Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 24 hits in this display
BDBM29755(hydroxyethylamine derivative, 4)
BDBM50231685(3-(ethylamino)-N-((2S,3R)-3-hydroxy-1-phenyl-4-(2-...)
BDBM29756(CHEMBL403429 | hydroxyethylamine derivative, 6)
BDBM29756(CHEMBL403429 | hydroxyethylamine derivative, 6)
IC50: 49nMpH: 4.5 T: 2°CAssay Description:Enzyme activity and inhibition were assayed using a fluorescent FAM-[SEVNLDAEFK]-TAMRA substrate. Control reactions with no enzyme were included in e...More data for this Ligand-Target Pair
BDBM29757(hydroxyethylamine derivative, 7)
IC50: 63nMpH: 4.5 T: 2°CAssay Description:Enzyme activity and inhibition were assayed using a fluorescent FAM-[SEVNLDAEFK]-TAMRA substrate. Control reactions with no enzyme were included in e...More data for this Ligand-Target Pair
BDBM29756(CHEMBL403429 | hydroxyethylamine derivative, 6)
BDBM29756(CHEMBL403429 | hydroxyethylamine derivative, 6)
BDBM50231697(3-(ethylamino)-N-((2S,3R)-3-hydroxy-4-(phenethylam...)
BDBM50231685(3-(ethylamino)-N-((2S,3R)-3-hydroxy-1-phenyl-4-(2-...)
BDBM50231699(CHEMBL252860 | N-((2S,3R)-4-(benzylamino)-3-hydrox...)
BDBM50231685(3-(ethylamino)-N-((2S,3R)-3-hydroxy-1-phenyl-4-(2-...)
BDBM50231697(3-(ethylamino)-N-((2S,3R)-3-hydroxy-4-(phenethylam...)
BDBM50231675(CHEMBL402122 | N-((2S,3R)-4-(cyclopentylamino)-3-h...)
BDBM50231697(3-(ethylamino)-N-((2S,3R)-3-hydroxy-4-(phenethylam...)
BDBM29756(CHEMBL403429 | hydroxyethylamine derivative, 6)
BDBM29757(hydroxyethylamine derivative, 7)
BDBM29756(CHEMBL403429 | hydroxyethylamine derivative, 6)
IC50: 4.49E+3nMpH: 4.5 T: 2°CAssay Description:Enzyme activity and inhibition were assayed using a fluorescent FAM-[SEVNLDAEFK]-TAMRA substrate. Control reactions with no enzyme were included in e...More data for this Ligand-Target Pair
BDBM29756(CHEMBL403429 | hydroxyethylamine derivative, 6)
BDBM29756(CHEMBL403429 | hydroxyethylamine derivative, 6)
IC50: 6.58E+3nMAssay Description:Enzyme activity and inhibition were assayed using a fluorescent FAM-[SEVNLDAEFK]-TAMRA substrate. Control reactions with no enzyme were included in e...More data for this Ligand-Target Pair
BDBM29757(hydroxyethylamine derivative, 7)
IC50: 9.12E+3nMpH: 4.5 T: 2°CAssay Description:Enzyme activity and inhibition were assayed using a fluorescent FAM-[SEVNLDAEFK]-TAMRA substrate. Control reactions with no enzyme were included in e...More data for this Ligand-Target Pair
BDBM50231675(CHEMBL402122 | N-((2S,3R)-4-(cyclopentylamino)-3-h...)
BDBM50231699(CHEMBL252860 | N-((2S,3R)-4-(benzylamino)-3-hydrox...)
BDBM50231675(CHEMBL402122 | N-((2S,3R)-4-(cyclopentylamino)-3-h...)
BDBM50231699(CHEMBL252860 | N-((2S,3R)-4-(benzylamino)-3-hydrox...)