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| Wt: 375.4 BDBM27713  |
| Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kcal/mole | IC50 nM | Kd nM | EC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| poly-ADP-ribose polymerase 2 (PARP2) (Mus musculus (Mouse)) | BDBM27713 (1-[4-(4-phenyl-1,2,3,6-tetrahydropyridin-1-yl)buty...) | PDB MMDB Reactome pathway UniProtKB/SwissProt GoogleScholar | PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 70 | n/a | n/a | n/a | n/a | n/a | 25 |
Fujisawa Pharmaceutical Co., Ltd | Assay Description To assess the inhibitory activity of novel inhibitors, the PARP enzyme assay was carried out in reaction mixture consisting of activated salmon teste... | Bioorg Med Chem 14: 1378-90 (2006) Article DOI: 10.1016/j.bmc.2005.09.061 BindingDB Entry DOI: 10.7270/Q2610XPZ | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Poly [ADP-ribose] polymerase 1 (Homo sapiens (Human)) | BDBM27713 (1-[4-(4-phenyl-1,2,3,6-tetrahydropyridin-1-yl)buty...) | PDB MMDB Reactome pathway UniProtKB/SwissProt UniProtKB/TrEMBL antibodypedia GoogleScholar | PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 120 | n/a | n/a | n/a | n/a | 8.0 | 23 |
Fujisawa Pharmaceutical Co., Ltd | Assay Description To assess the inhibitory activity of novel inhibitors, the PARP enzyme assay was carried out in reaction mixture consisting of activated salmon teste... | Bioorg Med Chem 14: 1378-90 (2006) Article DOI: 10.1016/j.bmc.2005.09.061 BindingDB Entry DOI: 10.7270/Q2610XPZ | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
