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Found 262 with Last Name = 'yun' and Initial = 'm'
TargetProthrombin(Homo sapiens (Human))
Biotech Research Institute

Curated by ChEMBL
LigandPNGBDBM50069294((S)-3-[4-(carbohydrazonamidol)-phenyl]-N-cyclopent...)
Affinity DataKi:  0.380nMAssay Description:Compound was evaluated for its inhibitory activity against human thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Biotech Research Institute

Curated by ChEMBL
LigandPNGBDBM50069294((S)-3-[4-(carbohydrazonamidol)-phenyl]-N-cyclopent...)
Affinity DataKi:  0.380nMAssay Description:Compound was tested for inhibitory activity against human thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Biotech Research Institute

Curated by ChEMBL
LigandPNGBDBM50070780((S)-3-(5-Carbamimidoyl-thiophen-2-yl)-N-cyclopenty...)
Affinity DataKi:  0.490nMAssay Description:Compound was evaluated for its inhibitory activity against human thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Biotech Research Institute

Curated by ChEMBL
LigandPNGBDBM50070785((S)-3-(5-Carbamimidoyl-thiophen-2-yl)-N-cyclopenty...)
Affinity DataKi:  0.600nMAssay Description:Compound was evaluated for its inhibitory activity against human thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Biotech Research Institute

Curated by ChEMBL
LigandPNGBDBM50070782((S)-3-(4-Carbamimidoyl-phenyl)-N-cyclopentyl-N-met...)
Affinity DataKi:  0.840nMAssay Description:Compound was evaluated for its inhibitory activity against human thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Bos taurus (Bovine))
TBA

Curated by ChEMBL
LigandPNGBDBM50291355(1-[3-[4-amino(amineimino)methylphenyl]-2-(2-anthry...)
Affinity DataKi:  1nMAssay Description:Inhibitory effect against bovine thrombinMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProthrombin(Bos taurus (Bovine))
TBA

Curated by ChEMBL
LigandPNGBDBM50069294((S)-3-[4-(carbohydrazonamidol)-phenyl]-N-cyclopent...)
Affinity DataKi:  1.10nMAssay Description:Compound was tested for inhibitory activity against bovine thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Bos taurus (Bovine))
TBA

Curated by ChEMBL
LigandPNGBDBM50069297(1-[3-[4-amino(amineimino)methylphenyl]-2-(2-naphth...)
Affinity DataKi:  1.5nMAssay Description:Inhibitory effect against bovine thrombinMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProthrombin(Homo sapiens (Human))
Biotech Research Institute

Curated by ChEMBL
LigandPNGBDBM50070784((S)-3-(5-Carbamimidoyl-thiophen-2-yl)-N-cyclopenty...)
Affinity DataKi:  3nMAssay Description:Compound was evaluated for its inhibitory activity against human thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Bos taurus (Bovine))
TBA

Curated by ChEMBL
LigandPNGBDBM50069292(CHEMBL156082 | N-ethyl-N-cyclopentyl-3-(4-hydrazon...)
Affinity DataKi:  4nMAssay Description:Compound was tested for inhibitory activity against bovine thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Bos taurus (Bovine))
TBA

Curated by ChEMBL
LigandPNGBDBM50037996(1-[N-(naphthalen-2-ylsulfonyl)glycyl-4-carbamimido...)
Affinity DataKi:  6.5nMAssay Description:Inhibitory effect against bovine thrombinMore data for this Ligand-Target Pair
TargetProthrombin(Homo sapiens (Human))
Biotech Research Institute

Curated by ChEMBL
LigandPNGBDBM50070783((S)-3-(4-Carbamimidoyl-phenyl)-N-cyclopentyl-N-met...)
Affinity DataKi:  6.80nMAssay Description:Compound was evaluated for its inhibitory activity against human thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Bos taurus (Bovine))
TBA

Curated by ChEMBL
LigandPNGBDBM50291363(CHEMBL354307 | N-[(R)-2-Azepan-1-yl-1-(4-carbamimi...)
Affinity DataKi:  20nMAssay Description:Inhibitory effect against bovine thrombinMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProthrombin(Bos taurus (Bovine))
TBA

