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14 similar compounds to monomer 50005582

Compile data set for download or QSAR
Wt: 434.4
BDBM50005567
Wt: 318.3
BDBM50005570
Wt: 450.5
BDBM50005574
Wt: 408.4
BDBM50005575
Wt: 393.4
BDBM50005546
Wt: 434.4
BDBM50008052
Wt: 393.4
BDBM50008038
Wt: 450.5
BDBM50008042
Wt: 408.4
BDBM50008047
Wt: 438.4
BDBM50008048
Wt: 393.4
BDBM50035768
Wt: 393.4
BDBM50042484
Wt: 408.4
BDBM50042489
Wt: 536.5
BDBM50130353

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 22 hits for monomerid = 50005567,50005570,50005574,50005575,50005546,50008052,50008038,50008042,50008047,50008048,50035768,50042484,50042489,50130353   
Target/Host
(Institution)
LigandTarget/Host
Links
Ligand
Links
Trg + Lig
Links
Ki
nM
ΔG°
kcal/mole
IC50
nM
Kd
nM
EC50/IC50
nM
koff
s-1
kon
M-1s-1
pHTemp
°C
Dopamine Transporter (DAT)


(Rattus norvegicus (rat))
BDBM50130353
PNG
(3-[Bis-(4-fluoro-phenyl)-methoxy]-8-methyl-8-aza-b...)
Show SMILES CN1C2CCC1[C@H]([C@H](C2)OC(c1ccc(F)cc1)c1ccc(F)cc1)C(=O)OCCc1ccc(cc1)[N+]([O-])=O
Show InChI InChI=1S/C30H30F2N2O5/c1-33-25-14-15-26(33)28(30(35)38-17-16-19-2-12-24(13-3-19)34(36)37)27(18-25)39-29(20-4-8-22(31)9-5-20)21-6-10-23(32)11-7-21/h2-13,25-29H,14-18H2,1H3/t25?,26?,27-,28+/m0/s1
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97.7n/an/an/an/an/an/an/an/a



National Institute on Drug Abuse

Curated by ChEMBL


Assay Description
In vitro dopamine transporter binding affinity using [3H]WIN-35428 as radioligand was determined


J Med Chem 46: 2908-16 (2003)


Article DOI: 10.1021/jm0300375
BindingDB Entry DOI: 10.7270/Q2BG2PQ0
More data for this
Ligand-Target Pair
Monoamine transporters; Norepininephrine & dopamine


(Rattus norvegicus (rat))
BDBM50005570
PNG
(3-(4-Amino-benzoyloxy)-8-methyl-8-aza-bicyclo[3.2....)
Show SMILES COC(=O)C1C2CC[C@H](C[C@@H]1OC(=O)c1ccc(N)cc1)N2C
Show InChI InChI=1S/C17H22N2O4/c1-19-12-7-8-13(19)15(17(21)22-2)14(9-12)23-16(20)10-3-5-11(18)6-4-10/h3-6,12-15H,7-9,18H2,1-2H3/t12-,13?,14+,15?/m1/s1
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n/an/a 1.23E+3n/an/an/an/an/an/a



Research Triangle Institute

Curated by ChEMBL


Assay Description
Potency for the inhibition of [3H]WIN-35428 binding to the dopamine transporter


J Med Chem 35: 969-81 (1992)


Article DOI: 10.1021/jm00084a001
BindingDB Entry DOI: 10.7270/Q24T6K0F
More data for this
Ligand-Target Pair
Dopamine Transporter (DAT)


(Rattus norvegicus (rat))
BDBM50008047
PNG
(3-Benzoyloxy-8-methyl-8-aza-bicyclo[3.2.1]octane-2...)
Show SMILES CN1[C@@H]2CCC1C([C@H](C2)OC(=O)c1ccccc1)C(=O)OCCc1ccc(N)cc1
Show InChI InChI=1S/C24H28N2O4/c1-26-19-11-12-20(26)22(21(15-19)30-23(27)17-5-3-2-4-6-17)24(28)29-14-13-16-7-9-18(25)10-8-16/h2-10,19-22H,11-15,25H2,1H3/t19-,20?,21+,22?/m1/s1
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n/an/a 72n/an/an/an/an/an/a



Research Triangle Institute

Curated by ChEMBL


Assay Description
Inhibition of [3H]3-beta-(p-fluorophenyl)tropane-2beta-carboxylic acid methyl ester binding to Dopamine transporter in rat striatal membranes.


