TargetEpidermal growth factor receptor(Homo sapiens (Human))
Mcgill University Health Center/Royal Victoria Hospital
Curated by ChEMBL
Mcgill University Health Center/Royal Victoria Hospital
Curated by ChEMBL
Affinity DataIC50: 4.40nMAssay Description:Inhibition of EGFR tyrosine kinase expressed in A431 cellsMore data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Mcgill University Health Center/Royal Victoria Hospital
Curated by ChEMBL
Mcgill University Health Center/Royal Victoria Hospital
Curated by ChEMBL
Affinity DataIC50: 10nMAssay Description:Inhibition of poly(L-glutamic acid-L-tyrosine) phosphorylation by EGFR tyrosine kinase of A431 carcinoma cellsMore data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Mcgill University Health Center/Royal Victoria Hospital
Curated by ChEMBL
Mcgill University Health Center/Royal Victoria Hospital
Curated by ChEMBL
Affinity DataIC50: 11nMAssay Description:In vitro inhibition of Epidermal growth factor receptor tyrosine kinase isolated from A431 (human carcinoma).More data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Mcgill University Health Center/Royal Victoria Hospital
Curated by ChEMBL
Mcgill University Health Center/Royal Victoria Hospital
Curated by ChEMBL
Affinity DataIC50: 14nMAssay Description:In vitro inhibition of Epidermal growth factor receptor tyrosine kinase isolated from A431 (human carcinoma).More data for this Ligand-Target Pair
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Mcgill University/Royal Victoria Hospital
Curated by ChEMBL
Mcgill University/Royal Victoria Hospital
Curated by ChEMBL
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Mcgill University Health Center/Royal Victoria Hospital
Curated by ChEMBL
Mcgill University Health Center/Royal Victoria Hospital
Curated by ChEMBL
Affinity DataIC50: 24nMAssay Description:In vitro inhibition of Epidermal growth factor receptor tyrosine kinase isolated from A431 (human carcinoma).More data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Mcgill University Health Center/Royal Victoria Hospital
Curated by ChEMBL
Mcgill University Health Center/Royal Victoria Hospital
Curated by ChEMBL
Affinity DataIC50: 25nMAssay Description:In vitro inhibition of Epidermal growth factor receptor tyrosine kinase isolated from A431 (human carcinoma).More data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Mcgill University Health Center/Royal Victoria Hospital
Curated by ChEMBL
Mcgill University Health Center/Royal Victoria Hospital
Curated by ChEMBL
Affinity DataIC50: 26nMAssay Description:Inhibition of poly(L-glutamic acid-L-tyrosine) phosphorylation by EGFR tyrosine kinase of A431 carcinoma cellsMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Mcgill University/Royal Victoria Hospital
Curated by ChEMBL
Mcgill University/Royal Victoria Hospital
Curated by ChEMBL
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Mcgill University/Royal Victoria Hospital
Curated by ChEMBL
Mcgill University/Royal Victoria Hospital
Curated by ChEMBL
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Mcgill University Health Center/Royal Victoria Hospital
Curated by ChEMBL
Mcgill University Health Center/Royal Victoria Hospital
Curated by ChEMBL
Affinity DataIC50: 33nMAssay Description:Inhibition of EGFR-mediated poly(L-glutamic acid L-tyrosine) phosphorylationMore data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Mcgill University Health Center/Royal Victoria Hospital
Curated by ChEMBL
Mcgill University Health Center/Royal Victoria Hospital
Curated by ChEMBL
Affinity DataIC50: 37nMAssay Description:Inhibition of EGFR tyrosine kinase expressed in A431 cellsMore data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Mcgill University Health Center/Royal Victoria Hospital
Curated by ChEMBL
Mcgill University Health Center/Royal Victoria Hospital
Curated by ChEMBL
Affinity DataIC50: 38nMAssay Description:In vitro inhibition of Epidermal growth factor receptor tyrosine kinase isolated from A431 (human carcinoma).More data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Mcgill University Health Center/Royal Victoria Hospital
Curated by ChEMBL
Mcgill University Health Center/Royal Victoria Hospital
Curated by ChEMBL
Affinity DataIC50: 39nMAssay Description:In vitro inhibition of Epidermal growth factor receptor tyrosine kinase isolated from A431 (human carcinoma).More data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Mus musculus)
Mcgill University Health Center/Royal Victoria Hospital
Curated by ChEMBL
Mcgill University Health Center/Royal Victoria Hospital
Curated by ChEMBL
Affinity DataIC50: 40nMAssay Description:Inhibition of epidermal growth factor receptor tyrosine kinase (EGFR TK)More data for this Ligand-Target Pair
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Mcgill University/Royal Victoria Hospital
Curated by ChEMBL
Mcgill University/Royal Victoria Hospital
Curated by ChEMBL
TargetTyrosine-protein kinase ABL1/ABL2(Homo sapiens (Human))
Mcgill University/Royal Victoria Hospital
Curated by ChEMBL
Mcgill University/Royal Victoria Hospital
Curated by ChEMBL
Affinity DataIC50: 40nMAssay Description:Inhibition of Abl tyrosine kinaseMore data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Mcgill University Health Center/Royal Victoria Hospital
Curated by ChEMBL
Mcgill University Health Center/Royal Victoria Hospital
Curated by ChEMBL
Affinity DataIC50: 44nMAssay Description:Inhibition of poly(L-glutamic acid-L-tyrosine) phosphorylation by EGFR tyrosine kinase of A431 carcinoma cellsMore data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Mcgill University Health Center/Royal Victoria Hospital
Curated by ChEMBL
Mcgill University Health Center/Royal Victoria Hospital
Curated by ChEMBL
Affinity DataIC50: 44nMT: 2°CAssay Description:EGFR kinase assay was perform using Nunc MaxiSorp purchased from Nalge Nunc Interantional.More data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Mcgill University Health Center/Royal Victoria Hospital
Curated by ChEMBL
Mcgill University Health Center/Royal Victoria Hospital
Curated by ChEMBL
Affinity DataIC50: 44nMAssay Description:In vitro inhibition of Epidermal growth factor receptor tyrosine kinase isolated from A431 (human carcinoma).More data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Mcgill University Health Center/Royal Victoria Hospital
Curated by ChEMBL
Mcgill University Health Center/Royal Victoria Hospital
Curated by ChEMBL
Affinity DataIC50: 64nMAssay Description:In vitro inhibition of Epidermal growth factor receptor tyrosine kinase isolated from A431 (human carcinoma).More data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Mus musculus)
Mcgill University Health Center/Royal Victoria Hospital
Curated by ChEMBL
Mcgill University Health Center/Royal Victoria Hospital
Curated by ChEMBL
Affinity DataIC50: 70nMAssay Description:Inhibition of epidermal growth factor receptor tyrosine kinase (EGFR TK)More data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Mcgill University Health Center/Royal Victoria Hospital
Curated by ChEMBL
Mcgill University Health Center/Royal Victoria Hospital
Curated by ChEMBL
Affinity DataIC50: 71nMAssay Description:In vitro inhibition of Epidermal growth factor receptor tyrosine kinase isolated from A431 (human carcinoma).More data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Mcgill University Health Center/Royal Victoria Hospital
Curated by ChEMBL
Mcgill University Health Center/Royal Victoria Hospital
Curated by ChEMBL
Affinity DataIC50: 71nMAssay Description:Inhibition of EGFR tyrosine kinase expressed in A431 cellsMore data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Mcgill University Health Center/Royal Victoria Hospital
Curated by ChEMBL
Mcgill University Health Center/Royal Victoria Hospital
Curated by ChEMBL
Affinity DataIC50: 100nMAssay Description:In vitro inhibition of Epidermal growth factor receptor tyrosine kinase isolated from A431 (human carcinoma).More data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Mus musculus)
