Compile Data Set for Download or QSAR
maximum 50k data
Found 39 with Last Name = 'vella-rountree' and Initial = 'l'
LigandPNGBDBM86231(ATR | ATROPINE | Atropine,(-) | CAS_51-55-8 | CHEM...)
Affinity DataKi:  0.520nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
LigandPNGBDBM86231(ATR | ATROPINE | Atropine,(-) | CAS_51-55-8 | CHEM...)
Affinity DataKi:  1.10nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
LigandPNGBDBM50176065(4-DAMP | 4-Diphenylacetoxy-1,1-dimethyl-piperidini...)
Affinity DataKi:  1.40nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
LigandPNGBDBM81800(CAS_57558-44-8 | NSC_42470 | Secoverine)
Affinity DataKi:  5.90nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
LigandPNGBDBM81800(CAS_57558-44-8 | NSC_42470 | Secoverine)
Affinity DataKi:  7.80nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
LigandPNGBDBM39341(11-[(4-methylpiperazin-1-yl)acetyl]-5,11-dihydro-6...)
In DepthDetails PubMed
TargetMuscarinic acetylcholine receptor M2(RAT)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50005854(1-(4-Azetidin-1-yl-but-2-ynyl)-pyrrolidin-2-one | ...)
Affinity DataKi:  27nMAssay Description:Compound was evaluated for its binding affinity towards muscarinic acetylcholine receptor M2 in rat brainstemMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM81799(CAS_98299-40-2 | HHSiD | NSC_3602 | hexahydrosilad...)
Affinity DataKi:  47nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
LigandPNGBDBM81799(CAS_98299-40-2 | HHSiD | NSC_3602 | hexahydrosilad...)
Affinity DataKi:  60nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMuscarinic acetylcholine receptor M2(RAT)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50004665((oxotremorine)1-(4-Pyrrolidin-1-yl-but-2-ynyl)-pyr...)
Affinity DataKi:  84nMAssay Description:Compound was evaluated for its binding affinity towards muscarinic acetylcholine receptor M2 in rat brainstemMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50004665((oxotremorine)1-(4-Pyrrolidin-1-yl-but-2-ynyl)-pyr...)
Affinity DataKi:  196nMAssay Description:Compound was evaluated for its binding affinity towards muscarinic acetylcholine receptor in rat cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM39341(11-[(4-methylpiperazin-1-yl)acetyl]-5,11-dihydro-6...)
Affinity DataKi:  214nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
LigandPNGBDBM50064176(CHEMBL27673 | CHEMBL500996 | METHOCTRAMINE | N,N''...)
Affinity DataKi:  410nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
LigandPNGBDBM50064176(CHEMBL27673 | CHEMBL500996 | METHOCTRAMINE | N,N''...)
Affinity DataKi:  600nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
LigandPNGBDBM50018056((AF-DX 116) 11-[2-(2-Diethylaminomethyl-piperidin-...)
Affinity DataKi:  614nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMuscarinic acetylcholine receptor M2(RAT)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50455987(CHEMBL2115360)
Affinity DataKi:  636nMAssay Description:Compound was evaluated for its binding affinity towards M2 receptor in rat brainstemMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(RAT)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50005851(1-[4-(Ethyl-methyl-amino)-but-2-ynyl]-pyrrolidin-2...)
Affinity DataKi:  813nMAssay Description:Compound was evaluated for its binding affinity towards muscarinic acetylcholine receptor M2 in rat brainstemMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(RAT)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50005856(1-(4-Dimethylamino-but-2-ynyl)-pyrrolidin-2-one | ...)
Affinity DataKi:  926nMAssay Description:Compound was evaluated for its binding affinity towards Muscarinic acetylcholine receptor M2 in rat brainstemMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50018056((AF-DX 116) 11-[2-(2-Diethylaminomethyl-piperidin-...)
Affinity DataKi:  1.20E+3nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
LigandPNGBDBM50455986(CHEMBL2115361)
Affinity DataKi:  1.20E+3nMAssay Description:Compound was evaluated for its binding affinity towards M1 receptor in rat cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50005854(1-(4-Azetidin-1-yl-but-2-ynyl)-pyrrolidin-2-one | ...)
Affinity DataKi:  2.25E+3nMAssay Description:Compound was evaluated for its binding affinity towards muscarinic acetylcholine receptor in rat cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(RAT)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50455988(CHEMBL2115359)
Affinity DataKi:  2.46E+3nMAssay Description:Compound was evaluated for its binding affinity towards M2 receptor in rat brainstemMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50005851(1-[4-(Ethyl-methyl-amino)-but-2-ynyl]-pyrrolidin-2...)
Affinity DataKi:  2.69E+3nMAssay Description:Compound was evaluated for its binding affinity towards muscarinic acetylcholine receptor in rat cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50455987(CHEMBL2115360)
Affinity DataKi:  3.03E+3nMAssay Description:Compound was evaluated for its binding affinity towards M1 receptor in rat cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50455988(CHEMBL2115359)
Affinity DataKi:  3.07E+3nMAssay Description:Compound was evaluated for its binding affinity towards M1 receptor in rat cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(RAT)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50455986(CHEMBL2115361)
Affinity DataKi:  3.66E+3nMAssay Description:Compound was evaluated for its binding affinity towards M2 receptor in rat brainstemMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50455982(CHEMBL2114427)
Affinity DataKi:  5.38E+3nMAssay Description:Compound was evaluated for its binding affinity towards M1 receptor in rat cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50455985(CHEMBL2115362)
Affinity DataKi:  5.46E+3nMAssay Description:Compound was evaluated for its binding affinity towards M1 receptor in rat cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(RAT)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50455983(CHEMBL2114425)
Affinity DataKi:  5.64E+3nMAssay Description:Compound was evaluated for its binding affinity towards M2 receptor in rat brainstemMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(RAT)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50455985(CHEMBL2115362)
Affinity DataKi:  5.86E+3nMAssay Description:Compound was evaluated for its binding affinity towards M2 receptor in rat brainstemMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(RAT)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50455982(CHEMBL2114427)
Affinity DataKi:  7.06E+3nMAssay Description:Compound was evaluated for its binding affinity towards M2 receptor in rat brainstemMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50455984(CHEMBL2114430)
Affinity DataKi:  1.05E+4nMAssay Description:Compound was evaluated for its binding affinity towards M1 receptor in rat cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(RAT)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50455984(CHEMBL2114430)
Affinity DataKi:  1.08E+4nMAssay Description:Compound was evaluated for its binding affinity towards M2 receptor in rat brainstemMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(RAT)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50455981(CHEMBL2114426)
Affinity DataKi:  1.58E+4nMAssay Description:Compound was evaluated for its binding affinity towards M2 receptor in rat brainstemMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50005856(1-(4-Dimethylamino-but-2-ynyl)-pyrrolidin-2-one | ...)
Affinity DataKi:  1.59E+4nMAssay Description:Compound was evaluated for its binding affinity towards Muscarinic acetylcholine receptor M1 in rat cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50455981(CHEMBL2114426)
Affinity DataKi:  2.76E+4nMAssay Description:Compound was evaluated for its binding affinity towards M1 receptor in rat cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(RAT)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50005855(1-(4-Methylamino-but-2-ynyl)-pyrrolidin-2-one | CH...)
Affinity DataKi:  3.81E+4nMAssay Description:Compound was evaluated for its binding affinity towards muscarinic acetylcholine receptor M2 in rat brainstemMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50455983(CHEMBL2114425)
Affinity DataKi:  4.05E+4nMAssay Description:Compound was evaluated for its binding affinity towards M1 receptor in rat cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50005855(1-(4-Methylamino-but-2-ynyl)-pyrrolidin-2-one | CH...)
Affinity DataKi:  6.55E+4nMAssay Description:Compound was evaluated for its binding affinity towards muscarinic acetylcholine receptor in rat cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed