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Found 48 with Last Name = 'takimizu' and Initial = 'h'
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Homo sapiens (Human))
Minase Research Institute

Curated by ChEMBL
LigandPNGBDBM50111944((R)-4-[(R)-2-Cyclohexylmethylsulfanyl-1-(4-phenoxy...)
Affinity DataIC50:  120nMAssay Description:In vitro inhibition of N-type calcium channels in IMR-32 cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Homo sapiens (Human))
Minase Research Institute

Curated by ChEMBL
LigandPNGBDBM50111936((R)-3-(2-Methoxy-acetyl)-thiazolidine-4-carboxylic...)
Affinity DataIC50:  120nMAssay Description:In vitro inhibition of N-type calcium channels in IMR-32 cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Homo sapiens (Human))
Minase Research Institute

Curated by ChEMBL
LigandPNGBDBM50111940((R)-4-[(R)-2-Cyclohexylmethylsulfanyl-1-(4-phenoxy...)
Affinity DataIC50:  140nMAssay Description:In vitro inhibition of N-type calcium channel influx in IMR-32 human neuroblastoma cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Homo sapiens (Human))
Minase Research Institute

Curated by ChEMBL
LigandPNGBDBM50111940((R)-4-[(R)-2-Cyclohexylmethylsulfanyl-1-(4-phenoxy...)
Affinity DataIC50:  140nMAssay Description:In vitro inhibition of N-type calcium channels in IMR-32 cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Homo sapiens (Human))
Minase Research Institute

Curated by ChEMBL
LigandPNGBDBM50116658((R)-4-[(R)-2-Cyclohexylmethylsulfanyl-1-(1-phenyl-...)
Affinity DataIC50:  150nMAssay Description:In vitro inhibition of N-type calcium channel influx in IMR-32 human neuroblastoma cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Homo sapiens (Human))
Minase Research Institute

Curated by ChEMBL
LigandPNGBDBM50111945((R)-3-(2-Methoxy-ethyl)-thiazolidine-4-carboxylic ...)
Affinity DataIC50:  200nMAssay Description:In vitro inhibition of N-type calcium channels in IMR-32 cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Homo sapiens (Human))
Minase Research Institute

Curated by ChEMBL
LigandPNGBDBM50111935((R)-Thiazolidine-4-carboxylic acid [(R)-2-cyclohex...)
Affinity DataIC50:  290nMAssay Description:In vitro inhibition of N-type calcium channels in IMR-32 cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Homo sapiens (Human))
Minase Research Institute

Curated by ChEMBL
LigandPNGBDBM50111949((R)-4-[(R)-2-Cyclohexylmethylsulfanyl-1-(4-phenoxy...)
Affinity DataIC50:  330nMAssay Description:In vitro inhibition of N-type calcium channels in IMR-32 cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Homo sapiens (Human))
Minase Research Institute

Curated by ChEMBL
LigandPNGBDBM50116653((R)-4-[(R)-1-(1-Benzyl-piperidin-4-ylcarbamoyl)-2-...)
Affinity DataIC50:  330nMAssay Description:In vitro inhibition of N-type calcium channel influx in IMR-32 human neuroblastoma cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Homo sapiens (Human))
Minase Research Institute

Curated by ChEMBL
LigandPNGBDBM50111938((R)-3-(2-Hydroxy-ethyl)-thiazolidine-4-carboxylic ...)
Affinity DataIC50:  350nMAssay Description:In vitro inhibition of N-type calcium channels in IMR-32 cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Homo sapiens (Human))
Minase Research Institute

Curated by ChEMBL
LigandPNGBDBM50111948((R)-4-[(R)-2-Cyclohexylmethylsulfanyl-1-(4-phenoxy...)
Affinity DataIC50:  360nMAssay Description:In vitro inhibition of N-type calcium channels in IMR-32 cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Homo sapiens (Human))
Minase Research Institute

Curated by ChEMBL
LigandPNGBDBM50116657((R)-4-[(R)-2-(4-Benzyl-piperazin-1-yl)-1-cyclohexy...)
Affinity DataIC50:  370nMAssay Description:In vitro inhibition of N-type calcium channel influx in IMR-32 human neuroblastoma cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Homo sapiens (Human))
Minase Research Institute

Curated by ChEMBL
LigandPNGBDBM50116652((R)-4-[(R)-1-(2-Benzylamino-ethylcarbamoyl)-2-cycl...)
Affinity DataIC50:  380nMAssay Description:In vitro inhibition of N-type calcium channel influx in IMR-32 human neuroblastoma cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Homo sapiens (Human))
Minase Research Institute

Curated by ChEMBL
LigandPNGBDBM50111950((R)-4-[(R)-2-Cyclohexylmethylsulfanyl-1-(4-methoxy...)
Affinity DataIC50:  390nMAssay Description:In vitro inhibition of N-type calcium channels in IMR-32 cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Homo sapiens (Human))
Minase Research Institute

