Compile Data Set for Download or QSAR
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 6 hits in this display   

TargetRenin(Rattus norvegicus)
Massachusetts General Hospital

Curated by ChEMBL
LigandPNGBDBM50022021(1-(2-Acetylamino-3-phenyl-propionyl)-pyrrolidine-2...)
Affinity DataIC50:  42nMAssay Description:Inhibitory activity against rat plasma renin in vitro.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRenin(Rattus norvegicus)
Massachusetts General Hospital

Curated by ChEMBL
LigandPNGBDBM50022015(1-(2-Acetylamino-3-naphthalen-1-yl-propionyl)-pyrr...)
Affinity DataIC50:  50nMAssay Description:Inhibitory activity against rat plasma renin in vitro.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRenin(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50279761(3-Hydroxy-4-[2-(3-hydroxy-6-methyl-4-{2-[2-(3-meth...)
Affinity DataIC50:  190nMAssay Description:In vitro inhibitory activity against human plasma reninMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRenin(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50022994(CHEMBL286316 | Pro-Phe-Phe-Statine-Ile-Phe-NH2)
Affinity DataIC50:  430nMAssay Description:Inhibitory activity against human plasma reninMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-secretase 1/2(Homo sapiens (Human))
Affymax Research Institute

Curated by ChEMBL
LigandPNGBDBM50470133(CHEMBL277046)
Affinity DataIC50:  1.40E+3nMAssay Description:Inhibitory activity against aspartyl proteaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetRenin(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50022975(CHEMBL23991 | Phe-Statine-Ile-Phe-NH2)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibitory activity against human plasma reninMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed