Compile Data Set for Download or QSAR
maximum 50k data
Found 7 with Last Name = 'sernissi' and Initial = 'l'
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
University Of Florence

Curated by ChEMBL
LigandPNGBDBM50235980(2-((2S,5R,8S,11S)-5-benzyl-11-(3-guanidinopropyl)-...)
Affinity DataIC50:  0.400nMAssay Description:Binding affinity to integrin alphav/beta3 heterodimer in human M21 cells assessed as inhibition of integrin-mediated human M21 cell adhesion to vitro...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
University Of Florence

Curated by ChEMBL
LigandPNGBDBM50140178(CHEMBL3754350)
Affinity DataIC50:  2.40nMAssay Description:Binding affinity to integrin alphav/beta3 heterodimer in human M21 cells assessed as inhibition of integrin-mediated human M21 cell adhesion to vitro...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-5/beta-1(Homo sapiens (Human))
University Of Florence

Curated by ChEMBL
LigandPNGBDBM50140179(CHEMBL3753748)
Affinity DataIC50:  15nMAssay Description:Binding affinity to integrin alpha5/beta1 heterodimer in human K562 cells assessed as inhibition of integrin-mediated human K562 cell adhesion to fib...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
University Of Florence

Curated by ChEMBL
LigandPNGBDBM50140177(CHEMBL3752070)
Affinity DataIC50:  20nMAssay Description:Binding affinity to integrin alphav/beta3 heterodimer (unknown origin) assessed as inhibition of integrin-mediated cell adhesion to vitronectinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-5/beta-1(Homo sapiens (Human))
University Of Florence

Curated by ChEMBL
LigandPNGBDBM50140178(CHEMBL3754350)
Affinity DataIC50:  26nMAssay Description:Binding affinity to integrin alpha5/beta1 heterodimer in human K562 cells assessed as inhibition of integrin-mediated human K562 cell adhesion to fib...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
University Of Florence

Curated by ChEMBL
LigandPNGBDBM50140179(CHEMBL3753748)
Affinity DataIC50:  34nMAssay Description:Binding affinity to integrin alphav/beta3 heterodimer in human M21 cells assessed as inhibition of integrin-mediated human M21 cell adhesion to vitro...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-5/beta-1(Homo sapiens (Human))
University Of Florence

Curated by ChEMBL
LigandPNGBDBM50140177(CHEMBL3752070)
Affinity DataIC50:  1.50E+3nMAssay Description:Binding affinity to integrin alpha5/beta1 heterodimer (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed