TargetRetinoic acid receptor alpha [200-419]/gamma [183-417](Homo sapiens (Human))
Institute Of Genetics And Molecular And Cellular Biology (Igbmc)
Institute Of Genetics And Molecular And Cellular Biology (Igbmc)
Affinity DataKi: 1nM ΔG°: -47.8kJ/molepH: 8.0 T: 2°CAssay Description:Competitive assay were perform with 5nM tritiated all-trans retinoic acid (t-RA; 5nM) with or without 100-fold excess of non-radioactive t-RA (500nM)...More data for this Ligand-Target Pair
TargetRetinoic acid receptor alpha [200-419]/gamma [183-417](Homo sapiens (Human))
Institute Of Genetics And Molecular And Cellular Biology (Igbmc)
Institute Of Genetics And Molecular And Cellular Biology (Igbmc)
Affinity DataKi: 1nM ΔG°: -47.8kJ/molepH: 8.0 T: 2°CAssay Description:Competitive assay were perform with 5nM tritiated all-trans retinoic acid (t-RA; 5nM) with or without 100-fold excess of non-radioactive t-RA (500nM)...More data for this Ligand-Target Pair
TargetRetinoic acid receptor gamma [183-417](Homo sapiens (Human))
Institute Of Genetics And Molecular And Cellular Biology (Igbmc)
Institute Of Genetics And Molecular And Cellular Biology (Igbmc)
Affinity DataKi: 1.5nM ΔG°: -46.8kJ/molepH: 8.0 T: 2°CAssay Description:Competitive assay were perform with 5nM tritiated all-trans retinoic acid (t-RA; 5nM) with or without 100-fold excess of non-radioactive t-RA (500nM)...More data for this Ligand-Target Pair
TargetRetinoic acid receptor alpha [200-419](Homo sapiens (Human))
Institute Of Genetics And Molecular And Cellular Biology (Igbmc)
Institute Of Genetics And Molecular And Cellular Biology (Igbmc)
Affinity DataKi: 2nM ΔG°: -46.2kJ/molepH: 8.0 T: 2°CAssay Description:Competitive assay were perform with 5nM tritiated all-trans retinoic acid (t-RA; 5nM) with or without 100-fold excess of non-radioactive t-RA (500nM)...More data for this Ligand-Target Pair
TargetRetinoic acid receptor alpha [200-419](Homo sapiens (Human))
Institute Of Genetics And Molecular And Cellular Biology (Igbmc)
Institute Of Genetics And Molecular And Cellular Biology (Igbmc)
Affinity DataKi: 2.5nM ΔG°: -45.6kJ/molepH: 8.0 T: 2°CAssay Description:Competitive assay were perform with 5nM tritiated all-trans retinoic acid (t-RA; 5nM) with or without 100-fold excess of non-radioactive t-RA (500nM)...More data for this Ligand-Target Pair
Affinity DataIC50: 33nMAssay Description:Displacement of MR121-Nrf2 from human N-terminal His-tagged Kelch-DC domain of Keap1 (321 to 609) expressed in Escherichia coli BL21 (DE3) after 40 m...More data for this Ligand-Target Pair
Affinity DataIC50: 2.70E+3nMAssay Description:Displacement of MR121-Nrf2 from human N-terminal His-tagged Kelch-DC domain of Keap1 (321 to 609) expressed in Escherichia coli BL21 (DE3) after 40 m...More data for this Ligand-Target Pair
Affinity DataIC50: 1.18E+5nMAssay Description:Displacement of MR121-Nrf2 from human N-terminal His-tagged Kelch-DC domain of Keap1 (321 to 609) expressed in Escherichia coli BL21 (DE3) after 40 m...More data for this Ligand-Target Pair