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Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
8
hits in this display
Target
Platelet-activating factor receptor
(Homo sapiens (Human))
Broad Institute Of Mit And Harvard
Curated by
ChEMBL
Ligand
BDBM85035
(CAS_65154-06-5 | PAF | bloodplatelet-activatingfac...)
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Affinity Data
Ki: 0.150nM
Assay Description:
Displacement of [3H]PAF from platelet activating factor receptor in human platelets after 3 hrs
More data for this Ligand-Target Pair
Target Info
PDB
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KEGG
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antibodypedia
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Target
Beta-arrestin-1
(RABBIT)
Janssen Research Foundation
Curated by
PDSP K
i
Database
Ligand
BDBM85035
(CAS_65154-06-5 | PAF | bloodplatelet-activatingfac...)
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Affinity Data
Ki: 0.550nM
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
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Target
Nuclear receptor subfamily 5 group A member 2
(Homo sapiens (Human))
Emory University
Curated by
ChEMBL
Ligand
BDBM50467998
(CHEMBL4288877)
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Affinity Data
Ki: 81nM
Assay Description:
Displacement of 6N-FAM from human LRH1 LBD (299 to 541 residues) expressed in Escherichia coli BL21 pLysS by competitive binding based fluorescence p...
More data for this Ligand-Target Pair
Target Info
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MMDB
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KEGG
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antibodypedia
GoogleScholar
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Target
Steroidogenic factor 1
(Homo sapiens (Human))
Emory University
Curated by
ChEMBL
Ligand
BDBM50467998
(CHEMBL4288877)
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Affinity Data
Ki: 850nM
Assay Description:
Displacement of 6N-FAM from SF1 LBD (218 to 461 residues) (unknown origin) expressed in Escherichia coli BL21 pLysS by competitive binding based fluo...
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Target Info
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KEGG
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Target
Platelet-activating factor receptor
(Homo sapiens (Human))
Broad Institute Of Mit And Harvard
Curated by
ChEMBL
Ligand
BDBM85035
(CAS_65154-06-5 | PAF | bloodplatelet-activatingfac...)
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Copy InChI
Affinity Data
IC50: 0.280nM
Assay Description:
Displacement of [3H]PAF from platelet activating factor receptor in human platelets after 3 hrs
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
Purchase
ChEBI
DrugBank
KEGG
PC cid
PC sid
PDB
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In Depth
Details
Article
PubMed
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Target
Bile salt export pump
(Homo sapiens (Human))
Astrazeneca
Curated by
ChEMBL
Ligand
BDBM50238366
(CHEMBL4081726)
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Affinity Data
IC50: <1.60E+4nM
Assay Description:
Inhibition of human BSEP expressed in baculovirus transfected fall armyworm Sf21 cell membranes vesicles assessed as reduction in ATP-dependent [3H]-...
More data for this Ligand-Target Pair
Target Info
PDB
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UniProtKB/SwissProt
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CHEMBL
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In Depth
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Article
PubMed
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Target
Nuclear receptor subfamily 5 group A member 2
(Homo sapiens (Human))
Emory University
Curated by
ChEMBL
Ligand
BDBM50467998
(CHEMBL4288877)
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Affinity Data
EC50: >1.00E+5nM
Assay Description:
Agonist activity at recombinant full length human LRH1 expressed in HeLa cells after 24 hrs by dual-glo luciferase reporter gene assay
More data for this Ligand-Target Pair
Target Info
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Target
Fatty acid-binding protein, heart
(Homo sapiens (Human))
Osaka University
Curated by
ChEMBL
Ligand
BDBM50448440
(CHEMBL1235508)
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Affinity Data
Kd: 3.60nM
Assay Description:
Binding affinity to human FABP3 expressed in Escherichia coli BL21 (DE3) at 60 uM by surface plasmon resonance analysis
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
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antibodypedia
GoogleScholar
Ligand Info
CHEMBL
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In Depth
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Article
PubMed
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