Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 103 hits in this display
BDBM13212((3S,6S,9aS)-N-(diphenylmethyl)-6-[(2S)-2-(methylam...)
BDBM13212((3S,6S,9aS)-N-(diphenylmethyl)-6-[(2S)-2-(methylam...)
Ki: 4.80nM ΔG°: -47.0kJ/molepH: 7.5 T: 2°CAssay Description:Fluorescence polarization was measured on an Ultra plate reader at excitation and emission wavelengths of 485 and 530 nm, respectively. The equilibri...More data for this Ligand-Target Pair
BDBM13211((3S,6S,9aS)-6-[(2S)-2-aminobutanamido]-N-(diphenyl...)
BDBM13211((3S,6S,9aS)-6-[(2S)-2-aminobutanamido]-N-(diphenyl...)
BDBM13211((3S,6S,9aS)-6-[(2S)-2-aminobutanamido]-N-(diphenyl...)
BDBM26212((3S,6S,9aS)-6-[(2S)-2-aminopropanamido]-N-(dipheny...)Ki: 60nM ΔG°: -40.8kJ/molepH: 7.5 T: 2°CAssay Description:Fluorescence polarization was measured on an Ultra plate reader at excitation and emission wavelengths of 485 and 530 nm, respectively. The equilibri...More data for this Ligand-Target Pair
BDBM13212((3S,6S,9aS)-N-(diphenylmethyl)-6-[(2S)-2-(methylam...)
Ki: 61nM ΔG°: -40.9kJ/mole IC50: 530nMpH: 7.5 T: 2°CAssay Description:Fluorescence polarization was measured on an Ultra plate reader (Tecan) at excitation and emission wavelengths of 485 and 530 nm, respectively. The e...More data for this Ligand-Target Pair
BDBM13212((3S,6S,9aS)-N-(diphenylmethyl)-6-[(2S)-2-(methylam...)
Ki: 61nM ΔG°: -40.8kJ/molepH: 7.5 T: 2°CAssay Description:Fluorescence polarization was measured on an Ultra plate reader at excitation and emission wavelengths of 485 and 530 nm, respectively. The equilibri...More data for this Ligand-Target Pair
BDBM13212((3S,6S,9aS)-N-(diphenylmethyl)-6-[(2S)-2-(methylam...)
Ki: 61nM ΔG°: -40.8kJ/molepH: 7.5 T: 2°CAssay Description:A quantitative in vitro binding assay using the fluorescence polarization (FP) based method was developed and used to determine the binding affinity ...More data for this Ligand-Target Pair
BDBM13212((3S,6S,9aS)-N-(diphenylmethyl)-6-[(2S)-2-(methylam...)
Ki: 61nM ΔG°: -40.8kJ/molepH: 7.5 T: 2°CAssay Description:Fluorescence polarization was measured on an Ultra plate reader at excitation and emission wavelengths of 485 and 530 nm, respectively. The equilibri...More data for this Ligand-Target Pair
BDBM26205((3S,6S,7R,9aS)-6-[(2S)-2-aminobutanamido]-7-(2-ami...)
BDBM13211((3S,6S,9aS)-6-[(2S)-2-aminobutanamido]-N-(diphenyl...)
Ki: 420nM ΔG°: -36.0kJ/mole IC50: 460nMpH: 7.5 T: 2°CAssay Description:Fluorescence polarization was measured on an Ultra plate reader (Tecan) at excitation and emission wavelengths of 485 and 530 nm, respectively. The e...More data for this Ligand-Target Pair
BDBM26204((3S,6S,7R,9aS)-6-[(2S)-2-aminobutanamido]-7-(amino...)Ki: 870nM ΔG°: -34.2kJ/mole IC50: 970nMpH: 7.5 T: 2°CAssay Description:Fluorescence polarization was measured on an Ultra plate reader (Tecan) at excitation and emission wavelengths of 485 and 530 nm, respectively. The e...More data for this Ligand-Target Pair
BDBM13213((3S,6S,9aS)-6-[(2S)-2-(dimethylamino)butanamido]-N...)Ki: 1.44E+4nM ΔG°: -27.4kJ/molepH: 7.5 T: 2°CAssay Description:Fluorescence polarization was measured on an Ultra plate reader at excitation and emission wavelengths of 485 and 530 nm, respectively. The equilibri...More data for this Ligand-Target Pair
BDBM13213((3S,6S,9aS)-6-[(2S)-2-(dimethylamino)butanamido]-N...)