Curated by ChEMBL
LigandPNGBDBM50116655((R)-4-[(R)-1-Cyclohexylmethylsulfanylmethyl-2-oxo-...)
Affinity DataIC50:  390nMAssay Description:In vitro inhibition of N-type calcium channel influx in IMR-32 human neuroblastoma cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Homo sapiens (Human))
Minase Research Institute

Curated by ChEMBL
LigandPNGBDBM50111939((R)-4-[(R)-1-(4-Benzyloxy-benzylcarbamoyl)-2-cyclo...)
Affinity DataIC50:  500nMAssay Description:In vitro inhibition of N-type calcium channels in IMR-32 cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Homo sapiens (Human))
Minase Research Institute

Curated by ChEMBL
LigandPNGBDBM50116654((R)-4-[(R)-2-(4-Benzylamino-piperidin-1-yl)-1-cycl...)
Affinity DataIC50:  500nMAssay Description:In vitro inhibition of N-type calcium channel influx in IMR-32 human neuroblastoma cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Homo sapiens (Human))
Minase Research Institute

Curated by ChEMBL
LigandPNGBDBM50111947((R)-4-[(R)-2-Cyclohexylmethylsulfanyl-1-(4-nitro-b...)
Affinity DataIC50:  600nMAssay Description:In vitro inhibition of N-type calcium channels in IMR-32 cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Homo sapiens (Human))
Minase Research Institute

Curated by ChEMBL
LigandPNGBDBM50111933((R)-4-[(R)-2-Cyclohexylmethylsulfanyl-1-(4-dimethy...)
Affinity DataIC50:  610nMAssay Description:In vitro inhibition of N-type calcium channels in IMR-32 cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Homo sapiens (Human))
Minase Research Institute

Curated by ChEMBL
LigandPNGBDBM50451199(CHEMBL65110)
Affinity DataIC50:  610nMAssay Description:In vitro inhibition against N-type calcium influx in IMR-32 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Homo sapiens (Human))
Minase Research Institute

Curated by ChEMBL
LigandPNGBDBM50111946((R)-2-tert-Butoxycarbonylamino-3-cyclohexylmethyls...)
Affinity DataIC50:  610nMAssay Description:In vitro inhibition of N-type calcium channels in IMR-32 cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Homo sapiens (Human))
Minase Research Institute

Curated by ChEMBL
LigandPNGBDBM50102915(CHEMBL431324 | [(R)-2-Cyclopentylmethylsulfanyl-1-...)
Affinity DataIC50:  630nMAssay Description:In vitro inhibition against N-type calcium influx in IMR-32 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Homo sapiens (Human))
Minase Research Institute

Curated by ChEMBL
LigandPNGBDBM50102915(CHEMBL431324 | [(R)-2-Cyclopentylmethylsulfanyl-1-...)
Affinity DataIC50:  640nMAssay Description:In vitro inhibition of N-type calcium channels in IMR-32 cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Homo sapiens (Human))
Minase Research Institute

Curated by ChEMBL
LigandPNGBDBM50116656((R)-4-[(R)-1-Cyclohexylmethylsulfanylmethyl-2-oxo-...)
Affinity DataIC50:  660nMAssay Description:In vitro inhibition of N-type calcium channel influx in IMR-32 human neuroblastoma cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Homo sapiens (Human))
Minase Research Institute

Curated by ChEMBL
LigandPNGBDBM50111937((R)-3-Cyclohexylmethylsulfanyl-2-isobutoxycarbonyl...)
Affinity DataIC50:  720nMAssay Description:In vitro inhibition of N-type calcium channels in IMR-32 cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Homo sapiens (Human))
Minase Research Institute

Curated by ChEMBL
LigandPNGBDBM50111941((S)-2-[(R)-2-Cyclohexylmethylsulfanyl-1-(4-methoxy...)
Affinity DataIC50:  880nMAssay Description:In vitro inhibition of N-type calcium channels in IMR-32 cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Homo sapiens (Human))
Minase Research Institute

Curated by ChEMBL
LigandPNGBDBM50111953((R)-3-Cyclohexylmethylsulfanyl-2-(cyclopentanecarb...)
Affinity DataIC50:  920nMAssay Description:In vitro inhibition of N-type calcium channels in IMR-32 cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Homo sapiens (Human))
Minase Research Institute

Curated by ChEMBL
LigandPNGBDBM50451201(CHEMBL65360)
Affinity DataIC50:  950nMAssay Description:In vitro inhibition against N-type calcium influx in IMR-32 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Homo sapiens (Human))
Minase Research Institute

Curated by ChEMBL
LigandPNGBDBM50451196(CHEMBL305303)
Affinity DataIC50:  1.20E+3nMAssay Description:In vitro inhibition against N-type calcium influx in IMR-32 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Homo sapiens (Human))
Minase Research Institute

Curated by ChEMBL
LigandPNGBDBM50111943((R)-3-Cyclohexylmethylsulfanyl-2-(3-methyl-butyryl...)
Affinity DataIC50:  1.20E+3nMAssay Description:In vitro inhibition of N-type calcium channels in IMR-32 cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Homo sapiens (Human))
Minase Research Institute

