TargetNEDD8-activating enzyme E1 regulatory subunit(Homo sapiens (Human))
University Of Toronto Mississauga
Curated by ChEMBL
University Of Toronto Mississauga
Curated by ChEMBL
Affinity DataIC50: 4.70nMAssay Description:Inhibition of NAE (unknown origin)More data for this Ligand-Target Pair
TargetNEDD8-activating enzyme E1 regulatory subunit(Homo sapiens (Human))
University Of Toronto Mississauga
Curated by ChEMBL
University Of Toronto Mississauga
Curated by ChEMBL
Affinity DataIC50: 10nMAssay Description:Inhibition of NAE (unknown origin) in presence of ATPMore data for this Ligand-Target Pair
TargetNEDD8-activating enzyme E1 regulatory subunit(Homo sapiens (Human))
University Of Toronto Mississauga
Curated by ChEMBL
University Of Toronto Mississauga
Curated by ChEMBL
Affinity DataIC50: 800nMAssay Description:Inhibition of NAE (unknown origin)-catalyzed NEDD8-Ubcl2 intermediate formation by densitometric analysisMore data for this Ligand-Target Pair
TargetUbiquitin-like modifier-activating enzyme 6(Homo sapiens (Human))
University Of Toronto Mississauga
Curated by ChEMBL
University Of Toronto Mississauga
Curated by ChEMBL
Affinity DataIC50: 920nMAssay Description:Inhibition of UBA6 (unknown origin) in presence of ATPMore data for this Ligand-Target Pair
TargetUbiquitin-like modifier-activating enzyme 6(Homo sapiens (Human))
University Of Toronto Mississauga
Curated by ChEMBL
University Of Toronto Mississauga
Curated by ChEMBL
Affinity DataIC50: 1.80E+3nMAssay Description:Inhibition of UBA6 (unknown origin)More data for this Ligand-Target Pair
TargetSUMO-activating enzyme subunit 1(Homo sapiens (Human))
University Of Toronto Mississauga
Curated by ChEMBL
University Of Toronto Mississauga
Curated by ChEMBL
Affinity DataIC50: 2.20E+3nMAssay Description:Inhibition of recombinant SAE1(unknown origin)-mediated SUMOylation of RanGAP1-C2More data for this Ligand-Target Pair
TargetSUMO-activating enzyme subunit 1(Homo sapiens (Human))
University Of Toronto Mississauga
Curated by ChEMBL
University Of Toronto Mississauga
Curated by ChEMBL
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibition of recombinant SAE1(unknown origin)-mediated SUMOylation of RanGAP1-C2More data for this Ligand-Target Pair
TargetUbiquitin-like modifier-activating enzyme 7(Homo sapiens (Human))
University Of Toronto Mississauga
Curated by ChEMBL
University Of Toronto Mississauga
Curated by ChEMBL
Affinity DataIC50: 4.00E+3nMAssay Description:Inhibition of UBA7 (unknown origin) in presence of ATPMore data for this Ligand-Target Pair
TargetNEDD8-activating enzyme E1 regulatory subunit(Homo sapiens (Human))
University Of Toronto Mississauga
Curated by ChEMBL
University Of Toronto Mississauga
Curated by ChEMBL
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of NAE (unknown origin) assessed as decrease in NEDD8-Ubcl2 formationMore data for this Ligand-Target Pair
TargetSUMO-activating enzyme subunit 1(Homo sapiens (Human))
University Of Toronto Mississauga
Curated by ChEMBL
University Of Toronto Mississauga
Curated by ChEMBL
Affinity DataIC50: 6.40E+3nMAssay Description:Inhibition of SAE (unknown origin) in presence of ATPMore data for this Ligand-Target Pair
TargetSUMO-activating enzyme subunit 1(Homo sapiens (Human))
University Of Toronto Mississauga
Curated by ChEMBL
University Of Toronto Mississauga
Curated by ChEMBL
Affinity DataIC50: 8.20E+3nMAssay Description:Inhibition of SAE (unknown origin)More data for this Ligand-Target Pair
TargetUbiquitin-like modifier-activating enzyme ATG7(Homo sapiens (Human))
University Of Toronto Mississauga
Curated by ChEMBL
University Of Toronto Mississauga
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of ATG7 (unknown origin)More data for this Ligand-Target Pair
TargetSUMO-activating enzyme subunit 1(Homo sapiens (Human))
University Of Toronto Mississauga
Curated by ChEMBL
University Of Toronto Mississauga
Curated by ChEMBL
Affinity DataIC50: 1.17E+4nMAssay Description:Inhibition of recombinant His-tagged SAE1(unknown origin)-mediated SUMOylation of RanGAP1-C2 by immunoblotting analysisMore data for this Ligand-Target Pair
TargetNEDD8-activating enzyme E1 regulatory subunit(Homo sapiens (Human))
University Of Toronto Mississauga
Curated by ChEMBL
University Of Toronto Mississauga
Curated by ChEMBL
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of NAE (unknown origin)-catalyzed transthiolation of NEDD8 from NAE to Ubc12More data for this Ligand-Target Pair
TargetUbiquitin-like modifier-activating enzyme ATG7(Homo sapiens (Human))
University Of Toronto Mississauga
Curated by ChEMBL
University Of Toronto Mississauga
Curated by ChEMBL
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of ATG7 (unknown origin) in presence of ATPMore data for this Ligand-Target Pair
TargetSUMO-activating enzyme subunit 1(Homo sapiens (Human))
University Of Toronto Mississauga
Curated by ChEMBL
University Of Toronto Mississauga
Curated by ChEMBL
Affinity DataIC50: 4.50E+5nMAssay Description:Inhibition of human SAE by fluorescence assayMore data for this Ligand-Target Pair