Compile Data Set for Download or QSAR
maximum 50k data
Found 58 with Last Name = 'vice' and Initial = 'sf'
TargetMuscarinic acetylcholine receptor M2(RAT)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50121132((4-{2-[4-(Benzo[1,3]dioxole-5-sulfonyl)-phenyl]-[1...)
Affinity DataKi:  0.0650nMAssay Description:Binding affinity towards Muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(RAT)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50121130((2-Amino-3-methyl-phenyl)-(4-{2-[4-(4-methoxy-benz...)
Affinity DataKi:  0.390nMAssay Description:Binding affinity towards Muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(RAT)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50121134((3-Amino-2-methyl-phenyl)-(4-{2-[4-(4-methoxy-benz...)
Affinity DataKi:  0.400nMAssay Description:Binding affinity towards Muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(RAT)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50121126((2-Amino-4-fluoro-phenyl)-(4-{2-[4-(4-methoxy-benz...)
Affinity DataKi:  0.440nMAssay Description:Binding affinity towards Muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(RAT)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50121138((2-Amino-3-fluoro-phenyl)-(4-{2-[4-(4-methoxy-benz...)
Affinity DataKi:  0.510nMAssay Description:Binding affinity towards Muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(RAT)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50121139((5-Amino-2-chloro-phenyl)-(4-{2-[4-(4-methoxy-benz...)
Affinity DataKi:  0.530nMAssay Description:Binding affinity towards Muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(RAT)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50121127((3-Amino-2-chloro-phenyl)-(4-{2-[4-(4-methoxy-benz...)
Affinity DataKi:  0.530nMAssay Description:Binding affinity towards Muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(RAT)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50121124((4-{2-[4-(4-Methoxy-benzenesulfonyl)-phenyl]-[1,3]...)
Affinity DataKi:  0.540nMAssay Description:Binding affinity towards Muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(RAT)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50121125((2-Amino-5-fluoro-phenyl)-(4-{2-[4-(4-methoxy-benz...)
Affinity DataKi:  0.680nMAssay Description:Binding affinity towards Muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50123438((3,5-Dichloro-pyridin-4-yl)-(4-methyl-4-{(S)-3-met...)
Affinity DataKi:  0.700nMAssay Description:Ability to inhibit [125I]-labeled RANTES binding to the CCR5 receptor expressed in membrane preparations from CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(RAT)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50121131((3-Chloro-2-methyl-phenyl)-(4-{2-[4-(4-methoxy-ben...)
Affinity DataKi:  0.720nMAssay Description:Binding affinity towards Muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(RAT)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50121144((3-Amino-phenyl)-(4-{2-[4-(4-methoxy-benzenesulfon...)
Affinity DataKi:  0.780nMAssay Description:Binding affinity towards Muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(RAT)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50121140((4-{2-[4-(4-Methoxy-benzenesulfonyl)-phenyl]-[1,3]...)
Affinity DataKi:  0.860nMAssay Description:Binding affinity towards Muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(RAT)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50121142((4-{2-[4-(4-Methoxy-benzenesulfonyl)-phenyl]-[1,3]...)
Affinity DataKi:  0.900nMAssay Description:Binding affinity towards Muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(RAT)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50121129((4-{2-[4-(4-Methoxy-benzenesulfonyl)-phenyl]-[1,3]...)
Affinity DataKi:  1nMAssay Description:Binding affinity towards Muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(RAT)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50121121((2-Amino-3-chloro-phenyl)-(4-{2-[4-(4-methoxy-benz...)
Affinity DataKi:  1.10nMAssay Description:Binding affinity towards Muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(RAT)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50121135((4-{2-[4-(4-Methoxy-benzenesulfonyl)-phenyl]-[1,3]...)
Affinity DataKi:  1.20nMAssay Description:Binding affinity towards Muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(RAT)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50121136((2,3-Dimethyl-phenyl)-(4-{2-[4-(4-methoxy-benzenes...)
Affinity DataKi:  1.40nMAssay Description:Binding affinity towards Muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(RAT)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50121120((2-Amino-phenyl)-(4-{2-[4-(4-methoxy-benzenesulfon...)
Affinity DataKi:  1.5nMAssay Description:Binding affinity towards Muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(RAT)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50121123((2-Chloro-phenyl)-(4-{2-[4-(4-methoxy-benzenesulfo...)
Affinity DataKi:  1.60nMAssay Description:Binding affinity towards Muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(RAT)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50121143((2-Bromo-phenyl)-(4-{2-[4-(4-methoxy-benzenesulfon...)
Affinity DataKi:  1.80nMAssay Description:Binding affinity towards Muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50104946((2,4-Dimethyl-pyridin-3-yl)-(4-methyl-4-{(S)-3-met...)
Affinity DataKi:  2nMAssay Description:Ability to inhibit [125I]-labeled RANTES binding to the CCR5 receptor expressed in membrane preparations from CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(RAT)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50121133((2,6-Dichloro-phenyl)-(4-{2-[4-(4-methoxy-benzenes...)
Affinity DataKi:  2.30nMAssay Description:Binding affinity towards Muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(RAT)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50121128((4-{2-[4-(4-Methoxy-benzenesulfinyl)-phenyl]-[1,3]...)
Affinity DataKi:  2.5nMAssay Description:Binding affinity towards Muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50123436((3,5-Dichloro-1-oxy-pyridin-4-yl)-(4-methyl-4-{(S)...)
Affinity DataKi:  2.70nMAssay Description:Ability to inhibit [125I]-labeled RANTES binding to the CCR5 receptor expressed in membrane preparations from CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50123435((4,6-Dimethyl-pyrimidin-5-yl)-(4-methyl-4-{(S)-3-m...)
Affinity DataKi:  3nMAssay Description:Ability of compound to inhibit [125I]-labeled RANTES binding to the CCR5 receptor expressed in membrane preparations from CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(RAT)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50121141((2-Fluoro-phenyl)-(4-{2-[4-(4-methoxy-benzenesulfo...)
Affinity DataKi:  4.80nMAssay Description:Binding affinity towards Muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50123445((3,5-Dimethyl-pyridin-4-yl)-(4-methyl-4-{(S)-3-met...)
Affinity DataKi:  5.20nMAssay Description:Ability to inhibit [125I]-labeled RANTES binding to the CCR5 receptor expressed in membrane preparations from CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50104956((2,4-Dimethyl-1-oxy-pyridin-3-yl)-(4-methyl-4-{(S)...)
Affinity DataKi:  7nMAssay Description:Ability to inhibit [125I]-labeled RANTES binding to the CCR5 receptor expressed in membrane preparations from CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50123444((4,6-Dimethyl-2-trifluoromethyl-pyrimidin-5-yl)-(4...)
Affinity DataKi:  10nMAssay Description:Ability to inhibit [125I]-labeled RANTES binding to the CCR5 receptor expressed in membrane preparations from CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50123442((4-Methyl-4-{(S)-3-methyl-4-[(S)-1-(4-trifluoromet...)
Affinity DataKi:  10nMAssay Description:Ability to inhibit [125I]-labeled RANTES binding to the CCR5 receptor expressed in membrane preparations from CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50123446((4,6-Dimethyl-pyrimidin-5-yl)-(4-methyl-4-{(S)-3-m...)
Affinity DataKi:  11nMAssay Description:Ability to inhibit [125I]-labeled RANTES binding to the CCR5 receptor expressed in membrane preparations from CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50123437((2-Methoxy-4,6-dimethyl-pyrimidin-5-yl)-(4-methyl-...)
Affinity DataKi:  11nMAssay Description:Ability to inhibit [125I]-labeled RANTES binding to the CCR5 receptor expressed in membrane preparations from CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50123443((4,6-Dimethyl-pyrimidin-5-yl)-(4-{(S)-4-[(S)-1-(4-...)
Affinity DataKi:  11nMAssay Description:Ability to inhibit [125I]-labeled RANTES binding to the CCR5 receptor expressed in membrane preparations from CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50123439((4,6-Dimethyl-2-phenyl-pyrimidin-5-yl)-(4-methyl-4...)
Affinity DataKi:  12nMAssay Description:Ability to inhibit [125I]-labeled RANTES binding to the CCR5 receptor expressed in membrane preparations from CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50123447((3,5-Dimethyl-1-oxy-pyridin-4-yl)-(4-methyl-4-{(S)...)
Affinity DataKi:  18nMAssay Description:Ability to inhibit [125I]-labeled RANTES binding to the CCR5 receptor expressed in membrane preparations from CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(RAT)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50121122((4-{(4R,5R)-2-[4-(4-Methoxy-benzenesulfonyl)-pheny...)
Affinity DataKi:  18nMAssay Description:Binding affinity towards Muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50123440(4-((S)-1-{(S)-4-[1-(4,6-Dimethyl-pyrimidine-5-carb...)
Affinity DataKi:  20nMAssay Description:Ability to inhibit [125I]-labeled RANTES binding to the CCR5 receptor expressed in membrane preparations from CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50123441((2-Amino-4,6-dimethyl-pyrimidin-5-yl)-(4-methyl-4-...)
Affinity DataKi:  38nMAssay Description:Ability to inhibit [125I]-labeled RANTES binding to the CCR5 receptor expressed in membrane preparations from CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(RAT)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50121137((4-{(4R,5R)-2-[4-(4-Methoxy-benzenesulfinyl)-pheny...)
Affinity DataKi:  51nMAssay Description:Binding affinity towards Muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50123446((4,6-Dimethyl-pyrimidin-5-yl)-(4-methyl-4-{(S)-3-m...)
Affinity DataKi:  68nMAssay Description:Binding affinity towards muscarinic receptor M2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50123440(4-((S)-1-{(S)-4-[1-(4,6-Dimethyl-pyrimidine-5-carb...)
Affinity DataKi:  164nMAssay Description:Binding affinity towards muscarinic receptor M2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50123443((4,6-Dimethyl-pyrimidin-5-yl)-(4-{(S)-4-[(S)-1-(4-...)
Affinity DataKi:  169nMAssay Description:Binding affinity towards muscarinic receptor M2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50123437((2-Methoxy-4,6-dimethyl-pyrimidin-5-yl)-(4-methyl-...)
Affinity DataKi:  202nMAssay Description:Binding affinity towards muscarinic receptor M2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50104956((2,4-Dimethyl-1-oxy-pyridin-3-yl)-(4-methyl-4-{(S)...)
Affinity DataKi:  250nMAssay Description:Binding affinity towards muscarinic receptor M2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50123447((3,5-Dimethyl-1-oxy-pyridin-4-yl)-(4-methyl-4-{(S)...)
Affinity DataKi:  255nMAssay Description:Binding affinity towards muscarinic receptor M2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50123436((3,5-Dichloro-1-oxy-pyridin-4-yl)-(4-methyl-4-{(S)...)
Affinity DataKi:  348nMAssay Description:Binding affinity towards muscarinic receptor M2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50104956((2,4-Dimethyl-1-oxy-pyridin-3-yl)-(4-methyl-4-{(S)...)
Affinity DataKi:  350nMAssay Description:Binding affinity of the compound towards muscarinic receptor M1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50123435((4,6-Dimethyl-pyrimidin-5-yl)-(4-methyl-4-{(S)-3-m...)
Affinity DataKi:  456nMAssay Description:Inhibition of binding affinity of the compound to muscarinic receptor M2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50123435((4,6-Dimethyl-pyrimidin-5-yl)-(4-methyl-4-{(S)-3-m...)
Affinity DataKi:  575nMAssay Description:Binding affinity towards muscarinic receptor M2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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