Compile Data Set for Download or QSAR
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 3 hits in this display   

TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50386475(CHEMBL2047879)
Affinity DataIC50:  22nMAssay Description:Inhibition of wild type B-raf in presence of 1 mM ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAF proto-oncogene serine/threonine-protein kinase(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50386475(CHEMBL2047879)
Affinity DataIC50:  73nMAssay Description:Inhibition of wild type C-raf in presence of 1 mM ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2C9(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50386475(CHEMBL2047879)
Affinity DataIC50:  9.00E+3nMAssay Description:Inhibition of CYP2C9More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed