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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 6 hits in this display   

TargetHeat shock protein HSP 90-alpha(Homo sapiens (Human))
Fermentas

Curated by ChEMBL
LigandPNGBDBM50276570(4-chloro-6-(5-(4-methoxyphenyl)-1,2,3-thiadiazol-4...)
Affinity DataKd:  13nMAssay Description:Binding affinity to human full length Histidine6-tagged Hsp90alpha expressed in Escherichia coli BL21 DE3 by ITCMore data for this Ligand-Target Pair
TargetHeat shock protein HSP 90-alpha(Homo sapiens (Human))
Fermentas

Curated by ChEMBL
LigandPNGBDBM50276571(4-(5-chloro-2,4-dihydroxyphenyl)-5-(4-ethoxyphenyl...)
Affinity DataKd:  6.30nMAssay Description:Binding affinity to human full length Histidine6-tagged Hsp90alpha expressed in Escherichia coli BL21 DE3 by ITCMore data for this Ligand-Target Pair
TargetHeat shock protein HSP 90-alpha(Homo sapiens (Human))
Fermentas

Curated by ChEMBL
LigandPNGBDBM50276629(2-chloro-4-(5-(4-ethoxyphenyl)-1,2,3-thiadiazol-4-...)
Affinity DataKd: >2.00E+4nMAssay Description:Binding affinity to human full length Histidine6-tagged Hsp90alpha expressed in Escherichia coli BL21 DE3 by ITCMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHeat shock protein HSP 90-alpha(Homo sapiens (Human))
Fermentas

Curated by ChEMBL
LigandPNGBDBM50276573(4-chloro-6-(5-(3,4-dimethoxyphenyl)-1,2,3-thiadiaz...)
Affinity DataKd:  34nMAssay Description:Binding affinity to human full length Histidine6-tagged Hsp90alpha expressed in Escherichia coli BL21 DE3 by ITCMore data for this Ligand-Target Pair
TargetHeat shock protein HSP 90-alpha(Homo sapiens (Human))
Fermentas

Curated by ChEMBL
LigandPNGBDBM50276628(2,4-dichloro-6-(5-(4-methoxyphenyl)-1,2,3-thiadiaz...)
Affinity DataKd: >2.00E+4nMAssay Description:Binding affinity to human full length Histidine6-tagged Hsp90alpha expressed in Escherichia coli BL21 DE3 by ITCMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHeat shock protein HSP 90-alpha(Homo sapiens (Human))
Fermentas

Curated by ChEMBL
LigandPNGBDBM50276572(4-chloro-6-(5-p-tolyl-1,2,3-thiadiazol-4-yl)benzen...)
Affinity DataKd:  17nMAssay Description:Binding affinity to human full length Histidine6-tagged Hsp90alpha expressed in Escherichia coli BL21 DE3 by ITCMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed