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8 similar compounds to monomer 50010271

Compile data set for download or QSAR
Wt: 644.7
BDBM50010259
Wt: 630.7
BDBM50010262
Wt: 602.7
BDBM50010265
Wt: 658.8
BDBM50010266
Wt: 531.6
BDBM50010269
Wt: 658.8
BDBM50010272
Wt: 672.8
BDBM50010273
Wt: 602.7
BDBM50010275

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 18 hits for monomerid = 50010259,50010262,50010265,50010266,50010269,50010272,50010273,50010275   
Target/Host
(Institution)
LigandTarget/Host
Links
Ligand
Links
Trg + Lig
Links
Ki
nM
ΔG°
kcal/mole
IC50
nM
Kd
nM
EC50/IC50
nM
koff
s-1
kon
M-1s-1
pHTemp
°C
Glucose Transporter 1 (hGLUT1)


(Homo sapiens (Human))
BDBM50010259
PNG
(Acetic acid 10,10b-dihydroxy-6-{2-[3-(4-hydroxy-ph...)
Show SMILES CC(=O)O[C@H]1[C@@H](OC(=O)NCCNC(=O)CCc2ccc(O)cc2)[C@H]2C(C)(C)CC[C@H](O)[C@]2(C)[C@@]2(O)C(=O)C[C@@](C)(O[C@]12C)C=C
Show InChI InChI=1S/C34H48N2O10/c1-8-31(5)19-24(40)34(43)32(6)23(39)15-16-30(3,4)27(32)26(28(44-20(2)37)33(34,7)46-31)45-29(42)36-18-17-35-25(41)14-11-21-9-12-22(38)13-10-21/h8-10,12-13,23,26-28,38-39,43H,1,11,14-19H2,2-7H3,(H,35,41)(H,36,42)/t23-,26-,27-,28-,31-,32-,33+,34-/m0/s1
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n/an/an/a 2.80E+3n/an/an/an/an/a



Food and Drug Administration

Curated by ChEMBL


Assay Description
Inhibition of [125I]-7-IHPP-Fsk binding to glucose transporter of human erythrocyte membrane


J Med Chem 34: 3204-12 (1991)


Article DOI: 10.1021/jm00115a009
BindingDB Entry DOI: 10.7270/Q20C4TRQ
More data for this
Ligand-Target Pair
Adenylate cyclase


(Homo sapiens)
BDBM50010269
PNG
(CHEMBL327672 | [2-(4-Hydroxy-phenyl)-ethyl]-carbam...)
Show SMILES CC1(C)CC[C@H](O)[C@@]2(C)[C@H]1[C@H](O)[C@H](OC(=O)NCCc1ccc(O)cc1)[C@@]1(C)O[C@](C)(CC(=O)[C@]21O)C=C
Show InChI InChI=1S/C29H41NO8/c1-7-26(4)16-20(33)29(36)27(5)19(32)12-14-25(2,3)22(27)21(34)23(28(29,6)38-26)37-24(35)30-15-13-17-8-10-18(31)11-9-17/h7-11,19,21-23,31-32,34,36H,1,12-16H2,2-6H3,(H,30,35)/t19-,21-,22-,23-,26-,27-,28+,29-/m0/s1
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n/an/a 95n/an/an/an/an/an/a



Food and Drug Administration

Curated by ChEMBL


Assay Description
Inhibition of [125 I]-6-IHPP-forskolin binding to adenylate cyclase 1


J Med Chem 39: 2745-52 (1996)


Article DOI: 10.1021/jm960191+
BindingDB Entry DOI: 10.7270/Q2X34WJG
More data for this
Ligand-Target Pair
Adenylate cyclase type I


(Bos taurus)
BDBM50010259
PNG
(Acetic acid 10,10b-dihydroxy-6-{2-[3-(4-hydroxy-ph...)
Show SMILES CC(=O)O[C@H]1[C@@H](OC(=O)NCCNC(=O)CCc2ccc(O)cc2)[C@H]2C(C)(C)CC[C@H](O)[C@]2(C)[C@@]2(O)C(=O)C[C@@](C)(O[C@]12C)C=C
Show InChI InChI=1S/C34H48N2O10/c1-8-31(5)19-24(40)34(43)32(6)23(39)15-16-30(3,4)27(32)26(28(44-20(2)37)33(34,7)46-31)45-29(42)36-18-17-35-25(41)14-11-21-9-12-22(38)13-10-21/h8-10,12-13,23,26-28,38-39,43H,1,11,14-19H2,2-7H3,(H,35,41)(H,36,42)/t23-,26-,27-,28-,31-,32-,33+,34-/m0/s1
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Food and Drug Administration