J Med Chem 35: 135-40 (1992)


Article DOI: 10.1021/jm00079a017
BindingDB Entry DOI: 10.7270/Q2FQ9X7M
More data for this
Ligand-Target Pair
Dopamine Transporter (DAT)


(Rattus norvegicus (rat))
BDBM50008048
PNG
(3-Benzoyloxy-8-methyl-8-aza-bicyclo[3.2.1]octane-2...)
Show SMILES CN1[C@@H]2CCC1C([C@H](C2)OC(=O)c1ccccc1)C(=O)OCCc1ccc(cc1)[N+]([O-])=O
Show InChI InChI=1S/C24H26N2O6/c1-25-19-11-12-20(25)22(21(15-19)32-23(27)17-5-3-2-4-6-17)24(28)31-14-13-16-7-9-18(10-8-16)26(29)30/h2-10,19-22H,11-15H2,1H3/t19-,20?,21+,22?/m1/s1
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n/an/a 601n/an/an/an/an/an/a



Research Triangle Institute

Curated by ChEMBL


Assay Description
Inhibition of [3H]3-beta-(p-fluorophenyl)tropane-2beta-carboxylic acid methyl ester binding to Dopamine transporter in rat striatal membranes.


J Med Chem 35: 135-40 (1992)


Article DOI: 10.1021/jm00079a017
BindingDB Entry DOI: 10.7270/Q2FQ9X7M
More data for this
Ligand-Target Pair
Dopamine Transporter (DAT)


(Rattus norvegicus (rat))
BDBM50008052
PNG
(3-Benzoyloxy-8-methyl-8-aza-bicyclo[3.2.1]octane-2...)
Show SMILES CN1[C@@H]2CCC1C([C@H](C2)OC(=O)c1ccccc1)C(=O)OCCc1ccc(cc1)N=[N+]=[N-]
Show InChI InChI=1S/C24H26N4O4/c1-28-19-11-12-20(28)22(21(15-19)32-23(29)17-5-3-2-4-6-17)24(30)31-14-13-16-7-9-18(10-8-16)26-27-25/h2-10,19-22H,11-15H2,1H3/t19-,20?,21+,22?/m1/s1
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n/an/a 227n/an/an/an/an/an/a



Research Triangle Institute

Curated by ChEMBL


Assay Description
Inhibition of [3H]3-beta-(p-fluorophenyl)tropane-2beta-carboxylic acid methyl ester binding to Dopamine transporter in rat striatal membranes.


J Med Chem 35: 135-40 (1992)


Article DOI: 10.1021/jm00079a017
BindingDB Entry DOI: 10.7270/Q2FQ9X7M
More data for this
Ligand-Target Pair
Dopamine Transporter (DAT)


(Rattus norvegicus (rat))
BDBM50005546
PNG
(3-Benzoyloxy-8-methyl-8-aza-bicyclo[3.2.1]octane-2...)
Show SMILES CN1[C@@H]2CCC1C([C@H](C2)OC(=O)c1ccccc1)C(=O)OCCc1ccccc1
Show InChI InChI=1S/C24H27NO4/c1-25-19-12-13-20(25)22(24(27)28-15-14-17-8-4-2-5-9-17)21(16-19)29-23(26)18-10-6-3-7-11-18/h2-11,19-22H,12-16H2,1H3/t19-,20?,21+,22?/m1/s1
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n/an/a 248n/an/an/an/an/an/a



Research Triangle Institute

Curated by ChEMBL


Assay Description
Inhibition of [3H]WIN-35428 binding to the dopamine transporter


J Med Chem 35: 969-81 (1992)


Article DOI: 10.1021/jm00084a001
BindingDB Entry DOI: 10.7270/Q24T6K0F
More data for this
Ligand-Target Pair
Dopamine Transporter (DAT)


(Rattus norvegicus (rat))
BDBM50005567
PNG
(3-Benzoyloxy-8-methyl-8-aza-bicyclo[3.2.1]octane-2...)
Show SMILES CN1[C@@H]2CCC1C([C@H](C2)OC(=O)c1ccccc1)C(=O)OCCc1ccc(cc1)N=[N+]=[N-]
Show InChI InChI=1S/C24H26N4O4/c1-28-19-11-12-20(28)22(21(15-19)32-23(29)17-5-3-2-4-6-17)24(30)31-14-13-16-7-9-18(10-8-16)26-27-25/h2-10,19-22H,11-15H2,1H3/t19-,20?,21+,22?/m1/s1
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n/an/a 227n/an/an/an/an/an/a



