Affinity DataKi: 540nMAssay Description:Time dependent inhibition of CYP3A4 in human liver microsomesMore data for this Ligand-Target Pair
Affinity DataIC50: 0.340nMAssay Description:Activated Akt isoforms and pleckstrin homology domain deletion constructs were assayed utilizing a GSK-derived biotinylated peptide substrate. The e...More data for this Ligand-Target Pair
Affinity DataIC50: 0.380nMpH: 7.5Assay Description:Activated Akt isoforms and pleckstrin homology domain deletion constructs were assayed utilizing a GSK-derived biotinylated peptide substrate. The e...More data for this Ligand-Target Pair
Affinity DataIC50: 0.700nMAssay Description:Activated Akt isoforms and pleckstrin homology domain deletion constructs were assayed utilizing a GSK-derived biotinylated peptide substrate. The e...More data for this Ligand-Target Pair
Affinity DataIC50: 1.70nMpH: 7.5Assay Description:Activated Akt isoforms and pleckstrin homology domain deletion constructs were assayed utilizing a GSK-derived biotinylated peptide substrate. The e...More data for this Ligand-Target Pair
Affinity DataIC50: 2.30nMpH: 7.5Assay Description:Activated Akt isoforms and pleckstrin homology domain deletion constructs were assayed utilizing a GSK-derived biotinylated peptide substrate. The e...More data for this Ligand-Target Pair
Affinity DataIC50: 2.60nMAssay Description:Inhibition of human cloned Akt1 expressed in Drosophila S2 cells by HTRF assayMore data for this Ligand-Target Pair
Affinity DataIC50: 2.80nMAssay Description:Inhibition of human cloned Akt1 expressed in Drosophila S2 cells by HTRF assayMore data for this Ligand-Target Pair
Affinity DataIC50: 2.80nMAssay Description:Inhibition of human cloned Akt2 expressed in Drosophila S2 cells by HTRF assayMore data for this Ligand-Target Pair
Affinity DataIC50: 3.30nMAssay Description:Inhibition of human cloned Akt1 expressed in Drosophila S2 cells by HTRF assayMore data for this Ligand-Target Pair
Affinity DataIC50: 4nMAssay Description:Inhibition of human cloned Akt1 expressed in Drosophila S2 cells by HTRF assayMore data for this Ligand-Target Pair
Affinity DataIC50: 4.60nMAssay Description:Inhibition of human cloned Akt1 expressed in Drosophila S2 cells by HTRF assayMore data for this Ligand-Target Pair
Affinity DataIC50: 5nMAssay Description:Inhibition of Akt1 (unknown origin) by cell based assayMore data for this Ligand-Target Pair
Affinity DataIC50: 6.10nMpH: 7.5Assay Description:Activated Akt isoforms and pleckstrin homology domain deletion constructs were assayed utilizing a GSK-derived biotinylated peptide substrate. The e...More data for this Ligand-Target Pair
Affinity DataIC50: 6.70nMAssay Description:Inhibition of human cloned Akt2 expressed in Drosophila S2 cells by HTRF assayMore data for this Ligand-Target Pair
Affinity DataIC50: 8.20nMpH: 7.5Assay Description:Activated Akt isoforms and pleckstrin homology domain deletion constructs were assayed utilizing a GSK-derived biotinylated peptide substrate. The e...More data for this Ligand-Target Pair
Affinity DataIC50: 8.5nMAssay Description:Inhibition of human cloned Akt1 expressed in Drosophila S2 cells by HTRF assayMore data for this Ligand-Target Pair
Affinity DataIC50: 9.40nMAssay Description:Inhibition of human cloned Akt2 expressed in Drosophila S2 cells by HTRF assayMore data for this Ligand-Target Pair
Affinity DataIC50: 9.90nMAssay Description:Inhibition of human cloned Akt1 expressed in Drosophila S2 cells by HTRF assayMore data for this Ligand-Target Pair
Affinity DataIC50: 10nMpH: 7.5Assay Description:Activated Akt isoforms and pleckstrin homology domain deletion constructs were assayed utilizing a GSK-derived biotinylated peptide substrate. The e...More data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Inhibition of human cloned Akt2 expressed in Drosophila S2 cells by HTRF assayMore data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Inhibition of human cloned Akt1 expressed in Drosophila S2 cells by HTRF assayMore data for this Ligand-Target Pair
Affinity DataIC50: 10.4nMAssay Description:Inhibition of human cloned Akt2 expressed in Drosophila S2 cells by HTRF assayMore data for this Ligand-Target Pair
Affinity DataIC50: 10.5nMAssay Description:Inhibition of human cloned Akt2 expressed in Drosophila S2 cells by HTRF assayMore data for this Ligand-Target Pair
