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Found 120 with Last Name = 'yang' and Initial = 'jl'
TargetTGF-beta receptor type-1(Homo sapiens (Human))
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50151347(2-(3-(6-methylpyridin-2-yl)-1H-pyrazol-4-yl)-1,5-n...)
Affinity DataIC50:  4nMAssay Description:Inhibition of TGFR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTGF-beta receptor type-1(Homo sapiens (Human))
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50301158(4-(3-methylpyridin-2-yl)-5-(1,5-naphthyridin-2-yl)...)
Affinity DataIC50:  6nMAssay Description:Inhibition of TGFR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTGF-beta receptor type-1(Homo sapiens (Human))
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50214864(3-((5-(6-methylpyridin-2-yl)-4-(quinoxalin-6-yl)-1...)
Affinity DataIC50:  10nMAssay Description:Inhibition of TGFR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTGF-beta receptor type-1(Homo sapiens (Human))
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50151353(4-(4-Fluoro-phenyl)-5-[1,5]naphthyridin-2-yl-thiaz...)
Affinity DataIC50:  11nMAssay Description:Inhibition of TGFR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTGF-beta receptor type-1(Homo sapiens (Human))
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50151363(4-(3-Chloro-phenyl)-5-[1,5]naphthyridin-2-yl-thiaz...)
Affinity DataIC50:  13nMAssay Description:Inhibition of TGFR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTGF-beta receptor type-1(Homo sapiens (Human))
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50301167(CHEMBL567706 | N,N-dimethyl-3-(3-(4-(3-(pyridin-2-...)
Affinity DataIC50:  15nMAssay Description:Inhibition of TGFR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTGF-beta receptor type-1(Homo sapiens (Human))
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50301159(1-(2-(dimethylamino)ethyl)-3-(4-(2-(pyridin-2-yl)-...)
Affinity DataIC50:  18nMAssay Description:Inhibition of TGFR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTGF-beta receptor type-1(Homo sapiens (Human))
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50184872(4-(4-(3-(pyridin-2-yl)-1H-pyrazol-4-yl)pyridin-2-y...)
Affinity DataIC50:  18nMAssay Description:Inhibition of TGFR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTGF-beta receptor type-1(Homo sapiens (Human))
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50151357(2-(3-(pyridin-2-yl)-1H-pyrazol-4-yl)-1,5-naphthyri...)
Affinity DataIC50:  19nMAssay Description:Inhibition of TGFR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTGF-beta receptor type-1(Homo sapiens (Human))
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50151346(5-(1,5-naphthyridin-2-yl)-4-(pyridin-2-yl)thiazol-...)
Affinity DataIC50:  20nMAssay Description:Inhibition of TGFR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTGF-beta receptor type-1(Homo sapiens (Human))
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50301168(4-((4-(3a,4-dihydrobenzo[d][1,3]dioxol-5-yl)-5-(6-...)
Affinity DataIC50:  21nMAssay Description:Inhibition of TGFR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTGF-beta receptor type-1(Homo sapiens (Human))
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50301160(4-((4-(3a,4-dihydrobenzo[d][1,3]dioxol-5-yl)-5-(6-...)
Affinity DataIC50:  24nMAssay Description:Inhibition of TGFR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTGF-beta receptor type-1(Homo sapiens (Human))
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50184886(2-[4-(trifluoromethyl)phenyl]-4-(3-pyridin-2-yl-1H...)
Affinity DataIC50:  24nMAssay Description:Inhibition of TGFR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTGF-beta receptor type-1(Homo sapiens (Human))
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50301169(4-(4-(2-isopropyl-4-(6-methylpyridin-2-yl)-1H-imid...)
Affinity DataIC50:  25nMAssay Description:Inhibition of TGFR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTGF-beta receptor type-1(Homo sapiens (Human))
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50184880(1-(4-(4-(3-(pyridin-2-yl)-1H-pyrazol-4-yl)pyridin-...)
Affinity DataIC50:  25nMAssay Description:Inhibition of TGFR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTGF-beta receptor type-1(Homo sapiens (Human))
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50301170(4-(4-(3-(pyridin-2-yl)-1H-pyrazol-4-yl)pyridin-2-y...)
Affinity DataIC50:  27nMAssay Description:Inhibition of TGFR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTGF-beta receptor type-1(Homo sapiens (Human))
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50184896(2-(4-(2-(1H-imidazol-1-yl)ethoxy)phenyl)-4-(3-(pyr...)
