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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 5 hits in this display   

TargetBeta-mannosidase(Bacteroides thetaiotaomicron)
The Medical School, Newcastle University

LigandPNGBDBM36391(5-Hydroxymethyl-7-isopropoxy-6-oxa-bicyclo[3.2.2]n...)
Affinity DataKi: >4.00E+8nM ΔG°: >-2.36kJ/molepH: 5.6 T: 2°CAssay Description:Putative mannosidase assay using wild-type protein Btman2A. Enzyme inhibition assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRibonuclease HI(Escherichia coli (strain K12))
Chungnam National University

Curated by ChEMBL
LigandPNGBDBM50343047(CHEMBL1770694 | iso-dihydrodendranthemoside A)
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibition of Escherichia coli recombinant ribonuclease H after 30 mins by FRET quenching assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRibonuclease HI(Escherichia coli (strain K12))
Chungnam National University

Curated by ChEMBL
LigandPNGBDBM50343045((1R,2R,4S)-p-menthane-1,2,8-triol-1-O-beta-D-gluco...)
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibition of Escherichia coli recombinant ribonuclease H after 30 mins by FRET quenching assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRibonuclease HI(Escherichia coli (strain K12))
Chungnam National University

Curated by ChEMBL
LigandPNGBDBM50343045((1R,2R,4S)-p-menthane-1,2,8-triol-1-O-beta-D-gluco...)
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibition of Escherichia coli recombinant ribonuclease H after 30 mins by FRET quenching assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRibonuclease HI(Escherichia coli (strain K12))
Chungnam National University

Curated by ChEMBL
LigandPNGBDBM50343047(CHEMBL1770694 | iso-dihydrodendranthemoside A)
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibition of Escherichia coli recombinant ribonuclease H after 30 mins by FRET quenching assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed