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Found 65 with Last Name = 'yaksh' and Initial = 'tl'
TargetNicotinic acetylcholine receptor(RAT)
University Of California

Curated by PDSP Ki Database
LigandPNGBDBM50107863((-)-cytisine | (1R,9R)-7,11-diazatricyclo[7.3.1.0~...)
Affinity DataKi:  0.400nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50117263((3R,6S,12S)-12-[(S)-2-Amino-3-(4-hydroxy-phenyl)-p...)
Affinity DataKi:  0.630nMAssay Description:Inhibition of binding of [3H]diprenorphine to cloned human Opioid receptor delta 1 expressed in CHO cell membrane;Range is in between (0.62-0.65)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNicotinic acetylcholine receptor(RAT)
University Of California

Curated by PDSP Ki Database
LigandPNGBDBM50107863((-)-cytisine | (1R,9R)-7,11-diazatricyclo[7.3.1.0~...)
Affinity DataKi:  0.710nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50117262(12-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-6...)
Affinity DataKi:  0.790nMAssay Description:Inhibition of binding of [3H]-diprenorphine to cloned human Opioid receptor delta 1 expressed in CHO cell membrane;Range is between (0.66-0.95)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50117264(12-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-6...)
Affinity DataKi:  0.930nMAssay Description:Inhibition of binding of [3H]-diprenorphine to cloned human Opioid receptor delta 1 expressed in CHO cell membrane;Range is between (0.35-2.5)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNicotinic acetylcholine receptor(RAT)
University Of California

Curated by PDSP Ki Database
LigandPNGBDBM82070(CAS_29790-52-1 | NICOTINE-L (BASE) | Nicotine-D sa...)
Affinity DataKi:  1.5nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
University Of California San Diego

Curated by ChEMBL
LigandPNGBDBM50065353((S)-2-Amino-N-((6S,12R)-6-benzyl-1-methyl-5,8,11-t...)
Affinity DataKi:  1.60nMAssay Description:In vitro potency was measured against human Opioid receptor mu 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50117261(12-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-6...)
Affinity DataKi:  2nMAssay Description:Inhibition of binding of [3H]-diprenorphine to cloned human Opioid receptor delta 1 expressed in CHO cell membrane;Range is between (1.7-2.3)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
University Of California San Diego

Curated by ChEMBL
LigandPNGBDBM50117261(12-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-6...)
Affinity DataKi:  2nMAssay Description:Inhibition of binding of [3H]-diprenorphine to cloned human Opioid receptor mu 1 expressed in CHO cell membrane;Range is in between (1.8-2.2)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50065353((S)-2-Amino-N-((6S,12R)-6-benzyl-1-methyl-5,8,11-t...)
Affinity DataKi:  2.10nMAssay Description:In vitro potency was measured against human Opioid receptor delta 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50001683(13-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-7...)
Affinity DataKi:  2.20nMAssay Description:Inhibition of binding of [3H]diprenorphine to cloned human Opioid receptor delta 1 expressed in CHO cell membrane;Range is between (1-3.9)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50001683(13-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-7...)
Affinity DataKi:  2.20nMAssay Description:In vitro potency was measured against human Opioid receptor delta 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
University Of California San Diego

Curated by ChEMBL
LigandPNGBDBM50117263((3R,6S,12S)-12-[(S)-2-Amino-3-(4-hydroxy-phenyl)-p...)
Affinity DataKi:  2.30nMAssay Description:Inhibition of binding of [3H]-diprenorphine to cloned human Opioid receptor mu 1 expressed in CHO cell membrane;Range is in between (1.3-3.7)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNicotinic acetylcholine receptor(RAT)
University Of California

Curated by PDSP Ki Database
LigandPNGBDBM82070(CAS_29790-52-1 | NICOTINE-L (BASE) | Nicotine-D sa...)
Affinity DataKi:  2.31nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetNicotinic acetylcholine receptor(RAT)
University Of California

Curated by PDSP Ki Database
LigandPNGBDBM82546(CAS_14721-69-8 | MCC | N-methylcarbamylcholine | N...)
Affinity DataKi:  5.20nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetNicotinic acetylcholine receptor(RAT)
University Of California

Curated by PDSP Ki Database
LigandPNGBDBM50061562((12R,13aR)-12-Methoxy-1,4,5,6,9,11,12,13-octahydro...)
Affinity DataKi:  6.60nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetNicotinic acetylcholine receptor(RAT)
University Of California

Curated by PDSP Ki Database
LigandPNGBDBM50054820(Methyllycaconitine | [(1S,4S,5R,6S,8R,9R,13S,16S,1...)
Affinity DataKi:  8.90nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
University Of California San Diego

Curated by ChEMBL
LigandPNGBDBM21015((2S)-2-{2-[(2R)-2-[(2S)-2-amino-3-(4-hydroxyphenyl...)
Affinity DataKi:  14nMAssay Description:In vitro potency was measured against human Opioid receptor mu 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNicotinic acetylcholine receptor(RAT)
University Of California

Curated by PDSP Ki Database
LigandPNGBDBM50047021(2-(6-(2-hydroxy-2-phenylethyl)-1-methylpiperidin-2...)
Affinity DataKi:  15.5nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
University Of California San Diego

Curated by ChEMBL
LigandPNGBDBM50000092((-)-(etorphine) | (-)-morphine | (1S,5R,13R,14S)-1...)
Affinity DataKi:  17nMAssay Description:Inhibition of binding of [3H]-diprenorphine to cloned human Opioid receptor mu 1 expressed in CHO cell membrane;Range is in between (6.8-43)More data for this Ligand-Target Pair
TargetMu-type opioid receptor(Homo sapiens (Human))
University Of California San Diego

Curated by ChEMBL
LigandPNGBDBM50000092((-)-(etorphine) | (-)-morphine | (1S,5R,13R,14S)-1...)
Affinity DataKi:  17nMAssay Description:In vitro potency was measured against human Opioid receptor mu 1More data for this Ligand-Target Pair
TargetNicotinic acetylcholine receptor(RAT)
University Of California

Curated by PDSP Ki Database
LigandPNGBDBM50061562((12R,13aR)-12-Methoxy-1,4,5,6,9,11,12,13-octahydro...)
Affinity DataKi:  28nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetNicotinic acetylcholine receptor(RAT)
University Of California

Curated by PDSP Ki Database
LigandPNGBDBM50061567(1,1-Dimethyl-4-phenyl-piperazin-1-ium | CHEMBL1347...)
Affinity DataKi:  28.8nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetNicotinic acetylcholine receptor(RAT)
University Of California

Curated by PDSP Ki Database
LigandPNGBDBM82068(CHEMBL9732 | Nicotine-D salicylate | Nicotine-L sa...)
Affinity DataKi:  35nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
University Of California San Diego

Curated by ChEMBL
LigandPNGBDBM50117262(12-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-6...)
Affinity DataKi:  130nMAssay Description:Inhibition of binding of [3H]-diprenorphine to cloned human Opioid receptor mu 1 expressed in CHO cell membrane;Range is in between (110-150)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNicotinic acetylcholine receptor(RAT)
University Of California

Curated by PDSP Ki Database
LigandPNGBDBM82068(CHEMBL9732 | Nicotine-D salicylate | Nicotine-L sa...)
Affinity DataKi:  145nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50000092((-)-(etorphine) | (-)-morphine | (1S,5R,13R,14S)-1...)
Affinity DataKi:  150nMAssay Description:In vitro potency was measured against human Opioid receptor delta 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetDelta-type opioid receptor(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50000092((-)-(etorphine) | (-)-morphine | (1S,5R,13R,14S)-1...)
Affinity DataKi:  150nMAssay Description:Inhibition of binding of [3H]-diprenorphine to cloned human Opioid receptor delta 1 expressed in CHO cell membrane;Range is between (63-360)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetKappa-type opioid receptor(Homo sapiens (Human))
University Of California San Diego

Curated by ChEMBL
LigandPNGBDBM50000092((-)-(etorphine) | (-)-morphine | (1S,5R,13R,14S)-1...)
Affinity DataKi:  260nMAssay Description:In vitro potency was measured against human Opioid receptor kappa 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetKappa-type opioid receptor(Homo sapiens (Human))
University Of California San Diego

Curated by ChEMBL
LigandPNGBDBM50000092((-)-(etorphine) | (-)-morphine | (1S,5R,13R,14S)-1...)
Affinity DataKi:  260nMAssay Description:Inhibition of binding of [3H]diprenorphine to cloned human Opioid receptor kappa 1 expressed in CHO cell membrane;Range is in between (1400-1900)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetNicotinic acetylcholine receptor(RAT)
University Of California

Curated by PDSP Ki Database
LigandPNGBDBM50054820(Methyllycaconitine | [(1S,4S,5R,6S,8R,9R,13S,16S,1...)
Affinity DataKi:  261nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetNicotinic acetylcholine receptor(RAT)
University Of California

Curated by PDSP Ki Database
LigandPNGBDBM50000690(10,25-dimethoxy-15,15,30-trimethyl-(1S,16R)-7,23-d...)
Affinity DataKi:  282nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetNicotinic acetylcholine receptor(RAT)
University Of California

