Affinity DataKi: 0.380nMAssay Description:Compound was evaluated for its inhibitory activity against human thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 0.380nMAssay Description:Compound was tested for inhibitory activity against human thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 0.490nMAssay Description:Compound was evaluated for its inhibitory activity against human thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 0.600nMAssay Description:Compound was evaluated for its inhibitory activity against human thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 0.840nMAssay Description:Compound was evaluated for its inhibitory activity against human thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Inhibitory effect against bovine thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 1.10nMAssay Description:Compound was tested for inhibitory activity against bovine thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 1.5nMAssay Description:Inhibitory effect against bovine thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 3nMAssay Description:Compound was evaluated for its inhibitory activity against human thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 4nMAssay Description:Compound was tested for inhibitory activity against bovine thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 6.5nMAssay Description:Inhibitory effect against bovine thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 6.80nMAssay Description:Compound was evaluated for its inhibitory activity against human thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 20nMAssay Description:Inhibitory effect against bovine thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 41nMAssay Description:Compound was tested for inhibitory activity against bovine thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 46nMAssay Description:Inhibitory effect against bovine thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 50nMAssay Description:Inhibitory effect against bovine thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 52nMAssay Description:Inhibitory effect against bovine thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 91nMAssay Description:Compound was evaluated for its inhibitory activity against human thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 93nMAssay Description:Compound was tested for inhibitory activity against bovine thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 134nMAssay Description:Compound was evaluated for its inhibitory activity against bovine trypsinMore data for this Ligand-Target Pair
Affinity DataKi: 150nMAssay Description:Compound was evaluated for its inhibitory activity against bovine trypsinMore data for this Ligand-Target Pair
Affinity DataKi: 152nMAssay Description:Compound was tested for inhibitory activity against bovine thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 153nMAssay Description:Compound was evaluated for its inhibitory activity against bovine trypsinMore data for this Ligand-Target Pair
Affinity DataKi: 231nMAssay Description:Compound was tested for inhibitory activity against bovine thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 247nMAssay Description:Compound was tested for inhibitory activity against bovine thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 325nMAssay Description:Inhibitory effect of compound was measured in bovine trypsinMore data for this Ligand-Target Pair
Affinity DataKi: 367nMAssay Description:Compound was tested for inhibitory activity against bovine thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 1.10E+3nMAssay Description:The compound was tested for inhibitory activity against Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 1.14E+3nMAssay Description:Inhibitory effect against bovine thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 1.47E+3nMAssay Description:Compound was tested for inhibitory activity against bovine thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 2.44E+3nMAssay Description:Compound was evaluated for its inhibitory activity against bovine trypsinMore data for this Ligand-Target Pair
Affinity DataKi: 2.70E+3nMAssay Description:Inhibitory effect against bovine thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 3.20E+3nMAssay Description:Compound was evaluated for its inhibitory activity against bovine trypsinMore data for this Ligand-Target Pair
Affinity DataKi: 3.29E+3nMAssay Description:Compound was tested for inhibitory activity against bovine trypsinMore data for this Ligand-Target Pair
Affinity DataKi: 3.73E+3nMAssay Description:Inhibitory effect of compound was measured in bovine trypsinMore data for this Ligand-Target Pair
Affinity DataKi: 4.32E+3nMAssay Description:Inhibitory effect against bovine thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 5.37E+3nMAssay Description:Inhibitory effect against bovine thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 7.04E+3nMAssay Description:Compound was tested for inhibitory activity against bovine thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 8.65E+3nMAssay Description:Inhibitory effect of compound was measured in bovine trypsinMore data for this Ligand-Target Pair
Affinity DataKi: 1.36E+4nMAssay Description:Inhibitory effect against bovine thrombinMore data for this Ligand-Target Pair
Affinity DataKi: 1.62E+4nMAssay Description:Compound was evaluated for its inhibitory activity against bovine trypsinMore data for this Ligand-Target Pair
TargetTissue-type plasminogen activator(Homo sapiens (Human))
Biotech Research Institute
Curated by ChEMBL
Biotech Research Institute
Curated by ChEMBL
Affinity DataKi: 2.72E+4nMAssay Description:The compound was tested for inhibitory activity against tissue plasminogen activatorMore data for this Ligand-Target Pair
Affinity DataKi: 4.79E+4nMAssay Description:The compound was tested for inhibitory activity against human plasminMore data for this Ligand-Target Pair
Affinity DataKi: 8.15E+4nMAssay Description:Inhibitory effect of compound was measured in bovine trypsinMore data for this Ligand-Target Pair
Affinity DataKi: 1.92E+5nMAssay Description:Inhibitory effect of compound was measured in bovine trypsinMore data for this Ligand-Target Pair
Affinity DataKi: 3.16E+5nMAssay Description:Inhibitory effect of compound was measured in bovine trypsinMore data for this Ligand-Target Pair
Affinity DataKi: 5.45E+5nMAssay Description:Inhibitory effect of compound was measured in bovine trypsinMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Korea Institute Of Science And Technology (Kaist)
Curated by ChEMBL
Korea Institute Of Science And Technology (Kaist)
Curated by ChEMBL
Affinity DataIC50: 0.0150nMAssay Description:Inhibition of breakpoint cluster region-Abelson tyrosine kinase T315I mutant (unknown origin) using [gamma-33P]ATP as substrate by radiometric kinase...More data for this Ligand-Target Pair
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Korea Institute Of Science And Technology (Kaist)
Curated by ChEMBL
Korea Institute Of Science And Technology (Kaist)
Curated by ChEMBL
Affinity DataIC50: 0.0210nMAssay Description:Inhibition of breakpoint cluster region-Abelson tyrosine kinase T315I mutant (unknown origin) using [gamma-33P]ATP as substrate by radiometric kinase...More data for this Ligand-Target Pair
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Korea Institute Of Science And Technology (Kaist)
Curated by ChEMBL
Korea Institute Of Science And Technology (Kaist)
Curated by ChEMBL
Affinity DataIC50: 0.0640nMAssay Description:Inhibition of breakpoint cluster region-Abelson tyrosine kinase T315I mutant (unknown origin) using [gamma-33P]ATP as substrate by radiometric kinase...More data for this Ligand-Target Pair