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Found 176 with Last Name = 'scott' and Initial = 'ee'
TargetD(3) dopamine receptor(Homo sapiens (Human))
Smithkline Beecham Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50132022(Biphenyl-4-carboxylic acid [4-((4aS,10bS)-7-hydrox...)
Affinity DataKi:  1nMAssay Description:Binding affinity at Dopamine receptor D3 expressed in CHO cells by [125I]iodosulpiride displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Smithkline Beecham Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50216344(CHEMBL319116)
Affinity DataKi:  2nMAssay Description:Binding affinity at Dopamine receptor D3 expressed in CHO cells by [125I]iodosulpiride displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhenylethanolamine N-methyltransferase(Homo sapiens (Human))
University Of Kansas

Curated by ChEMBL
LigandPNGBDBM50554691(CHEMBL4764318)
Affinity DataKi:  2.10nMAssay Description:Competitive inhibition of C-terminal hexahistidine tag in human recombinant PNMT expressed in Escherichia coli assessed as inhibition constant using ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPhenylethanolamine N-methyltransferase(Homo sapiens (Human))
University Of Kansas

Curated by ChEMBL
LigandPNGBDBM50554692(CHEMBL4751862)
Affinity DataKi:  3.20nMAssay Description:Competitive inhibition of C-terminal hexahistidine tag in human recombinant PNMT expressed in Escherichia coli assessed as inhibition constant using ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPhenylethanolamine N-methyltransferase(Homo sapiens (Human))
University Of Kansas

Curated by ChEMBL
LigandPNGBDBM50554690(CHEMBL4782649)
Affinity DataKi:  3.30nMAssay Description:Competitive inhibition of C-terminal hexahistidine tag in human recombinant PNMT expressed in Escherichia coli assessed as inhibition constant using ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPhenylethanolamine N-methyltransferase(Homo sapiens (Human))
University Of Kansas

Curated by ChEMBL
LigandPNGBDBM50554695(CHEMBL4760727)
Affinity DataKi:  3.5nMAssay Description:Competitive inhibition of C-terminal hexahistidine tag in human recombinant PNMT expressed in Escherichia coli assessed as inhibition constant using ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPhenylethanolamine N-methyltransferase(Homo sapiens (Human))
University Of Kansas

Curated by ChEMBL
LigandPNGBDBM50554693(CHEMBL4800292)
Affinity DataKi:  3.80nMAssay Description:Competitive inhibition of C-terminal hexahistidine tag in human recombinant PNMT expressed in Escherichia coli assessed as inhibition constant using ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPhenylethanolamine N-methyltransferase(Homo sapiens (Human))
University Of Kansas

Curated by ChEMBL
LigandPNGBDBM50554689(CHEMBL4754656)
Affinity DataKi:  3.90nMAssay Description:Competitive inhibition of C-terminal hexahistidine tag in human recombinant PNMT expressed in Escherichia coli assessed as inhibition constant using ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Smithkline Beecham Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50470855(CHEMBL60708)
Affinity DataKi:  4nMAssay Description:Binding affinity against cloned human Dopamine receptor D4 using [3H]nemonapride as radioligandMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Smithkline Beecham Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50216340(CHEMBL99876)
Affinity DataKi:  5nMAssay Description:Binding affinity at Dopamine receptor D3 expressed in CHO cells by [125I]iodosulpiride displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Smithkline Beecham Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50470850(CHEMBL59326)
Affinity DataKi:  5nMAssay Description:Binding affinity against cloned human Dopamine receptor D4 using [3H]nemonapride as radioligandMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Smithkline Beecham Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50470854(CHEMBL433255)
Affinity DataKi:  6.30nMAssay Description:Binding affinity against cloned human Dopamine receptor D4 using [3H]nemonapride as radioligandMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Smithkline Beecham Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50216355(CHEMBL318925)
Affinity DataKi:  6.30nMAssay Description:Binding affinity at Dopamine receptor D3 expressed in CHO cells by [125I]iodosulpiride displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Smithkline Beecham Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50216339(CHEMBL2111591)
Affinity DataKi:  7.90nMAssay Description:Binding affinity at Dopamine receptor D3 expressed in CHO cells by [125I]iodosulpiride displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Smithkline Beecham Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50216348(CHEMBL95759)
Affinity DataKi:  7.90nMAssay Description:Binding affinity at Dopamine receptor D3 expressed in CHO cells by [125I]iodosulpiride displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Smithkline Beecham Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50216351(CHEMBL2111592)
Affinity DataKi:  10nMAssay Description:Binding affinity at Dopamine receptor D3 expressed in CHO cells by [125I]iodosulpiride displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Smithkline Beecham Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50216360(CHEMBL97856)
Affinity DataKi:  13nMAssay Description:Binding affinity at Dopamine receptor D3 expressed in CHO cells by [125I]iodosulpiride displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Smithkline Beecham Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50216350(CHEMBL97118)
Affinity DataKi:  16nMAssay Description:Binding affinity at Dopamine receptor D3 expressed in CHO cells by [125I]iodosulpiride displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Smithkline Beecham Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50216346(CHEMBL95743)
Affinity DataKi:  16nMAssay Description:Binding affinity at Dopamine receptor D3 expressed in CHO cells by [125I]iodosulpiride displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Smithkline Beecham Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50216353(CHEMBL98452)
Affinity DataKi:  16nMAssay Description:Binding affinity at Dopamine receptor D3 expressed in CHO cells by [125I]iodosulpiride displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhenylethanolamine N-methyltransferase(Homo sapiens (Human))
University Of Kansas

