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Found 583 with Last Name = 'smith' and Initial = 'ec'
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50065468(2-(4-Chloro-phenoxymethyl)-4-(3-piperidin-1-yl-pro...)
Affinity DataKi:  2nMAssay Description:Binding affinity of the compound at cloned Neuropeptide Y receptor type 1 expressed in AV-12 cells is evaluated.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50069414(2-(4-Chloro-phenoxymethyl)-4-methyl-1-{3-[1-(3-pip...)
Affinity DataKi:  4.5nMAssay Description:Binding affinity at cloned Neuropeptide Y-1 receptor expressed in AV-12 cells is evaluated.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50069417(2-(4-Chloro-phenoxymethyl)-4-methyl-1-{3-[1-(3-met...)
Affinity DataKi:  11nMAssay Description:Binding affinity at cloned Neuropeptide Y-1 receptor expressed in AV-12 cells is evaluated.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1(RAT)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50001265(3-(4-Amino-phenyl)-5,7-dichloro-4-hydroxy-1H-quino...)
Affinity DataKi:  18nMAssay Description:Ability to displace strychnine-insensitive [3H]-glycine binding to rat cortical membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50069423(4-(4-{3-[2-(4-Chloro-phenoxymethyl)-4-methyl-benzo...)
Affinity DataKi:  21nMAssay Description:Binding affinity at cloned Neuropeptide Y-1 receptor expressed in AV-12 cells is evaluated.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50069424(4-(4-{3-[2-(4-Chloro-phenoxymethyl)-4-methyl-benzo...)
Affinity DataKi:  29nMAssay Description:Binding affinity at cloned Neuropeptide Y-1 receptor expressed in AV-12 cells is evaluated.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50069421(2-(4-Chloro-phenoxymethyl)-4-methyl-1-[3-(1-phenet...)
Affinity DataKi:  29nMAssay Description:Binding affinity at cloned Neuropeptide Y-1 receptor expressed in AV-12 cells is evaluated.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50069427(2-(4-Chloro-phenoxymethyl)-4-methyl-1-[3-(1-propyl...)
Affinity DataKi:  29nMAssay Description:Binding affinity at cloned Neuropeptide Y-1 receptor expressed in AV-12 cells is evaluated.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50069412(2-(4-Chloro-phenoxymethyl)-4-methyl-1-{3-[1-(2-pip...)
Affinity DataKi:  37nMAssay Description:Binding affinity at cloned Neuropeptide Y-1 receptor expressed in AV-12 cells is evaluated.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1(RAT)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50001266(5,7-DICHLORO-4-HYDROXYQUINOLINE-2-CARBOXYLIC ACID ...)
Affinity DataKi:  40nMAssay Description:Tested for the ability to displace [3H]-glycine, by greater than 50%, from NMDA receptor of rat cortical membranes at a dose of 10 microMMore data for this Ligand-Target Pair
TargetGlutamate receptor ionotropic, NMDA 1(RAT)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50001266(5,7-DICHLORO-4-HYDROXYQUINOLINE-2-CARBOXYLIC ACID ...)
Affinity DataKi:  40nMAssay Description:Displacement of [3H]glycine from glycine site on the NMDA receptor.More data for this Ligand-Target Pair
TargetGlutamate receptor ionotropic, NMDA 1(RAT)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50001266(5,7-DICHLORO-4-HYDROXYQUINOLINE-2-CARBOXYLIC ACID ...)
Affinity DataKi:  40nMAssay Description:Ability to displace strychnine-insensitive [3H]-glycine binding to rat cortical membranes.More data for this Ligand-Target Pair
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50069415(2-(4-Chloro-phenoxymethyl)-4-methyl-1-{3-[1-(4-pip...)
Affinity DataKi:  52nMAssay Description:Binding affinity at cloned Neuropeptide Y-1 receptor expressed in AV-12 cells is evaluated.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50069415(2-(4-Chloro-phenoxymethyl)-4-methyl-1-{3-[1-(4-pip...)
Affinity DataKi:  52nMAssay Description:Binding affinity at cloned Neuropeptide Y-1 receptor expressed in AV-12 cells is evaluated.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50069418(2-(4-Chloro-phenoxymethyl)-4-methyl-1-[3-(1-methyl...)
Affinity DataKi:  52nMAssay Description:Binding affinity at cloned Neuropeptide Y-1 receptor expressed in AV-12 cells is evaluated.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50069420(2-(4-Chloro-phenoxymethyl)-4-methyl-1-{3-[1-(3-phe...)
