TargetSigma non-opioid intracellular receptor 1(RAT)
The University Of Mississippi
Curated by PDSP Ki Database
The University Of Mississippi
Curated by PDSP Ki Database
Affinity DataKi: 0.120nMAssay Description:Displacement of [3H](+)-pentazocine from opioid sigma1 receptor in rat brain homogenateMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(RAT)
The University Of Mississippi
Curated by PDSP Ki Database
The University Of Mississippi
Curated by PDSP Ki Database
Affinity DataKi: 0.350nMAssay Description:Displacement of [3H](+)-pentazocine from sigma 1 opioid receptor in rat brain cerebellumMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(RAT)
The University Of Mississippi
Curated by PDSP Ki Database
The University Of Mississippi
Curated by PDSP Ki Database
Affinity DataKi: 0.380nMAssay Description:Displacement of [3H](+)-pentazocine from sigma 1 opioid receptor in rat brain cerebellumMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(RAT)
The University Of Mississippi
Curated by PDSP Ki Database
The University Of Mississippi
Curated by PDSP Ki Database
Affinity DataKi: 0.410nMAssay Description:Displacement of [3H](+)-pentazocine from sigma 1 opioid receptor in rat brain cerebellumMore data for this Ligand-Target Pair
Affinity DataKi: 0.700nMAssay Description:Inhibition of N-terminal GST-tagged human PARP2 (2 to 583 residues) expressed in baculovirus infected Sf9 cells using histone mixture (H2A and H2B) a...More data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(RAT)
The University Of Mississippi
Curated by PDSP Ki Database
The University Of Mississippi
Curated by PDSP Ki Database
Affinity DataKi: 1.28nMAssay Description:Displacement of [3H](+)-pentazocine from opioid sigma1 receptor in rat brain homogenateMore data for this Ligand-Target Pair
Affinity DataKi: 1.40nMAssay Description:Inhibition of N-terminal GST-tagged human full length PARP1 (2 to 1041 residues) expressed in baculovirus infected Sf9 cells using histone mixture (H...More data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(RAT)
The University Of Mississippi
Curated by PDSP Ki Database
The University Of Mississippi
Curated by PDSP Ki Database
Affinity DataKi: 1.48nMAssay Description:Displacement of [3H](+)-pentazocine from opioid sigma1 receptor in rat brain homogenateMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(RAT)
The University Of Mississippi
Curated by PDSP Ki Database
The University Of Mississippi
Curated by PDSP Ki Database
Affinity DataKi: 1.70nMAssay Description:Displacement of [3H](+)-pentazocine from sigma 1 opioid receptor in rat brain cerebellumMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(RAT)
The University Of Mississippi
Curated by PDSP Ki Database
The University Of Mississippi
Curated by PDSP Ki Database
Affinity DataKi: 2.20nMAssay Description:Displacement of [3H](+)-pentazocine from sigma 1 opioid receptor in rat brain cerebellumMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(RAT)
The University Of Mississippi
Curated by PDSP Ki Database
The University Of Mississippi
Curated by PDSP Ki Database
Affinity DataKi: 3.30nMAssay Description:Displacement of [3H](+)-pentazocine from sigma 1 opioid receptor in rat brain cerebellumMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(RAT)
The University Of Mississippi
Curated by PDSP Ki Database
The University Of Mississippi
Curated by PDSP Ki Database
Affinity DataKi: 3.35nMAssay Description:Displacement of [3H](+)-pentazocine from opioid sigma1 receptor in rat brain homogenateMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(RAT)
The University Of Mississippi
Curated by PDSP Ki Database
The University Of Mississippi
Curated by PDSP Ki Database
Affinity DataKi: 3.37nMAssay Description:Displacement of [3H](+)-pentazocine from opioid sigma1 receptor in rat brain homogenateMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(RAT)
The University Of Mississippi
Curated by PDSP Ki Database
The University Of Mississippi
Curated by PDSP Ki Database
Affinity DataKi: 3.70nMAssay Description:Displacement of [3H](+)-pentazocine from sigma 1 opioid receptor in rat brain cerebellumMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(RAT)
The University Of Mississippi
Curated by PDSP Ki Database
The University Of Mississippi
Curated by PDSP Ki Database
Affinity DataKi: 4.17nMAssay Description:Displacement of [3H](+)-pentazocine from opioid sigma1 receptor in rat brain homogenateMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(RAT)
The University Of Mississippi
Curated by PDSP Ki Database
The University Of Mississippi
Curated by PDSP Ki Database
Affinity DataKi: 4.60nMAssay Description:Displacement of [3H](+)-pentazocine from opioid sigma1 receptor in rat brain homogenateMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(RAT)
The University Of Mississippi
Curated by PDSP Ki Database
The University Of Mississippi
Curated by PDSP Ki Database
Affinity DataKi: 4.66nMAssay Description:Displacement of [3H](+)-pentazocine from opioid sigma1 receptor in rat brain homogenateMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(RAT)
The University Of Mississippi
Curated by PDSP Ki Database
The University Of Mississippi
Curated by PDSP Ki Database
Affinity DataKi: 4.90nMAssay Description:Displacement of [3H](+)-pentazocine from opioid sigma1 receptor in rat brain homogenateMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(RAT)
The University Of Mississippi
Curated by PDSP Ki Database
The University Of Mississippi
Curated by PDSP Ki Database
Affinity DataKi: 4.98nMAssay Description:Displacement of [3H](+)-pentazocine from opioid sigma1 receptor in rat brain homogenateMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(RAT)
The University Of Mississippi