Affinity DataIC50: 11nMAssay Description:Inhibition of 50% inactivated mouse Nav1.7alpha incubated for 5 mins measured at 10 secs interval by PatchXpress automated electrophysiology methodMore data for this Ligand-Target Pair
Affinity DataIC50: 11nMAssay Description:Inhibition of 50% inactivated human Nav1.5alpha expressed in HEK293 cells measured after 5 to 10 mins post compound washout by PatchXpress automated ...More data for this Ligand-Target Pair
Affinity DataIC50: 14.6nMAssay Description:Inhibition of human cloned Akt2 expressed in Drosophila S2 cells by HTRF assayMore data for this Ligand-Target Pair
Affinity DataIC50: 17nMAssay Description:Inhibition of Akt1 (unknown origin) by cell based assayMore data for this Ligand-Target Pair
Affinity DataIC50: 17nMAssay Description:Inhibition of human cloned Akt1 expressed in Drosophila S2 cells by HTRF assayMore data for this Ligand-Target Pair
Affinity DataIC50: 18.1nMAssay Description:Inhibition of Akt1 (unknown origin) by cell based assayMore data for this Ligand-Target Pair
Affinity DataIC50: 18.3nMAssay Description:Inhibition of Akt1 (unknown origin) by cell based assayMore data for this Ligand-Target Pair
Affinity DataIC50: 21nMAssay Description:Inhibition of 50% inactivated human Nav1.7alpha expressed in HEK293 cells incubated for 5 mins measured at 10 secs interval by PatchXpress automated ...More data for this Ligand-Target Pair
Affinity DataIC50: 24nMpH: 7.5Assay Description:Activated Akt isoforms and pleckstrin homology domain deletion constructs were assayed utilizing a GSK-derived biotinylated peptide substrate. The e...More data for this Ligand-Target Pair
Affinity DataIC50: 24.1nMAssay Description:Inhibition of human cloned Akt2 expressed in Drosophila S2 cells by HTRF assayMore data for this Ligand-Target Pair
Affinity DataIC50: 24.6nMAssay Description:Inhibition of Akt1 (unknown origin) by cell based assayMore data for this Ligand-Target Pair
Affinity DataIC50: 26.7nMAssay Description:Inhibition of human cloned Akt1 expressed in Drosophila S2 cells by HTRF assayMore data for this Ligand-Target Pair
Affinity DataIC50: 27nMAssay Description:Inhibition of Akt1 (unknown origin) by cell based assayMore data for this Ligand-Target Pair
Affinity DataIC50: 29nMAssay Description:Inhibition of Nav1.2 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 30nMAssay Description:Inhibition of [3H]PIA binding to rat cortical adenosine A1 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 31nMAssay Description:Inhibition of NaV1.7 channel in human DRG neurons assessed as reduction of TTX-sensitive current by whole cell patch clamp assayMore data for this Ligand-Target Pair
Affinity DataIC50: 32nMpH: 7.5Assay Description:Activated Akt isoforms and pleckstrin homology domain deletion constructs were assayed utilizing a GSK-derived biotinylated peptide substrate. The e...More data for this Ligand-Target Pair
Affinity DataIC50: 39nMAssay Description:Inhibition of 50% inactivated human Nav1.7alpha expressed in HEK293 cells incubated for 5 mins measured at 10 secs interval by PatchXpress automated ...More data for this Ligand-Target Pair
Affinity DataIC50: 39nMpH: 7.5Assay Description:Activated Akt isoforms and pleckstrin homology domain deletion constructs were assayed utilizing a GSK-derived biotinylated peptide substrate. The e...More data for this Ligand-Target Pair
Affinity DataIC50: 41nMAssay Description:Inhibition of Akt2 (unknown origin) by cell based assayMore data for this Ligand-Target Pair
Affinity DataIC50: 41.8nMAssay Description:Inhibition of Akt1 (unknown origin) by cell based assayMore data for this Ligand-Target Pair
Affinity DataIC50: 47.7nMAssay Description:Inhibition of Akt2 (unknown origin) by cell based assayMore data for this Ligand-Target Pair
Affinity DataIC50: 50nMpH: 7.5Assay Description:Activated Akt isoforms and pleckstrin homology domain deletion constructs were assayed utilizing a GSK-derived biotinylated peptide substrate. The e...More data for this Ligand-Target Pair
Affinity DataIC50: 55.1nMAssay Description:Inhibition of human cloned Akt2 expressed in Drosophila S2 cells by HTRF assayMore data for this Ligand-Target Pair
Affinity DataIC50: 62.5nMAssay Description:Inhibition of Akt1 (unknown origin) by cell based assayMore data for this Ligand-Target Pair
Affinity DataIC50: 74nMAssay Description:Inhibition of 50% inactivated human Nav1.7alpha expressed in HEK293 cells incubated for 5 mins measured at 10 secs interval by PatchXpress automated ...More data for this Ligand-Target Pair