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Found 61 with Last Name = 'tashiro' and Initial = 'e'
TargetProtein kinase C delta type(Homo sapiens (Human))
Keio University

Curated by ChEMBL
LigandPNGBDBM50348877(CHEMBL1807163)
Affinity DataKi:  87nMAssay Description:Inhibition of [3H]PDBu binding to PKCdelta-C1B domain peptideMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C eta type(Homo sapiens (Human))
Keio University

Curated by ChEMBL
LigandPNGBDBM50348877(CHEMBL1807163)
Affinity DataKi:  360nMAssay Description:Inhibition of [3H]PDBu binding to PKCeta-C1B domain peptideMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C epsilon type(Homo sapiens (Human))
Keio University

Curated by ChEMBL
LigandPNGBDBM50348877(CHEMBL1807163)
Affinity DataKi:  480nMAssay Description:Inhibition of [3H]PDBu binding to PKCepsilon-C1B domain peptideMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
Keio University

Curated by ChEMBL
LigandPNGBDBM50348877(CHEMBL1807163)
Affinity DataKi:  600nMAssay Description:Inhibition of [3H]PDBu binding to PKCalpha-C1A domain peptideMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C gamma type(Homo sapiens (Human))
Keio University

Curated by ChEMBL
LigandPNGBDBM50348877(CHEMBL1807163)
Affinity DataKi:  660nMAssay Description:Inhibition of [3H]PDBu binding to PKCgamma-C1A domain peptideMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C beta type(Homo sapiens (Human))
Keio University

Curated by ChEMBL
LigandPNGBDBM50348877(CHEMBL1807163)
Affinity DataKi:  730nMAssay Description:Inhibition of [3H]PDBu binding to PKCbeta-C1A domain peptideMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-protein thioesterase 2(Homo sapiens (Human))
Technical University Of Dortmund

LigandPNGBDBM50282567(3,4-Dichlorophenyl boronic acid | 3,4-dichloro ben...)
Affinity DataIC50:  138nMAssay Description:The enzyme activities were determined by measuring the release of fluorescent 6,8-difluoro-4-methylumbelliferone (DiFMU) by the APT hydrolysis of DiF...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-protein thioesterase 2(Homo sapiens (Human))
Technical University Of Dortmund

LigandPNGBDBM92722(Phenylboronic acid, 15)
Affinity DataIC50:  238nMAssay Description:The enzyme activities were determined by measuring the release of fluorescent 6,8-difluoro-4-methylumbelliferone (DiFMU) by the APT hydrolysis of DiF...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAcyl-protein thioesterase 2(Homo sapiens (Human))
Technical University Of Dortmund

LigandPNGBDBM92718(Phenylboronic acid, 10)
Affinity DataIC50:  418nMAssay Description:The enzyme activities were determined by measuring the release of fluorescent 6,8-difluoro-4-methylumbelliferone (DiFMU) by the APT hydrolysis of DiF...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-protein thioesterase 1(Homo sapiens (Human))
Technical University Of Dortmund

LigandPNGBDBM92717(Phenylboronic acid, 8)
Affinity DataIC50:  510nMAssay Description:The enzyme activities were determined by measuring the release of fluorescent 6,8-difluoro-4-methylumbelliferone (DiFMU) by the APT hydrolysis of DiF...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-protein thioesterase 2(Homo sapiens (Human))
Technical University Of Dortmund

LigandPNGBDBM26139(1-benzothiophen-2-ylboranediol | 1-benzothiophen-2...)
Affinity DataIC50:  529nMAssay Description:The enzyme activities were determined by measuring the release of fluorescent 6,8-difluoro-4-methylumbelliferone (DiFMU) by the APT hydrolysis of DiF...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-protein thioesterase 1(Homo sapiens (Human))
Technical University Of Dortmund

LigandPNGBDBM50282567(3,4-Dichlorophenyl boronic acid | 3,4-dichloro ben...)
Affinity DataIC50:  1.10E+3nMAssay Description:The enzyme activities were determined by measuring the release of fluorescent 6,8-difluoro-4-methylumbelliferone (DiFMU) by the APT hydrolysis of DiF...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-protein thioesterase 1(Homo sapiens (Human))
Technical University Of Dortmund

LigandPNGBDBM92718(Phenylboronic acid, 10)
Affinity DataIC50:  1.40E+3nMAssay Description:The enzyme activities were determined by measuring the release of fluorescent 6,8-difluoro-4-methylumbelliferone (DiFMU) by the APT hydrolysis of DiF...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-protein thioesterase 2(Homo sapiens (Human))
Technical University Of Dortmund

LigandPNGBDBM92719(Phenylboronic acid, 12)
Affinity DataIC50:  1.60E+3nMAssay Description:The enzyme activities were determined by measuring the release of fluorescent 6,8-difluoro-4-methylumbelliferone (DiFMU) by the APT hydrolysis of DiF...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-protein thioesterase 2(Homo sapiens (Human))
Technical University Of Dortmund

LigandPNGBDBM92721(Phenylboronic acid, 14)
Affinity DataIC50:  1.80E+3nMAssay Description:The enzyme activities were determined by measuring the release of fluorescent 6,8-difluoro-4-methylumbelliferone (DiFMU) by the APT hydrolysis of DiF...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-protein thioesterase 2(Homo sapiens (Human))
Technical University Of Dortmund

LigandPNGBDBM92717(Phenylboronic acid, 8)
Affinity DataIC50:  1.97E+3nMAssay Description:The enzyme activities were determined by measuring the release of fluorescent 6,8-difluoro-4-methylumbelliferone (DiFMU) by the APT hydrolysis of DiF...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-protein thioesterase 2(Homo sapiens (Human))
Technical University Of Dortmund

LigandPNGBDBM92727(Phenylboronic acid, 20)
Affinity DataIC50:  1.98E+3nMAssay Description:The enzyme activities were determined by measuring the release of fluorescent 6,8-difluoro-4-methylumbelliferone (DiFMU) by the APT hydrolysis of DiF...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-protein thioesterase 2(Homo sapiens (Human))
Technical University Of Dortmund

LigandPNGBDBM92726(Phenylboronic acid, 19)
Affinity DataIC50:  2.16E+3nMAssay Description:The enzyme activities were determined by measuring the release of fluorescent 6,8-difluoro-4-methylumbelliferone (DiFMU) by the APT hydrolysis of DiF...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-protein thioesterase 1(Homo sapiens (Human))
Technical University Of Dortmund

LigandPNGBDBM26139(1-benzothiophen-2-ylboranediol | 1-benzothiophen-2...)
Affinity DataIC50:  2.30E+3nMAssay Description:The enzyme activities were determined by measuring the release of fluorescent 6,8-difluoro-4-methylumbelliferone (DiFMU) by the APT hydrolysis of DiF...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-protein thioesterase 1(Homo sapiens (Human))
Technical University Of Dortmund

LigandPNGBDBM92719(Phenylboronic acid, 12)
Affinity DataIC50:  2.60E+3nMAssay Description:The enzyme activities were determined by measuring the release of fluorescent 6,8-difluoro-4-methylumbelliferone (DiFMU) by the APT hydrolysis of DiF...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-protein thioesterase 1(Homo sapiens (Human))
Technical University Of Dortmund

LigandPNGBDBM92720(Phenylboronic acid, 13)
Affinity DataIC50:  2.70E+3nMAssay Description:The enzyme activities were determined by measuring the release of fluorescent 6,8-difluoro-4-methylumbelliferone (DiFMU) by the APT hydrolysis of DiF...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAcyl-protein thioesterase 2(Homo sapiens (Human))
Technical University Of Dortmund

LigandPNGBDBM92724(Phenylboronic acid, 17)
Affinity DataIC50:  2.87E+3nMAssay Description:The enzyme activities were determined by measuring the release of fluorescent 6,8-difluoro-4-methylumbelliferone (DiFMU) by the APT hydrolysis of DiF...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-protein thioesterase 2(Homo sapiens (Human))
Technical University Of Dortmund

LigandPNGBDBM92723(Phenylboronic acid, 16)
Affinity DataIC50:  2.95E+3nMAssay Description:The enzyme activities were determined by measuring the release of fluorescent 6,8-difluoro-4-methylumbelliferone (DiFMU) by the APT hydrolysis of DiF...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-protein thioesterase 1(Homo sapiens (Human))
Technical University Of Dortmund

LigandPNGBDBM92721(Phenylboronic acid, 14)
Affinity DataIC50:  3.20E+3nMAssay Description:The enzyme activities were determined by measuring the release of fluorescent 6,8-difluoro-4-methylumbelliferone (DiFMU) by the APT hydrolysis of DiF...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-protein thioesterase 1(Homo sapiens (Human))
Technical University Of Dortmund

LigandPNGBDBM92722(Phenylboronic acid, 15)
Affinity DataIC50:  3.20E+3nMAssay Description:The enzyme activities were determined by measuring the release of fluorescent 6,8-difluoro-4-methylumbelliferone (DiFMU) by the APT hydrolysis of DiF...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAcyl-protein thioesterase 2(Homo sapiens (Human))
Technical University Of Dortmund

LigandPNGBDBM26132((4-phenylphenyl)boranediol | Phenylboronic Acid, 1...)
Affinity DataIC50:  3.55E+3nMAssay Description:The enzyme activities were determined by measuring the release of fluorescent 6,8-difluoro-4-methylumbelliferone (DiFMU) by the APT hydrolysis of DiF...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-protein thioesterase 1(Homo sapiens (Human))
Technical University Of Dortmund

LigandPNGBDBM92723(Phenylboronic acid, 16)
Affinity DataIC50:  3.70E+3nMAssay Description:The enzyme activities were determined by measuring the release of fluorescent 6,8-difluoro-4-methylumbelliferone (DiFMU) by the APT hydrolysis of DiF...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-protein thioesterase 1(Homo sapiens (Human))
Technical University Of Dortmund

LigandPNGBDBM92724(Phenylboronic acid, 17)
Affinity DataIC50:  3.90E+3nMAssay Description:The enzyme activities were determined by measuring the release of fluorescent 6,8-difluoro-4-methylumbelliferone (DiFMU) by the APT hydrolysis of DiF...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-protein thioesterase 2(Homo sapiens (Human))
Technical University Of Dortmund

LigandPNGBDBM92720(Phenylboronic acid, 13)
Affinity DataIC50:  4.10E+3nMAssay Description:The enzyme activities were determined by measuring the release of fluorescent 6,8-difluoro-4-methylumbelliferone (DiFMU) by the APT hydrolysis of DiF...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAcyl-protein thioesterase 2(Homo sapiens (Human))
Technical University Of Dortmund

LigandPNGBDBM92725(Phenylboronic acid, 18)
Affinity DataIC50:  4.18E+3nMAssay Description:The enzyme activities were determined by measuring the release of fluorescent 6,8-difluoro-4-methylumbelliferone (DiFMU) by the APT hydrolysis of DiF...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-protein thioesterase 1(Homo sapiens (Human))
Technical University Of Dortmund

LigandPNGBDBM92725(Phenylboronic acid, 18)
Affinity DataIC50:  4.60E+3nMAssay Description:The enzyme activities were determined by measuring the release of fluorescent 6,8-difluoro-4-methylumbelliferone (DiFMU) by the APT hydrolysis of DiF...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-protein thioesterase 1(Homo sapiens (Human))
Technical University Of Dortmund

LigandPNGBDBM92726(Phenylboronic acid, 19)
Affinity DataIC50:  6.30E+3nMAssay Description:The enzyme activities were determined by measuring the release of fluorescent 6,8-difluoro-4-methylumbelliferone (DiFMU) by the APT hydrolysis of DiF...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-protein thioesterase 1(Homo sapiens (Human))
Technical University Of Dortmund

LigandPNGBDBM92727(Phenylboronic acid, 20)
Affinity DataIC50:  1.02E+4nMAssay Description:The enzyme activities were determined by measuring the release of fluorescent 6,8-difluoro-4-methylumbelliferone (DiFMU) by the APT hydrolysis of DiF...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-protein thioesterase 2(Homo sapiens (Human))
Technical University Of Dortmund

LigandPNGBDBM26140(1-benzofuran-2-ylboranediol | 1-benzofuran-2-ylbor...)
Affinity DataIC50:  1.13E+4nMAssay Description:The enzyme activities were determined by measuring the release of fluorescent 6,8-difluoro-4-methylumbelliferone (DiFMU) by the APT hydrolysis of DiF...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-protein thioesterase 1(Homo sapiens (Human))
Technical University Of Dortmund

LigandPNGBDBM26140(1-benzofuran-2-ylboranediol | 1-benzofuran-2-ylbor...)
Affinity DataIC50:  1.35E+4nMAssay Description:The enzyme activities were determined by measuring the release of fluorescent 6,8-difluoro-4-methylumbelliferone (DiFMU) by the APT hydrolysis of DiF...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50483440(Moverastin A)
Affinity DataIC50:  1.47E+4nMAssay Description:Inhibition of protein farnesyltransferase from human EC17 cells using [3H]FPP and GTP-H-RasMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAcyl-protein thioesterase 1(Homo sapiens (Human))
Technical University Of Dortmund

LigandPNGBDBM26996(CHEMBL21485 | PhB(OH)2 | Phenyl-boronic acid | Phe...)
Affinity DataIC50:  1.48E+4nMAssay Description:The enzyme activities were determined by measuring the release of fluorescent 6,8-difluoro-4-methylumbelliferone (DiFMU) by the APT hydrolysis of DiF...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-protein thioesterase 1(Homo sapiens (Human))
Technical University Of Dortmund

LigandPNGBDBM26132((4-phenylphenyl)boranediol | Phenylboronic Acid, 1...)
Affinity DataIC50:  1.69E+4nMAssay Description:The enzyme activities were determined by measuring the release of fluorescent 6,8-difluoro-4-methylumbelliferone (DiFMU) by the APT hydrolysis of DiF...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-protein thioesterase 2(Homo sapiens (Human))
Technical University Of Dortmund

LigandPNGBDBM26996(CHEMBL21485 | PhB(OH)2 | Phenyl-boronic acid | Phe...)
Affinity DataIC50:  2.51E+4nMAssay Description:The enzyme activities were determined by measuring the release of fluorescent 6,8-difluoro-4-methylumbelliferone (DiFMU) by the APT hydrolysis of DiF...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-protein thioesterase 1(Homo sapiens (Human))
Technical University Of Dortmund

LigandPNGBDBM92728(Phenylboronic acid, 7)
Affinity DataIC50:  3.36E+4nMAssay Description:The enzyme activities were determined by measuring the release of fluorescent 6,8-difluoro-4-methylumbelliferone (DiFMU) by the APT hydrolysis of DiF...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAcyl-protein thioesterase 2(Homo sapiens (Human))
Technical University Of Dortmund

LigandPNGBDBM92728(Phenylboronic acid, 7)
Affinity DataIC50:  4.15E+4nMAssay Description:The enzyme activities were determined by measuring the release of fluorescent 6,8-difluoro-4-methylumbelliferone (DiFMU) by the APT hydrolysis of DiF...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAcyl-protein thioesterase 2(Homo sapiens (Human))
Technical University Of Dortmund

LigandPNGBDBM26137((2-phenylphenyl)boranediol | Phenylboronic Acid, 1...)
Affinity DataIC50: >5.00E+4nMAssay Description:The enzyme activities were determined by measuring the release of fluorescent 6,8-difluoro-4-methylumbelliferone (DiFMU) by the APT hydrolysis of DiF...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-protein thioesterase 1(Homo sapiens (Human))
Technical University Of Dortmund

LigandPNGBDBM26137((2-phenylphenyl)boranediol | Phenylboronic Acid, 1...)
Affinity DataIC50: >5.00E+4nMAssay Description:The enzyme activities were determined by measuring the release of fluorescent 6,8-difluoro-4-methylumbelliferone (DiFMU) by the APT hydrolysis of DiF...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50483445(CHEMBL1683670)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of protein farnesyltransferase from human EC17 cells using [3H]FPP and GTP-H-RasMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50483444(CHEMBL1683675)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of protein farnesyltransferase from human EC17 cells using [3H]FPP and GTP-H-RasMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50483443(CHEMBL1683672)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of protein farnesyltransferase from human EC17 cells using [3H]FPP and GTP-H-RasMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50483442(CHEMBL1683668)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of protein farnesyltransferase from human EC17 cells using [3H]FPP and GTP-H-RasMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50483441(CHEMBL1683664)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of protein farnesyltransferase from human EC17 cells using [3H]FPP and GTP-H-RasMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50483439(CHEMBL1683674)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of protein farnesyltransferase from human EC17 cells using [3H]FPP and GTP-H-RasMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50483438(CHEMBL1683673)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of protein farnesyltransferase from human EC17 cells using [3H]FPP and GTP-H-RasMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
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