Affinity DataKi: 100nMAssay Description:Binding affinity for human receptor subtype hSSTR4.More data for this Ligand-Target Pair
Affinity DataKi: 300nMAssay Description:Binding affinity for human receptor subtype hSSTR1More data for this Ligand-Target Pair
Affinity DataKi: 500nMAssay Description:Binding affinity for human receptor subtype hSSTR4.More data for this Ligand-Target Pair
Affinity DataKi: 600nMAssay Description:Binding affinity for human receptor subtype hSSTR2More data for this Ligand-Target Pair
Affinity DataKi: 600nMAssay Description:Binding affinity for human receptor subtype hSSTR3.More data for this Ligand-Target Pair
Affinity DataKi: 800nMAssay Description:Binding affinity for human receptor subtype hSSTR2More data for this Ligand-Target Pair
Affinity DataKi: 900nMAssay Description:Binding affinity for human receptor subtype hSSTR3.More data for this Ligand-Target Pair
Affinity DataKi: 1.10E+3nMAssay Description:Binding affinity for human receptor subtype hSSTR4.More data for this Ligand-Target Pair
Affinity DataKi: 1.30E+3nMAssay Description:Binding affinity for human receptor subtype hSSTR5.More data for this Ligand-Target Pair
Affinity DataKi: 1.70E+3nMAssay Description:Binding affinity for human receptor subtype hSSTR4.More data for this Ligand-Target Pair
Affinity DataKi: 1.80E+3nMAssay Description:Binding affinity for human receptor subtype hSSTR2More data for this Ligand-Target Pair
Affinity DataKi: 1.90E+3nMAssay Description:Binding affinity for human receptor subtype hSSTR4.More data for this Ligand-Target Pair
Affinity DataKi: 2.00E+3nMAssay Description:Binding affinity for human receptor subtype hSSTR4.More data for this Ligand-Target Pair
Affinity DataKi: 2.00E+3nMAssay Description:Binding affinity for human receptor subtype hSSTR4.More data for this Ligand-Target Pair
Affinity DataKi: 2.10E+3nMAssay Description:Binding affinity for human receptor subtype hSSTR1More data for this Ligand-Target Pair
Affinity DataKi: 2.40E+3nMAssay Description:Binding affinity for human receptor subtype hSSTR1More data for this Ligand-Target Pair
Affinity DataKi: 2.60E+3nMAssay Description:Binding affinity for human receptor subtype hSSTR2More data for this Ligand-Target Pair
Affinity DataKi: 2.70E+3nMAssay Description:Binding affinity for human receptor subtype hSSTR2More data for this Ligand-Target Pair
Affinity DataKi: 2.80E+3nMAssay Description:Binding affinity for human receptor subtype hSSTR3.More data for this Ligand-Target Pair
Affinity DataKi: 3.00E+3nMAssay Description:Binding affinity for human receptor subtype hSSTR3.More data for this Ligand-Target Pair
Affinity DataKi: 3.00E+3nMAssay Description:Binding affinity for human receptor subtype hSSTR5.More data for this Ligand-Target Pair
Affinity DataKi: 3.00E+3nMAssay Description:Binding affinity for human receptor subtype hSSTR4.More data for this Ligand-Target Pair
Affinity DataKi: 3.10E+3nMAssay Description:Binding affinity for human receptor subtype hSSTR2More data for this Ligand-Target Pair
Affinity DataKi: 3.30E+3nMAssay Description:Binding affinity for human receptor subtype hSSTR3.More data for this Ligand-Target Pair
Affinity DataKi: 3.30E+3nMAssay Description:Binding affinity for human receptor subtype hSSTR3.More data for this Ligand-Target Pair
Affinity DataKi: 3.40E+3nMAssay Description:Binding affinity for human receptor subtype hSSTR5.More data for this Ligand-Target Pair
Affinity DataKi: 3.70E+3nMAssay Description:Binding affinity for human receptor subtype hSSTR5.More data for this Ligand-Target Pair
Affinity DataKi: 3.90E+3nMAssay Description:Binding affinity for human receptor subtype hSSTR5.More data for this Ligand-Target Pair
Affinity DataKi: 4.00E+3nMAssay Description:Binding affinity for human receptor subtype hSSTR1More data for this Ligand-Target Pair
Affinity DataKi: 4.00E+3nMAssay Description:Binding affinity for human receptor subtype hSSTR5.More data for this Ligand-Target Pair
Affinity DataKi: 4.00E+3nMAssay Description:Binding affinity for human receptor subtype hSSTR1More data for this Ligand-Target Pair
Affinity DataKi: 4.10E+3nMAssay Description:Binding affinity for human receptor subtype hSSTR1More data for this Ligand-Target Pair
Affinity DataKi: 4.40E+3nMAssay Description:Binding affinity for human receptor subtype hSSTR1More data for this Ligand-Target Pair
Affinity DataKi: 4.60E+3nMAssay Description:Binding affinity for human receptor subtype hSSTR2More data for this Ligand-Target Pair
Affinity DataKi: 4.60E+3nMAssay Description:Binding affinity for human receptor subtype hSSTR2More data for this Ligand-Target Pair
Affinity DataKi: 5.10E+3nMAssay Description:Binding affinity for human receptor subtype hSSTR5.More data for this Ligand-Target Pair
Affinity DataKi: 6.20E+3nMAssay Description:Binding affinity for human receptor subtype hSSTR3.More data for this Ligand-Target Pair
Affinity DataKi: 6.40E+3nMAssay Description:Binding affinity for human receptor subtype hSSTR3.More data for this Ligand-Target Pair
Affinity DataKi: 6.80E+3nMAssay Description:Binding affinity for human receptor subtype hSSTR1More data for this Ligand-Target Pair
Affinity DataKi: 2.60E+4nMAssay Description:Inhibition of human LDH-AMore data for this Ligand-Target Pair
Affinity DataIC50: 0.0700nMAssay Description:Inhibition of human ALK using poly[Glu:Tyr] (4:1) as substrate and [gamma-33P]ATP measured after 1 hrMore data for this Ligand-Target Pair
TargetInsulin-like growth factor 1 receptor(Homo sapiens (Human))
Ariad Pharmaceuticals
Curated by ChEMBL
Ariad Pharmaceuticals
Curated by ChEMBL
Affinity DataIC50: 0.110nMAssay Description:Inhibition of human IGF1R using KKKSPGEYVNIEFG as substrate and [gamma-33P]ATP measured after 1 hrMore data for this Ligand-Target Pair
Affinity DataIC50: 0.120nMAssay Description:Inhibition of human ALK using poly[Glu:Tyr] (4:1) as substrate and [gamma-33P]ATP measured after 1 hrMore data for this Ligand-Target Pair
Affinity DataIC50: 0.150nMAssay Description:Inhibition of human ALK using poly[Glu:Tyr] (4:1) as substrate and [gamma-33P]ATP measured after 1 hrMore data for this Ligand-Target Pair
Affinity DataIC50: <0.150nMAssay Description:Inhibition of human LYN using poly[Glu:Tyr] by Hotspot assayMore data for this Ligand-Target Pair
Affinity DataIC50: 0.180nMAssay Description:Inhibition of human ALK using poly[Glu:Tyr] (4:1) as substrate and [gamma-33P]ATP measured after 1 hrMore data for this Ligand-Target Pair
Affinity DataIC50: 0.180nMAssay Description:Inhibition of human ALK using poly[Glu:Tyr] (4:1) as substrate and [gamma-33P]ATP measured after 1 hrMore data for this Ligand-Target Pair
Affinity DataIC50: 0.200nMAssay Description:Inhibition of wild type human ABL using [EAIYAAPFAKKK] peptide substrate by Hotspot assayMore data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase receptor Ret(Homo sapiens (Human))
Ariad Pharmaceuticals
Curated by ChEMBL
Ariad Pharmaceuticals
Curated by ChEMBL
Affinity DataIC50: 0.200nMAssay Description:Inhibition of human RET using KKKSPGEYVNIEFG by Hotspot assayMore data for this Ligand-Target Pair
Affinity DataIC50: 0.200nMAssay Description:Inhibition of wild type human ABL using [EAIYAAPFAKKK] peptide substrate by Hotspot assayMore data for this Ligand-Target Pair