Affinity DataKi: 90nMAssay Description:Inhibitory activity against L-arginine binding to Inducible nitric oxide synthaseMore data for this Ligand-Target Pair
Affinity DataIC50: 0.100nMAssay Description:Affinity for mu opioid receptor was measured by displacement of tritiated DAMGO from rat brain membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 0.130nMAssay Description:Inhibitory concentration of the compound was evaluated against mu opioid receptor by the displacement of tritiated DAMGO from rat brain membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 0.130nMAssay Description:Inhibitory concentration of the compound was evaluated against mu opioid receptor by the displacement of tritiated DAMGO from rat brain membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 0.200nMAssay Description:Inhibitory concentration of the compound was evaluated against mu opioid receptor by the displacement of tritiated DAMGO from rat brain membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 0.920nMAssay Description:Inhibitory concentration of the compound was evaluated against mu opioid receptor by the displacement of tritiated DAMGO from rat brain membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 1.10nMAssay Description:Inhibitory concentration of the compound was evaluated against mu opioid receptor by the displacement of tritiated DAMGO from rat brain membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 1.10nMAssay Description:Inhibitory concentration of the compound was evaluated against mu opioid receptor by the displacement of tritiated DAMGO from rat brain membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 3.5nMAssay Description:Affinity for mu opioid receptor was measured by displacement of tritiated DAMGO from rat brain membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 4nMAssay Description:Affinity for mu opioid receptor was measured by displacement of tritiated DAMGO from rat brain membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 4.40nMAssay Description:Displacement of [3H]-DSLET from rat brain membrane delta opioid receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 8nMAssay Description:Inhibitory concentration of the compound was evaluated against delta opioid receptor by the displacement of tritiated DSLET from rat brain membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 8.60nMAssay Description:Displacement of [3H]-DSLET from rat brain membrane delta opioid receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 8.70nMAssay Description:Inhibitory concentration of the compound was evaluated against mu opioid receptor by the displacement of tritiated DAMGO from rat brain membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 9.60nMAssay Description:Inhibitory concentration of the compound was evaluated against delta opioid receptor by the displacement of tritiated DSLET from rat brain membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 12.3nMAssay Description:Affinity for mu opioid receptor was measured by displacement of tritiated DAMGO from rat brain membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 17.5nMAssay Description:Affinity for mu opioid receptor was measured by displacement of tritiated DAMGO from rat brain membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 23.7nMAssay Description:Affinity for mu opioid receptor was measured by displacement of tritiated DAMGO from rat brain membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 23.7nMAssay Description:Affinity for mu opioid receptor was measured by displacement of tritiated DAMGO from rat brain membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 28.6nMAssay Description:Affinity for mu opioid receptor was measured by displacement of tritiated DAMGO from rat brain membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 32nMAssay Description:Inhibitory concentration of the compound was evaluated against mu opioid receptor by the displacement of tritiated DAMGO from rat brain membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 45nMAssay Description:Inhibitory concentration of the compound was evaluated against mu opioid receptor by the displacement of tritiated DAMGO from rat brain membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 55nMAssay Description:Displacement of [3H]-DSLET from rat brain membrane delta opioid receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 57nMAssay Description:Affinity for mu opioid receptor was measured by displacement of tritiated DAMGO from rat brain membranesMore data for this Ligand-Target Pair
TargetNitric oxide synthase, brain(Homo sapiens (Human))
G. D. Searle Research And Development
Curated by ChEMBL
G. D. Searle Research And Development
Curated by ChEMBL
Affinity DataIC50: 60nMAssay Description:Inhibition of human Neuronal nitric oxide synthaseMore data for this Ligand-Target Pair
Affinity DataIC50: 64nMAssay Description:Displacement of [3H]-DSLET from rat brain membrane delta opioid receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 80nMAssay Description:Inhibition of human Inducible nitric oxide synthaseMore data for this Ligand-Target Pair