Curated by ChEMBL


Assay Description
Displacement of [125I]-6-IHPP-Fsk from adenylate cyclase of bovine brain membrane


J Med Chem 34: 3204-12 (1991)


Article DOI: 10.1021/jm00115a009
BindingDB Entry DOI: 10.7270/Q20C4TRQ
More data for this
Ligand-Target Pair
Glucose Transporter 1 (hGLUT1)


(Homo sapiens (Human))
BDBM50010265
PNG
(CHEMBL327142 | {2-[3-(4-Hydroxy-phenyl)-propionyla...)
Show SMILES CC1(C)CC[C@H](O)[C@@]2(C)[C@H]1[C@H](O)[C@H](OC(=O)NCCNC(=O)CCc1ccc(O)cc1)[C@@]1(C)O[C@](C)(CC(=O)[C@]21O)C=C
Show InChI InChI=1S/C32H46N2O9/c1-7-29(4)18-22(37)32(41)30(5)21(36)14-15-28(2,3)25(30)24(39)26(31(32,6)43-29)42-27(40)34-17-16-33-23(38)13-10-19-8-11-20(35)12-9-19/h7-9,11-12,21,24-26,35-36,39,41H,1,10,13-18H2,2-6H3,(H,33,38)(H,34,40)/t21-,24-,25-,26-,29-,30-,31+,32-/m0/s1
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n/an/an/a 1.10E+3n/an/an/an/an/a



Food and Drug Administration

Curated by ChEMBL


Assay Description
Inhibition of [125I]-7-IHPP-Fsk binding to glucose transporter of human erythrocyte membrane


J Med Chem 34: 3204-12 (1991)


Article DOI: 10.1021/jm00115a009
BindingDB Entry DOI: 10.7270/Q20C4TRQ
More data for this
Ligand-Target Pair
Glucose Transporter 1 (hGLUT1)


(Homo sapiens (Human))
BDBM50010266
PNG
(CHEMBL324659 | {6-[3-(4-Hydroxy-phenyl)-propionyla...)
Show SMILES CC1(C)CC[C@H](O)[C@@]2(C)[C@H]1[C@H](O)[C@H](OC(=O)NCCCCCCNC(=O)CCc1ccc(O)cc1)[C@@]1(C)O[C@](C)(CC(=O)[C@]21O)C=C
Show InChI InChI=1S/C36H54N2O9/c1-7-33(4)22-26(41)36(45)34(5)25(40)18-19-32(2,3)29(34)28(43)30(35(36,6)47-33)46-31(44)38-21-11-9-8-10-20-37-27(42)17-14-23-12-15-24(39)16-13-23/h7,12-13,15-16,25,28-30,39-40,43,45H,1,8-11,14,17-22H2,2-6H3,(H,37,42)(H,38,44)/t25-,28-,29-,30-,33-,34-,35+,36-/m0/s1
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Food and Drug Administration

Curated by ChEMBL


Assay Description
Inhibition of [125I]-7-IHPP-Fsk binding to glucose transporter of human erythrocyte membrane


J Med Chem 34: 3204-12 (1991)


Article DOI: 10.1021/jm00115a009
BindingDB Entry DOI: 10.7270/Q20C4TRQ
More data for this
Ligand-Target Pair
Adenylate cyclase type I


(Bos taurus)
BDBM50010269
PNG
(CHEMBL327672 | [2-(4-Hydroxy-phenyl)-ethyl]-carbam...)
Show SMILES CC1(C)CC[C@H](O)[C@@]2(C)[C@H]1[C@H](O)[C@H](OC(=O)NCCc1ccc(O)cc1)[C@@]1(C)O[C@](C)(CC(=O)[C@]21O)C=C
Show InChI InChI=1S/C29H41NO8/c1-7-26(4)16-20(33)29(36)27(5)19(32)12-14-25(2,3)22(27)21(34)23(28(29,6)38-26)37-24(35)30-15-13-17-8-10-18(31)11-9-17/h7-11,19,21-23,31-32,34,36H,1,12-16H2,2-6H3,(H,30,35)/t19-,21-,22-,23-,26-,27-,28+,29-/m0/s1
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n/an/an/a 61n/an/an/an/an/a



Food and Drug Administration

Curated by ChEMBL


Assay Description
Displacement of [125I]-6-IHPP-Fsk from adenylate cyclase of bovine brain membrane


J Med Chem 34: 3204-12 (1991)


Article DOI: 10.1021/jm00115a009
BindingDB Entry DOI: 10.7270/Q20C4TRQ
More data for this
Ligand-Target Pair
Adenylate cyclase type I


(Bos taurus)
BDBM50010272
PNG
(CHEMBL322952 | {6-[3-(4-Hydroxy-phenyl)-propionyla...)
Show SMILES CC1(C)CC[C@H](O)[C@@]2(C)[C@H]1[C@H](OC(=O)NCCCCCCNC(=O)CCc1ccc(O)cc1)[C@H](O)[C@@]1(C)O[C@](C)(CC(=O)[C@]21O)C=C
Show InChI InChI=1S/C36H54N2O9/c1-7-33(4)22-26(41)36(45)34(5)25(40)18-19-32(2,3)29(34)28(30(43)35(36,6)47-33)46-31(44)38-21-11-9-8-10-20-37-27(42)17-14-23-12-15-24(39)16-13-23/h7,12-13,15-16,25,28-30,39-40,43,45H,1,8-11,14,17-22H2,2-6H3,(H,37,42)(H,38,44)/t25-,28-,29-,30-,33-,34-,35+,36-/m0/s1
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Food and Drug Administration

Curated by ChEMBL


Assay Description
Displacement of [125I]-6-IHPP-Fsk from adenylate cyclase of bovine brain membrane


J Med Chem 34: 3204-12 (1991)


Article DOI: 10.1021/jm00115a009
BindingDB Entry DOI: 10.7270/Q20C4TRQ
More data for this
Ligand-Target Pair
Glucose Transporter 1 (hGLUT1)


(Homo sapiens (Human))
BDBM50010273
PNG
(CHEMBL111738 | {7-[3-(4-Hydroxy-phenyl)-propionyla...)
Show SMILES CC1(C)CC[C@H](O)[C@@]2(C)[C@H]1[C@H](O)[C@H](OC(=O)NCCCCCCCNC(=O)CCc1ccc(O)cc1)[C@@]1(C)O[C@](C)(CC(=O)[C@]21O)C=C
Show InChI InChI=1S/C37H56N2O9/c1-7-34(4)23-27(42)37(46)35(5)26(41)19-20-33(2,3)30(35)29(44)31(36(37,6)48-34)47-32(45)39-22-12-10-8-9-11-21-38-28(43)18-15-24-13-16-25(40)17-14-24/h7,13-14,16-17,26,29-31,40-41,44,46H,1,8-12,15,18-23H2,2-6H3,(H,38,43)(H,39,45)/t26-,29-,30-,31-,34-,35-,36+,37-/m0/s1
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n/an/an/a 100n/an/an/an/an/a



Food and Drug Administration

Curated by ChEMBL


Assay Description
Inhibition of [125I]-7-IHPP-Fsk binding to glucose transporter of human erythrocyte membrane


J Med Chem 34: 3204-12 (1991)


Article DOI: 10.1021/jm00115a009
BindingDB Entry DOI: 10.7270/Q20C4TRQ
More data for this
Ligand-Target Pair
Adenylate cyclase type I


(Bos taurus)
BDBM50010266
PNG
(CHEMBL324659 | {6-[3-(4-Hydroxy-phenyl)-propionyla...)
Show SMILES CC1(C)CC[C@H](O)[C@@]2(C)[C@H]1[C@H](O)[C@H](OC(=O)NCCCCCCNC(=O)CCc1ccc(O)cc1)[C@@]1(C)O[C@](C)(CC(=O)[C@]21O)C=C
Show InChI InChI=1S/C36H54N2O9/c1-7-33(4)22-26(41)36(45)34(5)25(40)18-19-32(2,3)29(34)28(43)30(35(36,6)47-33)46-31(44)38-21-11-9-8-10-20-37-27(42)17-14-23-12-15-24(39)16-13-23/h7,12-13,15-16,25,28-30,39-40,43,45H,1,8-11,14,17-22H2,2-6H3,(H,37,42)(H,38,44)/t25-,28-,29-,30-,33-,34-,35+,36-/m0/s1
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n/an/an/a 82n/an/an/an/an/a



