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Found 391 with Last Name = 'salois' and Initial = 'd'
TargetDelta-type opioid receptor(Homo sapiens (Human))
Astrazeneca R & D Montr£Al

Curated by ChEMBL
LigandPNGBDBM50302760(CHEMBL568818 | N,N-diethyl-4-((1-(2-(furan-3-yl)et...)
Affinity DataKi:  0.220nMAssay Description:Displacement of [125I]-[D-Ala2]deltorphin 2 from human cloned delta opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Astrazeneca R & D Montr£Al

Curated by ChEMBL
LigandPNGBDBM50302755(CHEMBL569316 | N,N-diethyl-4-((3-hydroxyphenyl)(1-...)
Affinity DataKi:  0.240nMAssay Description:Displacement of [125I]-[D-Ala2]deltorphin 2 from human cloned delta opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Astrazeneca R & D Montr£Al

Curated by ChEMBL
LigandPNGBDBM50302759(CHEMBL584941 | N,N-diethyl-4-((3-hydroxyphenyl)(1-...)
Affinity DataKi:  0.270nMAssay Description:Displacement of [125I]-[D-Ala2]deltorphin 2 from human cloned delta opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Astrazeneca R & D Montr£Al

Curated by ChEMBL
LigandPNGBDBM50299393(4-((1-benzylpiperidin-4-yl)(3-carbamoylphenyl)amin...)
Affinity DataKi:  0.290nMAssay Description:Displacement of [125I]-[D-Ala2]deltorphin 2 from human cloned delta opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Astrazeneca R & D Montr£Al

Curated by ChEMBL
LigandPNGBDBM50302756(4-((1-(2-(1H-imidazol-2-yl)ethyl)piperidin-4-yl)(3...)
Affinity DataKi:  0.300nMAssay Description:Displacement of [125I]-[D-Ala2]deltorphin 2 from human cloned delta opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Astrazeneca R & D Montr£Al

Curated by ChEMBL
LigandPNGBDBM50299390(CHEMBL574640 | Methyl 3-((1-benzylpiperidin-4-yl)(...)
Affinity DataKi:  0.410nMAssay Description:Displacement of [125I]-[D-Ala2]deltorphin 2 from human cloned delta opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Astrazeneca R & D Montr£Al

Curated by ChEMBL
LigandPNGBDBM50299385(4-((1-benzylpiperidin-4-yl)(3-hydroxyphenyl)amino)...)
Affinity DataKi:  0.420nMAssay Description:Displacement of [125I]-[D-Ala2]deltorphin 2 from human cloned delta opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Astrazeneca R & D Montr£Al

Curated by ChEMBL
LigandPNGBDBM50302765(CHEMBL569755 | N,N-diethyl-4-((3-hydroxyphenyl)(1-...)
Affinity DataKi:  0.420nMAssay Description:Displacement of [125I]-[D-Ala2]deltorphin 2 from human cloned delta opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Astrazeneca R & D Montr£Al

Curated by ChEMBL
LigandPNGBDBM50302758(CHEMBL570000 | N,N-diethyl-4-((1-(2-(furan-2-yl)et...)
Affinity DataKi:  0.420nMAssay Description:Displacement of [125I]-[D-Ala2]deltorphin 2 from human cloned delta opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Astrazeneca R&D Montreal

Curated by ChEMBL
LigandPNGBDBM50364921(CHEMBL1950329)
Affinity DataKi:  0.560nMAssay Description:Binding affinity to human CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Astrazeneca R & D Montr£Al

Curated by ChEMBL
LigandPNGBDBM50302763(CHEMBL569728 | N,N-diethyl-4-((3-hydroxyphenyl)(1-...)
Affinity DataKi:  0.640nMAssay Description:Displacement of [125I]-[D-Ala2]deltorphin 2 from human cloned delta opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Astrazeneca R & D Montr£Al

Curated by ChEMBL
LigandPNGBDBM50302757(CHEMBL568803 | N,N-diethyl-4-((3-hydroxyphenyl)(1-...)
Affinity DataKi:  0.650nMAssay Description:Displacement of [125I]-[D-Ala2]deltorphin 2 from human cloned delta opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Astrazeneca R & D Montr£Al

Curated by ChEMBL
LigandPNGBDBM50302761(CHEMBL569006 | N,N-diethyl-4-((1-(3-fluorophenethy...)
Affinity DataKi:  0.700nMAssay Description:Displacement of [125I]-[D-Ala2]deltorphin 2 from human cloned delta opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Astrazeneca R & D Montr£Al

Curated by ChEMBL
LigandPNGBDBM50302762(CHEMBL576267 | N,N-diethyl-4-((1-(2-fluorophenethy...)
Affinity DataKi:  0.760nMAssay Description:Displacement of [125I]-[D-Ala2]deltorphin 2 from human cloned delta opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Astrazeneca R & D Montr£Al

