at pH 5.5.More data for this Ligand-Target Pair
Affinity DataKi: 1.80E+3nMAssay Description:Inhibition of thrombin (unknown origin) by chromogenic substrate assayMore data for this Ligand-Target Pair
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Novo Nordisk
Curated by ChEMBL
Novo Nordisk
Curated by ChEMBL
Affinity DataKi: 1.80E+3nMpH: 5.5Assay Description:Inhibitory effect against recombinant human protein-tyrosine phosphatase 1B (PTP1B), using p-nitrophenyl phosphate substrate at pH 5.5.More data for this Ligand-Target Pair
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Novo Nordisk
Curated by ChEMBL
Novo Nordisk
Curated by ChEMBL
Affinity DataKi: 2.00E+3nMpH: 5.5Assay Description:Inhibitory effect against recombinant human protein-tyrosine phosphatase 1B (PTP1B), using p-nitrophenyl phosphate substrate at pH 5.5.More data for this Ligand-Target Pair