Curated by PDSP Ki Database
LigandPNGBDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
Affinity DataKi:  325nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
University Of California San Diego

Curated by ChEMBL
LigandPNGBDBM50065353((S)-2-Amino-N-((6S,12R)-6-benzyl-1-methyl-5,8,11-t...)
Affinity DataKi:  340nMAssay Description:In vitro potency was measured against human Opioid receptor kappa 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
University Of California San Diego

Curated by ChEMBL
LigandPNGBDBM50117264(12-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-6...)
Affinity DataKi:  630nMAssay Description:Inhibition of binding of [3H]-diprenorphine to cloned human Opioid receptor mu 1 expressed in CHO cell membrane;Range is in between (580-680)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNicotinic acetylcholine receptor(RAT)
University Of California

Curated by PDSP Ki Database
LigandPNGBDBM50061565((+)Methyl-(2,3,3-trimethyl-bicyclo[2.2.1]hept-2-yl...)
Affinity DataKi:  1.00E+3nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
University Of California San Diego

Curated by ChEMBL
LigandPNGBDBM50117262(12-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-6...)
Affinity DataKi: >1.00E+3nMAssay Description:Inhibition of binding of [3H]diprenorphine to cloned human Opioid receptor kappa 1 expressed in CHO cell membrane;Range is in between (1400-1900)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNicotinic acetylcholine receptor(RAT)
University Of California

Curated by PDSP Ki Database
LigandPNGBDBM50000690(10,25-dimethoxy-15,15,30-trimethyl-(1S,16R)-7,23-d...)
Affinity DataKi:  1.00E+3nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetNicotinic acetylcholine receptor(RAT)
University Of California

Curated by PDSP Ki Database
LigandPNGBDBM50121739(Bungarotoxin Neuronal | Bungarotoxin,Alpha | CHEMB...)
Affinity DataKi:  1.00E+3nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
University Of California San Diego

Curated by ChEMBL
LigandPNGBDBM50117261(12-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-6...)
Affinity DataKi:  1.60E+3nMAssay Description:Inhibition of binding of [3H]-diprenorphine to cloned human Opioid receptor kappa 1 expressed in CHO cell membrane;Range is in between (1400-1900)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
University Of California San Diego

Curated by ChEMBL
LigandPNGBDBM50117263((3R,6S,12S)-12-[(S)-2-Amino-3-(4-hydroxy-phenyl)-p...)
Affinity DataKi:  6.40E+3nMAssay Description:Inhibition of binding of [3H]-diprenorphine to cloned human Opioid receptor kappa 1 expressed in CHO cell membrane; range is in between (4700-8500)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNicotinic acetylcholine receptor(RAT)
University Of California

Curated by PDSP Ki Database
LigandPNGBDBM82544(Alpha-Cobratoxin | CAS_69344-74-7 | COBRATOXIN)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetNicotinic acetylcholine receptor(RAT)
University Of California

Curated by PDSP Ki Database
LigandPNGBDBM50121739(Bungarotoxin Neuronal | Bungarotoxin,Alpha | CHEMB...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetNicotinic acetylcholine receptor(RAT)
University Of California

Curated by PDSP Ki Database
LigandPNGBDBM50121739(Bungarotoxin Neuronal | Bungarotoxin,Alpha | CHEMB...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetNicotinic acetylcholine receptor(RAT)
University Of California

Curated by PDSP Ki Database
LigandPNGBDBM50038416((1,6-trimethyl ammonium)hexane; dibromide | CHEMBL...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetNicotinic acetylcholine receptor(RAT)
University Of California

Curated by PDSP Ki Database
LigandPNGBDBM82545(CAS_441310 | NSC_441310 | Trimethaphan)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM21015((2S)-2-{2-[(2R)-2-[(2S)-2-amino-3-(4-hydroxyphenyl...)
Affinity DataKi: >1.00E+4nMAssay Description:In vitro potency was measured against human Opioid receptor delta 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
University Of California San Diego

Curated by ChEMBL
LigandPNGBDBM50001683(13-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-7...)
Affinity DataKi: >1.00E+4nMAssay Description:In vitro potency was measured against human Opioid receptor kappa 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
University Of California San Diego

Curated by ChEMBL
LigandPNGBDBM50001683(13-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-7...)
Affinity DataKi: >1.00E+4nMAssay Description:In vitro potency was measured against human Opioid receptor mu 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
University Of California San Diego

Curated by ChEMBL
LigandPNGBDBM50001683(13-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-7...)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of binding of [3H]diprenorphine to cloned human Opioid receptor mu 1 expressed in CHO cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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