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Found 926 with Last Name = 'de jesus' and Initial = 'r'
TargetMu-type opioid receptor(MOUSE)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50017233(CHEMBL592 | LEVO-DROMORAN | LEVORPHANOL)
Affinity DataKi:  0.300nMAssay Description:Binding affinity for mouse opioid receptor muMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 3(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50389603(CHEMBL2069499)
Affinity DataKi:  0.640nMAssay Description:Displacement of [125I]SS-14 from human SST3 receptor expressed in CHO cells after 60 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(MOUSE)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50017231((4aS,9aR)-4a-Ethyl-2-phenethyl-1,2,3,4,4a,9a-hexah...)
Affinity DataKi:  0.900nMAssay Description:Binding affinity for mouse opioid receptor muMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(MOUSE)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50017232(3-Cyclopropylmethyl-5-ethyl-8-hydroxy-11-methyl-3,...)
Affinity DataKi:  1.30nMAssay Description:Binding affinity for mouse opioid receptor muMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50094569(6-chloro-3,20-dioxo-1beta,2beta-dihydro-3'H-cyclop...)
Affinity DataKi:  1.30nMAssay Description:Adenosine A1 receptor binding was measured in adenosine deaminase (ADA) pretreated rat cortical membranes using [3H]cyclohexyladenosine in the presen...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 3(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50389592(CHEMBL2069500)
Affinity DataKi:  1.70nMAssay Description:Binding affinity to human SST3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Mus musculus (Mouse))
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50017233(CHEMBL592 | LEVO-DROMORAN | LEVORPHANOL)
Affinity DataKi:  1.90nMAssay Description:Binding affinity for mouse sigma opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Mus musculus (Mouse))
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50017232(3-Cyclopropylmethyl-5-ethyl-8-hydroxy-11-methyl-3,...)
Affinity DataKi:  2.30nMAssay Description:Binding affinity for mouse sigma opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(MOUSE)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50017238((4aS,9aR)-2-Cyclopropylmethyl-4a-ethyl-1,2,3,4,4a,...)
Affinity DataKi:  4nMAssay Description:Binding affinity for mouse opioid receptor muMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Mus musculus (Mouse))
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50017232(3-Cyclopropylmethyl-5-ethyl-8-hydroxy-11-methyl-3,...)
Affinity DataKi:  6nMAssay Description:Binding affinity for mouse opioid receptor kappaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a/A2b(Rattus norvegicus)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50015655((2S,3S,4R)-5-{(R)-6-Amino-2-[2-(4-chloro-phenyl)-e...)
Affinity DataKi:  7.5nMAssay Description:Binding to Adenosine A2 receptor was measured in ADA-pretreated rat striatal membranes using [3H]-CGS- 21680More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a/A2b(Rattus norvegicus)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50015648((2S,3S,4R)-5-{(R)-6-Amino-2-[2-(4-fluoro-phenyl)-e...)
Affinity DataKi:  7.70nMAssay Description:Binding to Adenosine A2 receptor was measured in ADA-pretreated rat striatal membranes using [3H]-CGS- 21680More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Mus musculus (Mouse))
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50017231((4aS,9aR)-4a-Ethyl-2-phenethyl-1,2,3,4,4a,9a-hexah...)
Affinity DataKi:  8nMAssay Description:Binding affinity for mouse sigma opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a/A2b(Rattus norvegicus)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50015649(3-(4-{2-[(R)-6-Amino-9-((3R,4S,5S)-5-ethylcarbamoy...)
Affinity DataKi:  9nMAssay Description:Binding to Adenosine A2 receptor was measured in ADA-pretreated rat striatal membranes using [3H]-CGS- 21680More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a/A2b(Rattus norvegicus)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM21220((2S,3S,4R,5R)-5-(6-amino-9H-purin-9-yl)-N-ethyl-3,...)
Affinity DataKi:  9nMAssay Description:Binding to Adenosine A2 receptor was measured in ADA-pretreated rat striatal membranes using [3H]-CGS- 21680More data for this Ligand-Target Pair
TargetAdenosine receptor A2a/A2b(Rattus norvegicus)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50385958(CHEMBL2042298)
Affinity DataKi:  9.70nMAssay Description:Binding to Adenosine A2 receptor was measured in ADA-pretreated rat striatal membranes using [3H]-CGS- 21680More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Mus musculus (Mouse))
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50017233(CHEMBL592 | LEVO-DROMORAN | LEVORPHANOL)
Affinity DataKi:  10nMAssay Description:Binding affinity for mouse opioid receptor kappaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a/A2b(Rattus norvegicus)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50015657((2S,3S,4R)-5-((R)-6-Amino-2-phenethylamino-purin-9...)
