TargetCalcitonin gene-related peptide type 1 receptor(Homo sapiens (Human))
Université
Curated by ChEMBL
Université
Curated by ChEMBL
Affinity DataIC50: 0.5nMAssay Description:Binding affinity of the compound against [125I]-hCalcitonin gene-related peptide type receptor binding sites in guinea pig vas deferens membrane prep...More data for this Ligand-Target Pair
TargetCalcitonin gene-related peptide type 1 receptor(Homo sapiens (Human))
Université
Curated by ChEMBL
Université
Curated by ChEMBL
Affinity DataIC50: 0.5nMAssay Description:Binding affinity of the compound against [125I]-hCalcitonin gene-related peptide type receptor binding sites in guinea pig vas deferens membrane prep...More data for this Ligand-Target Pair
Affinity DataIC50: 0.900nMAssay Description:Binding affinity against [125I]-hCalcitonin gene-related peptide type alpha receptor binding sites in rat brain membraneMore data for this Ligand-Target Pair
TargetCalcitonin gene-related peptide type 1 receptor(Homo sapiens (Human))
Université
Curated by ChEMBL
Université
Curated by ChEMBL
Affinity DataIC50: 1.70nMAssay Description:Binding affinity of the compound against [125I]-hCalcitonin gene-related peptide type receptor binding sites in guinea pig vas deferens membrane prep...More data for this Ligand-Target Pair
TargetCalcitonin gene-related peptide type 1 receptor(Homo sapiens (Human))
Université
Curated by ChEMBL
Université
Curated by ChEMBL
Affinity DataIC50: 1.70nMAssay Description:Binding affinity of the compound against [125I]-hCalcitonin gene-related peptide type receptor binding sites in guinea pig vas deferens membrane prep...More data for this Ligand-Target Pair
TargetCalcitonin gene-related peptide type 1 receptor(Homo sapiens (Human))
Université
Curated by ChEMBL
Université
Curated by ChEMBL
Affinity DataIC50: 2.30nMAssay Description:Binding affinity against [125I]-hCalcitonin gene-related peptide type receptor binding sites in guinea pig atrium membraneMore data for this Ligand-Target Pair
TargetCalcitonin gene-related peptide type 1 receptor(Homo sapiens (Human))
Université
Curated by ChEMBL
Université
Curated by ChEMBL
Affinity DataIC50: 2.30nMAssay Description:Binding affinity of the compound against [125I]-hCalcitonin gene-related peptide type receptor binding sites in guinea pig vas deferens membrane prep...More data for this Ligand-Target Pair
Affinity DataIC50: 2.30nMAssay Description:Binding affinity against [125I]-hCalcitonin gene-related peptide type alpha receptor binding sites in rat brain membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 2.40nMAssay Description:Binding affinity against [125I]-hCalcitonin gene-related peptide type alpha receptor binding sites in rat brain membraneMore data for this Ligand-Target Pair
TargetCalcitonin gene-related peptide type 1 receptor(Homo sapiens (Human))
Université
Curated by ChEMBL
Université
Curated by ChEMBL
Affinity DataIC50: 3nMAssay Description:Binding affinity of the compound against [125I]-hCalcitonin gene-related peptide type receptor binding sites in guinea pig vas deferens membrane prep...More data for this Ligand-Target Pair
TargetCalcitonin gene-related peptide type 1 receptor(Homo sapiens (Human))
Université
Curated by ChEMBL
Université
Curated by ChEMBL
Affinity DataIC50: 8nMAssay Description:Binding affinity of the compound against [125I]-hCalcitonin gene-related peptide type receptor binding sites in guinea pig vas deferens membrane prep...More data for this Ligand-Target Pair
Affinity DataIC50: 8nMAssay Description:Ability to induce 50% of maximal effect in mouse vas deferens expressing Opioid receptor delta 1More data for this Ligand-Target Pair
TargetCalcitonin gene-related peptide type 1 receptor(Homo sapiens (Human))
Université
Curated by ChEMBL
Université
Curated by ChEMBL
Affinity DataIC50: 8nMAssay Description:Binding affinity of the compound against [125I]-hCalcitonin gene-related peptide type receptor binding sites in guinea pig vas deferens membrane prep...More data for this Ligand-Target Pair
Affinity DataIC50: 8nMAssay Description:Binding affinity against [125I]-hCalcitonin gene-related peptide type alpha receptor binding sites in rat brain membraneMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor/Kappa-type opioid receptor/Mu-type opioid receptor/Sigma non-opioid intracellular receptor 1(Rattus norvegicus (rat))
TBA
Curated by ChEMBL
TBA
Curated by ChEMBL
Affinity DataIC50: 8.40nMAssay Description:Ability to displace 50% of (+/-) ethylketocyclazocine (2.8) in rat brain homogenateMore data for this Ligand-Target Pair
Affinity DataIC50: 8.60nMAssay Description:Ability to induce 50% of maximal effect in mouse vas deferens expressing Opioid receptor delta 1More data for this Ligand-Target Pair
TargetCalcitonin gene-related peptide type 1 receptor(Homo sapiens (Human))
Université
Curated by ChEMBL
Université
Curated by ChEMBL
Affinity DataIC50: 9nMAssay Description:Binding affinity of the compound against [125I]-hCalcitonin gene-related peptide type receptor binding sites in guinea pig vas deferens membrane prep...More data for this Ligand-Target Pair
Affinity DataIC50: 9nMAssay Description:Binding affinity against [125I]-hCalcitonin gene-related peptide type alpha receptor binding sites in rat brain membraneMore data for this Ligand-Target Pair
TargetCalcitonin gene-related peptide type 1 receptor(Homo sapiens (Human))
Université
Curated by ChEMBL
Université
Curated by ChEMBL
Affinity DataIC50: 9nMAssay Description:Binding affinity against [125I]-hCalcitonin gene-related peptide type receptor binding sites in guinea pig atrium membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 9.40nMAssay Description:Ability to induce 50% of maximal effect in mouse vas deferens expressing Opioid receptor delta 1More data for this Ligand-Target Pair
Affinity DataIC50: 9.80nMAssay Description:Ability to induce 50% of maximal effect in guinea pig ileum expressing Opioid receptor mu 1More data for this Ligand-Target Pair
Affinity DataIC50: 11nMAssay Description:Binding affinity against [125I]-hCalcitonin gene-related peptide type alpha receptor binding sites in rat brain membraneMore data for this Ligand-Target Pair
TargetCalcitonin gene-related peptide type 1 receptor(Homo sapiens (Human))
Université
Curated by ChEMBL
Université
Curated by ChEMBL
Affinity DataIC50: 11nMAssay Description:Binding affinity against [125I]-hCalcitonin gene-related peptide type receptor binding sites in guinea pig atrium membraneMore data for this Ligand-Target Pair
TargetCalcitonin gene-related peptide type 1 receptor(Homo sapiens (Human))
Université
Curated by ChEMBL
Université
Curated by ChEMBL
Affinity DataIC50: 12nMAssay Description:Binding affinity of the compound against [125I]-hCalcitonin gene-related peptide type receptor binding sites in guinea pig vas deferens membrane prep...More data for this Ligand-Target Pair
Affinity DataIC50: 12nMAssay Description:Ability to induce 50% of maximal effect in guinea pig ileum expressing Opioid receptor mu 1More data for this Ligand-Target Pair
Affinity DataIC50: 14.5nMAssay Description:Binding affinity against [125I]-hCalcitonin gene-related peptide type alpha receptor binding sites in rat brain membraneMore data for this Ligand-Target Pair
TargetCalcitonin gene-related peptide type 1 receptor(Homo sapiens (Human))
Université
Curated by ChEMBL
Université
Curated by ChEMBL
Affinity DataIC50: 15nMAssay Description:Binding affinity of the compound against [125I]-hCalcitonin gene-related peptide type receptor binding sites in guinea pig vas deferens membrane prep...More data for this Ligand-Target Pair
TargetCalcitonin gene-related peptide type 1 receptor(Homo sapiens (Human))
Université
Curated by ChEMBL
Université
Curated by ChEMBL
Affinity DataIC50: 20nMAssay Description:Binding affinity of the compound against [125I]-hCalcitonin gene-related peptide type receptor binding sites in guinea pig vas deferens membrane prep...More data for this Ligand-Target Pair
TargetCalcitonin gene-related peptide type 1 receptor(Homo sapiens (Human))
Université
Curated by ChEMBL
Université
Curated by ChEMBL
Affinity DataIC50: 20.2nMAssay Description:Binding affinity against [125I]-hCalcitonin gene-related peptide type receptor binding sites in guinea pig atrium membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 20.2nMAssay Description:Binding affinity against [125I]-hCalcitonin gene-related peptide type alpha receptor binding sites in rat brain membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 21.9nMAssay Description:Binding affinity against [125I]-hCalcitonin gene-related peptide type alpha receptor binding sites in rat brain membraneMore data for this Ligand-Target Pair
TargetCalcitonin gene-related peptide type 1 receptor(Homo sapiens (Human))
Université
Curated by ChEMBL
Université
Curated by ChEMBL
Affinity DataIC50: 22nMAssay Description:Binding affinity against [125I]-hCalcitonin gene-related peptide type receptor binding sites in guinea pig atrium membraneMore data for this Ligand-Target Pair
TargetCalcitonin gene-related peptide type 1 receptor(Homo sapiens (Human))
Université
Curated by ChEMBL
Université
Curated by ChEMBL
Affinity DataIC50: 25nMAssay Description:Binding affinity against [125I]-hCalcitonin gene-related peptide type receptor binding sites in guinea pig atrium membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 47nMAssay Description:Ability to induce 50% of maximal effect in rabbit vas deferens expressing Opioid receptor kappa 1More data for this Ligand-Target Pair
Affinity DataIC50: 77nMAssay Description:Ability to induce 50% of maximal effect in guinea pig ileum expressing Opioid receptor mu 1More data for this Ligand-Target Pair
Affinity DataIC50: 121nMAssay Description:Ability to induce 50% of maximal effect in rabbit vas deferens expressing Opioid receptor kappa 1More data for this Ligand-Target Pair
Affinity DataIC50: 157nMAssay Description:Ability to induce 50% of maximal effect in rabbit vas deferens expressing Opioid receptor kappa 1More data for this Ligand-Target Pair