Affinity DataKi:  57nMAssay Description:Binding affinity at cloned Neuropeptide Y-1 receptor expressed in AV-12 cells is evaluated.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50069413(4-(4-{3-[2-(4-Chloro-phenoxymethyl)-4-methyl-benzo...)
Affinity DataKi:  88nMAssay Description:Binding affinity at cloned Neuropeptide Y-1 receptor expressed in AV-12 cells is evaluated.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50069429(1-[3-(1-Benzyl-piperidin-4-yl)-propyl]-2-(4-chloro...)
Affinity DataKi:  109nMAssay Description:Binding affinity at cloned Neuropeptide Y-1 receptor expressed in AV-12 cells is evaluated.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50069426(2-(4-{3-[2-(4-Chloro-phenoxymethyl)-4-methyl-benzo...)
Affinity DataKi:  136nMAssay Description:Binding affinity at cloned Neuropeptide Y-1 receptor expressed in AV-12 cells is evaluated.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1(RAT)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50004952(3-(2-Carboxy-ethyl)-4,6-dichloro-1H-indole-2-carbo...)
Affinity DataKi:  140nMAssay Description:Tested for the ability to displace [3H]-glycine, by greater than 50%, from NMDA receptor of rat cortical membranes at a dose of 10 microMMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGlutamate receptor ionotropic, NMDA 1(RAT)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM22778(6,7-Dichloro-1,4-dihydro-quinoxaline-2,3-dione | 6...)
Affinity DataKi:  210nMAssay Description:Displacement of [3H]glycine from glycine site on the NMDA receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50069416(1-(4-{3-[2-(4-Chloro-phenoxymethyl)-4-methyl-benzo...)
Affinity DataKi:  260nMAssay Description:Binding affinity at cloned Neuropeptide Y-1 receptor expressed in AV-12 cells is evaluated.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1(RAT)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50001264(5,7-Dichloro-4-hydroxy-3-p-tolyl-1H-quinolin-2-one...)
Affinity DataKi:  300nMAssay Description:Ability to displace strychnine-insensitive [3H]-glycine binding to rat cortical membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50069428(2-(4-Chloro-phenoxymethyl)-4-methyl-1-(3-piperidin...)
Affinity DataKi:  335nMAssay Description:Binding affinity at cloned Neuropeptide Y-1 receptor expressed in AV-12 cells is evaluated.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1(RAT)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50129080(3-Carboxymethyl-4,6-dichloro-1H-indole-2-carboxyli...)
Affinity DataKi:  340nMAssay Description:Tested for the ability to displace [3H]-glycine, by greater than 50%, from NMDA receptor of rat cortical membranes at a dose of 10 microMMore data for this Ligand-Target Pair
In DepthDetails Article
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50069425((4-{3-[2-(4-Chloro-phenoxymethyl)-4-methyl-benzoim...)
Affinity DataKi:  427nMAssay Description:Binding affinity at cloned Neuropeptide Y-1 receptor expressed in AV-12 cells is evaluated.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1(RAT)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50002707(7,8-Dichloro-5H-[1,2,4]triazolo[4,3-a]quinoxalin-4...)
Affinity DataKi:  630nMAssay Description:Displacement of [3H]glycine from glycine site on the NMDA receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1(RAT)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50280807(3-Carboxymethyl-5,7-dichloro-4-oxo-1,4-dihydro-qui...)
Affinity DataKi:  650nMAssay Description:Tested for the ability to displace [3H]-glycine, by greater than 50%, from NMDA receptor of rat cortical membranes at a dose of 10 microMMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGlutamate receptor ionotropic, NMDA 1(RAT)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50001268(5,7-Dichloro-4-hydroxy-3-(4-nitro-phenyl)-1H-quino...)
Affinity DataKi:  860nMAssay Description:Ability to displace strychnine-insensitive [3H]-glycine binding to rat cortical membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1(RAT)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50004960(4,6-Dichloro-1H-indole-2-carboxylic acid | CHEMBL3...)
Affinity DataKi:  980nMAssay Description:Tested for the ability to displace [3H]-glycine, by greater than 50%, from NMDA receptor of rat cortical membranes at a dose of 10 microMMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGlutamate receptor ionotropic, NMDA 1(RAT)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50002696(7,8-Dichloro-5H-imidazo[1,2-a]quinoxalin-4-one | C...)
Affinity DataKi:  1.26E+3nMAssay Description:Displacement of [3H]glycine from glycine site on the NMDA receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1(RAT)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50002700(1-Butyl-7,8-dichloro-5H-[1,2,4]triazolo[4,3-a]quin...)