Affinity DataIC50:  30nMAssay Description:Inhibition of TGFR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTGF-beta receptor type-1(Homo sapiens (Human))
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50301171(5-(8-methylquinolin-2-yl)-4-(pyridin-2-yl)thiazol-...)
Affinity DataIC50:  30nMAssay Description:Inhibition of TGFR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTGF-beta receptor type-1(Homo sapiens (Human))
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50132992(4-(3-(6-methylpyridin-2-yl)-1H-pyrazol-4-yl)phenol...)
Affinity DataIC50:  31nMAssay Description:Inhibition of TGFR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTGF-beta receptor type-1(Homo sapiens (Human))
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50301172(3-hydroxy-N-(4-(2-(pyridin-2-yl)-5,6-dihydro-4H-py...)
Affinity DataIC50:  32nMAssay Description:Inhibition of TGFR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTGF-beta receptor type-1(Homo sapiens (Human))
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50301173(3-methoxy-N-(4-(2-(pyridin-2-yl)-5,6-dihydro-4H-py...)
Affinity DataIC50:  34nMAssay Description:Inhibition of TGFR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTGF-beta receptor type-1(Homo sapiens (Human))
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50184873(2-[4-cyanophenyl]-4-(3-pyridin-2-yl-1H-pyrazol-4-y...)
Affinity DataIC50:  35nMAssay Description:Inhibition of TGFR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTGF-beta receptor type-1(Homo sapiens (Human))
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50184874(2-[4-(2-pyrrolidin-1-ylethoxy)phenyl]-4-(3-pyridin...)
Affinity DataIC50:  40nMAssay Description:Inhibition of TGFR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTGF-beta receptor type-1(Homo sapiens (Human))
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50301174(CHEMBL584928 | methyl 4-(2-(pyridin-2-yl)-5,6-dihy...)
Affinity DataIC50:  40nMAssay Description:Inhibition of TGFR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTGF-beta receptor type-1(Homo sapiens (Human))
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50184489(3-(6-(2-(6-methylpyridin-2-yl)-5,6-dihydro-4H-pyrr...)
Affinity DataIC50:  41nMAssay Description:Inhibition of TGFR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTGF-beta receptor type-1(Homo sapiens (Human))
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50184877(4-(4-(4-(3-(pyridin-2-yl)-1H-pyrazol-4-yl)pyridin-...)
Affinity DataIC50:  42nMAssay Description:Inhibition of TGFR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTGF-beta receptor type-1(Homo sapiens (Human))
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50184900(2-(4-chlorophenyl)-4-(3-(pyridin-2-yl)-1H-pyrazol-...)
Affinity DataIC50:  43nMAssay Description:Inhibition of TGFR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTGF-beta receptor type-1(Homo sapiens (Human))
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50301176(4-((4-(3a,4-dihydrobenzo[d][1,3]dioxol-5-yl)-5-(6-...)
Affinity DataIC50:  46nMAssay Description:Inhibition of TGFR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTGF-beta receptor type-1(Homo sapiens (Human))
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50301175(4-((4-(3a,4-dihydrobenzo[d][1,3]dioxol-5-yl)-5-(6-...)
Affinity DataIC50:  46nMAssay Description:Inhibition of TGFR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTGF-beta receptor type-1(Homo sapiens (Human))
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50301177(CHEMBL566234 | N-(4-(4-(3-(pyridin-2-yl)-1H-pyrazo...)
Affinity DataIC50:  47nMAssay Description:Inhibition of TGFR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTGF-beta receptor type-1(Homo sapiens (Human))
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50148668(4-(2-(6-methylpyridin-2-yl)-5,6-dihydro-4H-pyrrolo...)
Affinity DataIC50:  47nMAssay Description:Inhibition of TGFR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTGF-beta receptor type-1(Homo sapiens (Human))
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50301178(4-((5-(6-ethylpyridin-2-yl)-4-(1,4,4a,8a-tetrahydr...)
Affinity DataIC50:  47nMAssay Description:Inhibition of TGFR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTGF-beta receptor type-1(Homo sapiens (Human))
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50184901(2-(4-fluorophenyl)-4-(3-(pyridin-2-yl)-1H-pyrazol-...)
Affinity DataIC50:  48nMAssay Description:Inhibition of TGFR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTGF-beta receptor type-1(Homo sapiens (Human))
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50148666(7-Chloro-4-[2-(6-methyl-pyridin-2-yl)-5,6-dihydro-...)
Affinity DataIC50:  48nMAssay Description:Inhibition of TGFR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTGF-beta receptor type-1(Homo sapiens (Human))
Sichuan University

Curated by ChEMBL
LigandPNGBDBM21492(4-[3-(pyridin-2-yl)-1H-pyrazol-4-yl]quinoline | CH...)
Affinity DataIC50:  51nMAssay Description:Inhibition of TGFR1More data for this Ligand-Target Pair
TargetTGF-beta receptor type-1(Homo sapiens (Human))
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50148655(7-Chloro-4-(2-pyridin-2-yl-5,6-dihydro-4H-pyrrolo[...)
Affinity DataIC50:  54nMAssay Description:Inhibition of TGFR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTGF-beta receptor type-1(Homo sapiens (Human))
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50301179(4-(2-(pyridin-2-yl)-5,6-dihydro-4H-pyrrolo[1,2-b]p...)
Affinity DataIC50:  59nMAssay Description:Inhibition of TGFR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTGF-beta receptor type-1(Homo sapiens (Human))
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50184883(2-(2-fluorophenyl)-4-(3-(pyridin-2-yl)-1H-pyrazol-...)
Affinity DataIC50:  59nMAssay Description:Inhibition of TGFR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTGF-beta receptor type-1(Homo sapiens (Human))
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50301180(2-(dimethylamino)-N-(4-(2-(pyridin-2-yl)-5,6-dihyd...)
Affinity DataIC50:  64nMAssay Description:Inhibition of TGFR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTGF-beta receptor type-1(Homo sapiens (Human))
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50184487(4-(3-(6-(2-(6-methylpyridin-2-yl)-5,6-dihydro-4H-p...)
Affinity DataIC50:  69nMAssay Description:Inhibition of TGFR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTGF-beta receptor type-1(Homo sapiens (Human))
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50148656(4-(2-(6-ethylpyridin-2-yl)-5,6-dihydro-4H-pyrrolo[...)
Affinity DataIC50:  71nMAssay Description:Inhibition of TGFR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTGF-beta receptor type-1(Homo sapiens (Human))
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50301181(3-((4-(3a,4-dihydrobenzo[d][1,3]dioxol-5-yl)-5-(6-...)
Affinity DataIC50:  73nMAssay Description:Inhibition of TGFR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTGF-beta receptor type-1(Homo sapiens (Human))
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50301182(4-((5-(6-methylpyridin-2-yl)-4-(1,4,4a,8a-tetrahyd...)
Affinity DataIC50:  75nMAssay Description:Inhibition of TGFR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTGF-beta receptor type-1(Homo sapiens (Human))
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50148661(4-(2-(6-methylpyridin-2-yl)-5,6-dihydro-4H-pyrrolo...)
Affinity DataIC50:  78nMAssay Description:Inhibition of TGFR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTGF-beta receptor type-1(Homo sapiens (Human))
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50301183(2-hydroxyethyl 4-(2-(pyridin-2-yl)-5,6-dihydro-4H-...)
Affinity DataIC50:  79nMAssay Description:Inhibition of TGFR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTGF-beta receptor type-1(Homo sapiens (Human))
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50184898(2-(4-(2-cyclohexylethoxy)phenyl)-4-(3-(pyridin-2-y...)
Affinity DataIC50:  81nMAssay Description:Inhibition of TGFR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTGF-beta receptor type-1(Homo sapiens (Human))
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50301184(CHEMBL565815 | N-(4-(2-(pyridin-2-yl)-5,6-dihydro-...)
Affinity DataIC50:  87nMAssay Description:Inhibition of TGFR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTGF-beta receptor type-1(Homo sapiens (Human))
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50148657(7-Ethoxy-4-[2-(6-methyl-pyridin-2-yl)-5,6-dihydro-...)
Affinity DataIC50:  88nMAssay Description:Inhibition of TGFR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTGF-beta receptor type-1(Homo sapiens (Human))
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50132980(4-(3-(5-fluoropyridin-2-yl)-1H-pyrazol-4-yl)quinol...)
Affinity DataIC50:  91nMAssay Description:Inhibition of TGFR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTGF-beta receptor type-1(Homo sapiens (Human))
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50184884(CHEMBL205151 | N-(2-methoxyethyl)-4-(4-(3-(pyridin...)
Affinity DataIC50:  91nMAssay Description:Inhibition of TGFR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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