Affinity DataKi: 0.400nMAssay Description:In vitro binding affinity for serotonin reuptake sites in rat frontal cortex membranes by [3H]-paroxetine displacement.More data for this Ligand-Target Pair
Affinity DataKi: 0.410nMAssay Description:Binding affinity for dopamine receptor D2 determined using [3H]-spiperoneMore data for this Ligand-Target Pair
Affinity DataKi: 0.420nMAssay Description:Binding affinity for dopamine receptor D2 determined using [3H]-spiperoneMore data for this Ligand-Target Pair
Affinity DataKi: 0.450nMAssay Description:Displacement of [3H]-Spiperone from Dopamine receptor D2 in rat striatumMore data for this Ligand-Target Pair
Affinity DataKi: 0.470nMAssay Description:Binding affinity for dopamine receptor D2 determined using [3H]-spiperoneMore data for this Ligand-Target Pair
Affinity DataKi: 0.600nMAssay Description:In vitro binding affinity for serotonin reuptake sites in rat frontal cortex membranes by [3H]-paroxetine displacement.More data for this Ligand-Target Pair
Affinity DataKi: 0.680nMAssay Description:Displacement of [3H]-Spiperone from Dopamine receptor D2 in rat striatumMore data for this Ligand-Target Pair
Affinity DataKi: 0.760nMAssay Description:Displacement of [3H]-Spiperone from Dopamine receptor D2 in rat striatumMore data for this Ligand-Target Pair
Affinity DataKi: 0.800nMAssay Description:In vitro binding affinity for serotonin reuptake sites in rat frontal cortex membranes by [3H]-paroxetine displacement.More data for this Ligand-Target Pair
Affinity DataKi: 0.800nMAssay Description:In vitro binding affinity for serotonin reuptake sites in rat frontal cortex membranes by [3H]-paroxetine displacement.More data for this Ligand-Target Pair
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Duphar Research Laboratories
Curated by ChEMBL
Duphar Research Laboratories
Curated by ChEMBL
Affinity DataKi: 0.870nMAssay Description:Ability to inhibit [3H]WB-4101 binding to alpha-1 adrenergic receptor was determined in ratMore data for this Ligand-Target Pair
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Duphar Research Laboratories
Curated by ChEMBL
Duphar Research Laboratories
Curated by ChEMBL
Affinity DataKi: 0.870nMAssay Description:Potency to displace [3H]- WB-4101 from alpha-1 adrenergic receptor in rat striatumMore data for this Ligand-Target Pair
Affinity DataKi: 0.910nMAssay Description:Ability to inhibit the [3H]spiperone binding to striatum Dopamine receptor D2 was determined in ratMore data for this Ligand-Target Pair
Affinity DataKi: 0.910nMAssay Description:Binding affinity for 5-hydroxytryptamine 1A receptor determined using [3H]-8-OH-DPAT as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 0.930nMAssay Description:Binding affinity for dopamine receptor D2 determined using [3H]-spiperoneMore data for this Ligand-Target Pair
Affinity DataKi: 0.960nMAssay Description:Displacement of [3H]-Spiperone from Dopamine receptor D2 in rat striatumMore data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:In vitro binding affinity for serotonin reuptake sites in rat frontal cortex membranes by [3H]-paroxetine displacement.More data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:In vitro binding affinity for serotonin reuptake sites in rat frontal cortex membranes by [3H]-paroxetine displacement.More data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Binding affinity for 5-hydroxytryptamine 1A receptor determined using [3H]-8-OH-DPAT as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Binding affinity for dopamine receptor D2 determined using [3H]-spiperoneMore data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Displacement of [3H]-Spiperone from Dopamine receptor D2 in rat striatumMore data for this Ligand-Target Pair
Affinity DataKi: 1.10nMAssay Description:Displacement of [3H]-Spiperone from Dopamine receptor D2 in rat striatumMore data for this Ligand-Target Pair
Affinity DataKi: 1.30nMAssay Description:In vitro binding affinity for serotonin reuptake sites in rat frontal cortex membranes by [3H]-paroxetine displacement.More data for this Ligand-Target Pair
Affinity DataKi: 1.30nMAssay Description:In vitro binding affinity for serotonin reuptake sites in rat frontal cortex membranes by [3H]-paroxetine displacement.More data for this Ligand-Target Pair
Affinity DataKi: 1.30nMAssay Description:Binding affinity for dopamine receptor D2 determined using [3H]-spiperoneMore data for this Ligand-Target Pair
Affinity DataKi: 1.40nMAssay Description:Ability to inhibit the [3H]spiperone binding to striatum Dopamine receptor D2 was determined in ratMore data for this Ligand-Target Pair
Affinity DataKi: 1.40nMAssay Description:Binding affinity for dopamine receptor D2 determined using [3H]-spiperoneMore data for this Ligand-Target Pair
Affinity DataKi: 1.40nMAssay Description:Displacement of [3H]-Spiperone from Dopamine receptor D2 in rat striatumMore data for this Ligand-Target Pair
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Duphar Research Laboratories
Curated by ChEMBL
Duphar Research Laboratories
Curated by ChEMBL
Affinity DataKi: 1.5nMAssay Description:Potency to displace [3H]- WB-4101 from alpha-1 adrenergic receptor in rat striatumMore data for this Ligand-Target Pair
Affinity DataKi: 1.5nMAssay Description:Binding affinity for 5-hydroxytryptamine 1A receptor determined using [3H]-8-OH-DPAT as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 1.70nMAssay Description:Binding affinity for dopamine receptor D2 determined using [3H]-spiperoneMore data for this Ligand-Target Pair
Affinity DataKi: 1.80nMAssay Description:Binding affinity for dopamine receptor D2 determined using [3H]-spiperoneMore data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:In vitro binding affinity for serotonin reuptake sites in rat frontal cortex membranes by [3H]-paroxetine displacement.More data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:In vitro binding affinity for serotonin reuptake sites in rat frontal cortex membranes by [3H]-paroxetine displacement.More data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Binding affinity for dopamine receptor D2 determined using [3H]-spiperoneMore data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:In vitro binding affinity for serotonin reuptake sites in rat frontal cortex membranes by [3H]-paroxetine displacement.More data for this Ligand-Target Pair
Affinity DataKi: 2.20nMAssay Description:Binding affinity for dopamine receptor D2 determined using [3H]-spiperoneMore data for this Ligand-Target Pair
Affinity DataKi: 2.20nMAssay Description:Binding affinity for dopamine receptor D2 determined using [3H]-spiperoneMore data for this Ligand-Target Pair
Affinity DataKi: 2.40nMAssay Description:Displacement of [3H]-Spiperone from Dopamine receptor D2 in rat striatumMore data for this Ligand-Target Pair
Affinity DataKi: 2.5nMAssay Description:In vitro binding affinity for serotonin reuptake sites in rat frontal cortex membranes by [3H]-paroxetine displacement.More data for this Ligand-Target Pair
Affinity DataKi: 2.5nMAssay Description:In vitro binding affinity for serotonin reuptake sites in rat frontal cortex membranes by [3H]-paroxetine displacement.More data for this Ligand-Target Pair
Affinity DataKi: 2.5nMAssay Description:In vitro binding affinity for serotonin reuptake sites in rat frontal cortex membranes by [3H]-paroxetine displacement.More data for this Ligand-Target Pair
Affinity DataKi: 2.90nMAssay Description:Binding affinity for dopamine receptor D2 determined using [3H]-spiperoneMore data for this Ligand-Target Pair
Affinity DataKi: 2.90nMAssay Description:Ability to inhibit the [3H]spiperone binding to striatum Dopamine receptor D2 was determined in ratMore data for this Ligand-Target Pair
Affinity DataKi: 3nMAssay Description:In vitro binding affinity for serotonin reuptake sites in rat frontal cortex membranes by [3H]-paroxetine displacement.More data for this Ligand-Target Pair
Affinity DataKi: 3nMAssay Description:In vitro binding affinity at human cloned dopamine receptor D2 (long) stably expressed in CHO cells by [3H]-Spiperone displacement.More data for this Ligand-Target Pair
Affinity DataKi: 3nMAssay Description:Binding affinity for dopamine receptor D2 determined using [3H]-spiperoneMore data for this Ligand-Target Pair
Affinity DataKi: 3.10nMAssay Description:Binding affinity for dopamine receptor D2 determined using [3H]-spiperoneMore data for this Ligand-Target Pair
Affinity DataKi: 4nMAssay Description:Binding affinity for dopamine receptor D2 determined using [3H]-spiperoneMore data for this Ligand-Target Pair
Affinity DataKi: 4.30nMAssay Description:Displacement of [3H]-Spiperone from Dopamine receptor D2 in rat striatumMore data for this Ligand-Target Pair