Affinity DataKi:  1.48E+3nMAssay Description:Displacement of [3H]glycine from glycine site on the NMDA receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50069422(4-(4-{3-[2-(4-Chloro-phenoxymethyl)-4-methyl-benzo...)
Affinity DataKi:  1.63E+3nMAssay Description:Binding affinity at cloned Neuropeptide Y-1 receptor expressed in AV-12 cells is evaluated.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50069419((4-{3-[2-(4-Chloro-phenoxymethyl)-4-methyl-benzoim...)
Affinity DataKi:  2.19E+3nMAssay Description:Binding affinity at cloned Neuropeptide Y-1 receptor expressed in AV-12 cells is evaluated.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1(RAT)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50002710(7,9-Dichloro-5H-[1,2,4]triazolo[4,3-a]quinoxalin-4...)
Affinity DataKi:  2.85E+3nMAssay Description:Displacement of [3H]glycine from glycine site on the NMDA receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1(RAT)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50002701(7,8-Dichloro-1-propyl-5H-[1,2,4]triazolo[4,3-a]qui...)
Affinity DataKi:  3.92E+3nMAssay Description:Displacement of [3H]glycine from glycine site on the NMDA receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1(RAT)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50001260(3-phenyl-4-hydroxyquinolin-2(1H)-one | 4-Hydroxy-3...)
Affinity DataKi:  4.50E+3nMAssay Description:Ability to displace strychnine-insensitive [3H]-glycine binding to rat cortical membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1(RAT)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50002711(7,8-Dichloro-1-ethyl-5H-[1,2,4]triazolo[4,3-a]quin...)
Affinity DataKi:  4.58E+3nMAssay Description:Displacement of [3H]glycine from glycine site on the NMDA receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1(RAT)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50009092(3-Carboxymethyl-1H-indole-2-carboxylic acid | CHEM...)
Affinity DataKi:  5.24E+3nMAssay Description:Tested for the ability to displace [3H]-glycine, by greater than 50%, from NMDA receptor of rat cortical membranes at a dose of 10 microMMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGlutamate receptor ionotropic, NMDA 1(RAT)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM81975(4-hydroxyquinoline-2-carboxylic acid | CAS_492-27-...)
Affinity DataKi:  5.40E+3nMAssay Description:Tested for the ability to displace [3H]-glycine, by greater than 50%, from NMDA receptor of rat cortical membranes at a dose of 10 microMMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGlutamate receptor ionotropic, NMDA 1(RAT)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM81975(4-hydroxyquinoline-2-carboxylic acid | CAS_492-27-...)
Affinity DataKi:  5.40E+3nMAssay Description:Ability to displace strychnine-insensitive [3H]-glycine binding to rat cortical membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1(RAT)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50280805(3-(2-Carboxy-ethyl)-5,7-dichloro-4-oxo-1,4-dihydro...)
Affinity DataKi:  7.04E+3nMAssay Description:Tested for the ability to displace [3H]-glycine, by greater than 50%, from NMDA receptor of rat cortical membranes at a dose of 10 microMMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGlutamate receptor ionotropic, NMDA 1(RAT)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50002704(7-Nitro-5H-[1,2,4]triazolo[4,3-a]quinoxalin-4-one ...)
Affinity DataKi:  7.35E+3nMAssay Description:Displacement of [3H]glycine from glycine site on the NMDA receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1(RAT)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50002709(8,9-Dichloro-6H-pyrazolo[1,5-c]quinazolin-5-one | ...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]glycine from glycine site on the NMDA receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1(RAT)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50002699(7,8-Difluoro-5H-[1,2,4]triazolo[4,3-a]quinoxalin-4...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]glycine from glycine site on the NMDA receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1(RAT)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50002708(7-Nitro-5H-1,2,3,5,9b-pentaaza-cyclopenta[a]naphth...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]glycine from glycine site on the NMDA receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1(RAT)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50002695(7,8-Dichloro-5H-1,2,3,5,9b-pentaaza-cyclopenta[a]n...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]glycine from glycine site on the NMDA receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1(RAT)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50002703(7,8-Dichloro-1-methyl-5H-[1,2,4]triazolo[4,3-a]qui...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]glycine from glycine site on the NMDA receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1(RAT)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50002702(7,8-Dichloro-1-trifluoromethyl-5H-[1,2,4]triazolo[...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]glycine from glycine site on the NMDA receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1(RAT)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50002705(8-Chloro-6H-pyrazolo[1,5-c]quinazolin-5-one | CHEM...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]glycine from glycine site on the NMDA receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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