Curated by PDSP Ki Database
The University Of Mississippi
Curated by PDSP Ki Database
Affinity DataKi: 5.22nMAssay Description:Displacement of [3H](+)-pentazocine from opioid sigma1 receptor in rat brain homogenateMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(RAT)
The University Of Mississippi
Curated by PDSP Ki Database
The University Of Mississippi
Curated by PDSP Ki Database
Affinity DataKi: 5.61nMAssay Description:Displacement of [3H](+)-pentazocine from opioid sigma1 receptor in rat brain homogenateMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(RAT)
The University Of Mississippi
Curated by PDSP Ki Database
The University Of Mississippi
Curated by PDSP Ki Database
Affinity DataKi: 6.55nMAssay Description:Displacement of [3H](+)-pentazocine from opioid sigma1 receptor in rat brain homogenateMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(RAT)
The University Of Mississippi
Curated by PDSP Ki Database
The University Of Mississippi
Curated by PDSP Ki Database
Affinity DataKi: 6.90nMAssay Description:Displacement of [3H](+)-pentazocine from opioid sigma1 receptor in rat brain homogenateMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(RAT)
The University Of Mississippi
Curated by PDSP Ki Database
The University Of Mississippi
Curated by PDSP Ki Database
Affinity DataKi: 10.6nMAssay Description:Displacement of [3H](+)-pentazocine from opioid sigma1 receptor in rat brain homogenateMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(RAT)
The University Of Mississippi
Curated by PDSP Ki Database
The University Of Mississippi
Curated by PDSP Ki Database
Affinity DataKi: 11.3nMAssay Description:Displacement of [3H](+)-pentazocine from opioid sigma1 receptor in rat brain homogenateMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(RAT)
The University Of Mississippi
Curated by PDSP Ki Database
The University Of Mississippi
Curated by PDSP Ki Database
Affinity DataKi: 30nMAssay Description:Displacement of [3H](+)-pentazocine from sigma 1 opioid receptor in rat brain cerebellumMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(RAT)
The University Of Mississippi
Curated by PDSP Ki Database
The University Of Mississippi
Curated by PDSP Ki Database
Affinity DataKi: 49nMAssay Description:Displacement of [3H](+)-pentazocine from sigma 1 opioid receptor in rat brain cerebellumMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(RAT)
The University Of Mississippi
Curated by PDSP Ki Database
The University Of Mississippi
Curated by PDSP Ki Database
Affinity DataKi: 113nMAssay Description:Displacement of [3H](+)-pentazocine from sigma 1 opioid receptor in rat brain cerebellumMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(RAT)
The University Of Mississippi
Curated by PDSP Ki Database
The University Of Mississippi
Curated by PDSP Ki Database
Affinity DataKi: 322nMAssay Description:Displacement of [3H](+)-pentazocine from sigma 1 opioid receptor in rat brain cerebellumMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
The University Of Mississippi
Curated by PDSP Ki Database
The University Of Mississippi
Curated by PDSP Ki Database
Affinity DataKi: 1.04E+3nMAssay Description:Displacement of [3H](-)-sulpiride from dopamine D2 receptor in rat brain homogenateMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
The University Of Mississippi
Curated by PDSP Ki Database
The University Of Mississippi
Curated by PDSP Ki Database
Affinity DataKi: 1.18E+3nMAssay Description:Displacement of [3H]WIN-35428 from dopamine transporter in rat brain homogenateMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
The University Of Mississippi
Curated by PDSP Ki Database
The University Of Mississippi
Curated by PDSP Ki Database
Affinity DataKi: 1.40E+3nMAssay Description:Displacement of [3H]paroxetine from serotonin transporter in rat brain homogenateMore data for this Ligand-Target Pair
Affinity DataKi: 5.00E+3nMAssay Description:Binding affinity to delta opioid receptorMore data for this Ligand-Target Pair
Affinity DataKi: 5.90E+3nMAssay Description:Binding affinity to mu opioid receptorMore data for this Ligand-Target Pair
Affinity DataKi: 9.80E+3nMAssay Description:Binding affinity to mu opioid receptorMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to delta opioid receptorMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to delta opioid receptorMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to delta opioid receptorMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to delta opioid receptorMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]nisoxetine from norepinephrine transporter in rat brain homogenateMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to mu opioid receptorMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to kappa opioid receptorMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to kappa opioid receptorMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to mu opioid receptorMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to mu opioid receptorMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to kappa opioid receptorMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to kappa opioid receptorMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to kappa opioid receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 0.110nMAssay Description:Inhibition of Nav1.7 (unknown origin) expressed in HEK293 cells assessed as reduction in veratridine-induced depolarization preincubated for 15 to 20...More data for this Ligand-Target Pair
Affinity DataIC50: 0.400nMAssay Description:Inhibition of N-terminal GST-tagged human full length PARP1 (2 to 1041 residues) expressed in baculovirus infected Sf9 cells using histone mixture (H...More data for this Ligand-Target Pair