Curated by ChEMBL
LigandPNGBDBM50302766(4-((1-(2-cyclopropylethyl)piperidin-4-yl)(3-hydrox...)
Affinity DataKi:  0.970nMAssay Description:Displacement of [125I]-[D-Ala2]deltorphin 2 from human cloned delta opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Astrazeneca R & D Montr£Al

Curated by ChEMBL
LigandPNGBDBM50302769(CHEMBL571324 | N,N-diethyl-4-((3-hydroxyphenyl)(1-...)
Affinity DataKi:  0.990nMAssay Description:Displacement of [125I]-[D-Ala2]deltorphin 2 from human cloned delta opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Astrazeneca R & D Montr£Al

Curated by ChEMBL
LigandPNGBDBM50302768(4-((1-(but-3-enyl)piperidin-4-yl)(3-hydroxyphenyl)...)
Affinity DataKi:  1nMAssay Description:Displacement of [125I]-[D-Ala2]deltorphin 2 from human cloned delta opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Astrazeneca R & D Montr£Al

Curated by ChEMBL
LigandPNGBDBM50302777(CHEMBL569529 | N,N-diethyl-4-((3-hydroxyphenyl)(1-...)
Affinity DataKi:  1nMAssay Description:Displacement of [125I]-[D-Ala2]deltorphin 2 from human cloned delta opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Astrazeneca R&D Montreal

Curated by ChEMBL
LigandPNGBDBM50244317(2-(4-ethoxybenzyl)-1-(cyclopentylmethyl)-N,N-dieth...)
Affinity DataKi:  1nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Astrazeneca R & D Montr£Al

Curated by ChEMBL
LigandPNGBDBM50039029((+)-4-((alpha R)-((2S,5R)-4-allyl-2,5-dimethylpipe...)
Affinity DataKi:  1.30nMAssay Description:Displacement of [125I]-[D-Ala2]deltorphin 2 from human cloned delta opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Astrazeneca R & D Montr£Al

Curated by ChEMBL
LigandPNGBDBM50302764(CHEMBL568865 | N,N-diethyl-4-((3-hydroxyphenyl)(1-...)
Affinity DataKi:  1.40nMAssay Description:Displacement of [125I]-[D-Ala2]deltorphin 2 from human cloned delta opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Astrazeneca R & D Montr£Al

Curated by ChEMBL
LigandPNGBDBM50299389(4-((1-benzylpiperidin-4-yl)(3-(methylsulfonamido)p...)
Affinity DataKi:  1.40nMAssay Description:Displacement of [125I]-[D-Ala2]deltorphin 2 from human cloned delta opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Astrazeneca R&D Montreal

Curated by ChEMBL
LigandPNGBDBM50244316(2-(4-ethoxybenzyl)-1-(cyclobutylmethyl)-N,N-diethy...)
Affinity DataKi:  1.60nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Astrazeneca R & D Montr£Al

Curated by ChEMBL
LigandPNGBDBM50302776(4-((1-(2-(1H-imidazol-4-yl)ethyl)piperidin-4-yl)(3...)
Affinity DataKi:  1.60nMAssay Description:Displacement of [125I]-[D-Ala2]deltorphin 2 from human cloned delta opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Astrazeneca R & D Montr£Al

Curated by ChEMBL
LigandPNGBDBM50302778(CHEMBL570448 | N,N-diethyl-4-((3-hydroxyphenyl)(1-...)
Affinity DataKi:  1.70nMAssay Description:Displacement of [125I]-[D-Ala2]deltorphin 2 from human cloned delta opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Astrazeneca R & D Montr£Al

Curated by ChEMBL
LigandPNGBDBM50299382(4-((3-acetylphenyl)(1-benzylpiperidin-4-yl)amino)-...)
Affinity DataKi:  1.70nMAssay Description:Displacement of [125I]-[D-Ala2]deltorphin 2 from human cloned delta opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Astrazeneca R & D Montr£Al

Curated by ChEMBL
LigandPNGBDBM50299388(4-((3-acetamidophenyl)(1-benzylpiperidin-4-yl)amin...)
Affinity DataKi:  1.80nMAssay Description:Displacement of [125I]-[D-Ala2]deltorphin 2 from human cloned delta opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Astrazeneca R & D Montr£Al

Curated by ChEMBL
LigandPNGBDBM50299391(4-((3-aminophenyl)(1-benzylpiperidin-4-yl)amino)-N...)
Affinity DataKi:  2nMAssay Description:Displacement of [125I]-[D-Ala2]deltorphin 2 from human cloned delta opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Astrazeneca R & D Montr£Al

Curated by ChEMBL
LigandPNGBDBM50302767(4-((1-(2-cyclohexylethyl)piperidin-4-yl)(3-hydroxy...)
Affinity DataKi:  2.30nMAssay Description:Displacement of [125I]-[D-Ala2]deltorphin 2 from human cloned delta opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Astrazeneca R&D Montreal

Curated by ChEMBL
LigandPNGBDBM50244060(2-(4-ethoxybenzyl)-1-(cyclopropylmethyl)-N,N-dipro...)
Affinity DataKi:  2.80nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Astrazeneca R&D Montreal

Curated by ChEMBL
LigandPNGBDBM50244319(1-adamantan-1-ylmethyl-2-(4-ethoxy-benzyl)-1H-benz...)
Affinity DataKi:  2.80nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Astrazeneca R&D MontréAl

Curated by ChEMBL
LigandPNGBDBM60994((10R,10aR)-6,6,9-Trimethyl-3-pentyl-6a,7,8,10a-tet...)
Affinity DataKi:  2.90nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetCannabinoid receptor 1(Homo sapiens (Human))
Astrazeneca R&D MontréAl

Curated by ChEMBL
LigandPNGBDBM50364921(CHEMBL1950329)
Affinity DataKi:  3nMAssay Description:Displacement of [3H]-CP55,940 from human CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Astrazeneca R & D Montr£Al

Curated by ChEMBL
LigandPNGBDBM50299384(4-((1-benzylpiperidin-4-yl)(3-formylphenyl)amino)-...)
Affinity DataKi:  3.40nMAssay Description:Displacement of [125I]-[D-Ala2]deltorphin 2 from human cloned delta opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Astrazeneca R&D Montreal

Curated by ChEMBL
LigandPNGBDBM50244318(2-(4-ethoxybenzyl)-1-(cyclohexylmethyl)-N,N-diethy...)
Affinity DataKi:  3.70nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Astrazeneca R&D Montreal

Curated by ChEMBL
LigandPNGBDBM50243706(2-(4-ethoxybenzyl)-N,N-diethyl-1-((tetrahydro-2H-p...)
Affinity DataKi:  3.90nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Astrazeneca R&D Montreal

Curated by ChEMBL
LigandPNGBDBM50244140(CHEMBL517283 | N-(2-(4-ethoxybenzyl)-1-(cyclopropy...)
Affinity DataKi:  4nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Astrazeneca R&D Montreal

Curated by ChEMBL
LigandPNGBDBM50244214(CHEMBL458142 | N-(2-(4-ethoxybenzyl)-1-(cyclopropy...)
Affinity DataKi:  4nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Astrazeneca R&D Montreal

Curated by ChEMBL
LigandPNGBDBM50244277(2-(4-ethoxybenzyl)-1-(cyclopropylmethyl)-N,N-dieth...)
Affinity DataKi:  4.10nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Astrazeneca R&D Montreal

Curated by ChEMBL
LigandPNGBDBM50243961(2-(4-isopropoxybenzyl)-N,N-diethyl-1-isopentyl-1H-...)
Affinity DataKi:  4.5nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Astrazeneca R&D Montreal

Curated by ChEMBL
LigandPNGBDBM50244276(2-(4-ethoxybenzyl)-N,N-diethyl-1-isopentyl-1H-benz...)
Affinity DataKi:  4.5nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Astrazeneca R&D Montreal

Curated by ChEMBL
LigandPNGBDBM50244010(2-(4-phenoxybenzyl)-N,N-diethyl-1-isopentyl-1H-ben...)
Affinity DataKi:  4.90nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Astrazeneca R&D Montreal

Curated by ChEMBL
LigandPNGBDBM50244178(CHEMBL518206 | N-(2-(4-ethoxybenzyl)-1-(cyclopropy...)
Affinity DataKi:  5nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Astrazeneca R&D Montreal

Curated by ChEMBL
LigandPNGBDBM50244098(2-(4-ethoxybenzyl)-1-(cyclopropylmethyl)-N,N-bis(2...)
Affinity DataKi:  5.60nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Astrazeneca R&D Montreal

Curated by ChEMBL
LigandPNGBDBM50244181(1-(2-(4-ethoxybenzyl)-1-(cyclopropylmethyl)-1H-ben...)
Affinity DataKi:  5.70nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Astrazeneca R&D Montreal

Curated by ChEMBL
LigandPNGBDBM50244180(1-(2-(4-ethoxybenzyl)-1-(cyclopropylmethyl)-1H-ben...)
Affinity DataKi:  5.90nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Astrazeneca R&D Montreal

Curated by ChEMBL
LigandPNGBDBM50244096((2-(4-ethoxybenzyl)-1-(cyclopropylmethyl)-1H-benzo...)
Affinity DataKi:  6.90nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Astrazeneca R&D Montreal

Curated by ChEMBL
LigandPNGBDBM50244059(2-(4-ethoxybenzyl)-1-(cyclopropylmethyl)-N-methyl-...)
Affinity DataKi:  7.60nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Astrazeneca R&D Montreal

Curated by ChEMBL
LigandPNGBDBM50243861((R)-2-(4-ethoxybenzyl)-N,N-diethyl-1-((1-methylpip...)
Affinity DataKi:  8.90nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Astrazeneca R&D MontréAl

Curated by ChEMBL
LigandPNGBDBM50364923(CHEMBL1950333)
Affinity DataKi:  9nMAssay Description:Displacement of [3H]-CP55,940 from human CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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