Food and Drug Administration

Curated by ChEMBL


Assay Description
Displacement of [125I]-6-IHPP-Fsk from adenylate cyclase of bovine brain membrane


J Med Chem 34: 3204-12 (1991)


Article DOI: 10.1021/jm00115a009
BindingDB Entry DOI: 10.7270/Q20C4TRQ
More data for this
Ligand-Target Pair
Adenylate cyclase type I


(Bos taurus)
BDBM50010273
PNG
(CHEMBL111738 | {7-[3-(4-Hydroxy-phenyl)-propionyla...)
Show SMILES CC1(C)CC[C@H](O)[C@@]2(C)[C@H]1[C@H](O)[C@H](OC(=O)NCCCCCCCNC(=O)CCc1ccc(O)cc1)[C@@]1(C)O[C@](C)(CC(=O)[C@]21O)C=C
Show InChI InChI=1S/C37H56N2O9/c1-7-34(4)23-27(42)37(46)35(5)26(41)19-20-33(2,3)30(35)29(44)31(36(37,6)48-34)47-32(45)39-22-12-10-8-9-11-21-38-28(43)18-15-24-13-16-25(40)17-14-24/h7,13-14,16-17,26,29-31,40-41,44,46H,1,8-12,15,18-23H2,2-6H3,(H,38,43)(H,39,45)/t26-,29-,30-,31-,34-,35-,36+,37-/m0/s1
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n/an/an/a 53n/an/an/an/an/a



Food and Drug Administration

Curated by ChEMBL


Assay Description
Displacement of [125I]-6-IHPP-Fsk from adenylate cyclase of bovine brain membrane


J Med Chem 34: 3204-12 (1991)


Article DOI: 10.1021/jm00115a009
BindingDB Entry DOI: 10.7270/Q20C4TRQ
More data for this
Ligand-Target Pair
Glucose Transporter 1 (hGLUT1)


(Homo sapiens (Human))
BDBM50010272
PNG
(CHEMBL322952 | {6-[3-(4-Hydroxy-phenyl)-propionyla...)
Show SMILES CC1(C)CC[C@H](O)[C@@]2(C)[C@H]1[C@H](OC(=O)NCCCCCCNC(=O)CCc1ccc(O)cc1)[C@H](O)[C@@]1(C)O[C@](C)(CC(=O)[C@]21O)C=C
Show InChI InChI=1S/C36H54N2O9/c1-7-33(4)22-26(41)36(45)34(5)25(40)18-19-32(2,3)29(34)28(30(43)35(36,6)47-33)46-31(44)38-21-11-9-8-10-20-37-27(42)17-14-23-12-15-24(39)16-13-23/h7,12-13,15-16,25,28-30,39-40,43,45H,1,8-11,14,17-22H2,2-6H3,(H,37,42)(H,38,44)/t25-,28-,29-,30-,33-,34-,35+,36-/m0/s1
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Food and Drug Administration

Curated by ChEMBL


Assay Description
Inhibition of [125I]-7-IHPP-Fsk binding to glucose transporter of human erythrocyte membrane


J Med Chem 34: 3204-12 (1991)


Article DOI: 10.1021/jm00115a009
BindingDB Entry DOI: 10.7270/Q20C4TRQ
More data for this
Ligand-Target Pair
Adenylate cyclase type I


(Bos taurus)
BDBM50010265
PNG
(CHEMBL327142 | {2-[3-(4-Hydroxy-phenyl)-propionyla...)
Show SMILES CC1(C)CC[C@H](O)[C@@]2(C)[C@H]1[C@H](O)[C@H](OC(=O)NCCNC(=O)CCc1ccc(O)cc1)[C@@]1(C)O[C@](C)(CC(=O)[C@]21O)C=C
Show InChI InChI=1S/C32H46N2O9/c1-7-29(4)18-22(37)32(41)30(5)21(36)14-15-28(2,3)25(30)24(39)26(31(32,6)43-29)42-27(40)34-17-16-33-23(38)13-10-19-8-11-20(35)12-9-19/h7-9,11-12,21,24-26,35-36,39,41H,1,10,13-18H2,2-6H3,(H,33,38)(H,34,40)/t21-,24-,25-,26-,29-,30-,31+,32-/m0/s1
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n/an/an/a 13n/an/an/an/an/a



Food and Drug Administration

Curated by ChEMBL


Assay Description
Displacement of [125I]-6-IHPP-Fsk from adenylate cyclase of bovine brain membrane


J Med Chem 34: 3204-12 (1991)


Article DOI: 10.1021/jm00115a009
BindingDB Entry DOI: 10.7270/Q20C4TRQ
More data for this
Ligand-Target Pair
Glucose Transporter 1 (hGLUT1)


(Homo sapiens (Human))
BDBM50010275
PNG
(CHEMBL324463 | {2-[3-(4-Hydroxy-phenyl)-propionyla...)
Show SMILES CC1(C)CC[C@H](O)[C@@]2(C)[C@H]1[C@H](OC(=O)NCCNC(=O)CCc1ccc(O)cc1)[C@H](O)[C@@]1(C)O[C@](C)(CC(=O)[C@]21O)C=C
Show InChI InChI=1S/C32H46N2O9/c1-7-29(4)18-22(37)32(41)30(5)21(36)14-15-28(2,3)25(30)24(26(39)31(32,6)43-29)42-27(40)34-17-16-33-23(38)13-10-19-8-11-20(35)12-9-19/h7-9,11-12,21,24-26,35-36,39,41H,1,10,13-18H2,2-6H3,(H,33,38)(H,34,40)/t21-,24-,25-,26-,29-,30-,31+,32-/m0/s1
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n/an/an/a>1.00E+5n/an/an/an/an/a



Food and Drug Administration

Curated by ChEMBL


Assay Description
Inhibition of [125I]-7-IHPP-Fsk binding to glucose transporter of human erythrocyte membrane


J Med Chem 34: 3204-12 (1991)


Article DOI: 10.1021/jm00115a009
BindingDB Entry DOI: 10.7270/Q20C4TRQ
More data for this
Ligand-Target Pair
Glucose Transporter 1 (hGLUT1)


(Homo sapiens (Human))
BDBM50010269
PNG
(CHEMBL327672 | [2-(4-Hydroxy-phenyl)-ethyl]-carbam...)
Show SMILES CC1(C)CC[C@H](O)[C@@]2(C)[C@H]1[C@H](O)[C@H](OC(=O)NCCc1ccc(O)cc1)[C@@]1(C)O[C@](C)(CC(=O)[C@]21O)C=C
Show InChI InChI=1S/C29H41NO8/c1-7-26(4)16-20(33)29(36)27(5)19(32)12-14-25(2,3)22(27)21(34)23(28(29,6)38-26)37-24(35)30-15-13-17-8-10-18(31)11-9-17/h7-11,19,21-23,31-32,34,36H,1,12-16H2,2-6H3,(H,30,35)/t19-,21-,22-,23-,26-,27-,28+,29-/m0/s1
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n/an/an/a 240n/an/an/an/an/a



Food and Drug Administration

Curated by ChEMBL


Assay Description
Inhibition of [125I]-7-IHPP-Fsk binding to glucose transporter of human erythrocyte membrane


J Med Chem 34: 3204-12 (1991)


Article DOI: 10.1021/jm00115a009
BindingDB Entry DOI: 10.7270/Q20C4TRQ
More data for this
Ligand-Target Pair
Adenylate cyclase type I


(Bos taurus)
BDBM50010275
PNG
(CHEMBL324463 | {2-[3-(4-Hydroxy-phenyl)-propionyla...)
Show SMILES CC1(C)CC[C@H](O)[C@@]2(C)[C@H]1[C@H](OC(=O)NCCNC(=O)CCc1ccc(O)cc1)[C@H](O)[C@@]1(C)O[C@](C)(CC(=O)[C@]21O)C=C
Show InChI InChI=1S/C32H46N2O9/c1-7-29(4)18-22(37)32(41)30(5)21(36)14-15-28(2,3)25(30)24(26(39)31(32,6)43-29)42-27(40)34-17-16-33-23(38)13-10-19-8-11-20(35)12-9-19/h7-9,11-12,21,24-26,35-36,39,41H,1,10,13-18H2,2-6H3,(H,33,38)(H,34,40)/t21-,24-,25-,26-,29-,30-,31+,32-/m0/s1
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Food and Drug Administration

Curated by ChEMBL


Assay Description
Displacement of [125I]-6-IHPP-Fsk from adenylate cyclase of bovine brain membrane


J Med Chem 34: 3204-12 (1991)


Article DOI: 10.1021/jm00115a009
BindingDB Entry DOI: 10.7270/Q20C4TRQ
More data for this
Ligand-Target Pair
Adenylate cyclase type I


(Bos taurus)
BDBM50010262
PNG
(CHEMBL326703 | {4-[3-(4-Hydroxy-phenyl)-propionyla...)
Show SMILES CC1(C)CC[C@H](O)[C@@]2(C)[C@H]1[C@H](OC(=O)NCCCCNC(=O)CCc1ccc(O)cc1)[C@H](O)[C@@]1(C)O[C@](C)(CC(=O)[C@]21O)C=C
Show InChI InChI=1S/C34H50N2O9/c1-7-31(4)20-24(39)34(43)32(5)23(38)16-17-30(2,3)27(32)26(28(41)33(34,6)45-31)44-29(42)36-19-9-8-18-35-25(40)15-12-21-10-13-22(37)14-11-21/h7,10-11,13-14,23,26-28,37-38,41,43H,1,8-9,12,15-20H2,2-6H3,(H,35,40)(H,36,42)/t23-,26-,27-,28-,31-,32-,33+,34-/m0/s1
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n/an/an/a 80n/an/an/an/an/a



Food and Drug Administration

Curated by ChEMBL


Assay Description
Displacement of [125I]-6-IHPP-Fsk from adenylate cyclase of bovine brain membrane


J Med Chem 34: 3204-12 (1991)


Article DOI: 10.1021/jm00115a009
BindingDB Entry DOI: 10.7270/Q20C4TRQ
More data for this
Ligand-Target Pair
Adenylate cyclase


(Homo sapiens)
BDBM50010269
PNG
(CHEMBL327672 | [2-(4-Hydroxy-phenyl)-ethyl]-carbam...)
Show SMILES CC1(C)CC[C@H](O)[C@@]2(C)[C@H]1[C@H](O)[C@H](OC(=O)NCCc1ccc(O)cc1)[C@@]1(C)O[C@](C)(CC(=O)[C@]21O)C=C
Show InChI InChI=1S/C29H41NO8/c1-7-26(4)16-20(33)29(36)27(5)19(32)12-14-25(2,3)22(27)21(34)23(28(29,6)38-26)37-24(35)30-15-13-17-8-10-18(31)11-9-17/h7-11,19,21-23,31-32,34,36H,1,12-16H2,2-6H3,(H,30,35)/t19-,21-,22-,23-,26-,27-,28+,29-/m0/s1
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n/an/an/an/a 1.40E+3n/an/an/an/a



Food and Drug Administration

Curated by ChEMBL


Assay Description
Conversion of [32P] ATP to [32P]-cyclic AMP mediated by adenylate cyclase 1


J Med Chem 39: 2745-52 (1996)


Article DOI: 10.1021/jm960191+
BindingDB Entry DOI: 10.7270/Q2X34WJG
More data for this
Ligand-Target Pair
Glucose Transporter 1 (hGLUT1)


(Homo sapiens (Human))
BDBM50010262
PNG
(CHEMBL326703 | {4-[3-(4-Hydroxy-phenyl)-propionyla...)
Show SMILES CC1(C)CC[C@H](O)[C@@]2(C)[C@H]1[C@H](OC(=O)NCCCCNC(=O)CCc1ccc(O)cc1)[C@H](O)[C@@]1(C)O[C@](C)(CC(=O)[C@]21O)C=C
Show InChI InChI=1S/C34H50N2O9/c1-7-31(4)20-24(39)34(43)32(5)23(38)16-17-30(2,3)27(32)26(28(41)33(34,6)45-31)44-29(42)36-19-9-8-18-35-25(40)15-12-21-10-13-22(37)14-11-21/h7,10-11,13-14,23,26-28,37-38,41,43H,1,8-9,12,15-20H2,2-6H3,(H,35,40)(H,36,42)/t23-,26-,27-,28-,31-,32-,33+,34-/m0/s1
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n/an/an/a>1.00E+5n/an/an/an/an/a



Food and Drug Administration

Curated by ChEMBL


Assay Description
Inhibition of [125I]-7-IHPP-Fsk binding to glucose transporter of human erythrocyte membrane


J Med Chem 34: 3204-12 (1991)


Article DOI: 10.1021/jm00115a009
BindingDB Entry DOI: 10.7270/Q20C4TRQ
More data for this
Ligand-Target Pair