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Found 30 with Last Name = 'segre' and Initial = 'g'
TargetBeta-1 adrenergic receptor(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50040072(4-Chloro-benzene-1,3-disulfonic acid 3-amide 1-({2...)
Affinity DataKi:  1.40nMAssay Description:Inhibition of [3H]-Dihydroalprenolol binding to beta 1 adrenoceptor from turkey erythrocyte membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50040065(5-[3-(tert-butylamino)-2-hydroxypropoxy]-3,4-dihyd...)
Affinity DataKi:  1.90nMAssay Description:Inhibition of [3H]-Dihydroalprenolol binding to beta 1 adrenoceptor from turkey erythrocyte membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetBeta-1 adrenergic receptor(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM25761(Anapriline | Avlocardyl | CHEMBL27 | PROPANOLOL(-)...)
Affinity DataKi:  2.30nMAssay Description:Inhibition of [3H]-Dihydroalprenolol binding to beta 1 adrenoceptor from turkey erythrocyte membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetBeta-1 adrenergic receptor(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50040076(4-Chloro-benzene-1,3-disulfonic acid 3-amide 1-({2...)
Affinity DataKi:  5.20nMAssay Description:Inhibition of [3H]-Dihydroalprenolol binding to beta 1 adrenoceptor from turkey erythrocyte membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50040073(4-Chloro-N-{2-[2-hydroxy-3-(3-oxo-3,4-dihydro-2H-b...)
Affinity DataKi:  7.40nMAssay Description:Inhibition of [3H]-Dihydroalprenolol binding to beta 1 adrenoceptor from turkey erythrocyte membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50040069(2-Chloro-5-{2-[2-hydroxy-3-(3-oxo-3,4-dihydro-2H-b...)
Affinity DataKi:  7.80nMAssay Description:Inhibition of [3H]-Dihydroalprenolol binding to beta 1 adrenoceptor from turkey erythrocyte membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50040074(2-Chloro-5-{2-[2-hydroxy-3-(naphthalen-1-yloxy)-pr...)
Affinity DataKi:  15nMAssay Description:Inhibition of [3H]-Dihydroalprenolol binding to beta 1 adrenoceptor from turkey erythrocyte membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50040070(8-tert-Butylamino-2-(3-hydroxy-propoxy)-4H-benzo[1...)
Affinity DataKi:  24nMAssay Description:Inhibition of [3H]-Dihydroalprenolol binding to beta 1 adrenoceptor from turkey erythrocyte membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50040071(2-Chloro-5-{4-[2-hydroxy-3-(naphthalen-1-yloxy)-pr...)
Affinity DataKi:  31nMAssay Description:Inhibition of [3H]-Dihydroalprenolol binding to beta 1 adrenoceptor from turkey erythrocyte membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50040066(2-Chloro-5-{4-[2-hydroxy-3-(3-oxo-3,4-dihydro-2H-b...)
Affinity DataKi:  140nMAssay Description:Inhibition of [3H]-Dihydroalprenolol binding to beta 1 adrenoceptor from turkey erythrocyte membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50040068(4-Chloro-benzene-1,3-disulfonic acid 3-amide 1-({2...)
Affinity DataKi:  160nMAssay Description:Inhibition of [3H]-Dihydroalprenolol binding to beta 1 adrenoceptor from turkey erythrocyte membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50040075(4-Chloro-N-{2-[2-hydroxy-3-(2-oxo-1,2,3,4-tetrahyd...)
Affinity DataKi:  300nMAssay Description:Inhibition of [3H]-Dihydroalprenolol binding to beta 1 adrenoceptor from turkey erythrocyte membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50040067(4-Chloro-N-{2-[2-hydroxy-3-(naphthalen-1-yloxy)-pr...)
Affinity DataKi:  820nMAssay Description:Inhibition of [3H]-Dihydroalprenolol binding to beta 1 adrenoceptor from turkey erythrocyte membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 1/12/13/14/2/3/4/5A, mitochondrial/5B, mitochondrial/6/7/9(Homo sapiens (Human))
Istituto Chimico Internazionale Dr. G. Rende

Curated by ChEMBL
LigandPNGBDBM50229834(CHEMBL328270)
Affinity DataIC50:  230nMAssay Description:Inhibition of Carbonic anhydrase enzyme in rabbitsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 1/12/13/14/2/3/4/5A, mitochondrial/5B, mitochondrial/6/7/9(Homo sapiens (Human))
Istituto Chimico Internazionale Dr. G. Rende

Curated by ChEMBL
LigandPNGBDBM50229838(CHEMBL88183)
Affinity DataIC50:  310nMAssay Description:Inhibition of Carbonic anhydrase enzyme in rabbitsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 1/12/13/14/2/3/4/5A, mitochondrial/5B, mitochondrial/6/7/9(Homo sapiens (Human))
Istituto Chimico Internazionale Dr. G. Rende

Curated by ChEMBL
LigandPNGBDBM50229841(CHEMBL420799)
Affinity DataIC50:  370nMAssay Description:Inhibition of Carbonic anhydrase enzyme in rabbitsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 1/12/13/14/2/3/4/5A, mitochondrial/5B, mitochondrial/6/7/9(Homo sapiens (Human))
Istituto Chimico Internazionale Dr. G. Rende

Curated by ChEMBL
LigandPNGBDBM50229842(CHEMBL90119)
Affinity DataIC50:  390nMAssay Description:Inhibition of Carbonic anhydrase enzyme in rabbitsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 1/12/13/14/2/3/4/5A, mitochondrial/5B, mitochondrial/6/7/9(Homo sapiens (Human))
Istituto Chimico Internazionale Dr. G. Rende

Curated by ChEMBL
LigandPNGBDBM50212309(CHEMBL91302)
Affinity DataIC50:  440nMAssay Description:Inhibition of Carbonic anhydrase enzyme in rabbitsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 1/12/13/14/2/3/4/5A, mitochondrial/5B, mitochondrial/6/7/9(Homo sapiens (Human))
Istituto Chimico Internazionale Dr. G. Rende

Curated by ChEMBL
LigandPNGBDBM10880(AZA | AZA2 | AZM acetazolamide | Acerazolamide, AA...)
Affinity DataIC50:  440nMAssay Description:Inhibition of Carbonic anhydrase enzyme in rabbitsMore data for this Ligand-Target Pair
TargetCarbonic anhydrase 1/12/13/14/2/3/4/5A, mitochondrial/5B, mitochondrial/6/7/9(Homo sapiens (Human))
Istituto Chimico Internazionale Dr. G. Rende

Curated by ChEMBL
LigandPNGBDBM50229847(CHEMBL91512)
Affinity DataIC50:  450nMAssay Description:Inhibition of Carbonic anhydrase enzyme in rabbitsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 1/12/13/14/2/3/4/5A, mitochondrial/5B, mitochondrial/6/7/9(Homo sapiens (Human))
Istituto Chimico Internazionale Dr. G. Rende

Curated by ChEMBL
LigandPNGBDBM50229846(CHEMBL264307)
Affinity DataIC50:  480nMAssay Description:Inhibition of Carbonic anhydrase enzyme in rabbitsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 1/12/13/14/2/3/4/5A, mitochondrial/5B, mitochondrial/6/7/9(Homo sapiens (Human))
Istituto Chimico Internazionale Dr. G. Rende

Curated by ChEMBL
LigandPNGBDBM50229839(CHEMBL91622)
Affinity DataIC50:  520nMAssay Description:Inhibition of Carbonic anhydrase enzyme in rabbitsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 1/12/13/14/2/3/4/5A, mitochondrial/5B, mitochondrial/6/7/9(Homo sapiens (Human))
Istituto Chimico Internazionale Dr. G. Rende

Curated by ChEMBL
LigandPNGBDBM50229835(CHEMBL90857)
Affinity DataIC50:  520nMAssay Description:Inhibition of Carbonic anhydrase enzyme in rabbitsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 1/12/13/14/2/3/4/5A, mitochondrial/5B, mitochondrial/6/7/9(Homo sapiens (Human))
Istituto Chimico Internazionale Dr. G. Rende

Curated by ChEMBL
LigandPNGBDBM50229845(CHEMBL91517)
Affinity DataIC50:  520nMAssay Description:Inhibition of Carbonic anhydrase enzyme in rabbitsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 1/12/13/14/2/3/4/5A, mitochondrial/5B, mitochondrial/6/7/9(Homo sapiens (Human))
Istituto Chimico Internazionale Dr. G. Rende

Curated by ChEMBL
LigandPNGBDBM50229843(CHEMBL91131)
Affinity DataIC50:  730nMAssay Description:Inhibition of Carbonic anhydrase enzyme in rabbitsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 1/12/13/14/2/3/4/5A, mitochondrial/5B, mitochondrial/6/7/9(Homo sapiens (Human))
Istituto Chimico Internazionale Dr. G. Rende

Curated by ChEMBL
LigandPNGBDBM50229837(CHEMBL89489)
Affinity DataIC50:  910nMAssay Description:Inhibition of Carbonic anhydrase enzyme in rabbitsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 1/12/13/14/2/3/4/5A, mitochondrial/5B, mitochondrial/6/7/9(Homo sapiens (Human))
Istituto Chimico Internazionale Dr. G. Rende

Curated by ChEMBL
LigandPNGBDBM50229844(CHEMBL328566)
Affinity DataIC50:  910nMAssay Description:Inhibition of Carbonic anhydrase enzyme in rabbitsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 1/12/13/14/2/3/4/5A, mitochondrial/5B, mitochondrial/6/7/9(Homo sapiens (Human))
Istituto Chimico Internazionale Dr. G. Rende

Curated by ChEMBL
LigandPNGBDBM50229840(CHEMBL329625)
Affinity DataIC50:  940nMAssay Description:Inhibition of Carbonic anhydrase enzyme in rabbitsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed