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Found 1203 with Last Name = 'tian' and Initial = 'm'
TargetMu-type opioid receptor(Homo sapiens (Human))
University Of Pennsylvania

Curated by PDSP Ki Database
LigandPNGBDBM82425(CAS_61677 | ETORPHINE - HCI | NSC_61677)
Affinity DataKi:  0.180nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
University Of Pennsylvania

Curated by PDSP Ki Database
LigandPNGBDBM21865((14beta)-17-(cyclopropylmethyl)-18-(1-hydroxy-1-me...)
Affinity DataKi:  0.180nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University Of Pennsylvania

Curated by PDSP Ki Database
LigandPNGBDBM82425(CAS_61677 | ETORPHINE - HCI | NSC_61677)
Affinity DataKi:  0.270nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
University Of Pennsylvania

Curated by PDSP Ki Database
LigandPNGBDBM94503(2-hydroxypropane-1,2,3-tricarboxylic acid;N-[4-(me...)
Affinity DataKi:  0.300nMMore data for this Ligand-Target Pair
In DepthDetails PubMedDrugBank

TargetMu-type opioid receptor(Rattus norvegicus (rat))
University Of Pennsylvania

Curated by PDSP Ki Database
LigandPNGBDBM50028147(2-[3-cyclopropylmethyl-11-hydroxy-15-methoxy-(14R)...)
Affinity DataKi:  0.420nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetCollagenase 3(Homo sapiens (Human))
University Of Notre Dame

Curated by ChEMBL
LigandPNGBDBM50268316(CHEMBL4080186)
Affinity DataKi:  0.470nMAssay Description:Inhibition of human recombinant MMP-13 catalytic domain (104 to 274 residues) expressed in Escherichia coli using fluorogenic Mca-KPLGL-Dpa-AR-NH2 as...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
University Of Pennsylvania

Curated by PDSP Ki Database
LigandPNGBDBM50028147(2-[3-cyclopropylmethyl-11-hydroxy-15-methoxy-(14R)...)
Affinity DataKi:  0.510nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetCollagenase 3(Homo sapiens (Human))
University Of Notre Dame

Curated by ChEMBL
LigandPNGBDBM50268309(CHEMBL4088060)
Affinity DataKi:  0.590nMAssay Description:Inhibition of human recombinant MMP-13 catalytic domain (104 to 274 residues) expressed in Escherichia coli using fluorogenic Mca-KPLGL-Dpa-AR-NH2 as...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil collagenase(Homo sapiens (Human))
University Of Notre Dame

Curated by ChEMBL
LigandPNGBDBM50268309(CHEMBL4088060)
Affinity DataKi:  0.710nMAssay Description:Inhibition of human recombinant MMP-8 catalytic domain (99 to 269 residues) expressed in Escherichia coli using fluorogenic Mca-KPLGL-Dpa-AR-NH2 as s...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
University Of Pennsylvania

Curated by PDSP Ki Database
LigandPNGBDBM81934(Beta-Endorphin)
Affinity DataKi:  0.940nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University Of Pennsylvania

Curated by PDSP Ki Database
LigandPNGBDBM50008984(4-(4-Chloro-benzyl)-2-(1-methyl-azepan-4-yl)-2H-ph...)
Affinity DataKi:  1.30nMMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Homo sapiens (Human))
University Of Pennsylvania

Curated by PDSP Ki Database
LigandPNGBDBM21015((2S)-2-{2-[(2R)-2-[(2S)-2-amino-3-(4-hydroxyphenyl...)
Affinity DataKi:  1.40nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
University Of Pennsylvania

Curated by PDSP Ki Database
LigandPNGBDBM50013388(6-Ethyl-3-(1-hydroxy-cyclopropylmethyl)-11,11-dime...)
Affinity DataKi:  1.40nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
University Of Pennsylvania

Curated by PDSP Ki Database
LigandPNGBDBM50000788((morphine)4-methyl-(1S,5R,13R,14S,17R)-12-oxa-4-az...)
Affinity DataKi:  1.40nMMore data for this Ligand-Target Pair
In DepthDetails PubMedDrugBank

TargetMu-type opioid receptor(Homo sapiens (Human))
University Of Pennsylvania

Curated by PDSP Ki Database
LigandPNGBDBM60212((4R,4aS,7aR,12bS)-3-(cyclopropylmethyl)-4a,9-bis(o...)
Affinity DataKi:  1.5nMMore data for this Ligand-Target Pair
In DepthDetails PubMedDrugBank

TargetMu-type opioid receptor(Rattus norvegicus (rat))
University Of Pennsylvania

Curated by PDSP Ki Database
LigandPNGBDBM81934(Beta-Endorphin)
Affinity DataKi:  1.70nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
University Of Pennsylvania

Curated by PDSP Ki Database
LigandPNGBDBM50008984(4-(4-Chloro-benzyl)-2-(1-methyl-azepan-4-yl)-2H-ph...)
Affinity DataKi:  1.90nMMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Homo sapiens (Human))
University Of Pennsylvania

Curated by PDSP Ki Database
LigandPNGBDBM82427(CAS_5985-38-6 | LEVORPHANOL-tartarate)
Affinity DataKi:  1.90nMMore data for this Ligand-Target Pair
In DepthDetails PubMedDrugBank

TargetMu-type opioid receptor(Homo sapiens (Human))
University Of Pennsylvania

Curated by PDSP Ki Database
LigandPNGBDBM50000092((-)-(etorphine) | (-)-morphine | (1S,5R,13R,14S)-1...)
TargetNeutrophil collagenase(Homo sapiens (Human))
University Of Notre Dame

Curated by ChEMBL
LigandPNGBDBM50268317(CHEMBL4076356)
Affinity DataKi:  3.30nMAssay Description:Inhibition of human recombinant MMP-8 catalytic domain (99 to 269 residues) expressed in Escherichia coli using fluorogenic Mca-KPLGL-Dpa-AR-NH2 as s...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
University Of Pennsylvania

Curated by PDSP Ki Database
LigandPNGBDBM50019574(CHEMBL406014 | CTOP | D-Phe-Cys-Tyr-D-Trp-Orn-Thr-...)
Affinity DataKi:  3.90nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
University Of Pennsylvania

Curated by PDSP Ki Database
LigandPNGBDBM82507((+/-)-Methadone | CAS_5967-73-7 | METHADONE | Meth...)
Affinity DataKi:  5.60nMMore data for this Ligand-Target Pair
In DepthDetails PubMedDrugBank

TargetMu-type opioid receptor(Homo sapiens (Human))
University Of Pennsylvania

Curated by PDSP Ki Database
LigandPNGBDBM50021560(4-allyl-(13R,14S)-12-oxa-4-azapentacyclo[9.6.1.01,...)
Affinity DataKi:  6.60nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
University Of Pennsylvania

Curated by PDSP Ki Database
LigandPNGBDBM50001465((S)-2-[(S)-2-(2-{2-[(S)-2-Amino-3-(4-hydroxy-pheny...)
Affinity DataKi:  6.60nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetGlycogen phosphorylase, muscle form(Homo sapiens (Human))
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50149297((S)-1-Ethyl-6-methyl-4-phenyl-1,4-dihydro-pyridine...)
Affinity DataKi:  11nMAssay Description:Inhibitory activity against rabbit muscle glycogen phosphorylase a in the absence of AMPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
University Of Pennsylvania

Curated by PDSP Ki Database
LigandPNGBDBM50059090(10-(4-Amino-butyl)-19-(2-amino-3-phenyl-propionyla...)
Affinity DataKi:  12nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University Of Pennsylvania

Curated by PDSP Ki Database
LigandPNGBDBM82507((+/-)-Methadone | CAS_5967-73-7 | METHADONE | Meth...)
Affinity DataKi:  19nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetNeutrophil collagenase(Homo sapiens (Human))
University Of Notre Dame

Curated by ChEMBL
LigandPNGBDBM50268316(CHEMBL4080186)
Affinity DataKi:  19nMAssay Description:Inhibition of human recombinant MMP-8 catalytic domain (99 to 269 residues) expressed in Escherichia coli using fluorogenic Mca-KPLGL-Dpa-AR-NH2 as s...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University Of Pennsylvania

Curated by PDSP Ki Database
LigandPNGBDBM50000092((-)-(etorphine) | (-)-morphine | (1S,5R,13R,14S)-1...)
Affinity DataKi:  22nMMore data for this Ligand-Target Pair
TargetCollagenase 3(Homo sapiens (Human))
University Of Notre Dame

Curated by ChEMBL
LigandPNGBDBM50268317(CHEMBL4076356)
Affinity DataKi:  25nMAssay Description:Inhibition of human recombinant MMP-13 catalytic domain (104 to 274 residues) expressed in Escherichia coli using fluorogenic Mca-KPLGL-Dpa-AR-NH2 as...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCollagenase 3(Homo sapiens (Human))
University Of Notre Dame

Curated by ChEMBL
LigandPNGBDBM50268310(CHEMBL4069479)
Affinity DataKi:  36nMAssay Description:Inhibition of human recombinant MMP-13 catalytic domain (104 to 274 residues) expressed in Escherichia coli using fluorogenic Mca-KPLGL-Dpa-AR-NH2 as...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
University Of Pennsylvania

Curated by PDSP Ki Database
LigandPNGBDBM82266(CAS_29485-83-4 | CODEINE SULFATE | Codeine | NSC_2...)
Affinity DataKi:  65nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University Of Pennsylvania

Curated by PDSP Ki Database
LigandPNGBDBM82266(CAS_29485-83-4 | CODEINE SULFATE | Codeine | NSC_2...)
Affinity DataKi:  168nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetCollagenase 3(Homo sapiens (Human))
University Of Notre Dame

Curated by ChEMBL
LigandPNGBDBM50268311(CHEMBL4104422)
Affinity DataKi:  190nMAssay Description:Inhibition of human recombinant MMP-13 catalytic domain (104 to 274 residues) expressed in Escherichia coli using fluorogenic Mca-KPLGL-Dpa-AR-NH2 as...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen phosphorylase, muscle form(Oryctolagus cuniculus (rabbit))
The National Hellenic Research Foundation

Curated by ChEMBL
LigandPNGBDBM50194701((2R,3R,4R)-2-Hydroxymethylpyrrolidin-3,4-diol hydr...)
Affinity DataKi:  342nMAssay Description:Inhibition of non-phosphorylated form of rabbit muscle glycogen phosphorylase in presence of glycogen and 45 mM phosphateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen phosphorylase, muscle form(Oryctolagus cuniculus (rabbit))
The National Hellenic Research Foundation

Curated by ChEMBL
LigandPNGBDBM50194701((2R,3R,4R)-2-Hydroxymethylpyrrolidin-3,4-diol hydr...)
Affinity DataKi:  396nMAssay Description:Inhibition of non-phosphorylated form of rabbit muscle glycogen phosphorylase in presence of 6.17 mM glycogen and phosphateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen phosphorylase, liver form(Homo sapiens (Human))
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50016703(2-Hydroxymethyl-pyrrolidine-3,4-diol | BDBM5003148...)
Affinity DataKi:  400nMAssay Description:Inhibitory activity against pig Liver glycogen phosphorylase aMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2B(Homo sapiens (Human))
University Of Utah

Curated by ChEMBL
LigandPNGBDBM50335603(CHEMBL1651095 | Pulicatin A)
Affinity DataKi:  505nMAssay Description:Binding affinity to human 5HT2B receptor by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
University Of Pennsylvania

Curated by PDSP Ki Database
LigandPNGBDBM50000788((morphine)4-methyl-(1S,5R,13R,14S,17R)-12-oxa-4-az...)
Affinity DataKi:  1.00E+3nMMore data for this Ligand-Target Pair
In DepthDetails PubMedDrugBank

TargetMu-type opioid receptor(Homo sapiens (Human))
University Of Pennsylvania

Curated by PDSP Ki Database
LigandPNGBDBM50003571((-)-3-Hydroxy-N-methylmorphinan hydrochloride (lev...)
Affinity DataKi:  1.00E+3nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
University Of Pennsylvania

Curated by PDSP Ki Database
LigandPNGBDBM82426(Beta-Endorphin, des-Tyr)
Affinity DataKi:  1.00E+3nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
University Of Pennsylvania

Curated by PDSP Ki Database
LigandPNGBDBM50028147(2-[3-cyclopropylmethyl-11-hydroxy-15-methoxy-(14R)...)
Affinity DataKi:  1.00E+3nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
Target5-hydroxytryptamine receptor 2B(Homo sapiens (Human))
University Of Utah

Curated by ChEMBL
LigandPNGBDBM50335599(CHEMBL1651091 | pulicatins F)
Affinity DataKi:  1.03E+3nMAssay Description:Binding affinity to human 5HT2B receptor by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2B(Homo sapiens (Human))
University Of Utah

Curated by ChEMBL
LigandPNGBDBM50335600(CHEMBL1651092 | pulicatins G)
Affinity DataKi:  1.26E+3nMAssay Description:Binding affinity to human 5HT2B receptor by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2B(Homo sapiens (Human))
University Of Utah

Curated by ChEMBL
LigandPNGBDBM50335598(CHEMBL1651090 | aerugine)
Affinity DataKi:  1.36E+3nMAssay Description:Binding affinity to human 5HT2B receptor by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2B(Homo sapiens (Human))
University Of Utah

Curated by ChEMBL
LigandPNGBDBM50335604(CHEMBL1651096 | pulicatin D)
Affinity DataKi:  1.54E+3nMAssay Description:Binding affinity to human 5HT2B receptor by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen phosphorylase, muscle form(Homo sapiens (Human))
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50149315((6S,7S,8R,9R)-6,7,8-Trihydroxy-9-hydroxymethyl-1,3...)
Affinity DataKi:  3.00E+3nMAssay Description:Inhibitory activity against rabbit Muscle glycogen phosphorylase bMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2B(Homo sapiens (Human))
University Of Utah

Curated by ChEMBL
LigandPNGBDBM50335601(CHEMBL1651093 | Watasemycins A)
Affinity DataKi:  3.92E+3nMAssay Description:Binding affinity to human 5HT2B receptor by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2B(Homo sapiens (Human))
University Of Utah

Curated by ChEMBL
LigandPNGBDBM50335602(CHEMBL1651094 | Watasemycins B)
Affinity DataKi:  4.70E+3nMAssay Description:Binding affinity to human 5HT2B receptor by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen phosphorylase, muscle form(Oryctolagus cuniculus (rabbit))
The National Hellenic Research Foundation

Curated by ChEMBL
LigandPNGBDBM50182801((3R,4R,5R)-5-(Hydroxymethyl)piperidine-3,4-diol, 8...)
Affinity DataKi:  5.20E+3nMAssay Description:Inhibition of non-phosphorylated form of rabbit muscle glycogen phosphorylase in presence of phosphateMore data for this Ligand-Target Pair
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