Curated by ChEMBL
LigandPNGBDBM50111954((R)-2-(Cyclohexanecarbonyl-amino)-3-cyclohexylmeth...)
Affinity DataIC50:  1.30E+3nMAssay Description:In vitro inhibition of N-type calcium channels in IMR-32 cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Homo sapiens (Human))
Minase Research Institute

Curated by ChEMBL
LigandPNGBDBM50451204(CHEMBL65402)
Affinity DataIC50:  1.60E+3nMAssay Description:In vitro inhibition against N-type calcium influx in IMR-32 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Homo sapiens (Human))
Minase Research Institute

Curated by ChEMBL
LigandPNGBDBM50111951((R)-4-[(R)-2-Cyclohexylmethylsulfanyl-1-(4-hydroxy...)
Affinity DataIC50:  1.80E+3nMAssay Description:In vitro inhibition of N-type calcium channels in IMR-32 cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Homo sapiens (Human))
Minase Research Institute

Curated by ChEMBL
LigandPNGBDBM50451207(CHEMBL65467)
Affinity DataIC50:  1.80E+3nMAssay Description:In vitro inhibition against N-type calcium influx in IMR-32 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Homo sapiens (Human))
Minase Research Institute

Curated by ChEMBL
LigandPNGBDBM50111952((R)-3-Cyclohexylmethylsulfanyl-2-[(thiazole-4-carb...)
Affinity DataIC50:  1.90E+3nMAssay Description:In vitro inhibition of N-type calcium channels in IMR-32 cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Homo sapiens (Human))
Minase Research Institute

Curated by ChEMBL
LigandPNGBDBM50451208(CHEMBL2114022)
Affinity DataIC50:  2.00E+3nMAssay Description:In vitro inhibition against N-type calcium influx in IMR-32 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Homo sapiens (Human))
Minase Research Institute

Curated by ChEMBL
LigandPNGBDBM50451198(CHEMBL66138)
Affinity DataIC50:  2.30E+3nMAssay Description:In vitro inhibition against N-type calcium influx in IMR-32 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Homo sapiens (Human))
Minase Research Institute

Curated by ChEMBL
LigandPNGBDBM50451209(CHEMBL65117)
Affinity DataIC50:  2.60E+3nMAssay Description:In vitro inhibition against N-type calcium influx in IMR-32 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Homo sapiens (Human))
Minase Research Institute

Curated by ChEMBL
LigandPNGBDBM50111942((R)-3-Cyclohexylmethylsulfanyl-2-[((R)-thiazolidin...)
Affinity DataIC50:  2.70E+3nMAssay Description:In vitro inhibition of N-type calcium channels in IMR-32 cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Homo sapiens (Human))
Minase Research Institute

Curated by ChEMBL
LigandPNGBDBM50451205(CHEMBL293426)
Affinity DataIC50:  3.30E+3nMAssay Description:In vitro inhibition against N-type calcium influx in IMR-32 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Homo sapiens (Human))
Minase Research Institute

Curated by ChEMBL
LigandPNGBDBM50451202(CHEMBL302628)
Affinity DataIC50:  3.40E+3nMAssay Description:In vitro inhibition against N-type calcium influx in IMR-32 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Homo sapiens (Human))
Minase Research Institute

Curated by ChEMBL
LigandPNGBDBM50451195(CHEMBL62518)
Affinity DataIC50:  3.40E+3nMAssay Description:In vitro inhibition against N-type calcium influx in IMR-32 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Homo sapiens (Human))
Minase Research Institute

Curated by ChEMBL
LigandPNGBDBM50451210(CHEMBL294369)
Affinity DataIC50:  3.80E+3nMAssay Description:In vitro inhibition against N-type calcium influx in IMR-32 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Homo sapiens (Human))
Minase Research Institute

Curated by ChEMBL
LigandPNGBDBM50451206(CHEMBL305133)
Affinity DataIC50:  4.00E+3nMAssay Description:In vitro inhibition against N-type calcium influx in IMR-32 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Homo sapiens (Human))
Minase Research Institute

Curated by ChEMBL
LigandPNGBDBM50451203(CHEMBL292090)
Affinity DataIC50:  5.40E+3nMAssay Description:In vitro inhibition against N-type calcium influx in IMR-32 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Homo sapiens (Human))
Minase Research Institute

Curated by ChEMBL
LigandPNGBDBM50111934((R)-2-Amino-3-cyclohexylmethylsulfanyl-propionic a...)
Affinity DataIC50:  5.80E+3nMAssay Description:In vitro inhibition of N-type calcium channels in IMR-32 cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Homo sapiens (Human))
Minase Research Institute

Curated by ChEMBL
LigandPNGBDBM50451197(CHEMBL62825)
Affinity DataIC50:  1.50E+4nMAssay Description:In vitro inhibition against N-type calcium influx in IMR-32 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent N-type calcium channel subunit alpha-1B(Homo sapiens (Human))
Minase Research Institute

Curated by ChEMBL
LigandPNGBDBM50451200(CHEMBL65145)
Affinity DataIC50:  2.60E+4nMAssay Description:In vitro inhibition against N-type calcium influx in IMR-32 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed