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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
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kcal/mol
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Found
1
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Target
Beta-secretase 1 [22-454]
(Homo sapiens (Human))
Sunesis
Ligand
BDBM16292
(3-N-[(2S,3S,5R)-3-amino-5-[(4-fluorophenyl)carbamo...)
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Affinity Data
Ki: 26nM ΔG°: -42.9kJ/mole
pH: 4.5 T: 2°C
Assay Description:
Compounds were tested for their ability to inhibit BACE-1 hydrolysis of the internally quenched fluorescent substrate FS-2. Reactions were initiated ...
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