Research Triangle Institute

Curated by ChEMBL


Assay Description
Inhibition of [3H]WIN-35428 binding to the dopamine transporter


J Med Chem 35: 969-81 (1992)


Article DOI: 10.1021/jm00084a001
BindingDB Entry DOI: 10.7270/Q24T6K0F
More data for this
Ligand-Target Pair
Dopamine Transporter (DAT)


(Rattus norvegicus (rat))
BDBM50005574
PNG
(3-Benzoyloxy-8-methyl-8-aza-bicyclo[3.2.1]octane-2...)
Show SMILES CN1[C@@H]2CCC1C([C@H](C2)OC(=O)c1ccccc1)C(=O)OCCc1ccc(cc1)N=C=S
Show InChI InChI=1S/C25H26N2O4S/c1-27-20-11-12-21(27)23(22(15-20)31-24(28)18-5-3-2-4-6-18)25(29)30-14-13-17-7-9-19(10-8-17)26-16-32/h2-10,20-23H,11-15H2,1H3/t20-,21?,22+,23?/m1/s1
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n/an/a 196n/an/an/an/an/an/a



Research Triangle Institute

Curated by ChEMBL


Assay Description
Inhibition of [3H]WIN-35428 binding to the dopamine transporter


J Med Chem 35: 969-81 (1992)


Article DOI: 10.1021/jm00084a001
BindingDB Entry DOI: 10.7270/Q24T6K0F
More data for this
Ligand-Target Pair
Dopamine Transporter (DAT)


(Rattus norvegicus (rat))
BDBM50005575
PNG
(3-Benzoyloxy-8-methyl-8-aza-bicyclo[3.2.1]octane-2...)
Show SMILES CN1[C@@H]2CCC1C([C@H](C2)OC(=O)c1ccccc1)C(=O)OCCc1ccc(N)cc1
Show InChI InChI=1S/C24H28N2O4/c1-26-19-11-12-20(26)22(21(15-19)30-23(27)17-5-3-2-4-6-17)24(28)29-14-13-16-7-9-18(25)10-8-16/h2-10,19-22H,11-15,25H2,1H3/t19-,20?,21+,22?/m1/s1
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n/an/a 71n/an/an/an/an/an/a



Research Triangle Institute

Curated by ChEMBL


Assay Description
Inhibition of [3H]WIN-35428 binding to the dopamine transporter


J Med Chem 35: 969-81 (1992)


Article DOI: 10.1021/jm00084a001
BindingDB Entry DOI: 10.7270/Q24T6K0F
More data for this
Ligand-Target Pair
Dopamine Transporter (DAT)


(Rattus norvegicus (rat))
BDBM50005570
PNG
(3-(4-Amino-benzoyloxy)-8-methyl-8-aza-bicyclo[3.2....)
Show SMILES COC(=O)C1C2CC[C@H](C[C@@H]1OC(=O)c1ccc(N)cc1)N2C
Show InChI InChI=1S/C17H22N2O4/c1-19-12-7-8-13(19)15(17(21)22-2)14(9-12)23-16(20)10-3-5-11(18)6-4-10/h3-6,12-15H,7-9,18H2,1-2H3/t12-,13?,14+,15?/m1/s1
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n/an/a 3.04E+3n/an/an/an/an/an/a



Research Triangle Institute

Curated by ChEMBL


Assay Description
Inhibition of [3H]mazindol binding to the dopamine transporter.


J Med Chem 35: 969-81 (1992)


Article DOI: 10.1021/jm00084a001
BindingDB Entry DOI: 10.7270/Q24T6K0F
More data for this
Ligand-Target Pair
Dopamine Transporter (DAT)


(Rattus norvegicus (rat))
BDBM50005575
PNG
(3-Benzoyloxy-8-methyl-8-aza-bicyclo[3.2.1]octane-2...)
Show SMILES CN1[C@@H]2CCC1C([C@H](C2)OC(=O)c1ccccc1)C(=O)OCCc1ccc(N)cc1
Show InChI InChI=1S/C24H28N2O4/c1-26-19-11-12-20(26)22(21(15-19)30-23(27)17-5-3-2-4-6-17)24(28)29-14-13-16-7-9-18(25)10-8-16/h2-10,19-22H,11-15,25H2,1H3/t19-,20?,21+,22?/m1/s1
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n/an/a 72n/an/an/an/an/an/a



Research Triangle Institute

Curated by ChEMBL


Assay Description
Inhibition of [3H]WIN-35248 binding to the dopamine transporter in rat striatal membranes.


J Med Chem 35: 1813-7 (1992)


Article DOI: 10.1021/jm00088a017
BindingDB Entry DOI: 10.7270/Q29024D6
More data for this
Ligand-Target Pair
Dopamine Transporter (DAT)


(Rattus norvegicus (rat))
BDBM50005567
PNG
(3-Benzoyloxy-8-methyl-8-aza-bicyclo[3.2.1]octane-2...)
Show SMILES CN1[C@@H]2CCC1C([C@H](C2)OC(=O)c1ccccc1)C(=O)OCCc1ccc(cc1)N=[N+]=[N-]
Show InChI InChI=1S/C24H26N4O4/c1-28-19-11-12-20(28)22(21(15-19)32-23(29)17-5-3-2-4-6-17)24(30)31-14-13-16-7-9-18(10-8-16)26-27-25/h2-10,19-22H,11-15H2,1H3/t19-,20?,21+,22?/m1/s1
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n/an/a 227n/an/an/an/an/an/a



Research Triangle Institute

Curated by ChEMBL


Assay Description
Inhibition of [3H]WIN-35248 binding to the dopamine transporter in rat striatal membranes.


J Med Chem 35: 1813-7 (1992)


Article DOI: 10.1021/jm00088a017
BindingDB Entry DOI: 10.7270/Q29024D6
More data for this
Ligand-Target Pair
Dopamine Transporter (DAT)


(Rattus norvegicus (rat))
BDBM50005574
PNG
(3-Benzoyloxy-8-methyl-8-aza-bicyclo[3.2.1]octane-2...)
Show SMILES CN1[C@@H]2CCC1C([C@H](C2)OC(=O)c1ccccc1)C(=O)OCCc1ccc(cc1)N=C=S
Show InChI InChI=1S/C25H26N2O4S/c1-27-20-11-12-21(27)23(22(15-20)31-24(28)18-5-3-2-4-6-18)25(29)30-14-13-17-7-9-19(10-8-17)26-16-32/h2-10,20-23H,11-15H2,1H3/t20-,21?,22+,23?/m1/s1
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n/an/a 196n/an/an/an/an/an/a



Research Triangle Institute

Curated by ChEMBL


Assay Description
Inhibition of [3H]WIN-35248 binding to the dopamine transporter in rat striatal membranes.


J Med Chem 35: 1813-7 (1992)


Article DOI: 10.1021/jm00088a017
BindingDB Entry DOI: 10.7270/Q29024D6
More data for this
Ligand-Target Pair
Dopamine Transporter (DAT)


(Rattus norvegicus (rat))
BDBM50005546
PNG
(3-Benzoyloxy-8-methyl-8-aza-bicyclo[3.2.1]octane-2...)
Show SMILES CN1[C@@H]2CCC1C([C@H](C2)OC(=O)c1ccccc1)C(=O)OCCc1ccccc1
Show InChI InChI=1S/C24H27NO4/c1-25-19-12-13-20(25)22(24(27)28-15-14-17-8-4-2-5-9-17)21(16-19)29-23(26)18-10-6-3-7-11-18/h2-11,19-22H,12-16H2,1H3/t19-,20?,21+,22?/m1/s1
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n/an/a 248n/an/an/an/an/an/a



Research Triangle Institute

Curated by ChEMBL


Assay Description
Inhibition of [3H]WIN-35248 binding to the dopamine transporter in rat striatal membranes.