Curated by ChEMBL
LigandPNGBDBM50554685(CHEMBL4749263)
Affinity DataKi:  18nMAssay Description:Competitive inhibition of C-terminal hexahistidine tag in human recombinant PNMT expressed in Escherichia coli assessed as inhibition constant using ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Smithkline Beecham Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50470852(CHEMBL57019)
Affinity DataKi:  20nMAssay Description:Binding affinity against cloned human Dopamine receptor D4 using [3H]nemonapride as radioligandMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Smithkline Beecham Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50203469(3-Methoxy-naphthalene-2-carboxylic acid (1-benzyl-...)
Affinity DataKi:  20nMAssay Description:Binding affinity against cloned human Dopamine receptor D4 using [3H]nemonapride as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Smithkline Beecham Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50470849(CHEMBL59075)
Affinity DataKi:  25nMAssay Description:Binding affinity against cloned human Dopamine receptor D4 using [3H]nemonapride as radioligandMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Smithkline Beecham Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50132022(Biphenyl-4-carboxylic acid [4-((4aS,10bS)-7-hydrox...)
Affinity DataKi:  25nMAssay Description:Binding affinity at Dopamine receptor D2 expressed in CHO cells by [125I]iodosulpiride displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Smithkline Beecham Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50470857(CHEMBL299479)
Affinity DataKi:  25nMAssay Description:Binding affinity against cloned human Dopamine receptor D4 using [3H]nemonapride as radioligandMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Smithkline Beecham Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50470851(CHEMBL57407)
Affinity DataKi:  32nMAssay Description:Binding affinity against cloned human Dopamine receptor D4 using [3H]nemonapride as radioligandMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Smithkline Beecham Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50470856(CHEMBL292186)
Affinity DataKi:  32nMAssay Description:Binding affinity against cloned human Dopamine receptor D4 using [3H]nemonapride as radioligandMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPhenylethanolamine N-methyltransferase(Homo sapiens (Human))
University Of Kansas

Curated by ChEMBL
LigandPNGBDBM50554694(CHEMBL4740168)
Affinity DataKi:  38nMAssay Description:Competitive inhibition of C-terminal hexahistidine tag in human recombinant PNMT expressed in Escherichia coli assessed as inhibition constant using ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Smithkline Beecham Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50470855(CHEMBL60708)
Affinity DataKi:  40nMAssay Description:Binding affinity against cloned human Dopamine receptor D2 (long) using [125I]iodosulpiride as radioligandMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCytochrome P450 2A13(Homo sapiens (Human))
University Of Kansas

Curated by ChEMBL
LigandPNGBDBM50041234(6-hydroxy-7-methoxy-5-benzofuranacrylic acid delta...)
Affinity DataKi:  40nMAssay Description:Mixed inhibition of CYP2A13 (unknown origin)More data for this Ligand-Target Pair
TargetPhenylethanolamine N-methyltransferase(Homo sapiens (Human))
University Of Kansas

Curated by ChEMBL
LigandPNGBDBM50554681(CHEMBL4795252)
Affinity DataKi:  46nMAssay Description:Competitive inhibition of C-terminal hexahistidine tag in human recombinant PNMT expressed in Escherichia coli assessed as inhibition constant using ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Smithkline Beecham Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50216357(CHEMBL329702)
Affinity DataKi:  50nMAssay Description:Binding affinity at Dopamine receptor D3 expressed in CHO cells by [125I]iodosulpiride displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Smithkline Beecham Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50216359(CHEMBL97107)
Affinity DataKi:  50nMAssay Description:Binding affinity at Dopamine receptor D3 expressed in CHO cells by [125I]iodosulpiride displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhenylethanolamine N-methyltransferase(Homo sapiens (Human))
University Of Kansas

Curated by ChEMBL
LigandPNGBDBM50554684(CHEMBL4796664)
Affinity DataKi:  57nMAssay Description:Competitive inhibition of C-terminal hexahistidine tag in human recombinant PNMT expressed in Escherichia coli assessed as inhibition constant using ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Smithkline Beecham Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50216344(CHEMBL319116)
Affinity DataKi:  63nMAssay Description:Binding affinity at Dopamine receptor D2 expressed in CHO cells by [125I]iodosulpiride displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhenylethanolamine N-methyltransferase(Homo sapiens (Human))
University Of Kansas

Curated by ChEMBL
LigandPNGBDBM50554682(CHEMBL4789060)
Affinity DataKi:  70nMAssay Description:Competitive inhibition of C-terminal hexahistidine tag in human recombinant PNMT expressed in Escherichia coli assessed as inhibition constant using ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPhenylethanolamine N-methyltransferase(Homo sapiens (Human))
University Of Kansas

Curated by ChEMBL
LigandPNGBDBM50554688(CHEMBL4791266)
Affinity DataKi:  71nMAssay Description:Competitive inhibition of C-terminal hexahistidine tag in human recombinant PNMT expressed in Escherichia coli assessed as inhibition constant using ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPhenylethanolamine N-methyltransferase(Homo sapiens (Human))
University Of Kansas

Curated by ChEMBL
LigandPNGBDBM50554680(CHEMBL4791373)
Affinity DataKi:  86nMAssay Description:Competitive inhibition of C-terminal hexahistidine tag in human recombinant PNMT expressed in Escherichia coli assessed as inhibition constant using ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Smithkline Beecham Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50203469(3-Methoxy-naphthalene-2-carboxylic acid (1-benzyl-...)
Affinity DataKi:  126nMAssay Description:Binding affinity against cloned human Dopamine receptor D2 (long) using [125I]iodosulpiride as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2A6(Homo sapiens (Human))
University Of Kansas

Curated by ChEMBL
LigandPNGBDBM50240772((1R,2S)-(-)-2-phenylcyclopropylamine | (1R,2S)-2-p...)
Affinity DataKi:  130nMAssay Description:Mixed inhibition of CYP2A6 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Smithkline Beecham Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50470853(CHEMBL61090)
Affinity DataKi:  200nMAssay Description:Binding affinity against cloned human Dopamine receptor D4 using [3H]nemonapride as radioligandMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Smithkline Beecham Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50216345(CHEMBL97440)
Affinity DataKi:  200nMAssay Description:Binding affinity at Dopamine receptor D3 expressed in CHO cells by [125I]iodosulpiride displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2A6(Homo sapiens (Human))
University Of Kansas

Curated by ChEMBL
LigandPNGBDBM50041234(6-hydroxy-7-methoxy-5-benzofuranacrylic acid delta...)
Affinity DataKi:  250nMAssay Description:Mixed inhibition of CYP2A6 (unknown origin)More data for this Ligand-Target Pair
TargetD(3) dopamine receptor(Homo sapiens (Human))
Smithkline Beecham Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50216358(CHEMBL317996)
Affinity DataKi:  251nMAssay Description:Binding affinity at Dopamine receptor D3 expressed in CHO cells by [125I]iodosulpiride displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Smithkline Beecham Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50216356(CHEMBL97840)
Affinity DataKi:  251nMAssay Description:Binding affinity at Dopamine receptor D3 expressed in CHO cells by [125I]iodosulpiride displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Smithkline Beecham Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50216355(CHEMBL318925)
Affinity DataKi:  251nMAssay Description:Binding affinity at Dopamine receptor D2 expressed in CHO cells by [125I]iodosulpiride displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Smithkline Beecham Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50216340(CHEMBL99876)
Affinity DataKi:  316nMAssay Description:Binding affinity at Dopamine receptor D2 expressed in CHO cells by [125I]iodosulpiride displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Smithkline Beecham Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50216360(CHEMBL97856)
Affinity DataKi:  316nMAssay Description:Binding affinity at Dopamine receptor D2 expressed in CHO cells by [125I]iodosulpiride displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Smithkline Beecham Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50216351(CHEMBL2111592)
Affinity DataKi:  316nMAssay Description:Binding affinity at Dopamine receptor D2 expressed in CHO cells by [125I]iodosulpiride displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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