Mcgill University Health Center/Royal Victoria Hospital
Curated by ChEMBL
Mcgill University Health Center/Royal Victoria Hospital
Curated by ChEMBL
Affinity DataIC50: 110nMAssay Description:Inhibition of epidermal growth factor receptor tyrosine kinase (EGFR TK)More data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Mcgill University Health Center/Royal Victoria Hospital
Curated by ChEMBL
Mcgill University Health Center/Royal Victoria Hospital
Curated by ChEMBL
Affinity DataIC50: 120nMT: 2°CAssay Description:EGFR kinase assay was perform using Nunc MaxiSorp purchased from Nalge Nunc Interantional.More data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Mus musculus)
Mcgill University Health Center/Royal Victoria Hospital
Curated by ChEMBL
Mcgill University Health Center/Royal Victoria Hospital
Curated by ChEMBL
Affinity DataIC50: 130nMAssay Description:Inhibition of epidermal growth factor receptor tyrosine kinase (EGFR TK)More data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Mcgill University Health Center/Royal Victoria Hospital
Curated by ChEMBL
Mcgill University Health Center/Royal Victoria Hospital
Curated by ChEMBL
Affinity DataIC50: 150nMT: 2°CAssay Description:EGFR kinase assay was perform using Nunc MaxiSorp purchased from Nalge Nunc Interantional.More data for this Ligand-Target Pair
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Mcgill University/Royal Victoria Hospital
Curated by ChEMBL
Mcgill University/Royal Victoria Hospital
Curated by ChEMBL
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Mcgill University Health Center/Royal Victoria Hospital
Curated by ChEMBL
Mcgill University Health Center/Royal Victoria Hospital
Curated by ChEMBL
Affinity DataIC50: 180nMAssay Description:Inhibition of EGFR-mediated poly(L-glutamic acid L-tyrosine) phosphorylationMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Mcgill University/Royal Victoria Hospital
Curated by ChEMBL
Mcgill University/Royal Victoria Hospital
Curated by ChEMBL
TargetTyrosine-protein kinase ABL1/ABL2(Homo sapiens (Human))
Mcgill University/Royal Victoria Hospital
Curated by ChEMBL
Mcgill University/Royal Victoria Hospital
Curated by ChEMBL
Affinity DataIC50: 195nMAssay Description:Inhibition of Abl tyrosine kinaseMore data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Mcgill University Health Center/Royal Victoria Hospital
Curated by ChEMBL
Mcgill University Health Center/Royal Victoria Hospital
Curated by ChEMBL
Affinity DataIC50: 200nMAssay Description:In vitro inhibition of Epidermal growth factor receptor tyrosine kinase isolated from A431 (human carcinoma).More data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Mcgill University Health Center/Royal Victoria Hospital
Curated by ChEMBL
Mcgill University Health Center/Royal Victoria Hospital
Curated by ChEMBL
Affinity DataIC50: 200nMT: 2°CAssay Description:EGFR kinase assay was perform using Nunc MaxiSorp purchased from Nalge Nunc Interantional.More data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Mcgill University Health Center/Royal Victoria Hospital
Curated by ChEMBL
Mcgill University Health Center/Royal Victoria Hospital
Curated by ChEMBL
Affinity DataIC50: 200nMAssay Description:Inhibition of EGFR tyrosine kinase expressed in A431 cellsMore data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Mcgill University Health Center/Royal Victoria Hospital
Curated by ChEMBL
Mcgill University Health Center/Royal Victoria Hospital
Curated by ChEMBL
Affinity DataIC50: 200nMAssay Description:Inhibition of poly(L-glutamic acid-L-tyrosine) phosphorylation by EGFR tyrosine kinase of A431 carcinoma cellsMore data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Mus musculus)
Mcgill University Health Center/Royal Victoria Hospital
Curated by ChEMBL
Mcgill University Health Center/Royal Victoria Hospital
Curated by ChEMBL
Affinity DataIC50: 200nMAssay Description:Inhibition of epidermal growth factor receptor tyrosine kinase (EGFR TK)More data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Mcgill University Health Center/Royal Victoria Hospital
Curated by ChEMBL
Mcgill University Health Center/Royal Victoria Hospital
Curated by ChEMBL
Affinity DataIC50: 200nMAssay Description:In vitro inhibition of Epidermal growth factor receptor tyrosine kinase isolated from A431 (human carcinoma).More data for this Ligand-Target Pair
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Mcgill University/Royal Victoria Hospital
Curated by ChEMBL
Mcgill University/Royal Victoria Hospital
Curated by ChEMBL
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Mcgill University Health Center/Royal Victoria Hospital
Curated by ChEMBL
Mcgill University Health Center/Royal Victoria Hospital
Curated by ChEMBL
Affinity DataIC50: 238nMAssay Description:In vitro inhibition of Epidermal growth factor receptor tyrosine kinase isolated from A431 (human carcinoma).More data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Mcgill University Health Center/Royal Victoria Hospital
Curated by ChEMBL
Mcgill University Health Center/Royal Victoria Hospital
Curated by ChEMBL
Affinity DataIC50: 240nMAssay Description:Inhibition of EGFR-mediated poly(L-glutamic acid L-tyrosine) phosphorylationMore data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Mcgill University Health Center/Royal Victoria Hospital
Curated by ChEMBL
Mcgill University Health Center/Royal Victoria Hospital
Curated by ChEMBL
Affinity DataIC50: 335nMAssay Description:In vitro inhibition of Epidermal growth factor receptor tyrosine kinase isolated from A431 (human carcinoma).More data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Mcgill University Health Center/Royal Victoria Hospital
Curated by ChEMBL
Mcgill University Health Center/Royal Victoria Hospital
Curated by ChEMBL
Affinity DataIC50: 390nMAssay Description:Inhibition of EGFR-mediated poly(L-glutamic acid L-tyrosine) phosphorylationMore data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Mcgill University Health Center/Royal Victoria Hospital
Curated by ChEMBL
Mcgill University Health Center/Royal Victoria Hospital
Curated by ChEMBL
Affinity DataIC50: 482nMAssay Description:In vitro inhibition of Epidermal growth factor receptor tyrosine kinase isolated from A431 (human carcinoma).More data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Mcgill University Health Center/Royal Victoria Hospital
Curated by ChEMBL
Mcgill University Health Center/Royal Victoria Hospital
Curated by ChEMBL
Affinity DataIC50: 500nMAssay Description:Inhibition of EGFR-mediated poly(L-glutamic acid L-tyrosine) phosphorylationMore data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Mcgill University Health Center/Royal Victoria Hospital
Curated by ChEMBL
Mcgill University Health Center/Royal Victoria Hospital
Curated by ChEMBL
Affinity DataIC50: 508nMAssay Description:In vitro inhibition of Epidermal growth factor receptor tyrosine kinase isolated from A431 (human carcinoma).More data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Mus musculus)
Mcgill University Health Center/Royal Victoria Hospital
Curated by ChEMBL
Mcgill University Health Center/Royal Victoria Hospital
Curated by ChEMBL
Affinity DataIC50: 578nMAssay Description:Inhibition of epidermal growth factor receptor tyrosine kinase (EGFR TK)More data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Mcgill University Health Center/Royal Victoria Hospital
Curated by ChEMBL
Mcgill University Health Center/Royal Victoria Hospital
Curated by ChEMBL
Affinity DataIC50: 630nMAssay Description:Inhibition of EGFR-mediated poly(L-glutamic acid L-tyrosine) phosphorylationMore data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Mcgill University Health Center/Royal Victoria Hospital
Curated by ChEMBL
Mcgill University Health Center/Royal Victoria Hospital
Curated by ChEMBL
Affinity DataIC50: 720nMAssay Description:Inhibition of EGFR-mediated poly(L-glutamic acid L-tyrosine) phosphorylationMore data for this Ligand-Target Pair