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Found 46 with Last Name = 'pevet' and Initial = 'i'
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Institut De Recherches Servier

Curated by ChEMBL
LigandPNGBDBM6471(4-Anilino-7,8-dialkoxybenzo[g]quinoline-3-carbonit...)
Affinity DataIC50:  0.460nMAssay Description:Inhibition of c-SRCMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Institut De Recherches Servier

Curated by ChEMBL
LigandPNGBDBM8((1R)-cyclohexane-1,2-diol | cis-1,2-cyclohexanedio...)
Affinity DataIC50:  0.600nMAssay Description:Inhibition of c-SRCMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Institut De Recherches Servier

Curated by ChEMBL
LigandPNGBDBM4552(4-[(2,4-Dichloro-5-methoxyphenyl)amino]-6-methoxy-...)
Affinity DataIC50:  1nMAssay Description:Inhibition of c-SRCMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Institut De Recherches Servier

Curated by ChEMBL
LigandPNGBDBM12255(AZD0530 | CHEMBL217092 | Compound 33 | N-(5-chloro...)
Affinity DataIC50:  2.70nMAssay Description:Inhibition of c-SRCMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Institut De Recherches Servier

Curated by ChEMBL
LigandPNGBDBM50303801(CHEMBL571546 | N-benzyl-2-(5-(4-(2-morpholinoethox...)
Affinity DataIC50:  20nMAssay Description:Inhibition of c-SRCMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Institut De Recherches Servier

Curated by ChEMBL
LigandPNGBDBM50342390(3-Amino-6-(2-dimethylamino-ethylamino)-4-phenylthi...)
Affinity DataIC50:  32nMAssay Description:Inhibition of c-SRC assessed as residual activity using KVEKIGEGYYGVVYK as peptide substrate after 20 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Institut De Recherches Servier

Curated by ChEMBL
LigandPNGBDBM50342392(3-Amino-4-benzyl-6-(2-dimethylamino-ethylamino)-th...)
Affinity DataIC50:  40nMAssay Description:Inhibition of c-SRC assessed as residual activity using KVEKIGEGYYGVVYK as peptide substrate after 20 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Institut De Recherches Servier

Curated by ChEMBL
LigandPNGBDBM50342393(3-Amino-6-(2-dimethylamino-ethylamino)-4-propylthi...)
Affinity DataIC50:  63nMAssay Description:Inhibition of c-SRC assessed as residual activity using KVEKIGEGYYGVVYK as peptide substrate after 20 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Institut De Recherches Servier

Curated by ChEMBL
LigandPNGBDBM50342391(3-Amino-6-(2-dimethylamino-ethylamino)-4-phenylthi...)
Affinity DataIC50:  68nMAssay Description:Inhibition of c-SRC assessed as residual activity using KVEKIGEGYYGVVYK as peptide substrate after 20 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Institut De Recherches Servier

Curated by ChEMBL
LigandPNGBDBM50342389(3-Amino-6-(2-dimethylamino-ethylamino)-4-phenylthi...)
Affinity DataIC50:  107nMAssay Description:Inhibition of c-SRC assessed as residual activity using KVEKIGEGYYGVVYK as peptide substrate after 20 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Institut De Recherches Servier

Curated by ChEMBL
LigandPNGBDBM50342387(3-Amino-6-(2-dimethylamino-ethylamino)-4-methylthi...)
Affinity DataIC50:  230nMAssay Description:Inhibition of c-SRC assessed as residual activity using KVEKIGEGYYGVVYK as peptide substrate after 20 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Institut De Recherches Servier

Curated by ChEMBL
LigandPNGBDBM50342388(3-Amino-6-(2-dimethylamino-ethylamino)-4-methylthi...)
Affinity DataIC50:  246nMAssay Description:Inhibition of c-SRC assessed as residual activity using KVEKIGEGYYGVVYK as peptide substrate after 20 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Institut De Recherches Servier

Curated by ChEMBL
LigandPNGBDBM50342379(3-Amino-4,6-dimethyl-thieno[2,3-b]pyridine-2-carbo...)
Affinity DataIC50:  269nMAssay Description:Inhibition of c-SRC assessed as residual activity using KVEKIGEGYYGVVYK as peptide substrate after 20 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50223647(CHEMBL112366)
Affinity DataIC50:  270nMAssay Description:Inhibition of phosphodiesterase 4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Institut De Recherches Servier

Curated by ChEMBL
LigandPNGBDBM50342386(3-Amino-4-methyl-6-trifluoromethyl-thieno[2,3-b]py...)
Affinity DataIC50:  330nMAssay Description:Inhibition of c-SRC assessed as residual activity using KVEKIGEGYYGVVYK as peptide substrate after 20 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Institut De Recherches Servier

Curated by ChEMBL
LigandPNGBDBM50342381(3-Amino-4,6-dimethyl-thieno[2,3-b]pyridine-2-carbo...)
Affinity DataIC50:  769nMAssay Description:Inhibition of c-SRC assessed as residual activity using KVEKIGEGYYGVVYK as peptide substrate after 20 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Institut De Recherches Servier

Curated by ChEMBL
LigandPNGBDBM50342384(3-Amino-4,6-dimethyl-thieno[2,3-b]pyridine-2-carbo...)
Affinity DataIC50:  840nMAssay Description:Inhibition of c-SRC assessed as residual activity using KVEKIGEGYYGVVYK as peptide substrate after 20 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50217550(CHEMBL111925 | CI-1018)
Affinity DataIC50:  1.10E+3nMAssay Description:Inhibition of phosphodiesterase 4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Institut De Recherches Servier

