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Found 586 with Last Name = 'pettersson' and Initial = 'i'
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University Of Lund

Curated by ChEMBL
LigandPNGBDBM50005120(CHEMBL274491 | N-((2S,3S)-1-Benzyl-2-methyl-pyrrol...)
Affinity DataKi:  0.120nMAssay Description:Compound was evaluated for binding affinity towards DA D-2 receptor using radioligand [3H]SPIMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2/gamma-2(Homo sapiens (Human))
Lund University

Curated by ChEMBL
LigandPNGBDBM50185292(6-Benzyl-4-oxo-1,4-dihydroquinoline-3-carboxylic A...)
Affinity DataKi:  0.270nMAssay Description:Displacement of [3H]Flumazenil from human GABA-Aalpha1 receptor plus beta-2-gamma-2 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Homo sapiens (Human))
Royal Danish School Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM82247(8-Chloro-3-methyl-5-phenyl-2,3,4,5-tetrahydro-1H-b...)
Affinity DataKi:  0.300nMAssay Description:Binding affinity to displace [3H]- SCH 23390 against Dopamine receptor D1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Homo sapiens (Human))
Royal Danish School Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM82247(8-Chloro-3-methyl-5-phenyl-2,3,4,5-tetrahydro-1H-b...)
Affinity DataKi:  0.300nMAssay Description:Compound was tested for the displacement of [3H]-SCH- 23390 from dopamine receptor D1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Homo sapiens (Human))
Royal Danish School Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50010707(8-Chloro-3-methyl-5-m-tolyl-2,3,4,5-tetrahydro-1H-...)
Affinity DataKi:  0.400nMAssay Description:Binding affinity to displace [3H]- SCH 23390 against Dopamine receptor D1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Mus musculus (Mouse))
Royal Danish School Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM82247(8-Chloro-3-methyl-5-phenyl-2,3,4,5-tetrahydro-1H-b...)
Affinity DataKi:  0.400nMAssay Description:Binding affinity to displace [3H]- SCH 23390 against Dopamine receptor D1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Homo sapiens (Human))
Royal Danish School Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50010717(8-Chloro-3-methyl-5-o-tolyl-2,3,4,5-tetrahydro-1H-...)
Affinity DataKi:  0.800nMAssay Description:Binding affinity to displace [3H]- SCH 23390 against Dopamine receptor D1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Homo sapiens (Human))
Royal Danish School Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50010716(8-Chloro-3-methyl-5-p-tolyl-2,3,4,5-tetrahydro-1H-...)
Affinity DataKi:  1.60nMAssay Description:Binding affinity to displace [3H]- SCH 23390 against Dopamine receptor D1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Homo sapiens (Human))
Royal Danish School Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50004823((6aS,13bR)-11-Chloro-7-methyl-5,6a,7,8,9,13b-hexah...)
Affinity DataKi:  1.90nMAssay Description:Compound was tested for the displacement of [3H]-SCH- 23390 from dopamine receptor D1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Homo sapiens (Human))
Royal Danish School Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50004823((6aS,13bR)-11-Chloro-7-methyl-5,6a,7,8,9,13b-hexah...)
Affinity DataKi:  1.90nMAssay Description:Binding affinity to displace [3H]-SCH- 23390 against Dopamine receptor D1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University Of Lund

Curated by ChEMBL
LigandPNGBDBM50132693(4-Amino-N-(1-benzyl-piperidin-4-yl)-5-chloro-2-met...)
Affinity DataKi:  2.20nMAssay Description:Compound was evaluated for binding affinity towards DA D-2 receptor using radioligand [3H]SPIMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2/gamma-2(Homo sapiens (Human))
Lund University

Curated by ChEMBL
LigandPNGBDBM50185296(6-ethyl-3-(3-methylbutoxycarbonyl)-4-quinolone | C...)
Affinity DataKi:  4.10nMAssay Description:Displacement of [3H]Flumazenil from human GABA-Aalpha1 receptor plus beta-2-gamma-2 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Homo sapiens (Human))
Royal Danish School Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50004822((R)-1-phenyl-2,3,4,5-tetrahydro-1H-benzo[d]azepine...)
Affinity DataKi:  5.10nMAssay Description:Binding affinity against Dopamine receptor D1 in rat radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Homo sapiens (Human))
Royal Danish School Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50010709(5-Benzofuran-7-yl-8-chloro-3-methyl-2,3,4,5-tetrah...)
Affinity DataKi:  6nMAssay Description:Binding affinity to displace [3H]-SCH- 23390 against Dopamine receptor D1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Homo sapiens (Human))
Royal Danish School Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50004820(3-Chloro-7-methyl-5,6,7,7a,8,12b-hexahydro-7-aza-d...)
Affinity DataKi:  7nMAssay Description:Binding affinity to displace [3H]- SCH 23390 against Dopamine receptor D1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Homo sapiens (Human))
Royal Danish School Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50004820(3-Chloro-7-methyl-5,6,7,7a,8,12b-hexahydro-7-aza-d...)
Affinity DataKi:  7nMAssay Description:Compound was tested for the displacement of [3H]-SCH- 23390 from dopamine receptor D1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGamma-aminobutyric acid receptor subunit alpha-3/beta-2/gamma-2(Homo sapiens (Human))
Lund University

Curated by ChEMBL
LigandPNGBDBM50185292(6-Benzyl-4-oxo-1,4-dihydroquinoline-3-carboxylic A...)
Affinity DataKi:  7.20nMAssay Description:Displacement of [3H]Flumazenil from human GABA-Aalpha3 receptor plus beta-2-gamma-2 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University Of Lund

Curated by ChEMBL
LigandPNGBDBM50005118((S)-3,5-Dichloro-N-(1-ethyl-pyrrolidin-2-ylmethyl)...)
Affinity DataKi:  9.5nMAssay Description:Compound was evaluated for binding affinity towards DA D-2 receptor using radioligand [3H]SPIMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2/gamma-2(Homo sapiens (Human))
Lund University

Curated by ChEMBL
LigandPNGBDBM50000766(CHEMBL12 | DIAZEPAM | US9271961, Diazepam)
Affinity DataKi:  12nMAssay Description:Displacement of [3H]Flumazenil from human GABA-Aalpha1 receptor plus beta-2-gamma-2 expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-3/beta-2/gamma-2(Homo sapiens (Human))
Lund University

Curated by ChEMBL
LigandPNGBDBM50000766(CHEMBL12 | DIAZEPAM | US9271961, Diazepam)
Affinity DataKi:  14nMAssay Description:Displacement of [3H]Flumazenil from human GABA-Aalpha3 receptor plus beta-2-gamma-2 expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2/gamma-2(Homo sapiens (Human))
Lund University

Curated by ChEMBL
LigandPNGBDBM50185293(6-bromo-3-ethoxycarbonyl-4-quinolone | CHEMBL20525...)
Affinity DataKi:  14nMAssay Description:Displacement of [3H]Flumazenil from human GABA-Aalpha1 receptor plus beta-2-gamma-2 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(RAT)
Royal Danish School Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50010708(6-Phenyl-2,6,7,8,9,9a-hexahydro-1H-8-aza-benzo[cd]...)
Affinity DataKi:  24nMAssay Description:Binding affinity against Dopamine receptor D1 in rat radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGamma-aminobutyric acid receptor subunit alpha-3/beta-2/gamma-2(Homo sapiens (Human))
Lund University

Curated by ChEMBL
LigandPNGBDBM50185293(6-bromo-3-ethoxycarbonyl-4-quinolone | CHEMBL20525...)
Affinity DataKi:  26nMAssay Description:Displacement of [3H]Flumazenil from human GABA-Aalpha3 receptor plus beta-2-gamma-2 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University Of Lund

Curated by ChEMBL
LigandPNGBDBM50005117((racemic)5'-(5-Ethanesulfonyl-2-methoxy-phenyl)-1-...)
Affinity DataKi:  29nMAssay Description:Compound was evaluated for binding affinity towards Dopamine receptor D2 using radioligand [3H]SPIMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University Of Lund

Curated by ChEMBL
LigandPNGBDBM81774(CAS_15676-16-1 | SULPIRIDE,(+) | Sulpiride-S | Sul...)
Affinity DataKi:  39nMAssay Description:Inhibitory concentration required for displacing radioligand [3H]SPI from DA D-2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2/gamma-2(Homo sapiens (Human))
Lund University

Curated by ChEMBL
LigandPNGBDBM26266(Ambien | CHEMBL911 | Dalparan | N,N-dimethyl-2-[6-...)
Affinity DataKi:  53nMAssay Description:Displacement of [3H]Flumazenil from human GABA-Aalpha1 receptor plus beta-2-gamma-2 expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-3/beta-2/gamma-2(Homo sapiens (Human))
Lund University

Curated by ChEMBL
LigandPNGBDBM50185296(6-ethyl-3-(3-methylbutoxycarbonyl)-4-quinolone | C...)
Affinity DataKi:  89nMAssay Description:Displacement of [3H]Flumazenil from human GABA-Aalpha3 receptor plus beta-2-gamma-2 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University Of Lund

Curated by ChEMBL
LigandPNGBDBM48320(4-amino-5-chloro-N-[2-(diethylamino)ethyl]-2-metho...)
Affinity DataKi:  104nMAssay Description:Inhibitory concentration required for displacing radioligand [3H]SPI from DA D-2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University Of Lund

Curated by ChEMBL
LigandPNGBDBM48320(4-amino-5-chloro-N-[2-(diethylamino)ethyl]-2-metho...)
Affinity DataKi:  104nMAssay Description:Compound was evaluated for binding affinity towards DA D-2 receptor using radioligand [3H]SPIMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Homo sapiens (Human))
Royal Danish School Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM55121(3-HYDROXYTYRAMINE HYDROCHLORIDE | 4-(2-aminoethyl)...)
Affinity DataKi:  192nMAssay Description:Binding affinity to displace [3H]- SCH 23390 against Dopamine receptor D1More data for this Ligand-Target Pair
TargetD(1A) dopamine receptor(Homo sapiens (Human))
Royal Danish School Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM82248(CAS_73445-63-3 | SCH 23388 (S-enantiomer))
Affinity DataKi:  192nMAssay Description:Compound was tested for the displacement of [3H]-SCH- 23390 from dopamine receptor D1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Homo sapiens (Human))
Royal Danish School Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50010715((6aS,13bS)11-Chloro-7-methyl-5,6a,7,8,9,13b-hexahy...)
Affinity DataKi:  513nMAssay Description:Binding affinity to displace [3H]-SCH- 23390 against Dopamine receptor D1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Homo sapiens (Human))
Royal Danish School Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50010711((6aR,13bS )11-Chloro-7-methyl-5,6a,7,8,9,13b-hexah...)
Affinity DataKi:  531nMAssay Description:Binding affinity to displace [3H]-SCH- 23390 against Dopamine receptor D1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Homo sapiens (Human))
Royal Danish School Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50010712((6aR,13bR)11-Chloro-7-methyl-5,6a,7,8,9,13b-hexahy...)
Affinity DataKi:  898nMAssay Description:Binding affinity to displace [3H]-SCH- 23390 against Dopamine receptor D1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(RAT)
Royal Danish School Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50010710(6-Phenyl-2,6,7,8,9,9a-hexahydro-1H-8-aza-benzo[cd]...)
Affinity DataKi:  1.22E+3nMAssay Description:Binding affinity against Dopamine receptor D1 in rat radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGamma-aminobutyric acid receptor subunit alpha-3/beta-2/gamma-2(Homo sapiens (Human))
Lund University

Curated by ChEMBL
LigandPNGBDBM26266(Ambien | CHEMBL911 | Dalparan | N,N-dimethyl-2-[6-...)
Affinity DataKi:  1.85E+3nMAssay Description:Displacement of [3H]Flumazenil from human GABA-Aalpha3 receptor plus beta-2-gamma-2 expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetGlucagon-like peptide 1 receptor(Homo sapiens (Human))
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50121523(CHEMBL3616742)
Affinity DataIC50:  0.0300nMAssay Description:Displacement of [125I]-GLP1 from human GLP1 receptor expressed in BHK cells after 2 hrs in absence of human serum albuminMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon-like peptide 1 receptor(Homo sapiens (Human))
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50120380(CHEMBL3616743)
Affinity DataIC50:  0.0400nMAssay Description:Displacement of [125I]-GLP1 from human GLP1 receptor expressed in BHK cells after 2 hrs in absence of human serum albuminMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon-like peptide 1 receptor(Homo sapiens (Human))
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50121405(CHEMBL3616767)
Affinity DataIC50:  0.0600nMAssay Description:Displacement of [125I]-GLP1 from human GLP1 receptor expressed in BHK cells after 2 hrs in absence of human serum albuminMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon-like peptide 1 receptor(Homo sapiens (Human))
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50121399(CHEMBL3616764)
Affinity DataIC50:  0.0600nMAssay Description:Displacement of [125I]-GLP1 from human GLP1 receptor expressed in BHK cells after 2 hrs in absence of human serum albuminMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon-like peptide 1 receptor(Homo sapiens (Human))
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50121527(CHEMBL3616718)
Affinity DataIC50:  0.0800nMAssay Description:Displacement of [125I]-GLP1 from human GLP1 receptor expressed in BHK cells after 2 hrs in presence of 2% human serum albuminMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon-like peptide 1 receptor(Homo sapiens (Human))
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50121402(CHEMBL3616772)
Affinity DataIC50:  0.0900nMAssay Description:Displacement of [125I]-GLP1 from human GLP1 receptor expressed in BHK cells after 2 hrs in absence of human serum albuminMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon-like peptide 1 receptor(Homo sapiens (Human))
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50121518(CHEMBL428139)
Affinity DataIC50:  0.100nMAssay Description:Displacement of [125I]-GLP1 from human GLP1 receptor expressed in BHK cells after 2 hrs in presence of 2% human serum albuminMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon-like peptide 1 receptor(Homo sapiens (Human))
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50121508(CHEMBL3616774)
Affinity DataIC50:  0.100nMAssay Description:Displacement of [125I]-GLP1 from human GLP1 receptor expressed in BHK cells after 2 hrs in absence of human serum albuminMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon-like peptide 1 receptor(Homo sapiens (Human))
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50121526(CHEMBL3616762)
Affinity DataIC50:  0.100nMAssay Description:Displacement of [125I]-GLP1 from human GLP1 receptor expressed in BHK cells after 2 hrs in absence of human serum albuminMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon-like peptide 1 receptor(Homo sapiens (Human))
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50121401(CHEMBL3616771)
Affinity DataIC50:  0.110nMAssay Description:Displacement of [125I]-GLP1 from human GLP1 receptor expressed in BHK cells after 2 hrs in absence of human serum albuminMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon-like peptide 1 receptor(Homo sapiens (Human))
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50121398(CHEMBL3616480)
Affinity DataIC50:  0.110nMAssay Description:Displacement of [125I]-GLP1 from human GLP1 receptor expressed in BHK cells after 2 hrs in absence of human serum albuminMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon-like peptide 1 receptor(Homo sapiens (Human))
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50121535(CHEMBL3616739)
Affinity DataIC50:  0.120nMAssay Description:Displacement of [125I]-GLP1 from human GLP1 receptor expressed in BHK cells after 2 hrs in absence of human serum albuminMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon-like peptide 1 receptor(Homo sapiens (Human))
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50121400(CHEMBL3616752)
Affinity DataIC50:  0.130nMAssay Description:Displacement of [125I]-GLP1 from human GLP1 receptor expressed in BHK cells after 2 hrs in absence of human serum albuminMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon-like peptide 1 receptor(Homo sapiens (Human))
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50121394(CHEMBL3616711)
Affinity DataIC50:  0.140nMAssay Description:Displacement of [125I]-GLP1 from human GLP1 receptor expressed in BHK cells after 2 hrs in presence of 2% human serum albuminMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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