TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)
Curated by ChEMBL
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)
Curated by ChEMBL
Affinity DataKi: 0.0300nMAssay Description:Displacement of [3H]-CGP-12177 from human beta2-adrenergic receptor expressed in CHO cells after 60 mins by radioligand competition binding assayMore data for this Ligand-Target Pair
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)
Curated by ChEMBL
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)
Curated by ChEMBL
Affinity DataKi: 0.0300nMAssay Description:Displacement of [3H]-CGP-12177 from human beta2-adrenergic receptor expressed in CHO cells after 60 mins by radioligand competition binding assayMore data for this Ligand-Target Pair
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)
Curated by ChEMBL
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)
Curated by ChEMBL
Affinity DataKi: 0.0340nMAssay Description:Displacement of [3H]CGP12177 from human beta2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetBeta-1 adrenergic receptor(Mus musculus)
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)
Curated by ChEMBL
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)
Curated by ChEMBL
Affinity DataKi: 0.0900nMAssay Description:Displacement of [3H]-CGP-12177 from murine beta1-adrenergic receptor expressed in HEK293T cells after 60 mins by radioligand competition binding assa...More data for this Ligand-Target Pair
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)
Curated by ChEMBL
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)
Curated by ChEMBL
Affinity DataKi: 0.180nMAssay Description:Displacement of [3H]CGP12177 from human beta2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetBeta-1 adrenergic receptor(Mus musculus)
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)
Curated by ChEMBL
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)
Curated by ChEMBL
Affinity DataKi: 0.210nMAssay Description:Displacement of [3H]-CGP-12177 from murine beta1-adrenergic receptor expressed in HEK293T cells after 60 mins by radioligand competition binding assa...More data for this Ligand-Target Pair
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)
Curated by ChEMBL
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)
Curated by ChEMBL
Affinity DataKi: 0.25nMAssay Description:Displacement of [3H]-CGP-12177 from human beta2-adrenergic receptor expressed in CHO cells after 60 mins by radioligand competition binding assayMore data for this Ligand-Target Pair
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)
Curated by ChEMBL
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)
Curated by ChEMBL
Affinity DataKi: 0.25nMAssay Description:Displacement of [3H]CGP12177 from human beta2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)
Curated by ChEMBL
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)
Curated by ChEMBL
Affinity DataKi: 0.480nMAssay Description:Displacement of [3H]CGP12177 from human beta2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)
Curated by ChEMBL
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)
Curated by ChEMBL
Affinity DataKi: 0.880nMAssay Description:Displacement of [3H]-CGP-12177 from human beta2-adrenergic receptor expressed in CHO cells after 60 mins by radioligand competition binding assayMore data for this Ligand-Target Pair
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)
Curated by ChEMBL
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)
Curated by ChEMBL
Affinity DataKi: 0.880nMAssay Description:Displacement of [3H]CGP12177 from human beta2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)
Curated by ChEMBL
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)
Curated by ChEMBL
Affinity DataKi: 2.80nMAssay Description:Displacement of [3H]CGP12177 from human beta2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)
Curated by ChEMBL
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)
Curated by ChEMBL
Affinity DataKi: 3.30nMAssay Description:Displacement of [3H]-CGP-12177 from human beta2-adrenergic receptor expressed in CHO cells after 60 mins by radioligand competition binding assayMore data for this Ligand-Target Pair
TargetBeta-1 adrenergic receptor(Mus musculus)
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)
Curated by ChEMBL
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)
Curated by ChEMBL
Affinity DataKi: 3.40nMAssay Description:Displacement of [3H]-CGP-12177 from murine beta1-adrenergic receptor expressed in HEK293T cells after 60 mins by radioligand competition binding assa...More data for this Ligand-Target Pair
Affinity DataKi: 3.5nMAssay Description:Displacement of [3H]spiperone from human D3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 4.5nMAssay Description:Displacement of [3H]spiperone from human D4.4 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetBeta-1 adrenergic receptor(Mus musculus)
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)
Curated by ChEMBL
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)
Curated by ChEMBL
Affinity DataKi: 5.10nMAssay Description:Displacement of [3H]CGP12177 from mouse beta1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)
Curated by ChEMBL
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)
Curated by ChEMBL
Affinity DataKi: 5.40nMAssay Description:Displacement of [3H]-CGP-12177 from human beta2-adrenergic receptor expressed in CHO cells after 60 mins by radioligand competition binding assayMore data for this Ligand-Target Pair
TargetBeta-1 adrenergic receptor(Mus musculus)
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)
Curated by ChEMBL
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)
Curated by ChEMBL
Affinity DataKi: 5.80nMAssay Description:Displacement of [3H]CGP12177 from mouse beta1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)
Curated by ChEMBL
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)
Curated by ChEMBL
Affinity DataKi: 6.30nMAssay Description:Displacement of [3H]CGP12177 from human beta2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetBeta-1 adrenergic receptor(Mus musculus)
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)
Curated by ChEMBL
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)
Curated by ChEMBL
Affinity DataKi: 6.5nMAssay Description:Displacement of [3H]-CGP-12177 from murine beta1-adrenergic receptor expressed in HEK293T cells after 60 mins by radioligand competition binding assa...More data for this Ligand-Target Pair
TargetBeta-1 adrenergic receptor(Mus musculus)
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)
Curated by ChEMBL
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)
Curated by ChEMBL
Affinity DataKi: 6.60nMAssay Description:Displacement of [3H]-CGP-12177 from murine beta1-adrenergic receptor expressed in HEK293T cells after 60 mins by radioligand competition binding assa...More data for this Ligand-Target Pair
Affinity DataKi: 7.10nMAssay Description:Displacement of [3H]spiperone from human D2S receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)
Curated by ChEMBL
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)
Curated by ChEMBL
Affinity DataKi: 7.20nMAssay Description:Displacement of [3H]-CGP-12177 from human beta2-adrenergic receptor expressed in CHO cells after 60 mins by radioligand competition binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 8.5nMAssay Description:Displacement of [3H]spiperone from human D4.4 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 12nMAssay Description:Displacement of [3H]spiperone from human D3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetBeta-1 adrenergic receptor(Mus musculus)
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)
Curated by ChEMBL
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)
Curated by ChEMBL
Affinity DataKi: 12nMAssay Description:Displacement of [3H]-CGP-12177 from murine beta1-adrenergic receptor expressed in HEK293T cells after 60 mins by radioligand competition binding assa...More data for this Ligand-Target Pair
Affinity DataKi: 12nMAssay Description:Displacement of [3H]spiperone from human D2L receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)
Curated by ChEMBL
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)
Curated by ChEMBL
Affinity DataKi: 12nMAssay Description:Displacement of [3H]-CGP-12177 from human beta2-adrenergic receptor expressed in CHO cells after 60 mins by radioligand competition binding assayMore data for this Ligand-Target Pair
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)
Curated by ChEMBL
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)
Curated by ChEMBL
Affinity DataKi: 13nMAssay Description:Displacement of [3H]CGP12177 from human beta2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetBeta-1 adrenergic receptor(Mus musculus)
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)
Curated by ChEMBL
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)
Curated by ChEMBL
Affinity DataKi: 14nMAssay Description:Displacement of [3H]-CGP-12177 from murine beta1-adrenergic receptor expressed in HEK293T cells after 60 mins by radioligand competition binding assa...More data for this Ligand-Target Pair
Affinity DataKi: 15nMAssay Description:Displacement of [3H]spiperone from human D3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 17nMAssay Description:Displacement of [3H]spiperone from human D2S receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 18nMAssay Description:Displacement of [3H]spiperone from human D3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)
Curated by ChEMBL
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)
Curated by ChEMBL
Affinity DataKi: 18nMAssay Description:Displacement of [3H]CGP12177 from human beta2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)
Curated by ChEMBL
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)
Curated by ChEMBL
Affinity DataKi: 18nMAssay Description:Displacement of [3H]-CGP-12177 from human beta2-adrenergic receptor expressed in CHO cells after 60 mins by radioligand competition binding assayMore data for this Ligand-Target Pair
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)
Curated by ChEMBL
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)
Curated by ChEMBL
Affinity DataKi: 21nMAssay Description:Displacement of [3H]-CGP-12177 from human beta2-adrenergic receptor expressed in CHO cells after 60 mins by radioligand competition binding assayMore data for this Ligand-Target Pair
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)
Curated by ChEMBL
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)
Curated by ChEMBL
Affinity DataKi: 23nMAssay Description:Displacement of [3H]CGP12177 from human beta2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetBeta-1 adrenergic receptor(Mus musculus)
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)
Curated by ChEMBL
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)
Curated by ChEMBL
Affinity DataKi: 24nMAssay Description:Displacement of [3H]-CGP-12177 from murine beta1-adrenergic receptor expressed in HEK293T cells after 60 mins by radioligand competition binding assa...More data for this Ligand-Target Pair
Affinity DataKi: 25nMAssay Description:Displacement of [3H]spiperone from human D3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)
Curated by ChEMBL
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)
Curated by ChEMBL
Affinity DataKi: 26nMAssay Description:Displacement of [3H]-CGP-12177 from human beta2-adrenergic receptor expressed in CHO cells after 60 mins by radioligand competition binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 26nMAssay Description:Displacement of [3H]spiperone from human D2S receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)
Curated by ChEMBL
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)
Curated by ChEMBL
Affinity DataKi: 26nMAssay Description:Displacement of [3H]CGP12177 from human beta2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)
Curated by ChEMBL
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)
Curated by ChEMBL
Affinity DataKi: 33nMAssay Description:Displacement of [3H]CGP12177 from human beta2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 38nMAssay Description:Displacement of [3H]spiperone from human D4.4 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 40nMAssay Description:Displacement of [3H]spiperone from human D2S receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)
Curated by ChEMBL
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)
Curated by ChEMBL
Affinity DataKi: 46nMAssay Description:Displacement of [3H]CGP12177 from human beta2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)
Curated by ChEMBL
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)
Curated by ChEMBL
Affinity DataKi: 46nMAssay Description:Displacement of [3H]-CGP-12177 from human beta2-adrenergic receptor expressed in CHO cells after 60 mins by radioligand competition binding assayMore data for this Ligand-Target Pair
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)
Curated by ChEMBL
Friedrich-Alexander University Erlangen-N£Rnberg (Fau)
Curated by ChEMBL
Affinity DataKi: 47nMAssay Description:Displacement of [3H]CGP12177 from human beta2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 48nMAssay Description:Displacement of [3H]spiperone from human D2S receptor expressed in CHO cellsMore data for this Ligand-Target Pair