Affinity DataIC50: 100nMAssay Description:Inhibition of human Inducible nitric oxide synthaseMore data for this Ligand-Target Pair
Affinity DataIC50: 124nMAssay Description:Inhibitory concentration of the compound was evaluated against delta opioid receptor by the displacement of tritiated DSLET from rat brain membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 127nMAssay Description:Displacement of [3H]-DSLET from rat brain membrane delta opioid receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 133nMAssay Description:Inhibitory concentration of the compound was evaluated against delta opioid receptor by the displacement of tritiated DSLET from rat brain membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 152nMAssay Description:Inhibition of inducible nitric oxide synthaseMore data for this Ligand-Target Pair
Affinity DataIC50: 160nMAssay Description:Inhibitory activity evaluated for soluble cell extract of human Inducible nitric oxide synthase and partially purified by DEAE-sepharose chromatograp...More data for this Ligand-Target Pair
TargetNitric oxide synthase, brain(Homo sapiens (Human))
G. D. Searle Research And Development
Curated by ChEMBL
G. D. Searle Research And Development
Curated by ChEMBL
Affinity DataIC50: 170nMAssay Description:Inhibition of cloned (from RNA) human Neuronal nitric oxide synthaseMore data for this Ligand-Target Pair
Affinity DataIC50: 170nMAssay Description:Inhibition of cloned (from RNA) human inducible nitric oxide synthase (hiNOS)More data for this Ligand-Target Pair
Affinity DataIC50: 190nMAssay Description:Inhibitory activity evaluated for soluble cell extract of human Inducible nitric oxide synthase and partially purified by DEAE-sepharose chromatograp...More data for this Ligand-Target Pair
TargetNitric oxide synthase, brain(Homo sapiens (Human))
G. D. Searle Research And Development
Curated by ChEMBL
G. D. Searle Research And Development
Curated by ChEMBL
Affinity DataIC50: 200nMAssay Description:Inhibition of human Neuronal nitric oxide synthaseMore data for this Ligand-Target Pair
Affinity DataIC50: 200nMAssay Description:Inhibition of human Inducible nitric oxide synthaseMore data for this Ligand-Target Pair
Affinity DataIC50: 221nMAssay Description:Inhibitory concentration of the compound was evaluated against kappa opioid receptor by displacement of tritiated U-69593 from rat brain membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 230nMAssay Description:Inhibition of cloned (from RNA) human inducible nitric oxide synthase (hiNOS)More data for this Ligand-Target Pair
Affinity DataIC50: 300nMAssay Description:Inhibition of cloned (from RNA) human inducible nitric oxide synthase (hiNOS)More data for this Ligand-Target Pair
TargetNitric oxide synthase, endothelial(Homo sapiens (Human))
G. D. Searle Research And Development
Curated by ChEMBL
G. D. Searle Research And Development
Curated by ChEMBL
Affinity DataIC50: 300nMAssay Description:inhibition of human endothelial constitutive Endothelial nitric oxide synthase (heNOS)More data for this Ligand-Target Pair
Affinity DataIC50: 316nMAssay Description:Inhibitory concentration of the compound was evaluated against kappa opioid receptor by displacement of tritiated U-69593 from rat brain membranesMore data for this Ligand-Target Pair
TargetNitric oxide synthase, brain(Homo sapiens (Human))
G. D. Searle Research And Development
Curated by ChEMBL
G. D. Searle Research And Development
Curated by ChEMBL
Affinity DataIC50: 339nMAssay Description:Inhibition of Neuronal nitric oxide synthaseMore data for this Ligand-Target Pair
Affinity DataIC50: 360nMAssay Description:Inhibition of cloned (from RNA) human inducible nitric oxide synthase (hiNOS)More data for this Ligand-Target Pair
Affinity DataIC50: 360nMAssay Description:Inhibition of cloned (from RNA) human inducible nitric oxide synthase (hiNOS)More data for this Ligand-Target Pair
Affinity DataIC50: 367nMAssay Description:Inhibitory concentration of the compound was evaluated against delta opioid receptor by the displacement of tritiated DSLET from rat brain membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 367nMAssay Description:Inhibitory concentration of the compound was evaluated against delta opioid receptor by the displacement of tritiated DSLET from rat brain membranesMore data for this Ligand-Target Pair
TargetNitric oxide synthase, brain(Homo sapiens (Human))
G. D. Searle Research And Development
Curated by ChEMBL
G. D. Searle Research And Development
Curated by ChEMBL
Affinity DataIC50: 390nMAssay Description:Inhibition of cloned (from RNA) human Neuronal nitric oxide synthaseMore data for this Ligand-Target Pair
TargetNitric oxide synthase, brain(Homo sapiens (Human))
G. D. Searle Research And Development
Curated by ChEMBL
G. D. Searle Research And Development
Curated by ChEMBL
Affinity DataIC50: 400nMAssay Description:Inhibition of human Neuronal nitric oxide synthaseMore data for this Ligand-Target Pair