Affinity DataKi:  14nMAssay Description:Binding to Adenosine A2 receptor was measured in ADA-pretreated rat striatal membranes using [3H]-CGS- 21680More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(MOUSE)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50017234((4aS,9aR)-2-Cyclobutylmethyl-4a-ethyl-1,2,3,4,4a,9...)
Affinity DataKi:  17nMAssay Description:Binding affinity for mouse opioid receptor muMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a/A2b(Rattus norvegicus)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM35804((CGS21680) 3-(4-{2-[6-Amino-9-(5-ethylcarbamoylmet...)
Affinity DataKi:  19nMAssay Description:Binding to Adenosine A2 receptor was measured in ADA-pretreated rat striatal membranes using [3H]-CGS- 21680More data for this Ligand-Target Pair
TargetMu-type opioid receptor(MOUSE)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50017236((4aS,9aR)-4a-Ethyl-2-methyl-1,2,3,4,4a,9a-hexahydr...)
Affinity DataKi:  19nMAssay Description:Binding affinity for mouse opioid receptor muMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(MOUSE)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50017237((4aS,9aR)-4a-Ethyl-2-propyl-1,2,3,4,4a,9a-hexahydr...)
Affinity DataKi:  30nMAssay Description:Binding affinity for mouse opioid receptor muMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(MOUSE)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50017239((4aS,9aR)-4a-Ethyl-2-furan-3-ylmethyl-1,2,3,4,4a,9...)
Affinity DataKi:  31nMAssay Description:Binding affinity for mouse opioid receptor muMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Mus musculus (Mouse))
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50017238((4aS,9aR)-2-Cyclopropylmethyl-4a-ethyl-1,2,3,4,4a,...)
Affinity DataKi:  34nMAssay Description:Binding affinity for mouse opioid receptor kappaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a/A2b(Rattus norvegicus)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50015650((4-{2-[(R)-6-Amino-9-((3R,4S,5S)-5-ethylcarbamoyl-...)
Affinity DataKi:  42nMAssay Description:Binding to Adenosine A2 receptor was measured in ADA-pretreated rat striatal membranes using [3H]-CGS- 21680More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a/A2b(Rattus norvegicus)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50015654((4-{2-[(R)-6-Amino-9-((3R,4S,5S)-5-ethylcarbamoyl-...)
Affinity DataKi:  45nMAssay Description:Binding to Adenosine A2 receptor was measured in ADA-pretreated rat striatal membranes using [3H]-CGS- 21680More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(MOUSE)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50017240((4aS,9aR)-2-Cyclopentylmethyl-4a-ethyl-1,2,3,4,4a,...)
Affinity DataKi:  50nMAssay Description:Binding affinity for mouse opioid receptor muMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Mus musculus (Mouse))
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50017238((4aS,9aR)-2-Cyclopropylmethyl-4a-ethyl-1,2,3,4,4a,...)
Affinity DataKi:  53nMAssay Description:Binding affinity for mouse sigma opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a/A2b(Rattus norvegicus)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50015651((2S,3S,4R)-5-[(R)-6-Amino-2-(methyl-phenethyl-amin...)
Affinity DataKi:  71nMAssay Description:Binding to Adenosine A2 receptor was measured in ADA-pretreated rat striatal membranes using [3H]-CGS- 21680More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a/A2b(Rattus norvegicus)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM82022(2-(Phenylamino)ado (CV-1808) | 2-[6-Amino-2-(3-cyc...)
Affinity DataKi:  71nMAssay Description:Binding to Adenosine A2 receptor was measured in ADA-pretreated rat striatal membranes using [3H]-CGS- 21680More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a/A2b(Rattus norvegicus)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50407975(CHEMBL519809)
Affinity DataKi:  71nMAssay Description:Binding to Adenosine A2 receptor was measured in ADA-pretreated rat striatal membranes using [3H]-CGS- 21680More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(MOUSE)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50017235((4aS,9aR)-4a-Ethyl-2-(tetrahydro-furan-2-ylmethyl)...)
Affinity DataKi:  73nMAssay Description:Binding affinity for mouse opioid receptor muMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a/A2b(Rattus norvegicus)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50015652((2S,3S,4R)-5-((R)-6-Amino-2-phenethylamino-purin-9...)
Affinity DataKi:  77nMAssay Description:Binding to Adenosine A2 receptor was measured in ADA-pretreated rat striatal membranes using [3H]-CGS- 21680More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(MOUSE)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50017241((4aS,9aR)-4a-Ethyl-2-furan-2-ylmethyl-1,2,3,4,4a,9...)
Affinity DataKi:  99nMAssay Description:Binding affinity for mouse opioid receptor muMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50407975(CHEMBL519809)
Affinity DataKi:  101nMAssay Description:Adenosine A1 receptor binding was measured in adenosine deaminase (ADA) pretreated rat cortical membranes using [3H]cyclohexyladenosine in the presen...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Mus musculus (Mouse))
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50017239((4aS,9aR)-4a-Ethyl-2-furan-3-ylmethyl-1,2,3,4,4a,9...)
Affinity DataKi:  115nMAssay Description:Binding affinity for mouse sigma opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(MOUSE)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50017242((4aS,9aR)-4a-Ethyl-2,9a-dimethyl-1,2,3,4,4a,9a-hex...)
Affinity DataKi:  126nMAssay Description:Binding affinity for mouse opioid receptor muMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Mus musculus (Mouse))
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50017239((4aS,9aR)-4a-Ethyl-2-furan-3-ylmethyl-1,2,3,4,4a,9...)
Affinity DataKi:  190nMAssay Description:Binding affinity for mouse opioid receptor kappaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Mus musculus (Mouse))
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50017236((4aS,9aR)-4a-Ethyl-2-methyl-1,2,3,4,4a,9a-hexahydr...)
Affinity DataKi:  212nMAssay Description:Binding affinity for mouse sigma opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Mus musculus (Mouse))
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50017237((4aS,9aR)-4a-Ethyl-2-propyl-1,2,3,4,4a,9a-hexahydr...)
Affinity DataKi:  231nMAssay Description:Binding affinity for mouse sigma opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Mus musculus (Mouse))
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50017234((4aS,9aR)-2-Cyclobutylmethyl-4a-ethyl-1,2,3,4,4a,9...)
Affinity DataKi:  270nMAssay Description:Binding affinity for mouse opioid receptor kappaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Mus musculus (Mouse))
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50017237((4aS,9aR)-4a-Ethyl-2-propyl-1,2,3,4,4a,9a-hexahydr...)
Affinity DataKi:  335nMAssay Description:Binding affinity for mouse opioid receptor kappaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Mus musculus (Mouse))
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50017240((4aS,9aR)-2-Cyclopentylmethyl-4a-ethyl-1,2,3,4,4a,...)
Affinity DataKi:  340nMAssay Description:Binding affinity for mouse sigma opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Mus musculus (Mouse))
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50017234((4aS,9aR)-2-Cyclobutylmethyl-4a-ethyl-1,2,3,4,4a,9...)
Affinity DataKi:  410nMAssay Description:Binding affinity for mouse sigma opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50385958(CHEMBL2042298)
Affinity DataKi:  473nMAssay Description:Adenosine A1 receptor binding was measured in adenosine deaminase (ADA) pretreated rat cortical membranes using [3H]cyclohexyladenosine in the presen...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Mus musculus (Mouse))
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50017235((4aS,9aR)-4a-Ethyl-2-(tetrahydro-furan-2-ylmethyl)...)
Affinity DataKi:  474nMAssay Description:Binding affinity for mouse sigma opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Mus musculus (Mouse))
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50017242((4aS,9aR)-4a-Ethyl-2,9a-dimethyl-1,2,3,4,4a,9a-hex...)
Affinity DataKi:  481nMAssay Description:Binding affinity for mouse sigma opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50015657((2S,3S,4R)-5-((R)-6-Amino-2-phenethylamino-purin-9...)
Affinity DataKi:  502nMAssay Description:Adenosine A1 receptor binding was measured in adenosine deaminase (ADA) pretreated rat cortical membranes using [3H]cyclohexyladenosine in the presen...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Mus musculus (Mouse))
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50017240((4aS,9aR)-2-Cyclopentylmethyl-4a-ethyl-1,2,3,4,4a,...)
Affinity DataKi:  550nMAssay Description:Binding affinity for mouse opioid receptor kappaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Mus musculus (Mouse))
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50017241((4aS,9aR)-4a-Ethyl-2-furan-2-ylmethyl-1,2,3,4,4a,9...)
Affinity DataKi:  571nMAssay Description:Binding affinity for mouse sigma opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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