J Med Chem 35: 1813-7 (1992)


Article DOI: 10.1021/jm00088a017
BindingDB Entry DOI: 10.7270/Q29024D6
More data for this
Ligand-Target Pair
Dopamine Transporter (DAT)


(Rattus norvegicus (rat))
BDBM50042484
PNG
(CHEMBL118380 | R-3-Benzoyloxy-8-methyl-8-aza-bicyc...)
Show SMILES CN1C2CCC1C([C@@H](C2)OC(=O)c1ccccc1)C(=O)OCCc1ccccc1
Show InChI InChI=1S/C24H27NO4/c1-25-19-12-13-20(25)22(24(27)28-15-14-17-8-4-2-5-9-17)21(16-19)29-23(26)18-10-6-3-7-11-18/h2-11,19-22H,12-16H2,1H3/t19?,20?,21-,22?/m1/s1
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n/an/a 248n/an/an/an/an/an/a



University of Michigan

Curated by ChEMBL


Assay Description
Inhibition of [3H]WIN-35428 binding to dopamine transporter in rat striatal membranes.


J Med Chem 36: 3572-9 (1994)


Article DOI: 10.1021/jm00075a012
BindingDB Entry DOI: 10.7270/Q24J0FQ5
More data for this
Ligand-Target Pair
Dopamine Transporter (DAT)


(Rattus norvegicus (rat))
BDBM50042489
PNG
(CHEMBL332452 | R-3-Benzoyloxy-8-methyl-8-aza-bicyc...)
Show SMILES CN1C2CCC1C([C@@H](C2)OC(=O)c1ccccc1)C(=O)OCCc1ccc(N)cc1
Show InChI InChI=1S/C24H28N2O4/c1-26-19-11-12-20(26)22(21(15-19)30-23(27)17-5-3-2-4-6-17)24(28)29-14-13-16-7-9-18(25)10-8-16/h2-10,19-22H,11-15,25H2,1H3/t19?,20?,21-,22?/m1/s1
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n/an/a 72n/an/an/an/an/an/a



University of Michigan

Curated by ChEMBL


Assay Description
Inhibition of [3H]WIN-35428 binding to dopamine transporter in rat striatal membranes.


J Med Chem 36: 3572-9 (1994)


Article DOI: 10.1021/jm00075a012
BindingDB Entry DOI: 10.7270/Q24J0FQ5
More data for this
Ligand-Target Pair
Sodium-dependent serotonin transporter


(Rattus norvegicus (rat))
BDBM50035768
PNG
(3-Benzoyloxy-8-methyl-8-aza-bicyclo[3.2.1]octane-2...)
Show SMILES CN1C2CCC1C(C(C2)OC(=O)c1ccccc1)C(=O)OCCc1ccccc1
Show InChI InChI=1S/C24H27NO4/c1-25-19-12-13-20(25)22(24(27)28-15-14-17-8-4-2-5-9-17)21(16-19)29-23(26)18-10-6-3-7-11-18/h2-11,19-22H,12-16H2,1H3
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n/an/a 615n/an/an/an/an/an/a



Research Triangle Institute

Curated by ChEMBL


Assay Description
Binding affinity at the Serotonin transporter in rat midbrain by inhibition of 0.5 nM [3H]-paroxetine binding


J Med Chem 38: 379-88 (1995)


Article DOI: 10.1021/jm00002a020
BindingDB Entry DOI: 10.7270/Q2D50NM0
More data for this
Ligand-Target Pair
Norepinephrine Monoamine transporters


(Rattus norvegicus)
BDBM50035768
PNG
(3-Benzoyloxy-8-methyl-8-aza-bicyclo[3.2.1]octane-2...)
Show SMILES CN1C2CCC1C(C(C2)OC(=O)c1ccccc1)C(=O)OCCc1ccccc1
Show InChI InChI=1S/C24H27NO4/c1-25-19-12-13-20(25)22(24(27)28-15-14-17-8-4-2-5-9-17)21(16-19)29-23(26)18-10-6-3-7-11-18/h2-11,19-22H,12-16H2,1H3
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n/an/a 1.99E+4n/an/an/an/an/an/a



Research Triangle Institute

Curated by ChEMBL


Assay Description
Binding affinity at the Norepinephrine transporter in rat frontal cortex by inhibition of 0.5 nM [3H]nisoxetine binding


J Med Chem 38: 379-88 (1995)


Article DOI: 10.1021/jm00002a020
BindingDB Entry DOI: 10.7270/Q2D50NM0
More data for this
Ligand-Target Pair
Dopamine Transporter (DAT)


(Rattus norvegicus (rat))
BDBM50035768
PNG
(3-Benzoyloxy-8-methyl-8-aza-bicyclo[3.2.1]octane-2...)
Show SMILES CN1C2CCC1C(C(C2)OC(=O)c1ccccc1)C(=O)OCCc1ccccc1
Show InChI InChI=1S/C24H27NO4/c1-25-19-12-13-20(25)22(24(27)28-15-14-17-8-4-2-5-9-17)21(16-19)29-23(26)18-10-6-3-7-11-18/h2-11,19-22H,12-16H2,1H3
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n/an/a 181n/an/an/an/an/an/a



Research Triangle Institute

Curated by ChEMBL


Assay Description
Binding affinity at the Dopamine transporter in rat striata by inhibition of 0.5 nM [3H]WIN-35428 binding


J Med Chem 38: 379-88 (1995)


Article DOI: 10.1021/jm00002a020
BindingDB Entry DOI: 10.7270/Q2D50NM0
More data for this
Ligand-Target Pair
Dopamine Transporter (DAT)


(Rattus norvegicus (rat))
BDBM50130353
PNG
(3-[Bis-(4-fluoro-phenyl)-methoxy]-8-methyl-8-aza-b...)
Show SMILES CN1C2CCC1[C@H]([C@H](C2)OC(c1ccc(F)cc1)c1ccc(F)cc1)C(=O)OCCc1ccc(cc1)[N+]([O-])=O
Show InChI InChI=1S/C30H30F2N2O5/c1-33-25-14-15-26(33)28(30(35)38-17-16-19-2-12-24(13-3-19)34(36)37)27(18-25)39-29(20-4-8-22(31)9-5-20)21-6-10-23(32)11-7-21/h2-13,25-29H,14-18H2,1H3/t25?,26?,27-,28+/m0/s1
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n/an/a 3.30n/an/an/an/an/an/a



National Institute on Drug Abuse

Curated by ChEMBL


Assay Description
In vitro potency for inhibiting [3H]- dopamine uptake was determined


J Med Chem 46: 2908-16 (2003)


Article DOI: 10.1021/jm0300375
BindingDB Entry DOI: 10.7270/Q2BG2PQ0
More data for this
Ligand-Target Pair
Dopamine Transporter (DAT)


(Rattus norvegicus (rat))
BDBM50008038
PNG
(3-Benzoyloxy-8-methyl-8-aza-bicyclo[3.2.1]octane-2...)
Show SMILES CN1[C@@H]2CCC1C([C@H](C2)OC(=O)c1ccccc1)C(=O)OCCc1ccccc1
Show InChI InChI=1S/C24H27NO4/c1-25-19-12-13-20(25)22(24(27)28-15-14-17-8-4-2-5-9-17)21(16-19)29-23(26)18-10-6-3-7-11-18/h2-11,19-22H,12-16H2,1H3/t19-,20?,21+,22?/m1/s1
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n/an/a 248n/an/an/an/an/an/a



Research Triangle Institute

Curated by ChEMBL


Assay Description
Inhibition of [3H]3-beta-(p-fluorophenyl)tropane-2beta-carboxylic acid methyl ester binding to Dopamine transporter in rat striatal membranes.


J Med Chem 35: 135-40 (1992)


Article DOI: 10.1021/jm00079a017
BindingDB Entry DOI: 10.7270/Q2FQ9X7M
More data for this
Ligand-Target Pair
Dopamine Transporter (DAT)


(Rattus norvegicus (rat))
BDBM50008042
PNG
(3-Benzoyloxy-8-methyl-8-aza-bicyclo[3.2.1]octane-2...)
Show SMILES CN1[C@@H]2CCC1C([C@H](C2)OC(=O)c1ccccc1)C(=O)OCCc1ccc(cc1)N=C=S
Show InChI InChI=1S/C25H26N2O4S/c1-27-20-11-12-21(27)23(22(15-20)31-24(28)18-5-3-2-4-6-18)25(29)30-14-13-17-7-9-19(10-8-17)26-16-32/h2-10,20-23H,11-15H2,1H3/t20-,21?,22+,23?/m1/s1
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n/an/a 196n/an/an/an/an/an/a



Research Triangle Institute

Curated by ChEMBL


Assay Description
Inhibition of [3H]3-beta-(p-fluorophenyl)tropane-2beta-carboxylic acid methyl ester binding to Dopamine transporter in rat striatal membranes.


J Med Chem 35: 135-40 (1992)


Article DOI: 10.1021/jm00079a017
BindingDB Entry DOI: 10.7270/Q2FQ9X7M
More data for this
Ligand-Target Pair