Curated by ChEMBL
LigandPNGBDBM50069293(CHEMBL440188 | N-methyl-N-n-butyl-3-(4-hydrazonofo...)
Affinity DataKi:  41nMAssay Description:Compound was tested for inhibitory activity against bovine thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Bos taurus (Bovine))
TBA

Curated by ChEMBL
LigandPNGBDBM50291361(4-[(S)-3-Azepan-1-yl-2-(naphthalene-2-sulfonylamin...)
Affinity DataKi:  46nMAssay Description:Inhibitory effect against bovine thrombinMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProthrombin(Bos taurus (Bovine))
TBA

Curated by ChEMBL
LigandPNGBDBM50291357(4-[(S)-2-(Anthracene-2-sulfonylamino)-3-azepan-1-y...)
Affinity DataKi:  50nMAssay Description:Inhibitory effect against bovine thrombinMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProthrombin(Bos taurus (Bovine))
TBA

Curated by ChEMBL
LigandPNGBDBM50291358(4-[(S)-3-Azepan-1-yl-2-(naphthalene-2-sulfonylamin...)
Affinity DataKi:  52nMAssay Description:Inhibitory effect against bovine thrombinMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProthrombin(Homo sapiens (Human))
Biotech Research Institute

Curated by ChEMBL
LigandPNGBDBM50070781(1N-cyclopentyl-1N-methyl-3-[5-amino(aminoimino)met...)
Affinity DataKi:  91nMAssay Description:Compound was evaluated for its inhibitory activity against human thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Bos taurus (Bovine))
TBA

Curated by ChEMBL
LigandPNGBDBM50069296(CHEMBL347371 | N-(n-propyl)-N-cyclopentyl-3-(4-hyd...)
Affinity DataKi:  93nMAssay Description:Compound was tested for inhibitory activity against bovine thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Bos taurus (bovine))
Biotech Research Institute

Curated by ChEMBL
LigandPNGBDBM50070780((S)-3-(5-Carbamimidoyl-thiophen-2-yl)-N-cyclopenty...)
Affinity DataKi:  134nMAssay Description:Compound was evaluated for its inhibitory activity against bovine trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Bos taurus (bovine))
Biotech Research Institute

Curated by ChEMBL
LigandPNGBDBM50070785((S)-3-(5-Carbamimidoyl-thiophen-2-yl)-N-cyclopenty...)
Affinity DataKi:  150nMAssay Description:Compound was evaluated for its inhibitory activity against bovine trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Bos taurus (Bovine))
TBA

Curated by ChEMBL
LigandPNGBDBM50069298(CHEMBL434678 | N-methyl-N-cyclohexyl-3-(4-hydrazon...)
Affinity DataKi:  152nMAssay Description:Compound was tested for inhibitory activity against bovine thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Bos taurus (bovine))
Biotech Research Institute

Curated by ChEMBL
LigandPNGBDBM50070784((S)-3-(5-Carbamimidoyl-thiophen-2-yl)-N-cyclopenty...)
Affinity DataKi:  153nMAssay Description:Compound was evaluated for its inhibitory activity against bovine trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Bos taurus (Bovine))
TBA

Curated by ChEMBL
LigandPNGBDBM50069299(CHEMBL155317 | N-(n-butyl)-N-cyclopentyl-3-(4-hydr...)
Affinity DataKi:  231nMAssay Description:Compound was tested for inhibitory activity against bovine thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Bos taurus (Bovine))
TBA

Curated by ChEMBL
LigandPNGBDBM50069295(CHEMBL348175 | N-methyl-N-cyclopropyl-3-(4-hydrazo...)
Affinity DataKi:  247nMAssay Description:Compound was tested for inhibitory activity against bovine thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Bos taurus (bovine))
Biotech Research Institute

Curated by ChEMBL
LigandPNGBDBM50037996(1-[N-(naphthalen-2-ylsulfonyl)glycyl-4-carbamimido...)
Affinity DataKi:  325nMAssay Description:Inhibitory effect of compound was measured in bovine trypsinMore data for this Ligand-Target Pair
TargetProthrombin(Bos taurus (Bovine))
TBA

Curated by ChEMBL
LigandPNGBDBM50069300(CHEMBL350901 | N-hydroxy-N-cyclopentyl-3-(4-hydraz...)
Affinity DataKi:  367nMAssay Description:Compound was tested for inhibitory activity against bovine thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Biotech Research Institute

Curated by ChEMBL
LigandPNGBDBM50069294((S)-3-[4-(carbohydrazonamidol)-phenyl]-N-cyclopent...)
Affinity DataKi:  1.10E+3nMAssay Description:The compound was tested for inhibitory activity against Coagulation factor XMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Bos taurus (Bovine))
TBA

Curated by ChEMBL
LigandPNGBDBM50291359(4-[(S)-3-Azepan-1-yl-2-(naphthalene-2-sulfonylamin...)
Affinity DataKi:  1.14E+3nMAssay Description:Inhibitory effect against bovine thrombinMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProthrombin(Bos taurus (Bovine))
TBA

Curated by ChEMBL
LigandPNGBDBM50069297(1-[3-[4-amino(amineimino)methylphenyl]-2-(2-naphth...)
Affinity DataKi:  1.47E+3nMAssay Description:Compound was tested for inhibitory activity against bovine thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Bos taurus (bovine))
Biotech Research Institute

Curated by ChEMBL
LigandPNGBDBM50070782((S)-3-(4-Carbamimidoyl-phenyl)-N-cyclopentyl-N-met...)
Affinity DataKi:  2.44E+3nMAssay Description:Compound was evaluated for its inhibitory activity against bovine trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Bos taurus (Bovine))
TBA

Curated by ChEMBL
LigandPNGBDBM50291362(1N-[1-[4-amino(aminoimino)methylbenzyl]-2-(1-azepa...)
Affinity DataKi:  2.70E+3nMAssay Description:Inhibitory effect against bovine thrombinMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSerine protease 1(Bos taurus (bovine))
Biotech Research Institute

Curated by ChEMBL
LigandPNGBDBM50069294((S)-3-[4-(carbohydrazonamidol)-phenyl]-N-cyclopent...)
Affinity DataKi:  3.20E+3nMAssay Description:Compound was evaluated for its inhibitory activity against bovine trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrypsin(Homo sapiens (Human))
Biotech Research Institute

Curated by ChEMBL
LigandPNGBDBM50069294((S)-3-[4-(carbohydrazonamidol)-phenyl]-N-cyclopent...)
Affinity DataKi:  3.29E+3nMAssay Description:Compound was tested for inhibitory activity against bovine trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Bos taurus (bovine))
Biotech Research Institute

Curated by ChEMBL
LigandPNGBDBM50069297(1-[3-[4-amino(amineimino)methylphenyl]-2-(2-naphth...)
Affinity DataKi:  3.73E+3nMAssay Description:Inhibitory effect of compound was measured in bovine trypsinMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProthrombin(Bos taurus (Bovine))
TBA

Curated by ChEMBL
LigandPNGBDBM50291364(CHEMBL424164 | N-{(R)-1-[4-(N-Methylcarbamimidoyl)...)
Affinity DataKi:  4.32E+3nMAssay Description:Inhibitory effect against bovine thrombinMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProthrombin(Bos taurus (Bovine))
TBA

Curated by ChEMBL
LigandPNGBDBM50291360(1N-[1-[4-amino(amineimino)methylbenzyl]-2-hexahydr...)
Affinity DataKi:  5.37E+3nMAssay Description:Inhibitory effect against bovine thrombinMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProthrombin(Bos taurus (Bovine))
TBA

Curated by ChEMBL
LigandPNGBDBM50069301(CHEMBL155311 | N-hydroxyethyl-N-cyclopentyl-3-(4-h...)
Affinity DataKi:  7.04E+3nMAssay Description:Compound was tested for inhibitory activity against bovine thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Bos taurus (bovine))
Biotech Research Institute

Curated by ChEMBL
LigandPNGBDBM50291358(4-[(S)-3-Azepan-1-yl-2-(naphthalene-2-sulfonylamin...)
Affinity DataKi:  8.65E+3nMAssay Description:Inhibitory effect of compound was measured in bovine trypsinMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProthrombin(Bos taurus (Bovine))
TBA

Curated by ChEMBL
LigandPNGBDBM50291356(4-[(S)-3-Azepan-1-yl-2-(naphthalene-2-sulfonylamin...)
Affinity DataKi:  1.36E+4nMAssay Description:Inhibitory effect against bovine thrombinMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSerine protease 1(Bos taurus (bovine))
Biotech Research Institute

Curated by ChEMBL
LigandPNGBDBM50070783((S)-3-(4-Carbamimidoyl-phenyl)-N-cyclopentyl-N-met...)
Affinity DataKi:  1.62E+4nMAssay Description:Compound was evaluated for its inhibitory activity against bovine trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTissue-type plasminogen activator(Homo sapiens (Human))
Biotech Research Institute

Curated by ChEMBL
LigandPNGBDBM50069294((S)-3-[4-(carbohydrazonamidol)-phenyl]-N-cyclopent...)
Affinity DataKi:  2.72E+4nMAssay Description:The compound was tested for inhibitory activity against tissue plasminogen activatorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen(Homo sapiens (Human))
Biotech Research Institute

Curated by ChEMBL
LigandPNGBDBM50069294((S)-3-[4-(carbohydrazonamidol)-phenyl]-N-cyclopent...)
Affinity DataKi:  4.79E+4nMAssay Description:The compound was tested for inhibitory activity against human plasminMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Bos taurus (bovine))
Biotech Research Institute

Curated by ChEMBL
LigandPNGBDBM50291364(CHEMBL424164 | N-{(R)-1-[4-(N-Methylcarbamimidoyl)...)
Affinity DataKi:  8.15E+4nMAssay Description:Inhibitory effect of compound was measured in bovine trypsinMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSerine protease 1(Bos taurus (bovine))
Biotech Research Institute

Curated by ChEMBL
LigandPNGBDBM50291360(1N-[1-[4-amino(amineimino)methylbenzyl]-2-hexahydr...)
Affinity DataKi:  1.92E+5nMAssay Description:Inhibitory effect of compound was measured in bovine trypsinMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSerine protease 1(Bos taurus (bovine))
Biotech Research Institute

Curated by ChEMBL
LigandPNGBDBM50291359(4-[(S)-3-Azepan-1-yl-2-(naphthalene-2-sulfonylamin...)
Affinity DataKi:  3.16E+5nMAssay Description:Inhibitory effect of compound was measured in bovine trypsinMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSerine protease 1(Bos taurus (bovine))
Biotech Research Institute

Curated by ChEMBL
LigandPNGBDBM50291361(4-[(S)-3-Azepan-1-yl-2-(naphthalene-2-sulfonylamin...)
Affinity DataKi:  5.45E+5nMAssay Description:Inhibitory effect of compound was measured in bovine trypsinMore data for this Ligand-Target Pair
In DepthDetails Article
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Korea Institute Of Science And Technology (Kaist)

Curated by ChEMBL
LigandPNGBDBM50490888(CHEMBL2347725)
Affinity DataIC50:  0.0150nMAssay Description:Inhibition of breakpoint cluster region-Abelson tyrosine kinase T315I mutant (unknown origin) using [gamma-33P]ATP as substrate by radiometric kinase...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Korea Institute Of Science And Technology (Kaist)

Curated by ChEMBL
LigandPNGBDBM50490916(CHEMBL2347722)
Affinity DataIC50:  0.0210nMAssay Description:Inhibition of breakpoint cluster region-Abelson tyrosine kinase T315I mutant (unknown origin) using [gamma-33P]ATP as substrate by radiometric kinase...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Korea Institute Of Science And Technology (Kaist)

Curated by ChEMBL
LigandPNGBDBM50490889(CHEMBL2347723)
Affinity DataIC50:  0.0640nMAssay Description:Inhibition of breakpoint cluster region-Abelson tyrosine kinase T315I mutant (unknown origin) using [gamma-33P]ATP as substrate by radiometric kinase...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
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