Ki: 1.44E+4nM ΔG°: -27.4kJ/molepH: 7.5 T: 2°CAssay Description:A quantitative in vitro binding assay using the fluorescence polarization (FP) based method was developed and used to determine the binding affinity ...More data for this Ligand-Target Pair
IC50: 1.40nMAssay Description:Displacement of FITC-Smac from human recombinant His-tagged cIAP-1 BIR3 domain (245 to 357 residues) after 3 hrs by fluorescent polarization assayMore data for this Ligand-Target Pair
BDBM32609(1-aza-2-oxobicyclo[5.3.0]decane scaffold, 36b)
IC50: <2nMAssay Description:Displacement of AbuRPF-K(5-Fam)-NH2 from human recombinant His-tagged-cIAP1 BIR3 domain after 3 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
IC50: <2nMAssay Description:Displacement of AbuRPF-K(5-Fam)-NH2 from human recombinant His-tagged-cIAP1 BIR3 domain after 3 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
IC50: <2nMAssay Description:Displacement of AbuRPF-K(5-Fam)-NH2 from human recombinant His-tagged-cIAP1 BIR3 domain after 3 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
IC50: <2nMAssay Description:Displacement of AbuRPF-K(5-Fam)-NH2 from human recombinant His-tagged-cIAP1 BIR3 domain after 3 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
IC50: <2nMAssay Description:Displacement of AbuRPF-K(5-Fam)-NH2 from human recombinant His-tagged-cIAP1 BIR3 domain after 3 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
IC50: <2nMAssay Description:Displacement of AbuRPF-K(5-Fam)-NH2 from human recombinant His-tagged-cIAP1 BIR3 domain after 3 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
IC50: <2nMAssay Description:Displacement of AbuRPF-K(5-Fam)-NH2 from human recombinant His-tagged-cIAP1 BIR3 domain after 3 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
IC50: <2nMAssay Description:Displacement of AbuRPF-K(5-Fam)-NH2 from human recombinant His-tagged-cIAP1 BIR3 domain after 3 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
IC50: <2nMAssay Description:Displacement of AbuRPF-K(5-Fam)-NH2 from human recombinant His-tagged-cIAP1 BIR3 domain after 3 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
IC50: <2nMAssay Description:Displacement of AbuRPF-K(5-Fam)-NH2 from human recombinant His-tagged-cIAP1 BIR3 domain after 3 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
IC50: <2nMAssay Description:Displacement of AbuRPF-K(5-Fam)-NH2 from human recombinant His-tagged-cIAP1 BIR3 domain after 3 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
IC50: <2nMAssay Description:Displacement of AbuRPF-K(5-Fam)-NH2 from human recombinant His-tagged-cIAP1 BIR3 domain after 3 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
IC50: <2nMAssay Description:Displacement of AbuRPF-K(5-Fam)-NH2 from human recombinant His-tagged-cIAP1 BIR3 domain after 3 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
IC50: <2nMAssay Description:Displacement of AbuRPF-K(5-Fam)-NH2 from human recombinant His-tagged-cIAP1 BIR3 domain after 3 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
IC50: 3.30nMAssay Description:Displacement of AbuRPF-K(5-Fam)-NH2 from human recombinant His-tagged-cIAP1 BIR3 domain after 3 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
IC50: 5.90nMAssay Description:Displacement of Smac-1F from human His-tagged XIAP linker BIR2-BIR3 linker (124 to 356 residues) after 3 hrs by fluorescent polarization assayMore data for this Ligand-Target Pair
BDBM32615(1-aza-2-oxobicyclo[5.3.0]decane scaffold, 40d)
BDBM32589(1-aza-2-oxobicyclo[5.3.0]decane scaffold, 18b | 1-...)IC50: 35nMAssay Description:Fluorescence polarization was measured on an Ultra plate reader (Tecan) at excitation and emission wavelengths of 485 and 530 nm, respectively. The e...More data for this Ligand-Target Pair
IC50: 41nMAssay Description:Displacement of AbuRPF-K(5-Fam)-NH2 from recombinant human His-tagged-XIAP BIR3 domain after 3 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
IC50: 44nMAssay Description:Displacement of AbuRPF-K(5-Fam)-NH2 from recombinant human His-tagged-XIAP BIR3 domain after 3 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
IC50: 47nMAssay Description:Displacement of AbuRPF-K(5-Fam)-NH2 from recombinant human His-tagged-XIAP BIR3 domain after 3 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
IC50: 47nMAssay Description:Displacement of AbuRPF-K(5-Fam)-NH2 from recombinant human His-tagged-XIAP BIR3 domain after 3 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
BDBM32589(1-aza-2-oxobicyclo[5.3.0]decane scaffold, 18b | 1-...)
IC50: 49nMAssay Description:Fluorescence polarization was measured on an Ultra plate reader (Tecan) at excitation and emission wavelengths of 485 and 530 nm, respectively. The e...More data for this Ligand-Target Pair
IC50: 52nMAssay Description:Displacement of AbuRPF-K(5-Fam)-NH2 from recombinant human His-tagged-XIAP BIR3 domain after 3 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
IC50: 52nMAssay Description:Displacement of AbuRPF-K(5-Fam)-NH2 from recombinant human His-tagged-XIAP BIR3 domain after 3 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
IC50: 53nMAssay Description:Displacement of AbuRPF-K(5-Fam)-NH2 from recombinant human His-tagged-XIAP BIR3 domain after 3 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
BDBM32582(1-aza-2-oxobicyclo[5.3.0]decane scaffold, 4b)
BDBM32609(1-aza-2-oxobicyclo[5.3.0]decane scaffold, 36b)
IC50: 55nMAssay Description:Fluorescence polarization was measured on an Ultra plate reader (Tecan) at excitation and emission wavelengths of 485 and 530 nm, respectively. The e...More data for this Ligand-Target Pair
BDBM32588(1-aza-2-oxobicyclo[5.3.0]decane scaffold, 18a | 1-...)IC50: 56nMAssay Description:Fluorescence polarization was measured on an Ultra plate reader (Tecan) at excitation and emission wavelengths of 485 and 530 nm, respectively. The e...More data for this Ligand-Target Pair
IC50: 57nMAssay Description:Displacement of AbuRPF-K(5-Fam)-NH2 from recombinant human His-tagged-XIAP BIR3 domain after 3 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
IC50: 57nMAssay Description:Displacement of AbuRPF-K(5-Fam)-NH2 from recombinant human His-tagged-XIAP BIR3 domain after 3 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
IC50: 58nMAssay Description:Displacement of AbuRPF-K(5-Fam)-NH2 from recombinant human His-tagged-XIAP BIR3 domain after 3 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
BDBM32595(1-aza-2-oxobicyclo[5.3.0]decane scaffold, 22c | 1-...)IC50: 58nMAssay Description:Fluorescence polarization was measured on an Ultra plate reader (Tecan) at excitation and emission wavelengths of 485 and 530 nm, respectively. The e...More data for this Ligand-Target Pair
IC50: 65nMAssay Description:Displacement of AbuRPF-K(5-Fam)-NH2 from recombinant human His-tagged-XIAP BIR3 domain after 3 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
BDBM32606(1-aza-2-oxobicyclo[5.3.0]decane scaffold, 34a)IC50: 70nMAssay Description:Fluorescence polarization was measured on an Ultra plate reader (Tecan) at excitation and emission wavelengths of 485 and 530 nm, respectively. The e...More data for this Ligand-Target Pair
BDBM32613(1-aza-2-oxobicyclo[5.3.0]decane scaffold, 40b)IC50: 70nMAssay Description:Fluorescence polarization was measured on an Ultra plate reader (Tecan) at excitation and emission wavelengths of 485 and 530 nm, respectively. The e...More data for this Ligand-Target Pair
BDBM32589(1-aza-2-oxobicyclo[5.3.0]decane scaffold, 18b | 1-...)
IC50: 72nMAssay Description:Fluorescence polarization was measured on an Ultra plate reader (Tecan) at excitation and emission wavelengths of 485 and 530 nm, respectively. The e...More data for this Ligand-Target Pair
IC50: 78nMAssay Description:Displacement of AbuRPF-K(5-Fam)-NH2 from recombinant human His-tagged-XIAP BIR3 domain after 3 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
BDBM32605(1-aza-2-oxobicyclo[5.3.0]decane scaffold, 32b)IC50: 85nMAssay Description:Fluorescence polarization was measured on an Ultra plate reader (Tecan) at excitation and emission wavelengths of 485 and 530 nm, respectively. The e...More data for this Ligand-Target Pair
BDBM26205((3S,6S,7R,9aS)-6-[(2S)-2-aminobutanamido]-7-(2-ami...)
IC50: 86nMAssay Description:Fluorescence polarization was measured on an Ultra plate reader (Tecan) at excitation and emission wavelengths of 485 and 530 nm, respectively. The e...More data for this Ligand-Target Pair
BDBM32613(1-aza-2-oxobicyclo[5.3.0]decane scaffold, 40b)
IC50: 86nMAssay Description:Fluorescence polarization was measured on an Ultra plate reader (Tecan) at excitation and emission wavelengths of 485 and 530 nm, respectively. The e...More data for this Ligand-Target Pair
BDBM32588(1-aza-2-oxobicyclo[5.3.0]decane scaffold, 18a | 1-...)
IC50: 92nMAssay Description:Fluorescence polarization was measured on an Ultra plate reader (Tecan) at excitation and emission wavelengths of 485 and 530 nm, respectively. The e...More data for this Ligand-Target Pair
BDBM32607(1-aza-2-oxobicyclo[5.3.0]decane scaffold, 34b)IC50: 100nMAssay Description:Fluorescence polarization was measured on an Ultra plate reader (Tecan) at excitation and emission wavelengths of 485 and 530 nm, respectively. The e...More data for this Ligand-Target Pair
BDBM32582(1-aza-2-oxobicyclo[5.3.0]decane scaffold, 4b)
IC50: 100nMpH: 7.5 T: 2°CAssay Description:Fluorescence polarization was measured on an Ultra plate reader (Tecan) at excitation and emission wavelengths of 485 and 530 nm, respectively. The e...More data for this Ligand-Target Pair
IC50: 110nMAssay Description:Displacement of AbuRPF-K(5-Fam)-NH2 from recombinant human His-tagged-XIAP BIR3 domain after 3 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
BDBM32595(1-aza-2-oxobicyclo[5.3.0]decane scaffold, 22c | 1-...)
IC50: 110nMAssay Description:Fluorescence polarization was measured on an Ultra plate reader (Tecan) at excitation and emission wavelengths of 485 and 530 nm, respectively. The e...More data for this Ligand-Target Pair
BDBM32592(1-aza-2-oxobicyclo[5.3.0]decane scaffold, 20c)IC50: 110nMAssay Description:Fluorescence polarization was measured on an Ultra plate reader (Tecan) at excitation and emission wavelengths of 485 and 530 nm, respectively. The e...More data for this Ligand-Target Pair
BDBM32591(1-aza-2-oxobicyclo[5.3.0]decane scaffold, 20b)IC50: 110nMAssay Description:Fluorescence polarization was measured on an Ultra plate reader (Tecan) at excitation and emission wavelengths of 485 and 530 nm, respectively. The e...More data for this Ligand-Target Pair
BDBM26204((3S,6S,7R,9aS)-6-[(2S)-2-aminobutanamido]-7-(amino...)
IC50: 110nMAssay Description:Fluorescence polarization was measured on an Ultra plate reader (Tecan) at excitation and emission wavelengths of 485 and 530 nm, respectively. The e...More data for this Ligand-Target Pair
BDBM32588(1-aza-2-oxobicyclo[5.3.0]decane scaffold, 18a | 1-...)
IC50: 110nMAssay Description:Fluorescence polarization was measured on an Ultra plate reader (Tecan) at excitation and emission wavelengths of 485 and 530 nm, respectively. The e...More data for this Ligand-Target Pair
BDBM32615(1-aza-2-oxobicyclo[5.3.0]decane scaffold, 40d)
IC50: 110nMAssay Description:Fluorescence polarization was measured on an Ultra plate reader (Tecan) at excitation and emission wavelengths of 485 and 530 nm, respectively. The e...More data for this Ligand-Target Pair
IC50: 111nMAssay Description:Displacement of AbuRPF-K(5-Fam)-NH2 from recombinant human His-tagged-XIAP BIR3 domain after 3 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
BDBM32595(1-aza-2-oxobicyclo[5.3.0]decane scaffold, 22c | 1-...)
IC50: 120nMAssay Description:Fluorescence polarization was measured on an Ultra plate reader (Tecan) at excitation and emission wavelengths of 485 and 530 nm, respectively. The e...More data for this Ligand-Target Pair
BDBM32609(1-aza-2-oxobicyclo[5.3.0]decane scaffold, 36b)
IC50: 120nMAssay Description:Fluorescence polarization was measured on an Ultra plate reader (Tecan) at excitation and emission wavelengths of 485 and 530 nm, respectively. The e...More data for this Ligand-Target Pair
BDBM32607(1-aza-2-oxobicyclo[5.3.0]decane scaffold, 34b)
IC50: 130nMAssay Description:Fluorescence polarization was measured on an Ultra plate reader (Tecan) at excitation and emission wavelengths of 485 and 530 nm, respectively. The e...More data for this Ligand-Target Pair
BDBM32605(1-aza-2-oxobicyclo[5.3.0]decane scaffold, 32b)
IC50: 140nMpH: 7.5 T: 2°CAssay Description:Fluorescence polarization was measured on an Ultra plate reader (Tecan) at excitation and emission wavelengths of 485 and 530 nm, respectively. The e...More data for this Ligand-Target Pair
BDBM32590(1-aza-2-oxobicyclo[5.3.0]decane scaffold, 20a)IC50: 150nMAssay Description:Fluorescence polarization was measured on an Ultra plate reader (Tecan) at excitation and emission wavelengths of 485 and 530 nm, respectively. The e...More data for this Ligand-Target Pair
BDBM32593(1-aza-2-oxobicyclo[5.3.0]decane scaffold, 22a)IC50: 150nMAssay Description:Fluorescence polarization was measured on an Ultra plate reader (Tecan) at excitation and emission wavelengths of 485 and 530 nm, respectively. The e...More data for this Ligand-Target Pair
IC50: 181nMAssay Description:Displacement of FITC-Smac from human His-tagged XIAP BIR3 domain (241 to 356 residues) after 3 hrs by fluorescent polarization assayMore data for this Ligand-Target Pair
IC50: 181nMAssay Description:Displacement of AbuRPF-K(5-Fam)-NH2 from recombinant human His-tagged-XIAP BIR3 domain after 3 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
BDBM32594(1-aza-2-oxobicyclo[5.3.0]decane scaffold, 22b)IC50: 190nMAssay Description:Fluorescence polarization was measured on an Ultra plate reader (Tecan) at excitation and emission wavelengths of 485 and 530 nm, respectively. The e...More data for this Ligand-Target Pair
BDBM32588(1-aza-2-oxobicyclo[5.3.0]decane scaffold, 18a | 1-...)
IC50: 240nMpH: 7.5 T: 2°CAssay Description:Fluorescence polarization was measured on an Ultra plate reader (Tecan) at excitation and emission wavelengths of 485 and 530 nm, respectively. The e...More data for this Ligand-Target Pair
BDBM32604(1-aza-2-oxobicyclo[5.3.0]decane scaffold, 31a)IC50: 240nMAssay Description:Fluorescence polarization was measured on an Ultra plate reader (Tecan) at excitation and emission wavelengths of 485 and 530 nm, respectively. The e...More data for this Ligand-Target Pair
BDBM32602(1-aza-2-oxobicyclo[5.3.0]decane scaffold, 28a)IC50: 240nMAssay Description:Fluorescence polarization was measured on an Ultra plate reader (Tecan) at excitation and emission wavelengths of 485 and 530 nm, respectively. The e...More data for this Ligand-Target Pair
BDBM26205((3S,6S,7R,9aS)-6-[(2S)-2-aminobutanamido]-7-(2-ami...)
IC50: 250nMpH: 7.5 T: 2°CAssay Description:Fluorescence polarization was measured on an Ultra plate reader (Tecan) at excitation and emission wavelengths of 485 and 530 nm, respectively. The e...More data for this Ligand-Target Pair
BDBM32595(1-aza-2-oxobicyclo[5.3.0]decane scaffold, 22c | 1-...)
IC50: 260nMpH: 7.5 T: 2°CAssay Description:Fluorescence polarization was measured on an Ultra plate reader (Tecan) at excitation and emission wavelengths of 485 and 530 nm, respectively. The e...More data for this Ligand-Target Pair
BDBM32606(1-aza-2-oxobicyclo[5.3.0]decane scaffold, 34a)
IC50: 280nMAssay Description:Fluorescence polarization was measured on an Ultra plate reader (Tecan) at excitation and emission wavelengths of 485 and 530 nm, respectively. The e...More data for this Ligand-Target Pair
BDBM32589(1-aza-2-oxobicyclo[5.3.0]decane scaffold, 18b | 1-...)
IC50: 320nMpH: 7.5 T: 2°CAssay Description:Fluorescence polarization was measured on an Ultra plate reader (Tecan) at excitation and emission wavelengths of 485 and 530 nm, respectively. The e...More data for this Ligand-Target Pair
BDBM32604(1-aza-2-oxobicyclo[5.3.0]decane scaffold, 31a)
IC50: 320nMpH: 7.5 T: 2°CAssay Description:Fluorescence polarization was measured on an Ultra plate reader (Tecan) at excitation and emission wavelengths of 485 and 530 nm, respectively. The e...More data for this Ligand-Target Pair
BDBM32594(1-aza-2-oxobicyclo[5.3.0]decane scaffold, 22b)
IC50: 330nMpH: 7.5 T: 2°CAssay Description:Fluorescence polarization was measured on an Ultra plate reader (Tecan) at excitation and emission wavelengths of 485 and 530 nm, respectively. The e...More data for this Ligand-Target Pair
BDBM32602(1-aza-2-oxobicyclo[5.3.0]decane scaffold, 28a)
IC50: 340nMpH: 7.5 T: 2°CAssay Description:Fluorescence polarization was measured on an Ultra plate reader (Tecan) at excitation and emission wavelengths of 485 and 530 nm, respectively. The e...More data for this Ligand-Target Pair
BDBM13211((3S,6S,9aS)-6-[(2S)-2-aminobutanamido]-N-(diphenyl...)
IC50: 360nMAssay Description:Fluorescence polarization was measured on an Ultra plate reader (Tecan) at excitation and emission wavelengths of 485 and 530 nm, respectively. The e...More data for this Ligand-Target Pair
BDBM32592(1-aza-2-oxobicyclo[5.3.0]decane scaffold, 20c)
IC50: 370nMpH: 7.5 T: 2°CAssay Description:Fluorescence polarization was measured on an Ultra plate reader (Tecan) at excitation and emission wavelengths of 485 and 530 nm, respectively. The e...More data for this Ligand-Target Pair
BDBM13212((3S,6S,9aS)-N-(diphenylmethyl)-6-[(2S)-2-(methylam...)
IC50: 420nMAssay Description:Fluorescence polarization was measured on an Ultra plate reader (Tecan) at excitation and emission wavelengths of 485 and 530 nm, respectively. The e...More data for this Ligand-Target Pair
BDBM32593(1-aza-2-oxobicyclo[5.3.0]decane scaffold, 22a)
IC50: 430nMpH: 7.5 T: 2°CAssay Description:Fluorescence polarization was measured on an Ultra plate reader (Tecan) at excitation and emission wavelengths of 485 and 530 nm, respectively. The e...More data for this Ligand-Target Pair
BDBM32591(1-aza-2-oxobicyclo[5.3.0]decane scaffold, 20b)
IC50: 440nMpH: 7.5 T: 2°CAssay Description:Fluorescence polarization was measured on an Ultra plate reader (Tecan) at excitation and emission wavelengths of 485 and 530 nm, respectively. The e...More data for this Ligand-Target Pair
BDBM32590(1-aza-2-oxobicyclo[5.3.0]decane scaffold, 20a)
IC50: 650nMpH: 7.5 T: 2°CAssay Description:Fluorescence polarization was measured on an Ultra plate reader (Tecan) at excitation and emission wavelengths of 485 and 530 nm, respectively. The e...More data for this Ligand-Target Pair
BDBM26204((3S,6S,7R,9aS)-6-[(2S)-2-aminobutanamido]-7-(amino...)
IC50: 970nMpH: 7.5 T: 2°CAssay Description:Fluorescence polarization was measured on an Ultra plate reader (Tecan) at excitation and emission wavelengths of 485 and 530 nm, respectively. The e...More data for this Ligand-Target Pair
BDBM44282((2S)-1-[(2R)-2-[[(2S)-2-amino-1-oxopropyl]amino]-2...)
BDBM44282((2S)-1-[(2R)-2-[[(2S)-2-amino-1-oxopropyl]amino]-2...)
BDBM44360(1-[2-cyclohexyl-2-[2-(methylamino)propanoylamino]e...)IC50: 9.30E+3nMAssay Description:Data Source: Sanford-Burnham Center for Chemical Genomics (SBCCG) Source Affiliation: Sanford-Burnham Medical Research Institute (SBMRI, San Diego, C...More data for this Ligand-Target Pair
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