Compile Data Set for Download or QSAR
maximum 50k data
Found 608 with Last Name = 'steinmetzer' and Initial = 'p'
TargetCoagulation factor X(Homo sapiens (Human))
Curacyte Discovery

Curated by ChEMBL
LigandPNGBDBM50211565((R)-N-[(S)-1-(2-aminomethyl-5-chloro-benzylcarbamo...)
Affinity DataKi:  0.0330nMAssay Description:Inhibition of factor 10aMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Curacyte Discovery

Curated by ChEMBL
LigandPNGBDBM50211578((S)-1-[(R)-4-(1-oxy-pyridin-2-yl)-2-phenylmethanes...)
Affinity DataKi:  0.0490nMAssay Description:Inhibition of factor 10aMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Curacyte Discovery

Curated by ChEMBL
LigandPNGBDBM50211567((R)-N-[(S)-1-(2-aminomethyl-5-chloro-benzylcarbamo...)
Affinity DataKi:  0.0590nMAssay Description:Inhibition of factor 10aMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSuppressor of tumorigenicity 14 protein(Homo sapiens (Human))
Curacyte Discovery

Curated by ChEMBL
LigandPNGBDBM50253952(3-{(S)-3-[4-(2-Amino-ethyl)-piperidin-1-yl]-2-[3-(...)
Affinity DataKi:  0.0800nMAssay Description:Inhibition of matriptase (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Curacyte Discovery

Curated by ChEMBL
LigandPNGBDBM50211585(CHEMBL389960 | [(R)-1-[(S)-2-(2-aminomethyl-5-chlo...)
Affinity DataKi:  0.0800nMAssay Description:Inhibition of factor 10aMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Curacyte Discovery

Curated by ChEMBL
LigandPNGBDBM50211571((R)-N-((S)-1-(2-(aminomethyl)-5-chlorobenzylamino)...)
Affinity DataKi:  0.0840nMAssay Description:Inhibition of factor 10aMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Curacyte Discovery

Curated by ChEMBL
LigandPNGBDBM50211564((R)-N-[(5-chloro-2-ethyl-benzylcarbamoyl)-methyl]-...)
Affinity DataKi:  0.0950nMAssay Description:Inhibition of factor 10aMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Curacyte Discovery

Curated by ChEMBL
LigandPNGBDBM50211563((S)-4-(2-aminomethyl-5-chloro-benzylcarbamoyl)-4-{...)
Affinity DataKi:  0.240nMAssay Description:Inhibition of factor 10aMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Curacyte Discovery

Curated by ChEMBL
LigandPNGBDBM50211570(CHEMBL228984 | N-((S)-1-(2-(aminomethyl)-5-chlorob...)
Affinity DataKi:  0.25nMAssay Description:Inhibition of factor 10aMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Curacyte Discovery

Curated by ChEMBL
LigandPNGBDBM50211582((R)-N-[(4-carbamimidoyl-benzylcarbamoyl)-methyl]-4...)
Affinity DataKi:  0.320nMAssay Description:Inhibition of factor 10aMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Curacyte Discovery

Curated by ChEMBL
LigandPNGBDBM50211552((4-{[1-{[(2-aminomethyl-5-chloro-benzylcarbamoyl)-...)
Affinity DataKi:  0.350nMAssay Description:Inhibition of factor 10aMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Curacyte Discovery

Curated by ChEMBL
LigandPNGBDBM50211572((4-{[1-{[(2-aminomethyl-5-chloro-benzylcarbamoyl)-...)
Affinity DataKi:  0.360nMAssay Description:Inhibition of factor 10aMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Curacyte Discovery

Curated by ChEMBL
LigandPNGBDBM50211586((s)-4-(2-aminomethyl-5-chloro-benzylcarbamoyl)-4-[...)
Affinity DataKi:  0.520nMAssay Description:Inhibition of factor 10aMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Curacyte Discovery

Curated by ChEMBL
LigandPNGBDBM50211578((S)-1-[(R)-4-(1-oxy-pyridin-2-yl)-2-phenylmethanes...)
Affinity DataKi:  0.560nMAssay Description:Inhibition of thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Curacyte Discovery

Curated by ChEMBL
LigandPNGBDBM50211587(CHEMBL427464 | N-[(R)-1-[(S)-2-(2-aminomethyl-5-ch...)
Affinity DataKi:  0.630nMAssay Description:Inhibition of factor 10aMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Curacyte Discovery

Curated by ChEMBL
LigandPNGBDBM50211584(CHEMBL231393 | [1-{[(2-aminomethyl-5-chloro-benzyl...)
Affinity DataKi:  0.760nMAssay Description:Inhibition of factor 10aMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Curacyte Discovery

Curated by ChEMBL
LigandPNGBDBM50211551(CHEMBL228285 | N-[1-[(S)-2-(2-aminomethyl-5-chloro...)
Affinity DataKi:  0.870nMAssay Description:Inhibition of factor 10aMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Curacyte Discovery

Curated by ChEMBL
LigandPNGBDBM50211576(CHEMBL228341 | [(R)-1-[(S)-2-(2-aminomethyl-5-chlo...)
Affinity DataKi:  0.920nMAssay Description:Inhibition of factor 10aMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Curacyte Discovery

Curated by ChEMBL
LigandPNGBDBM50211556(CHEMBL390402 | [(R)-1-[(S)-2-(2-aminomethyl-5-chlo...)
Affinity DataKi:  0.940nMAssay Description:Inhibition of factor 10aMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSuppressor of tumorigenicity 14 protein(Homo sapiens (Human))
Curacyte Discovery

Curated by ChEMBL
LigandPNGBDBM104908(CHEMBL468270 | US8569313, Inhibitor 16)
Affinity DataKi:  1nMAssay Description:Inhibition of matriptase (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Curacyte Discovery

Curated by ChEMBL
LigandPNGBDBM50211577(CHEMBL229036 | [(R)-1-[(S)-2-(2-aminomethyl-5-chlo...)
Affinity DataKi:  1nMAssay Description:Inhibition of factor 10aMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSuppressor of tumorigenicity 14 protein(Homo sapiens (Human))
Curacyte Discovery

Curated by ChEMBL
LigandPNGBDBM23921(3-amidinophenylalanine deriv., 63 | 3-amino-N-(3-{...)
Affinity DataKi:  1.5nMAssay Description:The measurements were carried out on a microplate reader. Two concentrations of the substrate and five concentrations of the inhibitor were used. Af...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Curacyte Discovery

Curated by ChEMBL
LigandPNGBDBM50211581(2-((R)-1-((S)-2-((2-(aminomethyl)-5-chlorobenzyl)c...)
Affinity DataKi:  1.5nMAssay Description:Inhibition of factor 10aMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Curacyte Discovery

Curated by ChEMBL
LigandPNGBDBM50211580(CHEMBL231494 | [1-{[(2-aminomethyl-5-chloro-benzyl...)
Affinity DataKi:  1.60nMAssay Description:Inhibition of factor 10aMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSuppressor of tumorigenicity 14 protein(Homo sapiens (Human))
Curacyte Discovery

Curated by ChEMBL
LigandPNGBDBM50254410(3-{(S)-3-[4-(2-Amino-ethyl)-piperidin-1-yl]-2-[3-(...)
Affinity DataKi:  1.60nMAssay Description:Inhibition of matriptase (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Curacyte Discovery

Curated by ChEMBL
LigandPNGBDBM50211566(CHEMBL228340 | [(R)-1-[(S)-2-(2-aminomethyl-5-chlo...)
Affinity DataKi:  1.70nMAssay Description:Inhibition of factor 10aMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSuppressor of tumorigenicity 14 protein(Homo sapiens (Human))
Curacyte Discovery

Curated by ChEMBL
LigandPNGBDBM23916(3-amidinophenylalanine deriv., 12 | 3-amino-N-(3-{...)
Affinity DataKi:  1.80nMAssay Description:Inhibition of matriptase (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSuppressor of tumorigenicity 14 protein(Homo sapiens (Human))
Curacyte Discovery

Curated by ChEMBL
LigandPNGBDBM23916(3-amidinophenylalanine deriv., 12 | 3-amino-N-(3-{...)
Affinity DataKi:  1.80nMAssay Description:The measurements were carried out on a microplate reader. Two concentrations of the substrate and five concentrations of the inhibitor were used. Af...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSuppressor of tumorigenicity 14 protein(Homo sapiens (Human))
Curacyte Discovery

Curated by ChEMBL
LigandPNGBDBM50254368((+/-)-3-[3-[4-(2-Amino-ethyl)-piperidin-1-yl]-2-(4...)
Affinity DataKi:  2.5nMAssay Description:Inhibition of matriptase (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Curacyte Discovery

Curated by ChEMBL
LigandPNGBDBM50211555(CHEMBL397679 | N-[(2,5-dichloro-benzylcarbamoyl)-m...)
Affinity DataKi:  2.55nMAssay Description:Inhibition of factor 10aMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Curacyte Discovery

Curated by ChEMBL
LigandPNGBDBM50211573(CHEMBL390403 | ethyl 2-((R)-1-((S)-2-((2-(aminomet...)
Affinity DataKi:  2.90nMAssay Description:Inhibition of factor 10aMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSuppressor of tumorigenicity 14 protein(Homo sapiens (Human))
Curacyte Discovery

Curated by ChEMBL
LigandPNGBDBM50254219(Azetidine-3-carboxylic acid {3-[(S)-2-[4-(2-amino-...)
Affinity DataKi:  3nMAssay Description:Inhibition of matriptase (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Curacyte Discovery

Curated by ChEMBL
LigandPNGBDBM50211562(2-((R)-1-((S)-2-((2-(aminomethyl)-5-chlorobenzyl)c...)
Affinity DataKi:  3.20nMAssay Description:Inhibition of thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Curacyte Discovery

Curated by ChEMBL
LigandPNGBDBM50211575((R)-N-[(3-chloro-benzylcarbamoyl)-methyl]-4-(1-oxy...)
Affinity DataKi:  3.30nMAssay Description:Inhibition of factor 10aMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Curacyte Discovery

Curated by ChEMBL
LigandPNGBDBM50211560(CHEMBL231292 | N-[(2-aminomethyl-5-chloro-benzylca...)
Affinity DataKi:  3.40nMAssay Description:Inhibition of factor 10aMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Curacyte Discovery

Curated by ChEMBL
LigandPNGBDBM50211581(2-((R)-1-((S)-2-((2-(aminomethyl)-5-chlorobenzyl)c...)
Affinity DataKi:  3.5nMAssay Description:Inhibition of thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Curacyte Discovery

Curated by ChEMBL
LigandPNGBDBM50211559(CHEMBL230360 | ethyl 2-((R)-1-((S)-2-((2-(aminomet...)
Affinity DataKi:  3.60nMAssay Description:Inhibition of thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSuppressor of tumorigenicity 14 protein(Homo sapiens (Human))
Curacyte Discovery

Curated by ChEMBL
LigandPNGBDBM23917(3-amidinophenylalanine deriv., 59 | 3-amino-N-(3-{...)
Affinity DataKi:  3.80nMAssay Description:Inhibition of matriptase (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Curacyte Discovery

Curated by ChEMBL
LigandPNGBDBM50211573(CHEMBL390403 | ethyl 2-((R)-1-((S)-2-((2-(aminomet...)
Affinity DataKi:  3.80nMAssay Description:Inhibition of thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSuppressor of tumorigenicity 14 protein(Homo sapiens (Human))
Curacyte Discovery

Curated by ChEMBL
LigandPNGBDBM23918(3-amidinophenylalanine deriv., 60 | 4-amino-N-(3-{...)
Affinity DataKi:  3.90nMAssay Description:The measurements were carried out on a microplate reader. Two concentrations of the substrate and five concentrations of the inhibitor were used. Af...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSuppressor of tumorigenicity 14 protein(Homo sapiens (Human))
Curacyte Discovery

Curated by ChEMBL
LigandPNGBDBM23915(3-amidinophenylalanine deriv., 58 | 3-carbamimidam...)
Affinity DataKi:  4.20nMAssay Description:The measurements were carried out on a microplate reader. Two concentrations of the substrate and five concentrations of the inhibitor were used. Af...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Curacyte Discovery

Curated by ChEMBL
LigandPNGBDBM50211566(CHEMBL228340 | [(R)-1-[(S)-2-(2-aminomethyl-5-chlo...)
Affinity DataKi:  4.90nMAssay Description:Inhibition of thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Curacyte Discovery

Curated by ChEMBL
LigandPNGBDBM50211557(CHEMBL231595 | N-[1-{[(2-aminomethyl-5-chloro-benz...)
Affinity DataKi:  4.90nMAssay Description:Inhibition of factor 10aMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Curacyte Discovery

Curated by ChEMBL
LigandPNGBDBM50211568(CHEMBL395773 | N-[1-{[(2-aminomethyl-5-chloro-benz...)
Affinity DataKi:  4.90nMAssay Description:Inhibition of factor 10aMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSuppressor of tumorigenicity 14 protein(Homo sapiens (Human))
Curacyte Discovery

Curated by ChEMBL
LigandPNGBDBM23920(3-amidinophenylalanine deriv., 62 | 3-amino-N-(3-{...)
Affinity DataKi:  5nMAssay Description:The measurements were carried out on a microplate reader. Two concentrations of the substrate and five concentrations of the inhibitor were used. Af...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSuppressor of tumorigenicity 14 protein(Homo sapiens (Human))
Curacyte Discovery

Curated by ChEMBL
LigandPNGBDBM50254367((+/-)-3-[3-[4-(2-Amino-ethyl)-piperidin-1-yl]-2-(3...)
Affinity DataKi:  5.40nMAssay Description:Inhibition of matriptase (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSuppressor of tumorigenicity 14 protein(Homo sapiens (Human))
Curacyte Discovery

Curated by ChEMBL
LigandPNGBDBM50254365((+/-)-3-[3-[4-(2-Amino-ethyl)-piperidin-1-yl]-2-(4...)
Affinity DataKi:  6nMAssay Description:Inhibition of matriptase (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSuppressor of tumorigenicity 14 protein(Homo sapiens (Human))
Curacyte Discovery

Curated by ChEMBL
LigandPNGBDBM50257511((S)-methyl 4-(1-(2-(3-(3-aminopropanamido)phenylsu...)
Affinity DataKi:  6.10nMAssay Description:Inhibition of matriptase (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSuppressor of tumorigenicity 14 protein(Homo sapiens (Human))
Curacyte Discovery

Curated by ChEMBL
LigandPNGBDBM50257512((S)-4-(1-(2-(3-(3-aminopropanamido)phenylsulfonami...)
Affinity DataKi:  6.30nMAssay Description:Inhibition of matriptase (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSuppressor of tumorigenicity 14 protein(Homo sapiens (Human))
Curacyte Discovery

Curated by ChEMBL
LigandPNGBDBM23917(3-amidinophenylalanine deriv., 59 | 3-amino-N-(3-{...)
Affinity DataKi:  6.60nMAssay Description:The measurements were carried out on a microplate reader. Two concentrations of the substrate and five concentrations of the inhibitor were used. Af...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Displayed 1 to 50 (of 608 total ) | Next | Last >>
Jump to: