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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 8 hits in this display   

TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Broad Institute Of Mit And Harvard

Curated by ChEMBL
LigandPNGBDBM85035(CAS_65154-06-5 | PAF | bloodplatelet-activatingfac...)
Affinity DataKi:  0.150nMAssay Description:Displacement of [3H]PAF from platelet activating factor receptor in human platelets after 3 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-arrestin-1(RABBIT)
Janssen Research Foundation

Curated by PDSP Ki Database
LigandPNGBDBM85035(CAS_65154-06-5 | PAF | bloodplatelet-activatingfac...)
Affinity DataKi:  0.550nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor subfamily 5 group A member 2(Homo sapiens (Human))
Emory University

Curated by ChEMBL
LigandPNGBDBM50467998(CHEMBL4288877)
Affinity DataKi:  81nMAssay Description:Displacement of 6N-FAM from human LRH1 LBD (299 to 541 residues) expressed in Escherichia coli BL21 pLysS by competitive binding based fluorescence p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteroidogenic factor 1(Homo sapiens (Human))
Emory University

Curated by ChEMBL
LigandPNGBDBM50467998(CHEMBL4288877)
Affinity DataKi:  850nMAssay Description:Displacement of 6N-FAM from SF1 LBD (218 to 461 residues) (unknown origin) expressed in Escherichia coli BL21 pLysS by competitive binding based fluo...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Broad Institute Of Mit And Harvard

Curated by ChEMBL
LigandPNGBDBM85035(CAS_65154-06-5 | PAF | bloodplatelet-activatingfac...)
Affinity DataIC50:  0.280nMAssay Description:Displacement of [3H]PAF from platelet activating factor receptor in human platelets after 3 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBile salt export pump(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50238366(CHEMBL4081726)
Affinity DataIC50: <1.60E+4nMAssay Description:Inhibition of human BSEP expressed in baculovirus transfected fall armyworm Sf21 cell membranes vesicles assessed as reduction in ATP-dependent [3H]-...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor subfamily 5 group A member 2(Homo sapiens (Human))
Emory University

Curated by ChEMBL
LigandPNGBDBM50467998(CHEMBL4288877)
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at recombinant full length human LRH1 expressed in HeLa cells after 24 hrs by dual-glo luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty acid-binding protein, heart(Homo sapiens (Human))
Osaka University

Curated by ChEMBL
LigandPNGBDBM50448440(CHEMBL1235508)
Affinity DataKd:  3.60nMAssay Description:Binding affinity to human FABP3 expressed in Escherichia coli BL21 (DE3) at 60 uM by surface plasmon resonance analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed