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Found 203 with Last Name = 'o''sullivan' and Initial = 'tj'
TargetStromelysin-1(Homo sapiens (Human))
Pharmacia And Upjohn

Curated by ChEMBL
LigandPNGBDBM50076372(1-[(S)-2-Oxo-1-pentafluorophenylmethyl-2-(4-pyridi...)
Affinity DataKi:  14nMAssay Description:Binding affinity for matrix metalloproteinase-3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
Pharmacia And Upjohn

Curated by ChEMBL
LigandPNGBDBM50076341((S)-N-Methyl-3-pentafluorophenyl-2-[3-(5-thioxo-4,...)
Affinity DataKi:  18nMAssay Description:Binding affinity for matrix metalloproteinase-3More data for this Ligand-Target Pair
TargetStromelysin-1(Homo sapiens (Human))
Pharmacia And Upjohn

Curated by ChEMBL
LigandPNGBDBM50076338((S)-3-(4-Fluoro-phenyl)-N-methyl-2-[3-(5-thioxo-4,...)
Affinity DataKi:  100nMAssay Description:Binding affinity for matrix metalloproteinase-3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Pharmacia

Curated by ChEMBL
LigandPNGBDBM13611(2-(carboxymethoxy)-5-[(2S)-2-[(2S)-2-(3-formamidop...)
Affinity DataKi:  220nMAssay Description:Inhibitory activity against human protein tyrosine phosphatase 1B (PTP1B)More data for this Ligand-Target Pair
TargetStromelysin-1(Homo sapiens (Human))
Pharmacia And Upjohn

Curated by ChEMBL
LigandPNGBDBM50076367(1-[(S)-1-(4-Fluoro-benzyl)-2-oxo-2-(4-pyridin-2-yl...)
Affinity DataKi:  270nMAssay Description:Binding affinity for matrix metalloproteinase-3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
Pharmacia And Upjohn

Curated by ChEMBL
LigandPNGBDBM50076357((S)-3-Phenyl-2-[3-(5-thioxo-4,5-dihydro-[1,3,4]thi...)
Affinity DataKi:  290nMAssay Description:Binding affinity for matrix metalloproteinase-3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50277957((R)-3-((2',4'-difluorobiphenyl-4-yl)methyl)-5-meth...)
Affinity DataKi:  323nMAssay Description:Binding affinity to human 5HT2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
Pharmacia And Upjohn

Curated by ChEMBL
LigandPNGBDBM50076366((S)-N-Methyl-3-(4-nitro-phenyl)-2-[3-(5-thioxo-4,5...)
Affinity DataKi:  330nMAssay Description:Binding affinity for matrix metalloproteinase-3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
Pharmacia And Upjohn

Curated by ChEMBL
LigandPNGBDBM50076374(1-((S)-1-Benzyl-2-oxo-2-thiomorpholin-4-yl-ethyl)-...)
Affinity DataKi:  380nMAssay Description:Binding affinity for matrix metalloproteinase-3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
Pharmacia And Upjohn

Curated by ChEMBL
LigandPNGBDBM50076339((S)-3-(4-Hydroxy-phenyl)-N-methyl-2-[3-(5-thioxo-4...)
Affinity DataKi:  400nMAssay Description:Binding affinity for matrix metalloproteinase-3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
Pharmacia And Upjohn

Curated by ChEMBL
LigandPNGBDBM50076336(1-[(S)-1-Benzyl-2-oxo-2-(4-pyrimidin-2-yl-piperazi...)
Affinity DataKi:  420nMAssay Description:Binding affinity for matrix metalloproteinase-3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
Pharmacia And Upjohn

Curated by ChEMBL
LigandPNGBDBM50076351((S)-3-(4-Methoxy-phenyl)-N-methyl-2-[3-(5-thioxo-4...)
Affinity DataKi:  460nMAssay Description:Binding affinity for matrix metalloproteinase-3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
Pharmacia And Upjohn

Curated by ChEMBL
LigandPNGBDBM50076334((S)-N-(3,4-Dimethoxy-benzyl)-3-phenyl-2-[3-(5-thio...)
Affinity DataKi:  490nMAssay Description:Binding affinity for matrix metalloproteinase-3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
Pharmacia And Upjohn

Curated by ChEMBL
LigandPNGBDBM50076382((S)-N-Benzyl-3-phenyl-2-[3-(5-thioxo-4,5-dihydro-[...)
Affinity DataKi:  510nMAssay Description:Binding affinity for matrix metalloproteinase-3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
Pharmacia And Upjohn

Curated by ChEMBL
LigandPNGBDBM50076342(1-[(S)-1-Benzyl-2-oxo-2-(4-pyridin-2-yl-piperazin-...)
Affinity DataKi:  520nMAssay Description:Binding affinity for matrix metalloproteinase-3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Pharmacia

Curated by ChEMBL
LigandPNGBDBM50124517(2-Carboxymethoxy-5-(2-pentylcarbamoyl-2-{(S)-(S)-3...)
Affinity DataKi:  590nMAssay Description:Inhibitory activity against human protein tyrosine phosphatase 1B (PTP1B)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
Pharmacia And Upjohn

Curated by ChEMBL
LigandPNGBDBM50076346(1-((S)-1-Benzyl-2-oxo-2-pyrrolidin-1-yl-ethyl)-3-(...)
Affinity DataKi:  660nMAssay Description:Binding affinity for matrix metalloproteinase-3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Pharmacia

Curated by ChEMBL
LigandPNGBDBM50124511(2-Carboxymethoxy-5-(2-{(S)-(S)-2-[2-(4-methoxy-phe...)
Affinity DataKi:  670nMAssay Description:Inhibitory activity against human protein tyrosine phosphatase 1B (PTP1B)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Pharmacia

Curated by ChEMBL
LigandPNGBDBM50124514(2-Carboxymethoxy-5-[2-{(S)-2-[2-(5-mercapto-tetraz...)
Affinity DataKi:  700nMAssay Description:Inhibitory activity against human protein tyrosine phosphatase 1B (PTP1B)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
Pharmacia And Upjohn

Curated by ChEMBL
LigandPNGBDBM50241372((S)-1-(1-(methylamino)-1-oxo-3-phenylpropan-2-yl)-...)
Affinity DataKi:  710nMAssay Description:Binding affinity for matrix metalloproteinase-3More data for this Ligand-Target Pair
TargetInterstitial collagenase(Homo sapiens (Human))
Pharmacia And Upjohn

Curated by ChEMBL
LigandPNGBDBM50076372(1-[(S)-2-Oxo-1-pentafluorophenylmethyl-2-(4-pyridi...)
Affinity DataKi:  770nMAssay Description:Binding affinity for matrix metalloproteinase-1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
Pharmacia And Upjohn

Curated by ChEMBL
LigandPNGBDBM50076348((S)-N-Cyclohexylmethyl-3-phenyl-2-[3-(5-thioxo-4,5...)
Affinity DataKi:  810nMAssay Description:Binding affinity for matrix metalloproteinase-3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
Pharmacia And Upjohn

Curated by ChEMBL
LigandPNGBDBM50076354(1-[(S)-1-Benzyl-2-(4-benzyl-piperazin-1-yl)-2-oxo-...)
Affinity DataKi:  860nMAssay Description:Binding affinity for matrix metalloproteinase-3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Pharmacia

Curated by ChEMBL
LigandPNGBDBM50124513(2-Carboxymethoxy-5-[(S)-2-pentylcarbamoyl-2-((S)-2...)
Affinity DataKi:  870nMAssay Description:Inhibitory activity against human protein tyrosine phosphatase 1B (PTP1B)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
Pharmacia And Upjohn

Curated by ChEMBL
LigandPNGBDBM50076364(1-((S)-1-Benzyl-2-morpholin-4-yl-2-oxo-ethyl)-3-(5...)
Affinity DataKi:  930nMAssay Description:Binding affinity for matrix metalloproteinase-3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
Pharmacia And Upjohn

Curated by ChEMBL
LigandPNGBDBM50076363(1-{(S)-1-Benzyl-2-[4-(4-methoxy-phenyl)-piperazin-...)
Affinity DataKi:  1.00E+3nMAssay Description:Binding affinity for matrix metalloproteinase-3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
Pharmacia And Upjohn

Curated by ChEMBL
LigandPNGBDBM50076358((S)-N-Isopropyl-3-phenyl-2-[3-(5-thioxo-4,5-dihydr...)
Affinity DataKi:  1.30E+3nMAssay Description:Binding affinity for matrix metalloproteinase-3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Pharmacia

Curated by ChEMBL
LigandPNGBDBM50124515(2-Carboxymethoxy-5-{2-pentylcarbamoyl-2-[(S)-(S)-3...)
Affinity DataKi:  1.40E+3nMAssay Description:Inhibitory activity against human protein tyrosine phosphatase 1B (PTP1B)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInterstitial collagenase(Homo sapiens (Human))
Pharmacia And Upjohn

Curated by ChEMBL
LigandPNGBDBM50076342(1-[(S)-1-Benzyl-2-oxo-2-(4-pyridin-2-yl-piperazin-...)
Affinity DataKi:  1.50E+3nMAssay Description:Binding affinity for matrix metalloproteinase-1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInterstitial collagenase(Homo sapiens (Human))
Pharmacia And Upjohn

Curated by ChEMBL
LigandPNGBDBM50076367(1-[(S)-1-(4-Fluoro-benzyl)-2-oxo-2-(4-pyridin-2-yl...)
Affinity DataKi:  1.80E+3nMAssay Description:Binding affinity for matrix metalloproteinase-1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Pharmacia

Curated by ChEMBL
LigandPNGBDBM50112101(5-[2-(2-tert-Butoxycarbonylamino-3-phenyl-propiony...)
Affinity DataKi:  2.00E+3nMAssay Description:Inhibitory activity against human protein tyrosine phosphatase 1B (PTP1B)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMedMMDB

TargetStromelysin-1(Homo sapiens (Human))
Pharmacia And Upjohn

Curated by ChEMBL
LigandPNGBDBM50241378((S)-1-(3-(benzyloxy)-1-(methylamino)-1-oxopropan-2...)
Affinity DataKi:  2.00E+3nMAssay Description:Binding affinity for matrix metalloproteinase-3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50277955((R)-3-((3'-chloro-4'-fluorobiphenyl-4-yl)methyl)-5...)
Affinity DataKi:  2.10E+3nMAssay Description:Binding affinity to human 5HT2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
Pharmacia And Upjohn

Curated by ChEMBL
LigandPNGBDBM50076370((S)-N,N-Dimethyl-3-phenyl-2-[3-(5-thioxo-4,5-dihyd...)
Affinity DataKi:  2.30E+3nMAssay Description:Binding affinity for matrix metalloproteinase-3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInterstitial collagenase(Homo sapiens (Human))
Pharmacia And Upjohn

Curated by ChEMBL
LigandPNGBDBM50076341((S)-N-Methyl-3-pentafluorophenyl-2-[3-(5-thioxo-4,...)
Affinity DataKi:  3.00E+3nMAssay Description:Binding affinity for matrix metalloproteinase-1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50277956((R)-3-((2'-fluoro-4'-(trifluoromethoxy)biphenyl-4-...)
Affinity DataKi: >3.10E+3nMAssay Description:Binding affinity to human 5HT2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50278007((R)-3-((6-(2-fluoro-4-(trifluoromethoxy)phenyl)pyr...)
Affinity DataKi: >3.10E+3nMAssay Description:Binding affinity to human 5HT2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50278009((R)-3-((6-(3,4-difluorophenyl)pyridin-3-yl)methyl)...)
Affinity DataKi: >3.10E+3nMAssay Description:Binding affinity to human 5HT2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50277846((5R)-3-(4-(1-cyclohexylethoxy)benzyl)-5-methyloxaz...)
Affinity DataKi: >3.20E+3nMAssay Description:Binding affinity to human 5HT2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
Pharmacia And Upjohn

Curated by ChEMBL
LigandPNGBDBM50076333((S)-3-Phenyl-2-[3-(5-thioxo-4,5-dihydro-[1,3,4]thi...)
Affinity DataKi:  3.20E+3nMAssay Description:Binding affinity for matrix metalloproteinase-3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
Pharmacia And Upjohn

Curated by ChEMBL
LigandPNGBDBM50076343((S)-3-Phenyl-2-[3-(5-thioxo-4,5-dihydro-[1,3,4]thi...)
Affinity DataKi:  3.30E+3nMAssay Description:Binding affinity for matrix metalloproteinase-3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
Pharmacia And Upjohn

Curated by ChEMBL
LigandPNGBDBM50241376((S)-1-(2-(methylamino)-2-oxo-1-phenylethyl)-3-(5-t...)
Affinity DataKi:  4.10E+3nMAssay Description:Binding affinity for matrix metalloproteinase-3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
Pharmacia And Upjohn

Curated by ChEMBL
LigandPNGBDBM50241374((S)-1-(3-cyclohexyl-1-(methylamino)-1-oxopropan-2-...)
Affinity DataKi:  4.10E+3nMAssay Description:Binding affinity for matrix metalloproteinase-3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Pharmacia

Curated by ChEMBL
LigandPNGBDBM13606((3S)-3-{[(1S)-1-{[(1S)-1-carbamoylpentyl]carbamoyl...)
Affinity DataKi:  5.00E+3nMAssay Description:Inhibitory activity against human protein tyrosine phosphatase 1B (PTP1B)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
Pharmacia And Upjohn

Curated by ChEMBL
LigandPNGBDBM50241373((R)-1-(1-(methylamino)-1-oxo-3-phenylpropan-2-yl)-...)
Affinity DataKi:  5.30E+3nMAssay Description:Binding affinity for matrix metalloproteinase-3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInterstitial collagenase(Homo sapiens (Human))
Pharmacia And Upjohn

Curated by ChEMBL
LigandPNGBDBM50076363(1-{(S)-1-Benzyl-2-[4-(4-methoxy-phenyl)-piperazin-...)
Affinity DataKi:  6.00E+3nMAssay Description:Binding affinity for matrix metalloproteinase-1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInterstitial collagenase(Homo sapiens (Human))
Pharmacia And Upjohn

Curated by ChEMBL
LigandPNGBDBM50076334((S)-N-(3,4-Dimethoxy-benzyl)-3-phenyl-2-[3-(5-thio...)
Affinity DataKi:  6.20E+3nMAssay Description:Binding affinity for matrix metalloproteinase-1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromelysin-1(Homo sapiens (Human))
Pharmacia And Upjohn

Curated by ChEMBL
LigandPNGBDBM50076369(1-Phenethyl-3-(5-thioxo-4,5-dihydro-[1,3,4]thiadia...)
Affinity DataKi:  7.00E+3nMAssay Description:Binding affinity for matrix metalloproteinase-3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInterstitial collagenase(Homo sapiens (Human))
Pharmacia And Upjohn

Curated by ChEMBL
LigandPNGBDBM50076338((S)-3-(4-Fluoro-phenyl)-N-methyl-2-[3-(5-thioxo-4,...)
Affinity DataKi:  8.90E+3nMAssay Description:Binding affinity for matrix metalloproteinase-1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Pharmacia

Curated by ChEMBL
LigandPNGBDBM50124512(2-{4-[(S)-2-((S)-2-tert-Butoxycarbonylamino-3-phen...)
Affinity DataKi:  9.00E+3nMAssay Description:Inhibitory activity against human protein tyrosine phosphatase 1B (PTP1B)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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