Curated by ChEMBL
LigandPNGBDBM50342382(3-Amino-thieno[2,3-b]pyridine-2-carboxylic acid(3-...)
Affinity DataIC50:  1.30E+3nMAssay Description:Inhibition of c-SRC assessed as residual activity using KVEKIGEGYYGVVYK as peptide substrate after 20 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Institut De Recherches Servier

Curated by ChEMBL
LigandPNGBDBM50342385(3-Amino-4-methyl-6-trifluoromethyl-thieno[2,3-b]py...)
Affinity DataIC50:  1.34E+3nMAssay Description:Inhibition of c-SRC assessed as residual activity using KVEKIGEGYYGVVYK as peptide substrate after 20 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Institut De Recherches Servier

Curated by ChEMBL
LigandPNGBDBM50342395(3-Amino-6-(2-dimethylamino-ethylamino)-5-propylthi...)
Affinity DataIC50:  2.08E+3nMAssay Description:Inhibition of c-SRC assessed as residual activity using KVEKIGEGYYGVVYK as peptide substrate after 20 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Institut De Recherches Servier

Curated by ChEMBL
LigandPNGBDBM50342394(3-Amino-5-benzyl-6-(2-dimethylamino-ethylamino)-th...)
Affinity DataIC50:  3.87E+3nMAssay Description:Inhibition of c-SRC assessed as residual activity using KVEKIGEGYYGVVYK as peptide substrate after 20 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50223646(CHEMBL418848)
Affinity DataIC50:  4.40E+3nMAssay Description:Inhibition of phosphodiesterase 4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50451952(CHEMBL2111730)
Affinity DataIC50:  6.10E+3nMAssay Description:Inhibition of phosphodiesterase 4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Institut De Recherches Servier

Curated by ChEMBL
LigandPNGBDBM50342383(3-Amino-4,6-dimethyl-thieno[2,3-b]pyridine-2-carbo...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of c-SRC assessed as residual activity using KVEKIGEGYYGVVYK as peptide substrate after 20 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Institut De Recherches Servier

Curated by ChEMBL
LigandPNGBDBM50342380(3-Amino-thieno[2,3-b]pyridine-2-carboxylic acid na...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of c-SRC assessed as residual activity using KVEKIGEGYYGVVYK as peptide substrate after 20 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A/3B(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50451952(CHEMBL2111730)
Affinity DataIC50:  1.20E+4nMAssay Description:Inhibition of phosphodiesterase 3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50451952(CHEMBL2111730)
Affinity DataIC50:  1.40E+4nMAssay Description:Inhibition of Phosphodiesterase 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50223646(CHEMBL418848)
Affinity DataIC50:  1.60E+4nMAssay Description:Inhibition of Phosphodiesterase 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50147632(4-Methoxy-6-phenyl-1,2-dihydro-8H-5,7,9a-triaza-be...)
Affinity DataIC50:  2.30E+4nMAssay Description:Inhibition of phosphodiesterase 4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50147630(CHEMBL112996 | N-(4-Methoxy-9-oxo-6-phenyl-1,2,8,9...)
Affinity DataIC50:  2.80E+4nMAssay Description:Inhibition of Phosphodiesterase 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50147630(CHEMBL112996 | N-(4-Methoxy-9-oxo-6-phenyl-1,2,8,9...)
Affinity DataIC50:  2.80E+4nMAssay Description:Inhibition of Phosphodiesterase 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A/3B(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50147630(CHEMBL112996 | N-(4-Methoxy-9-oxo-6-phenyl-1,2,8,9...)
Affinity DataIC50:  3.10E+4nMAssay Description:Inhibition of phosphodiesterase 3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50223645(CHEMBL109754)
Affinity DataIC50:  4.00E+4nMAssay Description:Inhibition of phosphodiesterase 4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A/3B(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50223646(CHEMBL418848)
Affinity DataIC50:  4.10E+4nMAssay Description:Inhibition of phosphodiesterase 3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50223645(CHEMBL109754)
Affinity DataIC50:  5.20E+4nMAssay Description:Inhibition of Phosphodiesterase 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50147630(CHEMBL112996 | N-(4-Methoxy-9-oxo-6-phenyl-1,2,8,9...)
Affinity DataIC50:  7.30E+4nMAssay Description:Inhibition of phosphodiesterase 4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50147630(CHEMBL112996 | N-(4-Methoxy-9-oxo-6-phenyl-1,2,8,9...)
Affinity DataIC50:  7.30E+4nMAssay Description:Inhibition of phosphodiesterase 4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A/3B(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50223645(CHEMBL109754)
Affinity DataIC50:  7.70E+4nMAssay Description:Inhibition of phosphodiesterase 3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50147632(4-Methoxy-6-phenyl-1,2-dihydro-8H-5,7,9a-triaza-be...)
Affinity DataIC50:  9.10E+4nMAssay Description:Inhibition of Phosphodiesterase 5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50147630(CHEMBL112996 | N-(4-Methoxy-9-oxo-6-phenyl-1,2,8,9...)
Affinity DataIC50:  9.50E+4nMAssay Description:Inhibition of Phosphodiesterase 5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A/3B(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50147630(CHEMBL112996 | N-(4-Methoxy-9-oxo-6-phenyl-1,2,8,9...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of phosphodiesterase 3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50147632(4-Methoxy-6-phenyl-1,2-dihydro-8H-5,7,9a-triaza-be...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of Phosphodiesterase 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50147630(CHEMBL112996 | N-(4-Methoxy-9-oxo-6-phenyl-1,2,8,9...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of Phosphodiesterase 5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50451952(CHEMBL2111730)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of Phosphodiesterase 5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A/3B(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50147632(4-Methoxy-6-phenyl-1,2-dihydro-8H-5,7,9a-triaza-be...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of phosphodiesterase 3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed