Compounds in cluster

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There are 5 purchasable compounds for target: ATP-dependent RNA helicase DDX1

Wt: 302.2
BDBM82820

Wt: 375.4
BDBM50379306

Wt: 242.2
BDBM50379301

Wt: 374.4
BDBM50379303

Wt: 353.3
BDBM50379304

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 5 hits for monomerid = 82820,50379306,50379301,50379303,50379304
Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kcal/mole	IC50 nM	Kd nM	EC50/IC50 nM	k_off s^-1	k_on M^-1s^-1	pH	Temp °C
ATP-dependent RNA helicase DDX1 (Homo sapiens)	BDBM82820 (1,3-bis(3-nitrophenyl)urea \| MLS000719904 \| N,N...) Show SMILES Show InChI	PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet	Purchase PC cid PC sid UniChem	Article PubMed	n/a	n/a	>5.00E+5	n/a	n/a	n/a	n/a	n/a	n/a
University of Siena Curated by ChEMBL					Assay Description Inhibition of human recombinant DDX1 helicase activity expressed in Escherichia coli assessed as conversion of a 6-FAM-labeled double stranded RNA in...				Bioorg Med Chem Lett 22: 2094-8 (2012) Article DOI: 10.1016/j.bmcl.2011.12.135 BindingDB Entry DOI: 10.7270/Q2930V51
University of Siena Curated by ChEMBL					More data for this Ligand-Target Pair
ATP-dependent RNA helicase DDX1 (Homo sapiens)	BDBM50379301 (CHEMBL2011809) Show SMILES Nc1cccc(NC(=O)Nc2cccc(N)c2)c1 Show InChI	PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet	Purchase CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	>5.00E+5	n/a	n/a	n/a	n/a	n/a	n/a
University of Siena Curated by ChEMBL					Assay Description Inhibition of human recombinant DDX1 helicase activity expressed in Escherichia coli assessed as conversion of a 6-FAM-labeled double stranded RNA in...				Bioorg Med Chem Lett 22: 2094-8 (2012) Article DOI: 10.1016/j.bmcl.2011.12.135 BindingDB Entry DOI: 10.7270/Q2930V51
University of Siena Curated by ChEMBL					More data for this Ligand-Target Pair
ATP-dependent RNA helicase DDX1 (Homo sapiens)	BDBM50379306 (CHEMBL2011806) Show SMILES Show InChI	PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet	Purchase CHEMBL PC cid PC sid UniChem	Article PubMed	n/a	n/a	>5.00E+5	n/a	n/a	n/a	n/a	n/a	n/a
University of Siena Curated by ChEMBL					Assay Description Inhibition of human recombinant DDX1 helicase activity expressed in Escherichia coli assessed as conversion of a 6-FAM-labeled double stranded RNA in...				Bioorg Med Chem Lett 22: 2094-8 (2012) Article DOI: 10.1016/j.bmcl.2011.12.135 BindingDB Entry DOI: 10.7270/Q2930V51
University of Siena Curated by ChEMBL					More data for this Ligand-Target Pair
ATP-dependent RNA helicase DDX1 (Homo sapiens)	BDBM50379304 (CHEMBL2011805) Show SMILES Show InChI	PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	>5.00E+5	n/a	n/a	n/a	n/a	n/a	n/a
University of Siena Curated by ChEMBL					Assay Description Inhibition of human recombinant DDX1 helicase activity expressed in Escherichia coli assessed as conversion of a 6-FAM-labeled double stranded RNA in...				Bioorg Med Chem Lett 22: 2094-8 (2012) Article DOI: 10.1016/j.bmcl.2011.12.135 BindingDB Entry DOI: 10.7270/Q2930V51
University of Siena Curated by ChEMBL					More data for this Ligand-Target Pair
ATP-dependent RNA helicase DDX1 (Homo sapiens)	BDBM50379303 (CHEMBL2011804) Show SMILES Show InChI	PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	>5.00E+5	n/a	n/a	n/a	n/a	n/a	n/a
University of Siena Curated by ChEMBL					Assay Description Inhibition of human recombinant DDX1 helicase activity expressed in Escherichia coli assessed as conversion of a 6-FAM-labeled double stranded RNA in...				Bioorg Med Chem Lett 22: 2094-8 (2012) Article DOI: 10.1016/j.bmcl.2011.12.135 BindingDB Entry DOI: 10.7270/Q2930V51
University of Siena Curated by ChEMBL					More data for this Ligand-Target Pair